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Небесная энциклопедия

Космические корабли и станции, автоматические КА и методы их проектирования, бортовые комплексы управления, системы и средства жизнеобеспечения, особенности технологии производства ракетно-космических систем

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Мониторинг СМИ

Мониторинг СМИ и социальных сетей. Сканирование интернета, новостных сайтов, специализированных контентных площадок на базе мессенджеров. Гибкие настройки фильтров и первоначальных источников.

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Форма поиска

Поддерживает ввод нескольких поисковых фраз (по одной на строку). При поиске обеспечивает поддержку морфологии русского и английского языка
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Применить Всего найдено 507. Отображено 102.
24-01-2003 дата публикации

RAILWAY VEHICLE COMPRISING a FEEDING ATTACHMENT WHILE RUNNING

Номер: FR0002769763B1
Автор: BRUGMANN, DOBROS, KERSTIN
Принадлежит: DAIMLERCHRYSLER RAIL SYSTEMS GMBH

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15-10-1983 дата публикации

SPINNING DISK

Номер: BG0000034549A1
Принадлежит:

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23-02-2012 дата публикации

SILOXANE POLYMER CONTAINING TETHERED FLUOROQUINOLONE

Номер: US20120046313A1
Принадлежит:

A polymer that is a polysiloxane polymer has fluoroquinolone antibiotic groups, or pharmaceutically acceptable salts thereof, attached via linkers. The linkers may be hydrolytically labile thereby providing a manner of releasing the fluoroquinolone antibiotic from the polymer. 1. A polymer formed by {'br': None, 'sup': 1', '2', '3', '4', '5', '6', '7', '8', '9', '10', '11, 'sub': y', 'x', 'z, 'RRRSiO—(SiRR—O)(SiRH—O)(SiRR—O)SiRRR'}, '(a) reaction of a polyhydrosiloxane of general formula'}with a reactive compound to provide a functionalized polysiloxane, wherein the reactive compound comprises (1) a first reactive group, which is capable of reacting with an Si—H group, at one end, and (2) a second reactive group, which is capable of reacting with a fluoroquinolone antibiotic, at its other end;(b) reaction of the functionalized polysiloxane with the fluoroquinolone antibiotic or a pharmaceutically acceptable salt thereof to provide a fluoroquinolone-functionalized polysiloxane;{'sup': 1', '2', '3', '4', '5', '6', '8', '9', '10', '11, 'sub': 1', '20, 'wherein R, R, R, R, R, R, R, R, R, and Rare independently C-Calkyl, benzyl, tolyl, xylyl, or phenyl;'}{'sup': '7', 'sub': 1', '20, 'Ris a C-Calkyl, benzyl, tolyl, xylyl, phenyl, texturizing moiety, a cross-linkable group, or a combination thereof;'}x is 1 to 100;y is 0 to 100;z is 0 to 100;at least one of y and z is greater than 0; andthe polymer contains at least one fluoroquinolone group.2. The polymer of claim 1 , wherein the fluoroquinolone antibiotic is ofloxacin.3. The polymer of claim 1 , wherein the polyhydrosiloxane is selected from the group consisting of poly(methylhydro-co-dimethyl)siloxane claim 1 , polymethylhydrosiloxane claim 1 , polyethylhydrosiloxane claim 1 , polyphenyl-(dimethylhydro) siloxane claim 1 , methylhydrosiloxane-phenylmethylsiloxane copolymer claim 1 , methylhydrosiloxane-octylmethylsiloxane copolymer claim 1 , or blends of any two or more thereof.4. The polymer of claim 1 , wherein the ...

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07-06-2012 дата публикации

Electronic Sales With Decreasing Price

Номер: US20120143711A1
Принадлежит:

A pricing method, having multiple buyers collaborating virtually to achieve a declining price schedule for a given product or service. The method invites buyers to commit at a certain price, which may or may not be the price they ultimately pay. The price may or may not decline as more buyers commit. All buyers pay the same (lowest) price, at the end of the finite sale period. 1. A computer-implemented method for making goods or services available to buyers , the method comprising:making available for purchase, by a computer server system at an on-line service and to a plurality of potential buyers, one or more goods or services in an on-line electronic marketplace, including by pricing the goods or services at an initial price;receiving requests to purchase the one or more goods or services from a plurality of actual buyers from among the plurality of potential buyers;determining at the end of a predetermined time period an actual price for the goods or service based on a number of actual buyers who request to purchase the one or more goods or services, andautomatically billing the plurality of actual buyers for the one or more goods or services at the determined actual price and causing the one or more goods or services to be made available to the plurality of actual buyers.2. The computer-implemented method of claim 1 , further comprising posting or announcing an initial price for the one or more goods or services to the plurality of potential buyers before receiving requests to purchase from the plurality of potential buyers claim 1 , the initial price serving as a maximum price any buyer will pay for the one or more goods or services.3. The computer-implemented method of claim 2 , further comprising periodically updating and posting a real-time price for the one or more goods or services to be shown to the plurality of potential buyers after initially making the one or more goods or services available for purchase claim 2 , the real-time price falling from the ...

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13-09-2012 дата публикации

PHASE CHANGE INKS

Номер: US20120227622A1
Принадлежит: XEROX CORPORATION

An ink composition that includes stearyl stearamide, N,N′-ethylene bisoleamide, at least one wax, at least one antioxidant, and at least one solvent dye colorant is useful as a phase change ink. 1. An ink composition comprising:stearyl stearamide,N,N′-ethylene bisoleamide,at least one wax,at least one antioxidant, andat least one solvent dye colorant.2. The ink composition according to claim 1 , wherein the at least one wax comprises a mixture of at least one Fischer-Tropsch wax and at least one fatty acid ester wax.5. The ink composition according to claim 1 , wherein the at least one solvent dye colorant is solvent black.6. The ink composition according to claim 2 , wherein the at least one solvent dye colorant is solvent black.7. The ink composition according to claim 3 , wherein the at least one solvent dye colorant is solvent black.8. The ink composition according to claim 1 , wherein the at least one solvent dye colorant is solvent yellow.9. The ink composition according to claim 2 , wherein the at least one solvent dye colorant is solvent yellow.10. The ink composition according to claim 3 , wherein the at least one solvent dye colorant is solvent yellow.11. A phase change ink composition comprising an ink vehicle and a colorant claim 3 , wherein the phase change ink is solid at temperatures of from about 20° C. to about 27° C. and exhibits a viscosity of from about 1 to about 20 centipoise (cP) at an elevated temperature at which the phase change ink is to be jetted claim 3 , wherein the ink vehicle comprisesstearyl stearamide,N,N′-ethylene bisoleamide,at least one wax, andat least one antioxidant, and wherein the colorant comprises at least one solvent dye colorant.12. The phase change ink composition according to claim 11 , wherein the at least one wax comprises a mixture of at least one Fischer-Tropsch wax and at least one fatty acid ester wax.15. The phase change ink composition according to claim 11 , wherein the at least one solvent dye colorant is ...

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11-10-2012 дата публикации

Method for mac addresses withdrawal in telecommunication networks

Номер: US20120257539A1
Принадлежит: ECI Telecom Ltd

A rationalized MAC withdrawal method for a multi-domain communication network, where at least one access node interconnects a remote node with two or more access networks. The method allows flushing, both in the access nodes and in the remote node, only MAC addresses being related to a specific access networks where a topological change has taken place, without affecting other access networks connected to the same access node.

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02-01-2014 дата публикации

ACTIVE COMPOUND COMBINATIONS

Номер: US20140005049A1
Принадлежит:

The invention relates to active compound combinations, in particular within a composition, which comprises (A) an amidine compound of formula (I) and a further fungicidally (B-1), insecticidally (B-2) active or plant growth regulating compound (B-3). Moreover, the invention relates to a method for curatively or preventively controlling the phytopathogenic fungi of plants or reducing the mycotoxin contamination of plant or plant parts, to the use of a combination according to the invention for the treatment of seed, to a method for protecting a seed and not at least to the treated seed. 3. The composition according to wherein the at least one further active compound (B-I) is selected from the group consisting of Cyproconazole claim 1 , Epoxiconazole claim 1 , Flusilazole claim 1 , Fluquinconazole Ipconazole claim 1 , Propiconazole claim 1 , Metconazole claim 1 , Tebuconazole claim 1 , Triadimenol claim 1 , Azoxystrobin claim 1 , Fluoxastrobin claim 1 , Kresoxim-methyl claim 1 , Picoxystrobin claim 1 , Pyraclostrobin claim 1 , Boscalid claim 1 , Chlorothalonil claim 1 , Cyprodinil claim 1 , Fludioxonil claim 1 , Fluopyram claim 1 , Thiophanat-methyl claim 1 , Penflufen claim 1 , Isopyrazam claim 1 , Sedaxane claim 1 , Myclobutonil claim 1 , Prochloraz claim 1 , Spiroxamine claim 1 , N-(3′ claim 1 ,4′-dichloro-5-fluoro[1 claim 1 ,1′-biphenyl]-2-yl)-3-(difluoromethyl)-1-methyl-1H-pyrazole-4-carboxamide claim 1 , Ametoctradin claim 1 , 5-Chlor-6-(2 claim 1 ,4 claim 1 ,6-trifluorphenyl)-7-(4-methylpiperidin-1-yl)[1 claim 1 ,2 claim 1 ,4]triazolo[1 claim 1 ,5-a]pyrimidin claim 1 , 1-methyl-N-{2-[1′-methyl-1 claim 1 ,1′-bi(cyclopropyl)-2-yl]phenyl}-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide claim 1 , N-{2-[1 claim 1 ,1′-bi(cyclopropyl)-2-yl]phenyl}-1-methyl-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide claim 1 , 1-methyl-N-{2-[1′-methyl-1 claim 1 ,1′-bi(cyclopropyl)-2-yl]phenyl}-3-(difluoromethyl)-1H-pyrazole-4-carboxamide claim 1 , and N-{2-[1 claim 1 ,1′-bi(cyclopropyl ...

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06-01-2022 дата публикации

NOVEL HETEROARYL-TRIAZOLE AND HETEROARYL-TETRAZOLE COMPOUNDS AS PESTICIDES

Номер: US20220002268A1
Принадлежит:

The present invention relates to novel heteroaryl-triazole and heteroaryl-tetrazole compounds of the general formula (I), in which the structural elements Y, Q, Q, R, R, R, R, Rand Rhave the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals. 2. Compound according to claim 1 , in whichX is O or S;{'sup': 1', '2', '5', '1', '2, 'Qand Qare independently CRor N, provided at least one of Qand Qis N;'}{'sub': '2', 'Y is a direct bond or CH;'}{'sup': '1', 'sub': 1', '6', '2', '2', '3', '3', '1', '6', '2', '6', '2', '6', '2', '6', '2', '6', '3', '4', '1', '2', '3', '4', '2', '1', '3, 'Ris hydrogen; C-Calkyl optionally substituted with one substituent selected from the group consisting of CN, CONH, COOH, NOand —Si(CH); C-Chaloalkyl; C-Calkenyl; C-Chaloalkenyl; C-Calkynyl; C-Chaloalkynyl; C-Ccycloalkyl-C-Calkyl- wherein the C-Ccycloalkyl is optionally substituted with one or two halogen atoms; oxetan-3-yl-CH—; or benzyl optionally substituted with halogen or C-Chaloalkyl;'}{'sup': '2', 'sub': 1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '2', '5', '2', '2, 'Ris phenyl, pyridine, pyrimidine, pyrazine or pyridazine, wherein the phenyl, pyridine, pyrimidine, pyrazine or pyridazine is optionally substituted with one to three substituents, provided the substituent(s) are not on either carbon adjacent to the carbon bonded to the —C(X)— group, each independently selected from the group consisting of C-Calkyl, C-Chaloalkyl, C-Chaloalkylthio, C-Calkoxy, C-Chaloalkoxy, halogen, NO, SF, CN, CONH, COOH and C(S)NH;'}{'sup': 3a', '3b, 'claim-text': [{'sub': 1', '6', '2', '2', '2', '3', '6', '1', '3', '1', '4', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '4', '1', '4', '2', '1', '4', '1', '4', '1', '4', '2', '1', '4', '1', '4', '1', '4', '2, 'C-Calkyl wherein ...

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07-01-2016 дата публикации

NOVEL HALOGEN-SUBSTITUTED COMPOUNDS

Номер: US20160002208A1
Принадлежит:

The invention relates inter alia to halogen-substituted compounds of the general formula (I) 7. A compound of formula (I) capable of being used for controlling insects , arachnids and nematodes.8. Pharmaceutical composition comprising at least one compound according to .9. Compound according to that comprises a medicament.10. A compound according to capable of being used for preparing a pharmaceutical composition for controlling parasites on animals.11. Process for preparing crop protection compositions comprising mixing a compound according to and one or more customary extenders and/or surfactants.12. Method for controlling pests claim 1 , comprising allowing a compound according to to act on the pests and/or a habitat thereof.13. A compound according to capable of being used for protecting propagation material of a plant. The present application relates to novel halogen-substituted compounds, to processes for their preparation and to their use for controlling animal pests, in particular arthropods and especially insects, arachnids and nematodes.It is known that certain halogen-substituted compounds have herbicidal action (cf. J. Org. Chem. 1997, 62(17), 5908-5919, J. Heterocycl. Chem. 1998, 35(6), 1493-1499, WO 2004/035545, WO 2004/106324, US 2006/069132, WO 2008/029084).Furthermore, it is known that certain halogen-substituted compounds are insecticidally active (EP1911751, WO2012-069366, WO2012-080376 & WO2012-107434).In addition, it is known that certain halogen-substituted compounds have FAAH-inhibitory activities (WO 2009/151991).Modern crop protection compositions have to meet many demands, for example in relation to efficacy, persistence and spectrum of their action and possible use. Questions of toxicity, the combinability with other active compounds or formulation auxiliaries play a role, as well as the question of the expense that the synthesis of an active compound requires. Furthermore, resistances may occur. For all these reasons, the search for novel ...

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04-01-2018 дата публикации

2-(HET)ARYL-SUBSTITUTED FUSED BICYCLIC HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20180002345A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. Compound of formula (I) according to wherein{'sup': 1', '+', '−', '4, 'Arepresents nitrogen, ═N—O or ═C—R,'}{'sup': 2', '5, 'Arepresents —N—R, oxygen or sulphur,'}{'sup': '3', 'Arepresents oxygen,'}{'sup': 4', '+', '−', '4, 'Arepresents nitrogen, ═N—O or ═C—R,'}{'sup': '1', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '3', '6', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Rrepresents (C-C)-alkyl, (C-C)-hydroxyalkyl, (C-C)-haloalkyl, (C-C)-cyanoalkyl, (C-C)-alkoxy-(C-C)-alkyl, (C-C)-haloalkoxy-(C-C)-alkyl, (C-C)-alkenyl, (C-C)-alkenyloxy-(C-C)-alkyl, (C-C)-haloalkenyloxy-(C-C)-alkyl, (C-C)-haloalkenyl, (C-C)-cyanoalkenyl, (C-C)-alkynyl, (C-C)-alkynyloxy-(C-C)-alkyl, (C-C)-haloalkynyloxy-(C-C)-alkyl, (C-C)-haloalkynyl, (C-C)-cyanoalkynyl, (C-C)-cycloalkyl, (C-C)-cycloalkyl-(C-C)-cycloalkyl, (C-C)-alkyl-(C-C)-cycloalkyl, halo-(C-C)-cycloalkyl, (C-C)-alkylamino, di-(C-C)-alkylamino, (C-C)-cycloalkylamino, (C-C)-alkylcarbonylamino, (C-C)-alkylthio-(C-C)-alkyl, (C-C)-haloalkylthio-(C-C)-alkyl, (C-C)-alkylsulphinyl-(C-C)-alkyl, (C-C)-haloalkylsulphinyl-(C-C)-alkyl, (C-C)-alkylsulphonyl-(C-C)-alkyl, (C-C)-alkylcarbonyl-(C-C)-alkyl, (C-C)-haloalkylcarbonyl-(C-C)-alkyl, (C-C)-alkylsulphonylamino,'}{'sub': 1', '4', '1', '4', '2', '4', '2', '4', '3', '6', '1', '4', '3', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'or represents (C-C)-alkyl, (C-C)-alkoxy, (C-C)-alkenyl, (C-C)-alkynyl, (C-C)cycloalkyl, each of which is optionally mono- or disubstituted by identical or different substituents from the group consisting of ...

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14-01-2016 дата публикации

ALKOXIMINO-SUBSTITUTED ANTHRANILIC ACID DIAMIDES AS PESTICIDES

Номер: US20160007603A1
Принадлежит:

The present invention relates to novel anthranilic acid diamide derivatives of the general formula (I) 2. The compound of formula (I) as claimed in claim 1 , wherein{'sup': 6', '7, 'A represents N(R)R,'}{'sub': 2', '4', '2', '4', '2', '4', '3', '4', '1', '4', '3', '4', '1', '4', '1', '4', '2', '4', '2', '4', '2', '4, 'G represents fluoromethyl, difluoromethyl, chlorodifluoromethyl, C-C-haloalkyl, C-C-haloalkenyl, C-C-haloalkynyl, C-C-halocycloalkyl, C-C-alkoxy, fluoromethoxy, fluoroethoxy, difluoroethoxy, tetrafluoroethoxy, chlorodifluoroethoxy, dichlorofluoroethoxy, C-C-haloalkoxy, C-C-haloalkoxy-C-C-alkyl, C-C-haloalkylthio, C-C-haloalkylsulfinyl, C-C-haloalkylsulfonyl or represents —W-Q,'}{'sup': '1', 'sub': 1', '6', '2', '6', '2', '6', '3', '6', '1', '6', '1', '6', '2', '6', '2', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Rrepresents hydrogen, C-C-alkyl, C-C-alkenyl, C-C-alkynyl, C-C-cycloalkyl, cyano(C-C-alkyl), C-C-haloalkyl, C-C-haloalkenyl, C-C-haloalkynyl, C-C-alkoxy-C-C-alkyl, C-C-alkylthio-C-C-alkyl, C-C-alkylsulfinyl-C-C-alkyl or C-C-alkylsulfonyl-C-C-alkyl,'}{'sup': '2', 'sub': 1', '4', '1', '4, 'Rrepresents hydrogen, C-C-alkyl, halogen, cyano, C-C-alkoxy,'}{'sup': '3', 'sub': 1', '6', '1', '4, 'Rrepresents hydrogen, C-C-alkyl, C-C-alkoxy, halogen, cyano or nitro,'}m represents 0 to 2,{'sup': '4', 'sub': 1', '4', '3', '6', '2', '4', '2', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Rrepresents C-C-alkyl, C-C-cycloalkyl, C-C-alkenyl, C-C-alkynyl, C-C-alkylsulfonyl, C-C-alkoxycarbonyl, C-C-alkylcarbonyl, aminocarbonyl, C-C-alkylaminocarbonyl which is optionally mono- or polysubstituted by identical or different substituents, where the substituents independently of one another may be selected from the group consisting of halogen, cyano, C-C-alkyl, C-C-alkoxy, C-C-alkylthio, C-C-alkylsulfinyl or C-C-alkylsulfonyl,'}{'sup': '5', 'sub': 1', '4', '1', '4', '1', '4', '1 ...

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14-01-2016 дата публикации

NOVEL HALOGEN-SUBSTITUTED COMPOUNDS

Номер: US20160007604A1
Принадлежит: Bayer Animal Health GmbH

The invention relates inter alia to halogen-substituted compounds of the general formula (II) 7. Use of compounds of the general formula (II) or the general formulae (IIa) to (IIh) according to for controlling insects claim 1 , arachnids and nematodes.8. Pharmaceutical compositions comprising at least one compound according to .9. Compounds according to for use as medicaments.10. Use of compounds according to for preparing pharmaceutical compositions for controlling parasites on animals.11. Process for preparing crop protection compositions comprising compounds according to and customary extenders and/or surfactants.12. Method for controlling pests claim 1 , characterized in that a compound according to is allowed to act on the pests and/or their habitat.13. Use of compounds according to for protecting the propagation material of plants. The present application relates to novel halogen-substituted compounds, to processes for their preparation and to their use for controlling animal pests, in particular arthropods and especially insects, arachnids and nematodes.It is known that certain halogen-substituted compounds have herbicidal action (cf. J. Org. Chem. 1997, 62(17), 5908-5919, J. Heterocycl. Chem. 1998, 35(6), 1493-1499, WO 2004/035545, WO 2004/106324, US 2006/069132, WO 2008/029084).Furthermore, it is known that certain halogen-substituted compounds are insecticidally active (EP1911751, WO2012-069366, WO2012-080376 & WO2012-107434).In addition, it is known that certain halogen-substituted compounds have FAAH-inhibitory activities (WO 2009/151991).Modern crop protection compositions have to meet many demands, for example in relation to efficacy, persistence and spectrum of their action and possible use. Questions of toxicity, the combinability with other active compounds or formulation auxiliaries play a role, as well as the question of the expense that the synthesis of an active compound requires. Furthermore, resistances may occur. For all these reasons, the ...

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10-01-2019 дата публикации

Method for Assisting During Execution of a Sequence of Cuttings in a Tree, and System for Assisting During Execution of a Sequence of Cuttings in a Tree

Номер: US20190008099A1
Принадлежит: Andreas Stihl AG and Co KG

A method assists during execution of a sequence of cuttings in a tree, wherein, during a cutting sequence, a first cut in the tree is followed by a second cut in the tree At least a part of an ideal course of the second cut depends on at least a part of a course of the first cut. The method includes the steps of: identifying at least the part of the course of the first cut in the tree; precalculating at least the part of the ideal course of the second cut in the tree based on the identified part of the course of the first cut; and outputting cutting information for executing the second cut based on the precalculated part of the ideal course of the second cut.

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21-01-2021 дата публикации

HETEROCYCLIC COMPOUNDS AS PESTICIDES

Номер: US20210017136A1
Принадлежит:

The present application relates to the use of heterocyclic compounds for controlling animal pests including arthropods, insects and nematodes, to novel heterocyclic compounds, to processes for their preparation and to intermediates for preparing the heterocyclic compounds. 1. 1-(2 ,6-difluorophenyl)-1H-pyrazole-3-amine.2. N-[1-[(2 ,6-difluorophenyl)-1H-pyrazol-3-yl]acetamide. This application is a divisional of U.S. patent application Ser. No. 16/536,902, filed 9 Aug. 2019, which is a divisional of U.S. patent application Ser. No. 15/645,814, filed 10 Jul. 2017 (now U.S. Pat. No. 10,435,374, issued 8 Oct. 2019), which is a continuation of U.S. patent application Ser. No. 14/432,501, filed 31 Mar. 2015 (now U.S. Pat. No. 9,802,899, issued 31 Oct. 2017), which is a § 371 National Stage Application of PCT/EP2013/070371, filed 30 Sep. 2013, which claims priority to EP 12186946.5, filed 2 Oct. 2012 and EP 13170565.9, filed 5 Jun. 2013, the contents of each are incorporated by reference herein in their entireties.The present application relates to the use of heterocyclic compounds for controlling animal pests including arthropods, insects and nematodes, to novel heterocyclic compounds, to processes for their preparation and to intermediates for preparing the heterocyclic compounds.The heterocyclic compounds of the formulae (W) and (W2) are known (cf. for the compounds of the formula (W) Registry Numbers 1189645-25-7, 1189474-83-6, 1193202-69-5, 1172407-07-6, 1185158-40-0, 1185036-12-7, 1170986-74-9, 1193179-17-7, 1189458-68-1, 1189956-23-7, 1189915-26-1, 1170047-96-7). A use of these compounds has not been described.Derivatives of pyrazole-4-carboxamides are known from JP 2010-202649. The compounds described therein have bactericidal action against plant-damaging bacteria. Intermediates for their preparation are described in JP2010-202648.Crop protection compositions, which also include pesticides, have to meet many demands, for example in relation to efficacy, ...

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21-01-2021 дата публикации

CONDENSED BICYCLIC HETEROCYCLIC DERIVATIVES AS PEST CONTROL AGENTS

Номер: US20210017193A1
Принадлежит:

The present invention relates to novel fused bicyclic heterocycle derivatives of formula (I) 2. The compound of formula (I) as claimed in claim 1 , wherein{'img': {'@id': 'CUSTOM-CHARACTER-00011', '@he': '4.91mm', '@wi': '6.35mm', '@file': 'US20210017193A1-20210121-P00001.TIF', '@alt': 'custom-character', '@img-content': 'character', '@img-format': 'tif'}, 'sub': 1', '4, 'in the case that both exclusively represent double bonds and Bto Bthus form an aromatic ring,'}{'sub': '1', 'Brepresents CH,'}{'sub': '2', 'sup': '12', 'Brepresents C(R),'}{'sub': '3', 'sup': '13', 'Brepresents C(R) and'}{'sub': '4', 'Brepresents CH and'}{'img': {'@id': 'CUSTOM-CHARACTER-00012', '@he': '4.91mm', '@wi': '6.35mm', '@file': 'US20210017193A1-20210121-P00001.TIF', '@alt': 'custom-character', '@img-content': 'character', '@img-format': 'tif'}, 'where in the case that both exclusively represent single bonds,'}{'sub': '1', 'sup': 11', '15, 'Brepresents C(R)(R),'}{'sub': '2', 'sup': 12', '16, 'Brepresents C(R)(R),'}{'sub': '3', 'sup': 13', '17, 'Brepresents C(R)(R) and'}{'sub': 4', '2, 'Brepresents CH,'}and furthermore{'sup': '1', 'sub': 1', '6', '1', '6', '2', '6', '2', '6', '2', '6', '2', '6', '3', '3', '1', '6', '3', '8', '3', '8', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6, 'Rrepresents (C-C)-alkyl, (C-C)-haloalkyl, (C-C)-alkenyl, (C-C)-haloalkenyl, (C-C)-alkynyl, (C-C)-haloalkynyl, (C-C)-cycloalkyl, (C-C)-alkyl-(C-C)-cycloalkyl, halo-(C-C)-cycloalkyl, (C-C)-alkylthio-(C-C)-alkyl, (C-C)-alkylsulfinyl-(C-C)-alkyl or (C-C)-alkylsulfonyl-(C-C)-alkyl,'}{'sup': 11', '12', '13', '15', '16', '17, 'sub': 3', '6', '3', '8', '3', '8', '1', '6', '3', '8', '3', '8', '3', '8', '1', '6', '1', '6', '3', '8', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '2', '6', '2', '6', '2', '6', '2', '6', '2', '6', '2', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1 ...

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24-01-2019 дата публикации

HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20190021329A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. Compound of formula (I) according to in which{'sup': 1', '+', '−', '4, 'Arepresents nitrogen, ═N(O)— or ═C(R)—,'}{'sup': '1', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '3', '6', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'claim-text': {'sub': 1', '4', '1', '4', '2', '4', '2', '4', '3', '6', '1', '4', '3', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'or represents (C-C)-alkyl, (C-C)-alkoxy, (C-C)-alkenyl, (C-C)-alkynyl, (C-C)-cycloalkyl, each of which is optionally mono- or disubstituted by identical or different substituents from the group consisting of aryl, hetaryl and heterocyclyl, where aryl, hetaryl or heterocyclyl may each optionally be mono- or disubstituted by identical or different substituents from the group consisting of halogen, cyano, carbamoyl, aminosulphonyl, (C-C)-alkyl, (C-C)-cycloalkyl, (C-C)-alkoxy, (C-C)-haloalkyl, (C-C)-haloalkoxy, (C-C)-alkylthio, (C-C)-alkylsulphinyl, (C-C)-alkylsulphonyl, (C-C)-alkylsulphimino, or'}, 'Rrepresents (C-C)-alkyl, (C-C)-hydroxyalkyl, (C-C)-haloalkyl, (C-C)-cyanoalkyl, (C-C)-alkoxy-(C-C)-alkyl, (C-C)-haloalkoxy-(C-C)-alkyl, (C-C)-alkenyl, (C-C)-alkenyloxy-(C-C)-alkyl, (C-C)-haloalkenyloxy-(C-C)-alkyl, (C-C)-haloalkenyl, (C-C)-cyanoalkenyl, (C-C)-alkynyl, (C-C)-alkynyloxy-(C-C)-alkyl, (C-C)-haloalkynyloxy-(C-C)-alkyl, (C-C)-haloalkynyl, (C-C)-cyanoalkynyl, (C-C)-cycloalkyl, (C-C)-cycloalkyl-(C-C)-cycloalkyl, (C-C)-alkyl-(C-C)-cycloalkyl, halo-(C-C)-cycloalkyl, (C-C)-alkylamino, di-(C-C)-alkylamino, (C-C)-cycloalkylamino, (C-C)-alkylcarbonylamino, (C-C ...

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26-01-2017 дата публикации

METHOD FOR PRODUCING CARBOXAMIDES

Номер: US20170022168A1
Принадлежит:

The present application relates to novel heterocyclic compounds, to the use thereof for controlling animal pests including arthropods, insects and , and to processes and intermediates for preparation of the heterocyclic compounds. 2. Composition claim 1 , comprising at least one compound of formula (I) according to .3. Method for controlling one or more pests claim 1 , comprising allowing a compound of the formula (I) according to or a composition thereof to act on the pests and/or a habitat thereof. The present application relates to novel heterocyclic compounds, to the use thereof for controlling animal pests including arthropods, insects and , and to processes and intermediates for preparation of the heterocyclic compounds.Derivatives of acylated 1-aryl-4-amino-1,2-pyrazoles are known from WO 2004/098528. The compounds described therein have activity as p38 kinase inhibitors.EP 2 674 423 A1 and WO 2012/061290 A2 describe pyrazole derivatives as pesticides.3-Aryl derivatives of acylated 1-aryl-4-amino-1,2-pyrazoles of the formulaare furthermore known from Journal of Pharmaceutical Sciences; 78; 6; 437-442. The compounds described therein are precursors of compounds which bind at the benzodiazepine receptor.Crop protection agents, which also include pesticides, have to meet many demands, for example in relation to efficacy, persistence, and spectrum of their action and possible use. Questions of toxicity and of combinability with other active compounds or formulation auxiliaries play a role, as does the question of the expense that the synthesis of an active compound requires. In addition, resistances can occur. For all these reasons, the search for novel crop protection compositions cannot be considered to be complete, and there is a constant need for novel compounds having properties which, compared to the known compounds, are improved at least in relation to individual aspects.It was an object of the present invention to provide compounds which widen the ...

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22-01-2015 дата публикации

PESTICIDAL ARYLPYRROLIDINES

Номер: US20150025253A1
Принадлежит: Bayer Intellectual Property GmbH

Arylpyrrolidines of formula (I): 2. Compound according to claim 1 , wherein{'sup': '1', 'sub': '3', 'Ris CF;'}{'sup': '2', 'Ris hydroxy;'}n is 1;{'sup': 1', '1, 'Bis C—Y;'}{'sup': 3', '3, 'Bis C—Y;'}{'sup': 4', '4, 'Bis C—Y; and'}{'sub': 1-3', '1', '6, 'E E is oxygen or a Calkandiyl-group which group can be optionally substituted by 1 or 2 C-Calkyl groups.'}3. Compound according to claim 1 , wherein{'sup': '1', 'sub': '3', 'Ris CF;'}{'sup': '2', 'Ris hydroxy;'}n is 1;{'sup': '1', 'Bis nitrogen;'}{'sup': 3', '3, 'Bis C—Y;'}{'sup': 4', '4, 'Bis C—Y; and'}{'sub': 1-3', '1', '6, 'E is oxygen or a Calkandiyl-group which group can be optionally substituted by 1 or 2 C-Calkyl groups.'}4. Compound according to claim 1 , wherein{'sup': '1', 'sub': '3', 'Ris CF;'}{'sup': '2', 'Ris hydroxy;'}n is 1;{'sup': 1', '1, 'Bis C—Y;'}{'sup': '3', 'Bis nitrogen;'}{'sup': 4', '4, 'Bis C—Y; and'}{'sub': 1-3', '1', '6, 'E is oxygen or a Calkandiyl-group which group can be optionally substituted by 1 or 2 C-Calkyl groups.'}5. Compound according to claim 1 , wherein{'sup': '1', 'sub': '3', 'Ris CF;'}{'sup': '2', 'Ris hydroxy;'}n is 1;{'sup': 1', '1, 'Bis C—Y;'}{'sup': 3', '3, 'Bis C—Y;'}{'sup': '4', 'Bis nitrogen; and'}{'sub': 1-3', '1', '6, 'E is oxygen or a Calkandiyl-group which group can be optionally substituted by 1 or 2 C-Calkyl groups.'}6. Compound according to claim 1 , wherein{'sup': '1', 'sub': '3', 'Ris CF;'}{'sup': '2', 'Ris an oxo group;'}n is 1;{'sup': 1', '1, 'Bis C—Y;'}{'sup': 3', '3, 'Bis C—Y;'}{'sup': 4', '4, 'Bis C—Y; and'}{'sub': 1-3', '1', '6, 'E is oxygen or a Calkandiyl-group which group can be optionally substituted by 1 or 2 C-Calkyl groups.'}7. Compound according to claim 1 , wherein{'sup': '1', 'sub': '3', 'Ris CF;'}{'sup': '2', 'Ris an oxo group;'}n is 1;{'sup': '1', 'Bis nitrogen;'}{'sup': 3', '3, 'Bis C—Y;'}{'sup': 4', '4, 'Bis C—Y; and'}{'sub': 1-3', '1', '6, 'E is oxygen or a Calkandiyl-group which group can be optionally substituted by 1 or 2 C-Calkyl groups ...

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30-01-2020 дата публикации

2-(Het)aryl-substituted fused heterocycle derivatives as pesticides

Номер: US20200029567A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 4. The compound of formula (I) according to wherein{'sup': 1', '4, 'Arepresents nitrogen or ═C—R,'}{'sup': '1', 'Rrepresents methyl, ethyl, n-propyl, isopropyl, cyclopropyl, n-butyl, isobutyl, tert-butyl, cyclobutyl, fluoromethyl, difluoromethyl, trifluoromethyl, fluoroethyl, difluoroethyl, trifluoroethyl, tetrafluoroethyl or pentafluoroethyl,'}{'sup': '2', 'Rrepresents a group selected from G1, G2, G3, G4 G10, G11, G12, G13, G14, G15, G18 or G19,'}{'sup': '3', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Rrepresents hydrogen, cyano, halogen, (C-C)alkyl, (C-C)haloalkyl, (C-C)haloalkoxy, (C-C)alkylthio, (C-C)alkylsulphinyl, (C-C)alkylsulphonyl, (C-C)haloalkylthio, (C-C)haloalkylsulphinyl, (C-C)haloalkylsulphonyl or NHCO—(C-C)alkyl ((C-C)alkylcarbonylamino),'}{'sup': '4', 'Rrepresents hydrogen, fluorine, chlorine, bromine or cyano,'}X represents a heteroaromatic 9-membered or 12-membered fused bicyclic or tricyclic ring system from the series H1, H2, H3, H4, H5, H7, H8, H10, H11, H12, H13, H15, H16, H17, H18, H19, or H20,{'sup': '5', 'sub': 1', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Rrepresents hydrogen, cyano, halogen, (C-C)alkyl, (C-C)haloalkyl, (C-C)alkenyl, (C-C)haloalkenyl, (C-C)alkynyl, (C-C)haloalkynyl, (C-C)cycloalkyl, (C-C)cycloalkyl-(C-C)cycloalkyl, (C-C)alkyl-(C-C)cycloalkyl, (C-C)alkoxy, (C-C)haloalkoxy, (C-C)alkoxyimino, (C-C)alkylthio, (C-C)haloalkylthio, (C-C)alkylsulphinyl, (C-C)haloalkylsulphinyl, (C-C)alkylsulphonyl, (C-C)haloalkylsulphonyl, (C-C)alkylcarbonyl, (C-C)haloalkylcarbonyl, (C-C)alkylaminocarbonyl, di-(C-C)alkylaminocarbonyl, (C-C)alkylsulphonylamino (C-C)alkylaminosulphonyl or di-(C-C) ...

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06-02-2020 дата публикации

MESOIONIC IMIDAZOPYRIDINES AS INSECTICIDES

Номер: US20200037600A1
Принадлежит:

Provided are compounds of the formula (I) 3. The compound according to claim 1 , in which{'sup': 5a', '5b', '5c, 'sub': 2', '4', '3', '4', '3', '6', '2', '4', '3', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'claim-text': 'or', 'T represents hydrogen, C(R)(R)(R), C-C-alkenyl, C-C-alkynyl or C-C-cycloalkyl, where C-C-alkenyl, C-C-alkynyl or C-C-cycloalkyl may each optionally be mono- to trisubstituted and the substituents independently of one another are selected from the group consisting of halogen, and/or may each optionally be monosubstituted and the substituent is selected from the group consisting of cyano, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-haloalkoxy, C-C-alkylthio, C-C-alkylsulfinyl and C-C-alkylsulfonyl,'}{'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'claim-text': 'or', 'T represents phenyl, C-C-alkylenedioxyphenyl, naphthyl, furanyl, thienyl, pyrrolyl, pyrazolyl, imidazolyl, 1,2,3-triazolyl, 1,2,4-triazolyl, 1,3-oxazolyl, 1,2-oxazolyl, thiazolyl, isothiazolyl, 1,2,3-oxadiazolyl, 1,2,4-oxadiazolyl, 1,3,4-oxadiazolyl, 1,2,5-oxadiazolyl, 1,2,3-thiadiazolyl, 1,2,4-thiadiazolyl, 1,3,4-thiadiazolyl, 1,2,5-thiadiazolyl, pyridyl, pyrimidyl, thiophenyl, pyridazinyl, pyrazinyl, 1,2,3-triazinyl, 1,2,4-triazinyl, 1,3,5-triazinyl, benzofuranyl, indolyl, benzothiazolyl, benzoxazolyl, benzimidazolyl, pyrazolopyridinyl, quinolinyl, isoquinolinyl, cinnolinyl, azetidinyl, azolidinyl, azinanyl, oxetanyl, oxolanyl, oxanyl, dioxanyl, thiethanyl, thiolanyl, thianyl, or dihydroisoxazolyl, where the radicals mentioned above may each optionally be mono- to tetrasubstituted and the substituents independently of one another are selected from the group consisting of fluorine and chlorine, and/or may each optionally be mono- to disubstituted and the substituents independently of one another are selected from the group consisting of bromine, nitro, ...

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07-02-2019 дата публикации

SUBSTITUTED 2-OXYIMIDAZOLYLCARBOXAMIDES AS PESTICIDES

Номер: US20190040042A1
Принадлежит:

The present invention relates to compounds of the general formula (I) 2. Compound according to claim 1 , whereinQ represents oxygen or sulphur,{'sub': 1', '4', '1', '4', '1', '4', '1', '4, 'V represents a radical from the series hydrogen, halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-haloalkoxy and cyano,'}{'sub': 1', '4', '1', '4', '1', '4', '1', '4, 'W represents a radical from the series hydrogen, halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-haloalkoxy and cyano,'}{'sub': 1', '8', '3', '8', '3', '8', '1', '4', '1', '4', 'm, 'sup': 2', '2', '3', '2, 'claim-text': [{'sub': 3', '8', '3', '8', 'm', '1', '4', '1', '4', '1', '4, 'sup': 2', '4, 'C-C-cycloalkyl or C-C-cycloalkenyl, optionally interrupted once or twice independently of one another by O, S(O), C(G)Ror NRand optionally mono- to tetrasubstituted independently of one another by halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy or cyano,'}, {'sub': 3', '8', '1', '4', '3', '8', '1', '4', 'm', '1', '4', '1', '4', '1', '4, 'sup': 2', '4, 'straight-chain or branched C-C-cycloalkyl-C-C-alkyl or C-C-cycloalkenyl-C-C-alkyl, optionally interrupted once or twice independently of one another by O, S(O), C(G)Ror NRand optionally mono- to tetrasubstituted independently of one another by halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy or cyano,'}, {'sub': 1', '4', '1', '4', '1', '4', '1', '4', 'm', '1', '4', '1', '4', 'm', '1', '4', '1', '4', '1', '4', '1', '4', 'm', '1', '4', '1', '4', 'm, 'aryl or hetaryl, optionally mono- to trisubstituted independently of one another by halogen, acylamido, oxime ether, nitro, cyano, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-alkyl-S(O)—, C-C-haloalkoxy, C-C-haloalkyl-S(O)— or by aryloxy, hetaryloxy, aryl or heteraryl, optionally mono- to trisubstituted independently of one another by halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-alkyl-S(O)—, C-C-haloalkoxy, C-C-haloalkyl-S(O)—, hetaryloxy, aryloxy, nitro or cyano and'}, {'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', ...

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16-02-2017 дата публикации

NEW PESTICIDAL COMPOUNDS AND USES

Номер: US20170044104A1
Принадлежит: Bayer Animal Health GmbH

The invention relates to the use of known and novel phenalkyl carboxamide derivatives of the formula (I) 5. A method of protecting crops comprising administering an effective amount of the compound of .6. A method of protecting animals comprising administering an effective amount of the compound of .10. An agrochemical formulation claim 1 , comprising the compound of .11. An agrochemical formulation comprising the compound of .12. The agrochemical formulation of claim 10 , further comprising at least one extender and/or at least one surfactant.13. The agrochemical formulation of claim 10 , wherein the compound of the formula (I) claim 10 , (Ia) claim 10 , (Ib) or (Ic) is present in a mixture with at least one other active compound.14. A method for controlling an animal pest claim 1 , comprising applying an effective amount of the compound of formula (I) as defined in to an animal pest and/or a habitat of the animal pest.15. The method of claim 14 , wherein the animal pest comprises a nematode or is a nematode.16. A method for protecting a seed and/or a germinating plant from attack by a pest comprising the step of contacting the seed with a compound of formula (I) as defined in .17. A seed obtained by the method of .18. A method for controlling an animal pest comprising administering an effective amount of the compound of .19. The method of claim 18 , wherein the animal pest comprises a nematode or is a nematode.20. A method of protecting crops or animals comprising administering an effective amount of the compound of . The present invention relates to the use of known and novel phenalkyl carboxamide derivatives for the control of nematodes and/or other helminths, particularly in agriculture and in the animal health field, formulations containing such compounds, particularly agrochemical formulations, and methods for the control of nematodes and helminths.The present invention further relates to certain phenalkyl carboxamide derivatives as to processes for their ...

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15-02-2018 дата публикации

NOVEL PYRAZOLYL DERIVATIVES AS PEST CONTROL AGENTS

Номер: US20180044298A1
Принадлежит: Bayer Animal Health GmbH

The invention comprises novel pyrazolyl derivatives of the general formula (I) Also described are processes for preparing the compounds of the formula (I). The compounds according to the invention are especially suitable for controlling insects and arachnids in agriculture, and ectoparasites in veterinary medicine. 2. The compound as claimed in claim 1 , wherein Bis CR claim 1 , Bis CR claim 1 , Bis CR claim 1 , Bis CRand Bis CR claim 1 ,and/or a salt, N-oxide and/or a tautomeric form thereof.3. The compound as claimed in claim 1 , wherein Ris halogen or optionally halogenated C-C-alkyl or optionally halogenated C-C-alkoxy claim 1 , Ris hydrogen claim 1 , Ris halogenated C-C-alkyl claim 1 , Ris hydrogen and Ris halogen or optionally halogenated C-C-alkyl or optionally halogenated C-C-alkoxy claim 1 ,and/or a salt, N-oxide and/or a tautomeric form thereof.4. The compound as claimed in claim 1 , wherein Rand Rare hydrogen and W is oxygen claim 1 ,and/or a salt, N-oxide and/or a tautomeric form thereof.5. The compound as claimed in claim 1 , wherein Ais CR claim 1 , Ais CRor N claim 1 , Ais CRor N and Ais CRand Ris hydrogen or C-C-alkyl and R claim 1 , Rand Rare each independently of one another hydrogen claim 1 , halogen claim 1 , CN claim 1 , optionally halogenated C-C-alkyl or optionally halogenated N claim 1 ,N-di-C-C-alkylamino claim 1 ,and/or a salt, N-oxide and/or a tautomeric form thereof.6. The compound as claimed in claim 1 , wherein Q is{'sub': 1', '6, 'C-C-alkyl optionally substituted by one, two or three substituents selected from the group consisting of oxo, cyano, nitro and amino,'}{'sub': 1', '6, 'halogenated (C-C)-alkyl,'}{'sub': 3', '6', '1', '3, 'C-C-cycloalkyl optionally substituted by one, two or three substituents selected from the group consisting of halogen, cyano, nitro, C-C-alkyl and amino,'}{'sub': 2', '5', '1', '3, 'C-C-heterocyclyl optionally substituted with one, two or three substituents selected from the group consisting of halogen, ...

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14-02-2019 дата публикации

SUBSTITUTED IMIDAZOLYLCARBOXAMIDES AS PESTICIDES

Номер: US20190045783A1
Принадлежит:

The present invention relates to compounds of the general formula (I) 8. Composition claim 1 , comprising at least one compound according to and one or more customary extenders and/or surfactants optionally for controlling animal pests.9. Method for controlling one or more animal pests claim 1 , comprising allowing at least one compound according to is allowed to act on the animal pests and/or a habitat thereof.10. A product comprising at least one compound according to for controlling one or more animal pests.11. Method according to claim 9 , where surgical claim 9 , therapeutic and diagnostic treatment of a human or animal body is excluded.12. A product comprising at least one compound according to for protecting propagation material of one or more plants.13. Agrochemical formulation comprising at least one compound according to in a biologically effective amount of from 0.00000001 to 98% by weight based on the weight of the agrochemical formulation claim 1 , and also one or more extenders and/or surfactants.14. Agrochemical formulation according to claim 13 , additionally comprising a further agrochemically active compound. The present application relates to novel heterocyclic compounds and their use for controlling animal pests.WO 2011/009804 A2 describes heterocyclic compounds including, inter alia, imidazolylcarboxamides which can be used as insecticides. However, imidazolylcarboxamides which are substituted directly at the imidazolyl ring by the functional groups X according to the invention are not described. The imidazolylcarboxamides listed in WO 2011/009804 A2 have considerable weaknesses in their insecticidal action.Modern insecticides have to meet many demands, for example in relation to extent, persistence and spectrum of their action and possible use. Questions of toxicity, sparing of beneficial species and pollinators, environmental properties, application rates, combinability with other active ingredients or formulation auxiliaries play a role, as ...

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13-02-2020 дата публикации

HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20200045976A1
Принадлежит:

The invention relates to novel compounds of the formula (I), 2. Compound of formula (I) according to claim 1 , in which{'sup': '1', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '3', '6, 'Ris (C-C)alkyl, (C-C)cyanoalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkyl, (C-C)alkenyl, (C-C)haloalkenyl, (C-C)alkynyl, (C-C)haloalkynyl or (C-C)cycloalkyl,'}{'sup': '2', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '3', '6', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Ris hydrogen, (C-C)alkyl, (C-C)haloalkyl, (C-C)cyanoalkyl, (C-C)hydroxyalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkoxy-(C-C)alkyl, (C-C)cycloalkyl, (C-C)cycloalkyl-(C-C)cycloalkyl, (C-C)alkyl-(C-C)cycloalkyl, halo(C-C)cycloalkyl, cyano(C-C)cycloalkyl, (C-C)alkylthio-(C-C)alkyl, (C-C)haloalkylthio-(C-C)alkyl, (C-C)alkylsulfinyl-(C-C)alkyl, (C-C)haloalkylsulfinyl-(C-C)alkyl, (C-C)alkylsulfonyl-(C-C)alkyl or (C-C)haloalkylsulfonyl-(C-C)alkyl,'}{'sup': '3', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '3', '6', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '3', '6', '3', '6', '1', '4', '2', '4', '2', '4', '2', '4', '3', '6', '2', '2', '4', '2', '4', '3', '6', '2', '3', '6', '1', '4', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4, 'Ris hydrogen, halogen, cyano, nitro, (C-C)alkyl, (C-C)haloalkyl, (C-C)alkoxy, (C-C)haloalkoxy, (C-C)alkylthio, (C-C)haloalkylthio, (C-C)alkylsulfinyl, (C-C)haloalkylsulfinyl, (C-C) ...

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14-02-2019 дата публикации

SUBSTITUTED IMIDAZOLYLCARBOXAMIDES AS PESTICIDES

Номер: US20190047987A1
Принадлежит:

The present invention relates to compounds of the general formula (I) 3. Compound according to in whichQ represents oxygen,V represents a radical from the group consisting of hydrogen, fluorine, chlorine, bromine, methyl and ethyl,W represents a radical from the group consisting of hydrogen, fluorine, chlorine, bromine, cyano and methyl,{'sub': 1', '4', '3', '4', '3', '4', '3', '6, 'Y represents a radical from the group consisting of hydrogen, C-C-alkyl, C-C-alkenyl or C-C-alkynyl, optionally mono- to pentasubstituted independently of one another by fluorine, chlorine, bromine, methoxy or ethoxy, and C-C-cycloalkyl, optionally mono- to disubstituted independently of one another by fluorine, chlorine, bromine, methyl, ethyl, trifluoromethyl, methoxy, ethoxy or cyano,'}{'sub': 1', '6', '3', '6', '3', '6', '3', '6, 'A represents a radical from the group consisting of hydrogen, C-C-alkyl, C-C-alkenyl or C-C-alkynyl, optionally mono- to pentasubstituted independently of one another by fluorine, chlorine, bromine, methoxy, ethoxy or cyano, and C-C-cycloalkyl, optionally mono- to disubstituted independently of one another by fluorine, chlorine, bromine, methyl, ethyl, trifluoromethyl, methoxy, ethoxy or cyano,'}T represents an electron pair,{'sup': 1', '2, 'Land Lrepresent, together with N, a heterocycle from the group U-1, U-2, U-3, U-4, U-5, U-6, U-7, U-25, U-26, U-27, U-28, U-29 and U-30,'}{'sup': 'b', 'sub': 1', '4', '3', '6', '1', '2', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '6', '1', '4', '1', '4', '1', '6', '1', '6', 'n', 'n', 'n', 'n', 'n, 'claim-text': 'or', 'Xrepresents a radical from the group consisting of halogen, nitro, cyano, amino, C-C-alkyl, C-C-cycloalkyl, C-C-haloalkyl, C-C-alkoxy, C-C-haloalkoxy, C-C-halocycloalkyl, C-C-alkoxy-C-C-alkyl, C-C-alkylthio, C-C-alkoxycarbonyl, C-C-alkylaminocarbonyl, C-C-alkylsulphonyl, C-C-alkylcarbonylamino and phenyl, where phenyl may optionally be mono- to trisubstituted by fluorine, chlorine, bromine, ...

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25-02-2021 дата публикации

HETEROCYCLIC COMPOUNDS AS PESTICIDES

Номер: US20210053924A1
Принадлежит:

The present application relates to the use of heterocyclic compounds for controlling animal pests including arthropods, insects and nematodes, to novel heterocyclic compounds, to processes for their preparation and to intermediates for preparing the heterocyclic compounds. 118-. (canceled)24. A composition comprising at least one compound of formula (I) according to .25. A method for controlling pests claim 19 , comprising allowing the compound of formula (I) according to to act on the pests and/or their habitat claim 19 , provided that treatments of humans are excluded.26. The method according to claim 25 , wherein the pests are insects claim 25 , arachnids claim 25 , or nematodes.27. The method according to claim 25 , wherein the pests are nematodes.28. The compound according to claim 19 , wherein A is 3-fluoropyrazin-2-yl claim 19 , B is 2-(trifluoromethyl)phenyl claim 19 , R3 claim 19 , R4 claim 19 , R5 are H claim 19 , and Z is oxygen.29. The compound according to claim 19 , wherein A is 3-fluoropyrazin-2-yl claim 19 , B is 2-chlorophenyl claim 19 , R3 claim 19 , R4 claim 19 , R5 are H claim 19 , and Z is oxygen.30. The compound according to claim 19 , wherein A is 3-fluoropyrazin-2-yl claim 19 , B is 2-bromophenyl claim 19 , R3 claim 19 , R4 claim 19 , R5 are H claim 19 , and Z is oxygen.31. The compound according to claim 19 , wherein A is 3-fluoropyrazin-2-yl claim 19 , B is 2-iodophenyl claim 19 , R3 claim 19 , R4 claim 19 , R5 are H claim 19 , and Z is oxygen.32. The compound according to claim 19 , wherein A is 3-fluoropyrazin-2-yl claim 19 , B is 2 claim 19 ,6-difluorophenyl claim 19 , R3 claim 19 , R4 claim 19 , R5 are H claim 19 , and Z is oxygen.33. The compound according to claim 19 , wherein A is 3-fluoropyrazin-2-yl claim 19 , B is 3-(trifluoromethyl)pyridine-2-yl claim 19 , R3 claim 19 , R4 claim 19 , R5 are H claim 19 , and Z is oxygen.34. The compound according to claim 19 , wherein A is 2-chloropyrazin-5-yl claim 19 , B is 2-(trifluoromethyl) ...

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13-02-2020 дата публикации

SUBSTITUTED 2-(HET)ARYLIMIDAZOLYLCARBOXYAMIDES AS PESTICIDES

Номер: US20200048221A1
Принадлежит:

The present invention relates to compounds of the general formula (I) 2. The intermediate of formula (X) according to claim 1 , wherein X is Cl.3. The intermediate of formula (X) according to claim 1 , wherein X is Br.4. The intermediate of formula (X) according to claim 1 , wherein X is I.5. The intermediate of formula (X) according to claim 1 , wherein X is ethinyl.6. The intermediate of formula (X) according to claim 1 , whereinQ represents oxygen or sulphur,{'sub': 1', '4', '1', '4', '1', '4', '1', '4, 'V represents a radical selected from the group consisting of hydrogen, halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-haloalkoxy and cyano,'}{'sub': 1', '4', '1', '4', '1', '4', '1', '4, 'W represents a radical selected from the group consisting of hydrogen, halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-haloalkoxy and cyano,'} [{'sub': 1', '6', '3', '6', '3', '6', '1', '4', '1', '4', 'm, 'C-C-alkyl, C-C-alkenyl or C-C-alkynyl, optionally mono- to polysubstituted independently of one another by halogen, C-C-alkoxy, C-C-alkyl-S(O)— or cyano,'}, {'sub': 3', '8', '1', '4', '4', '1', '4, 'b': '1', 'C-C-cycloalkyl, optionally mono- to disubstituted independently of one another by halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy or cyano,'}, {'sub': 3', '8', '1', '4', 'm', '1', '4', '1', '4', '1', '4, 'sup': '2', 'straight-chain or branched C-C-cycloalkyl-C-C-alkyl, optionally interrupted once to twice independently of one another by O, S(O), CO or NRand optionally mono- to tetrasubstituted independently of one another by halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy or cyano, and'}, {'sub': 1', '4', '1', '4', '1', '4', '1', '4', 'm', '1', '4', '1', '4', 'm, 'arylalkyl or hetarylalkyl, optionally mono- to trisubstituted independently of one another by halogen, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-alkyl-S(O)—, C-C-haloalkoxy, C-C-haloalkyl-S(O)—, nitro or cyano,'}], 'Y represents a radical selected from the group consisting of hydrogen, methyl, cyano,'}m ...

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21-02-2019 дата публикации

SUBSTITUTED PYRIDINE COMPOUNDS AS PESTICIDES

Номер: US20190053492A1
Принадлежит:

The present invention relates to novel substituted pyridine compounds of the formula (I) 2. Compound of formula (I) and/or salt thereof according to in which{'sup': '1', 'Qis in each case optionally singly or multiply, identically or differently substituted phenyl, 1,3-benzodioxolyl, 2,3-dihydro-1,4-benzodioxinyl, hetaryl or oxohetaryl,'}{'sub': 5', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '2', '4', '2', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '3', '6', '3', '6', '1', '4', '3', '6', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '3', '6', '3', '6', '3', '6', '3', '6', '3', '6', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '6', '1', '6', '1', '4', '1', '4, 'where the substituents are selected from cyano, halogen, nitro, amino, SF, (C-C)alkyl, (C-C)haloalkyl, (C-C)cyanoalkyl, (C-C)hydroxyalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)alkenyl, (C-C)haloalkenyl, (C-C)cyanoalkenyl, (C-C)alkynyl, (C-C)haloalkynyl, (C-C)cyanoalkynyl, (C-C)alkoxy, (C-C)haloalkoxy, (C-C)cyanoalkoxy, (C-C)alkoxy-(C-C)alkoxy, (C-C)cycloalkyl, (C-C)halocycloalkyl, (C-C)alkyl-(C-C)cycloalkyl, (C-C)haloalkyl-(C-C)cycloalkyl, (C-C)haloalkenoxy, (C-C)alkylhydroxyimino, (C-C)alkoxyimino, (C-C)alkyl-(C-C)alkoxyimino, (C-C)haloalkyl-(C-C)alkoxyimino, (C-C)alkylsulphanyl, (C-C)alkylsulphanyl-(C-C)alkyl, (C-C)alkylsulphinyl, (C-C)haloalkylsulphinyl, (C-C)alkylsulphinyl-(C-C)alkyl, (C-C)alkylsulphonyl, (C-C)haloalkylsulphonyl, (C-C)alkylsulphonyl-(C-C)alkyl, (C-C)alkylsulphonyloxy, (C-C)haloalkylsulphanyl, (C-C)cycloalkylsulphanyl, (C-C)halocycloalkylsulphanyl, (C-C)cycloalkylsulphonyl, (C-C)halocycloalkylsulphonyl, (C-C)cycloalkylsulphinyl, (C-C)halocycloalkylsulphinyl, (C-C)alkylcarbonyl, (C-C)haloalkylcarbonyl, aminocarbonyl, (C-C ...

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20-02-2020 дата публикации

HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20200054017A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. Compound of formula (I) according to in which{'sup': '1', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '3', '6, 'Ris (C-C)alkyl, (C-C)cyanoalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkyl, (C-C)alkenyl, (C-C)haloalkenyl, (C-C)alkynyl, (C-C)haloalkynyl or (C-C)cycloalkyl,'}{'sup': '2', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '3', '6', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Ris hydrogen, (C-C)alkyl, (C-C)haloalkyl, (C-C)cyanoalkyl, (C-C)hydroxyalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkoxy-(C-C)alkyl, (C-C)cycloalkyl, (C-C)cycloalkyl-(C-C)cycloalkyl, (C-C)alkyl-(C-C)cycloalkyl, halo(C-C)cycloalkyl, cyano(C-C)cycloalkyl, (C-C)alkylthio-(C-C)alkyl, (C-C)haloalkylthio-(C-C)alkyl, (C-C)alkylsulfinyl-(C-C)alkyl, (C-C)haloalkylsulfinyl-(C-C)alkyl, (C-C)alkylsulfonyl-(C-C)alkyl or (C-C)haloalkylsulfonyl-(C-C)alkyl,'}{'sup': '3', 'sub': 3', '6', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4, 'Ris optionally singly or multiply, identically or differently substituted (C-C)cycloalkyl, where possible substituents in each case are: (C-C)cycloalkyl, (C-C)alkyl, (C-C)haloalkyl, (C-C)alkoxy, (C-C)haloalkoxy, aminocarbonyl, aminothiocarbonyl, halogen or cyano,'}X is a heteroaromatic 9-membered or 12-membered fused bicyclic or tricyclic ring system from the group of Q1 to Q18,{'sup': '4', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '3', '6, 'Ris hydrogen, (C-C)alkyl, (C-C)haloalkyl, (C-C)cyanoalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkoxy-(C-C)alkyl, (C-C)alkenyl, (C-C)haloalkenyl, (C-C)alkynyl, (C-C)haloalkynyl or (C-C)cycloalkyl,'}{'sup': 5', '6, 'sub': 1', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '3', '6 ...

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02-03-2017 дата публикации

N-ARYLAMIDINE-SUBSTITUTED TRIFLUOROETHYL SULFIDE DERIVATIVES AS ACARICIDES AND INSECTICIDES

Номер: US20170057914A1
Принадлежит:

The present invention relates to novel N-arylamide-substituted trifluoroethyl sulfide derivatives of the formula (I) This application is a divisional application of U.S. application Ser. No. 14/366,715 (filed Jun. 19, 2014), which is a §371 National Stage Application of PCT/EP2012/075269 (filed Dec. 12, 2012), which claims priority to EP 11194855.0 (filed Dec. 21, 2011), the contents of each of which are incorporated herein by reference.Field of the InventionThe present invention relates to novel N-arylamidine-substituted trifluoroethyl sulfide derivatives, to their use as acaricides and insecticides for controlling animal pests and to processes and intermediates for their preparation.Description of Related ArtVarious substituted N-arylamidines and their insecticidal and acaricidal action have already been described in the literature in WO 2007/131680.On application, the active compounds already known from the publications mentioned above have disadvantages, be it that they may have no or else only insufficient insecticidal and/or acaricidal activity against animal pests, in particular at relatively low application rates.Accordingly, it is an object of the present invention to provide corresponding N-arylamidine-substituted trifluoroethyl sulfide derivatives which can be employed as insecticides and/or acaricides with satisfactory insecticidal and/or acaricidal activity against animal pests, in particular at relatively low application rates, with high selectivity and improved compatibility in crops of useful plants.The present invention now provides novel compounds of the formula (I)in whichIf appropriate, the compounds of the formula (I) may be present in various polymorphic forms or as mixtures of different polymorphic forms. Both the pure polymorphs and the polymorph mixtures are provided by the invention and can be used according to the invention.The compounds of the formula (I) optionally comprise diastereomers or enantiomers and also rotamers, tautomers and ...

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27-02-2020 дата публикации

NOVEL HETEROCYCLIC COMPOUNDS AS PESTICIDES

Номер: US20200062729A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. The compound according to claim 1 , wherein{'sup': 10', '11, 'Z represents optionally substituted naphthyl, dibenzo[b,d]furanyl, dibenzo[b,d]thiophenyl, indan-4-yl, benzothiophen-4-yl, benzofuran-4-yl, indol-4-yl or represents substituted phenyl of the substructure formula (II) and the phenyl of the substructure formula (II) carries no further substituents apart from Rand R,'}{'sup': '5', 'Y represents O, S, —NR,'}{'sup': 1', '2', '3', '4, 'sub': 1', '4', '2', '4', '2', '4', '3', '6', '1', '4', '2', '4', '2', '4', '3', '6', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '3', '6', '3', '6', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '3', '6', '3', '6, 'R, R, Rand Reach independently of one another represent a substituent selected from the group consisting of hydrogen, halogen, nitro, cyano, or represent (C-C)-alkyl, (C-C)-alkenyl, (C-C)-alkynyl, (C-C)-cycloalkyl, (C-C)-alkoxy, (C-C)-alkenyloxy, (C-C)-alkynyloxy, (C-C)-cycloalkoxy, (C-C)-alkoxycarbonyl, (C-C)-cycloalkoxycarbonyl, N-mono-(C-C)-alkylamino, N,N-di-(C-C)-alkylamino, (C-C)-alkylsulfanyl, (C-C)-alkylsulfinyl, (C-C)-alkylsulfonyl, (C-C)-cycloalkylsulfanyl, (C-C)-cycloalkylsulfinyl, (C-C)-cycloalkylsulfonyl, each of which is optionally mono- or polysubstituted by identical or different substituents from the group consisting of halogen, cyano, nitro, (C-C)-alkyl, (C-C)-haloalkyl, (C-C)-alkoxy, (C-C)-haloalkoxy, (C-C)-cycloalkyl, (C-C)-halocycloalkyl,'}{'sup': '5', 'sub': 1', '4', '3', '4', '1', '3, 'Rrepresents hydrogen or represents (C-C)-alkyl, (C-C)-cycloalkyl, (C-C)-alkanoyl, optionally mono- or polysubstituted by identical or different halogen substituents,'}{'sup': 6', '8, 'sub': 1', '4', '3', '4', '1', '4', '2, 'Rrepresents hydrogen or represents (C-C)-alkyl, (C-C)-cycloalkyl, (C-C)-alkanoyl, optionally mono- or polysubstituted by identical or different halogen substituents, or a ring closure with Rformed by 1 ...

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10-03-2016 дата публикации

Current-Mode Sense Amplifier and Reference Current Circuitry

Номер: US20160071555A1
Принадлежит: International Business Machines Corp

An electronic circuit comprising is provided with a current sense amplifier. The amplifier comprises a reference current input terminal, a sense current input terminal, and a first output terminal. The electronic circuit includes a reference current source. The reference current source includes two reference n-FET stacks connected in series, and the reference current input terminal is coupled to a ground terminal via the two reference n-FET stacks. The electronic circuit includes a plurality of memory cells each coupled in parallel via a respective sense n-FET stack to the sense current input terminal. The amplifier is configured to generate a first logical value at the first output terminal of the amplifier in response to a sense current of the sense current input terminal being lower than a reference current of the reference current input terminal. The amplifier is further configured to generate a second logical value at the first output terminal of the amplifier in response to the sense current being higher than the reference current.

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17-03-2016 дата публикации

N-(2-FLUORO-2-PHENETHYL)CARBOXAMIDES AS NEMATICIDES AND ENDOPARASITICIDES

Номер: US20160075637A1
Принадлежит:

The present invention relates to N-(2-halogen-2-phenethyl)carboxamides, a process for producing such compounds, their use for the control of nematodes in agricultures and their use as anthelmintics against endoparasites in animals or humans, compositions containing such compounds and methods for the control of nematodes and helminths. 4. Compound of as defined in for use as a medicament with the proviso that the following compounds are disclaimed:3-chloro-N-[2-(4-chlorophenyl)-2,2-difluoroethyl]thiophene-2-carboxamide, 3-bromo-N-[2-(4-chlorophenyl)-2,2-difluoroethyl]thiophene-2-carboxamide, N-[2-(4-chlorophenyl)-2,2-difluoroethyl]-2-(trifluoromethyl)nicotin-amide, N-[2-(2,4-dichlorophenyl)-2,2-difluoroethyl]-2-(trifluoromethyl)nicotin-amide, 2-chloro-N-[2-(4-chlorophenyl)-2,2-difluoroethyl]-4-(trifluoromethyl)nicotinamide, 2-chloro-N-[2-(2,4-dichlorophenyl)-2,2-difluoroethyl]-4-(trifluoromethyl)nicotinamide, 6-chloro-N-[2-(4-chloro-phenyl)-2,2-difluoroethyl]-4-(trifluoromethyl)nicotinamide and 6-chloro-N-[2-(2,4-dichloro phenyl)-2,2-difluoroethyl]-4-(trifluoromethyl)nicotinamide.5. Compound of according to capable for use as a medicament with the proviso that the following compounds are disclaimed:3-chloro-N-[2-(4-chlorophenyl)-2,2-difluoroethyl]thiophene-2-carboxamide, 3-bromo-N-[2-(4-chlorophenyl)-2,2-difluoroethyl]thiophene-2-carboxamide, N-[2-(4-chlorophenyl)-2,2-difluoroethyl]-2-(trifluoromethyl)nicotin-amide, N-[2-(2,4-dichlorophenyl)-2,2-difluoroethyl]-2-(trifluoromethyl)nicotin-amide, 2-chloro-N-[2-(4-chlorophenyl)-2,2-difluoroethyl]-4-(trifluoromethyl)nicotinamide, 2-chloro-N-[2-(2,4-dichlorophenyl)-2,2-difluoroethyl]-4-(trifluoromethyl)nicotinamide, 6-chloro-N-[2-(4-chloro-phenyl)-2,2-difluoroethyl]-4-(trifluoromethyl)nicotinamide and 6-chloro-N-[2-(2,4-dichloro phenyl)-2,2-difluoroethyl]-4-(trifluoromethyl)nicotinamide.6. Compound of as defined in capable for use in treatment of helminths in animals and humans.7. Compound of as defined in capable for use ...

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17-03-2016 дата публикации

NEMATICIDAL N-(PHENYLCYCLOALKYL)CARBOXAMIDES AND N-(PHENYLCYCLOALKYL)THIOCARBOXAMIDES

Номер: US20160075653A1
Принадлежит:

The present invention relates to the use of N-(Phenylcycloalkyl)carboxamides and N-(Phenylcycloalkyl)thiocarboxamides for the control of nematodes in agriculture and as anthelmintic agents against endoparasites in animals and humans, compositions containing such compounds and methods for the control of nematodes and helminths and furthermore to novel N-(Phenylcycloalkyl)carboxamides and N-(Phenylcycloalkyl)thiocarboxamides, processes and intermediate compounds for their preparation, their use as nematicides, compositions containing such compounds and methods for the control of nematodes. 3. A compound according to claim 1 , in which T represents sulphur claim 1 , capable of being used for controlling nematodes.6. Composition claim 1 , comprising an effective amount of at least one compound of formula (I-1) or (I-2) and at least one surfactant claim 1 , solid or liquid diluent.7. A compound according to capable of being used as an endoparasiticide.8. A compounds according to capable of being used as an anthelmintic.9. A compound according to capable of being used for preparation of an endoparasitic agent for combating one or more endoparasites. The present invention relates to the use of N-(Phenylcycloalkyl)carboxamides and N-(Phenylcycloalkyl)thiocarboxamides for the control of nematodes in agriculture and as anthelmintic agents against endoparasites in animals and humans, compositions containing such compounds and methods for the control of nematodes and helminths.The present invention further relates to novel N-(Phenylcycloalkyl)carboxamides and N-(Phenylcycloalkyl)thiocarboxamides, processes and intermediate compounds for their preparation, their use as nematicides, compositions containing such compounds and methods for the control of nematodes.Nematodes cause a substantial loss in agricultural product including food and industrial crops and are controlled with chemical compounds having nematicidal activity. To be useful in agriculture these compounds should have ...

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16-03-2017 дата публикации

HETEROCYCLIC COMPOUNDS AS PESTICIDES

Номер: US20170073318A1
Принадлежит: Bayer CropScience Aktiengesellschaft

The present application relates to novel heterocyclic compounds, to the use thereof for controlling animal pests including arthropods, insects and nematodes, and to processes and intermediates for preparation of the novel compounds. 6. Composition claim 1 , comprising a content of at least one compound of formula (I) according to .7. Method for controlling pests claim 1 , comprising allowing a compound of formula (I) according to or a composition thereof to act o none or more pests and/or their habitat.9. Compound of formula (IIa-1-a) according to claim 8 , in which R3 is hydrogen.11. Compound of formula (1-9) according to claim 10 , in which R3 is hydrogen. The present application relates to novel heterocyclic compounds, to the use thereof for controlling animal pests including arthropods, insects and nematodes, and to processes and intermediates for preparation of the novel compounds.Derivatives of 1-aryl-3-aroylamino-1,2,4-triazoles are known from WO 2012/006473.The compounds described therein have activity as phosphatase inhibitors.Moreover, the following compounds are known in Scifinder as “Commercial Source” (CAS No. of the 2-Cl compound=321434-03-1, that of the 4-Cl compound=303144-57-2), without description of any use:Crop protection agents, which also include pesticides, have to meet many demands, for example in relation to efficacy, persistence, and spectrum of action and possible use. Questions of toxicity and of combinability with other active ingredients or formulation auxiliaries play a role, as does the question of the expense that the synthesis of an active ingredient entails. In addition, resistances can occur. For all these reasons, the search for novel crop protection compositions cannot be considered to be complete, and there is a constant need for novel compounds having properties which, compared to the known compounds, are improved at least in relation to individual aspects.It was an object of the present invention to provide compounds which ...

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16-03-2017 дата публикации

2-(HET)ARYL-SUBSTITUTED FUSED BICYCLIC HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20170073342A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. Compound of formula (I) according to in which{'sup': 1', '+', '−', '4, 'Ais nitrogen, ═N—Oor ═C—R,'}{'sup': 2', '5, 'Ais —N—R, oxygen or sulphur,'}{'sup': '3', 'Ais oxygen,'}{'sup': 4', '+', '−', '4, 'Ais nitrogen, ═N—Oor ═C—R,'}{'sup': '5', 'Ais ═C—H,'}{'sup': '1', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '3', '6', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'claim-text': {'sub': 1', '4', '1', '4', '2', '4', '2', '4', '3', '6', '1', '4', '3', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'or is (C-C)alkyl, (C-C)alkoxy, (C-C)alkenyl, (C-C)alkynyl, (C-C)cycloalkyl, each of which is optionally mono- or disubstituted identically or differently by aryl, hetaryl or heterocyclyl, where aryl, hetaryl and heterocyclyl may each optionally be mono- or disubstituted identically or differently by halogen, cyano, carbamoyl, aminosulphonyl, (C-C)alkyl, (C-C)cycloalkyl, (C-C)alkoxy, (C-C)haloalkyl, (C-C)haloalkoxy, (C-C)alkylthio, (C-C)alkylsulphinyl, (C-C)alkylsulphonyl, (C-C)alkylsulphimino, or'}, 'Ris (C-C)alkyl, (C-C)hydroxyalkyl, (C-C)haloalkyl, (C-C)cyanoalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkoxy-(C-C)alkyl, (C-C)alkenyl, (C-C)alkenyloxy-(C-C)alkyl, (C-C)haloalkenyloxy-(C-C)alkyl, (C-C)haloalkenyl, (C-C)cyanoalkenyl, (C-C)alkynyl, (C-C)alkynyloxy-(C-C)alkyl, (C-C)haloalkynyloxy-(C-C)alkyl, (C-C)haloalkynyl, (C-C)cyanoalkynyl, (C-C)cycloalkyl, (C-C)cycloalkyl(C-C)cycloalkyl, (C-C)alkyl-(C-C)cycloalkyl, halo(C-C)cycloalkyl, (C-C)alkylamino, di(C-C)alkylamino, (C-C)cycloalkylamino, (C-C)alkylcarbonylamino, (C-C) ...

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24-03-2016 дата публикации

Sram array comprising multiple cell cores

Номер: US20160086659A1
Принадлежит: International Business Machines Corp

An SRAM array having multiple cell cores to store and retrieve data. A cell core includes a plurality of SRAM cells, and at least two corresponding cell cores build a cell core row. A word decoder is configured to decode incoming address signals. The word decoder includes a cell core select unit configured to generate a cell core row select signal from a combination of a first part of the incoming address signals and a received clock signal.

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30-03-2017 дата публикации

PYRAZOLOPYRIDINE SULFONAMIDES AS NEMATICIDES

Номер: US20170088548A1
Принадлежит: Bayer CropScience Aktiengesellschaft

Disclosed are compounds of formula (I) which possess nematicidal properties 2. A compound according to claim 1 , wherein{'sup': '1', 'each Ris independently'}{'sup': '4', 'sub': 1', '4', '1', '4, 'halogen, cyano, OR, C-C-alkyl, C-C-haloalkyl;'}{'sub': 3', '7', '1', '4', '1', '4, 'or C-C-cycloalkyl, optionally substituted with 1 to 4 substituents independently selected from the group consisting of halogen, cyano, C-C-alkyl and C-C-haloalkyl;'}{'sup': '2', 'Ris'}{'sub': m', '2, 'sup': 9', '11', '12, 'H, halogen, cyano, S(O)Ror S(O)NRR;'}{'sub': 3', '6', '1', '4', '1', '4, 'or C-C-cycloalkyl, optionally substituted with 1 to 4 substituents independently selected from the group consisting of halogen, cyano, C-C-alkyl and C-C-haloalkyl;'}{'sub': 1', '4', 'm, 'sup': 4', '9, 'or C-C-alkyl substituted with 1 to 2 substituents independently selected from the group consisting of cyano, ORand S(O)R;'}{'sup': '3', 'Ris'}{'sub': 1', '4', '2', '3, 'sup': 7', '8, 'H, C-C-alkyl, C-C-alkenyl, C(X)Ror C(O)OR;'}{'sub': 1', '2, 'sup': '4', 'or C-C-alkyl substituted with OR;'}{'sub': 1', '2, 'or C-C-alkyl substituted with phenyl;'}Q is{'sub': 1', '6', '1', '6', '3', '7', '1', '6', '1', '6', 'm', '2, 'sup': 4', '7', '8', '11', '12', '9', '11', '12, 'C-C-alkyl, C-C-haloalkyl, C-C-cycloalkyl, phenyl or a 5- or 6-membered heteroaromatic ring system, each optionally substituted with 1 to 5 substituents independently selected from the group consisting of halogen, cyano, nitro, OR, C-C-alkyl, C-C-haloalkyl, C(X)R, C(O)OR, C(X)NRR, S(O)Rand S(O)NRR;'}or Q is selected from the group consisting of (U-1) to (U-61), (U-81) to (U-87), (U-89) to (U-103) and (U-105) to (U-123);{'sup': 'v', 'each Ris independently'}{'sup': 4', '7', '8', '11', '12', '9', '11', '12, 'sub': 1', '6', '1', '6', 'm', '2, 'halogen, cyano, nitro, OR, C-C-alkyl, C-C-haloalkyl, C(X)R, C(O)OR, C(X)NRR, S(O)R, S(O)NRR;'}r is 0, 1, 2 or 3, limited by the number of available positions on each U group;{'sup': '4', 'each Ris ...

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01-04-2021 дата публикации

METHOD FOR PREPARING HALOGENATED IMIDAZOPYRIDINE DERIVATIVES

Номер: US20210094947A1
Принадлежит:

The present invention relates to a method for preparing halogenated imidazopyridine derivatives of the formula (II) proceeding from compounds of the formula (I) via intermediates of the formula (IVa) or (IVb) 2. Method according to claim 1 , whereinQ is chlorine, iodine or bromine,Z is bromine, fluorine or chlorine,{'sup': 'c', 'Ris —O-pivaloyl, chlorine, bromine or iodine,'}{'sup': 1', '+', '−', '5, 'Ais nitrogen, ═N—O or ═C—R,'}{'sup': 2', '6, 'Ais —N—Ror oxygen,'}{'sup': '1', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '3', '6', '3', '6', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '3', '6', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'claim-text': {'sub': 1', '4', '1', '4', '2', '4', '2', '4', '3', '6', '1', '4', '3', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'or is (C-C)alkyl, (C-C)alkoxy, (C-C)alkenyl, (C-C)alkynyl or (C-C)cycloalkyl, each of which is optionally mono- or disubstituted by identical or different substituents from the group consisting of aryl, hetaryl and heterocyclyl, where aryl, hetaryl or heterocyclyl may each optionally be mono- or disubstituted by identical or different substituents from the group consisting of halogen, cyano, carbamoyl, aminosulfonyl, (C-C)alkyl, (C-C)cycloalkyl, (C-C)alkoxy, (C-C)haloalkyl, (C-C)haloalkoxy, (C-C)alkylthio, (C-C)alkylsulfinyl, (C-C)alkylsulfonyl and (C-C)alkylsulfimino,'}, 'Ris (C-C)alkyl, (C-C)hydroxyalkyl, (C-C)haloalkyl, (C-C)cyanoalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkoxy-(C-C)alkyl, (C-C)alkenyl, (C-C)alkenyloxy-(C-C)alkyl, (C-C)haloalkenyloxy-(C-C)alkyl, (C-C)haloalkenyl, (C-C)cyanoalkenyl, (C-C)alkynyl, (C-C)alkynyloxy-(C-C)alkyl, (C-C) ...

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14-04-2016 дата публикации

NEMATICIDAL N-(2-SUBSTITUTED 2-PHENYLETHYL)CARBOXAMIDES AND N-(2-SUBSTITUTED 2-PHENYLETHYL)-THIOCARBOXAMIDES

Номер: US20160100579A1
Принадлежит:

The present invention relates to the use of known and novel N-(2-substituted 2-phenylethyl)carboxamides and N-(2-substituted 2-phenylethyl)thiocarboxamides, for the control of plant damaging nematodes in agriculture and further relates to novel N-(2-substituted 2-phenylethyl)carboxamides and N-(2-substituted 2-phenylethyl)thiocarboxamides, processes and intermediate compounds for their preparation, their use as nematicides and their use as anthelmintics against endoparasites in animals and humans, compositions containing such compounds and methods for the control of nematodes and helminths. 4. Composition claim 2 , comprising an effective amount of at least one compound according to and at least one surfactant claim 2 , solid or liquid diluent.5. A compounds as described in capable of being used for preparation of a medicament for control of one or more animal parasites.6. A compounds as described in capable of being used for preparation of a medicament for control of helminths.7. A compound according to capable of being used for preparation of a medicament for control of one or more animal parasites.8. A compound as described in capable of being used for preparation of a medicament for control of helminths.9. A compound according to capable of being used for preparation of a medicament for control of one or more animal parasites.10. A compounds as described in capable of being used for preparation of a medicament for control of helminths.11. Composition claim 3 , comprising an effective amount of at least one compound according to and at least one surfactant claim 3 , solid or liquid diluent The present invention relates to the use of known and novel N-(2-substituted 2-phenylethyl)carboxamides and N-(2-substituted 2-phenylethyl)thiocarboxamides, for the control of plant damaging nematodes predominantly in agriculture.The present invention further relates to novel N-(2-substituted 2-phenylethyl)carboxamides and N-(2-substituted 2-phenylethyl)thiocarboxamides, ...

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13-04-2017 дата публикации

Bicyclic compounds as pesticides

Номер: US20170101422A1
Принадлежит:

The present application relates to novel bicyclic compounds, to their use for controlling animal pests and to processes and intermediates for their preparation. 9. A compound of formula (I) according to wherein T represents an electron pair.10. A compound of formula (I) according to wherein Het represents pyridin-3-yl.11. A compound of formula (I) according to wherein Het represents 5-fluoropyridin-3-yl.13. A composition claim 1 , comprising at least one compound of formula (I) according to and one or more customary extenders and/or surfactants.14. A product comprising one or more compounds of the formula (I) according to . that has been adapted-for controlling pests. The present application relates to novel bicyclic compounds, to their use for controlling animal pests and to processes and intermediates for their preparation.WO 2012/102387 A1 describes heterocyclic compounds which can be used particularly as insecticides and acaricides.WO 2003/033476 A1, WO 2004/014916 A1, WO 2008/152390, MedChemComm (2013), 4(2), 456-462, Bioorganic & Medicinal Chemistry Letters (2006), 16(18), 4723-4727, Journal of the American Pharmaceutical Association (1912-1977) (1955), 44, 193-6 and Journal of the Chemical Society (1949), 1064-8 report on the synthesis and pharmacological properties of certain [1,3]thiazolo[4,5-d]pyrimidin-7(6H)-ones or [1,3]oxazolo [4,5-d]pyrimidin-7(6H)-ones.Modern crop protection compositions have to meet many demands, for example in relation to extent, persistence and spectrum of their action and possible use. Questions of toxicity and of combinability with other active compounds or formulation auxiliaries play a role, as does the question of the expense that the synthesis of an active compound requires. In addition, resistances can occur. For all these reasons alone, the search for novel crop protection compositions cannot be considered complete, and there is a constant need for novel compounds having improved properties compared to the known compounds, ...

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21-04-2016 дата публикации

KNOWN AND NEW HETEROCYCLIC COMPOUNDS AS PEST CONTROL AGENTS

Номер: US20160106102A1
Принадлежит:

The present application relates to the use of known and novel heterocyclic compounds for controlling animal pests, to novel heterocyclic compounds, to processes for preparation thereof and to the use thereof for controlling animal pests. 3. Composition claim 1 , comprising a content of at least one compound of formula (I) according to and one or more customary extenders and/or surfactants.4. Composition claim 2 , comprising a content of at least one compound of formula (I) according to and one or more customary extenders and/or surfactants.5. Method for controlling one or more pests claim 1 , comprising allowing a compound of formula (I) according to to act on the pests and/or a habitat thereof.6. A compound of formula (I) according to capable of being used for controlling one or more pests. The present application relates to the use of known and novel heterocyclic compounds for controlling animal pests, to novel heterocyclic compounds, to processes for preparation thereof and to the use thereof for controlling animal pests.WO 2011/049987 A2, WO 2011/106114 A1, WO 2009/025793 A2, US 2008/0103182 A1, WO 2007/055941 A2, WO 2006/114313 A1, US 2009/0163545 A1 and FR 2836915 A1 disclose heterocyclic compounds for which pharmaceutical uses are described. U.S. Pat. No. 2,511,231 and JP 63218665 A disclose heterocyclic compounds for use in photography. The literature describes particular substituted pyridines as insecticides; see, for example WO 2003/097604 A1. WO 2005/074686 A1 and WO 2008/014905 A2 disclose carboxamides for control of unwanted microorganisms.The heterocyclic compounds of the formulae (G1), (G2) and (G4) are known. No use for these compounds has been described.In the case of compounds G1-1, G1-5, G1-6, G1-17, G1-71, G1-79 to G1-82 and G1-96 to G1-98 and G1-103, the Yand Ycolumns also show the carbon atoms bonded to Yand Yand the nitrogen atom bonded to Z. The same applies to all the tables in this patent application in which Yand Yoccur together.Modern ...

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21-04-2016 дата публикации

BICYCLIC ARYL SULFIDE AND ARYL SULFOXIDE DERIVATIVES AS PEST CONTROL AGENT

Номер: US20160108038A1
Принадлежит:

The present application relates to novel heterocyclic compounds, to processes for their preparation, to their use for controlling animal pests including arthropods and in particular insects and acarids, and to intermediates for preparing the heterocyclic compounds. 2. Compound according to claim 1 , in whichV represents oxygen;Q represents C—R or nitrogen;R represents hydrogen, hydroxy, halogen, cyano, alkyl, cycloalkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, amino, monoalkylamino or dialkylamino;{'sup': 1', '1, 'Qrepresents C—Ror nitrogen;'}{'sup': 2', '2, 'Qrepresents C—Ror nitrogen;'}{'sup': 3', '3, 'Qrepresents C—Ror nitrogen;'}{'sup': 4', '4, 'claim-text': {'sup': 1', '2', '3', '4', '1', '2', '3', '4, 'where at least one of the structural elements Q, Q, Q, Qis nitrogen and at most two of the structural elements Q, Q, Q, Qare nitrogen;'}, 'Qrepresents C—Ror nitrogen;'}{'sup': 1', '2', '3', '4, 'R, R, R, Reach independently of one another represent hydrogen, hydroxy, halogen, cyano, alkyl, cycloalkyl, haloalkyl, alkoxy, haloalkoxy, hetaryl, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, amino, monoalkylamino or dialkylamino;'}W represents hydrogen or halogen;n represents the number 0 or 1; represents hydrogen, fluorine, chlorine, bromine, cyano, nitro, amino, hydroxyl, alkyl, haloalkyl, alkenyl, alkynyl, alkoxy, haloalkoxy or aminothiocarbonyl;', 'or represent benzyl, phenoxy, phenylthio, cyclopropylmethyl, cyclopropyloxy or cyclopropylthio, which is optionally mono- or polysubstituted identically or differently by fluorine, chlorine, bromine, cyano, nitro, hydroxyl, amino, methyl, ethyl, trifluoromethyl, difluoromethyl, trifluoroethyl, difluoroethyl, methoxy, ethoxy, trifluoromethoxy, trifluoroethoxy, or optionally methyl-, fluorine-, chlorine- or cyano-substituted cyclopropyl;', 'or represent cyclopropyl, cyclobutyl, cyclopentyl, ...

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27-04-2017 дата публикации

NOVEL PYRAZOLYLTRIAZOLYLPYRIDINES AS PESTICIDES

Номер: US20170112129A1
Принадлежит:

The invention encompasses novel pyrazolyltriazolylpyridines of the general formula (I) in which the radicals A-A, W, Q, R, Rand Z-Zhave the meanings given in the description. Also described are processes for preparing the compounds of the formula (I). The compounds according to the invention are especially suitable for controlling insects and arachnids in agriculture, and ectoparasites in veterinary medicine. 2. Compound of formula (I) according to in which{'sup': '1', 'sub': 1', '6', '2', '6', '2', '6', '3', '7', '3', '7', '1', '3', '1', '6', '1', '6', '1', '6', '1', '6', '1', '3', '1', '3, 'Rrepresents hydrogen, or C-C-alkyl, C-C-alkenyl, C-C-alkynyl, C-C-cycloalkyl, C-C-cycloalkyl-C-C-alkyl, C-C-alkylcarbonyl, C-C-alkoxycarbonyl, C-C-alkoxy-C-C-alkyl, aryl-(C-C)-alkyl, heteroaryl-(C-C)-alkyl, each of which is optionally mono- or polysubstituted independently of one another by halogen, cyano, alkoxy and alkoxycarbonyl;'}the chemical moieties{'sub': '1', 'sup': '2', 'Arepresents CRor nitrogen,'}{'sub': '2', 'Arepresents nitrogen,'}{'sub': '3', 'sup': '3', 'Arepresents CRor nitrogen, and'}{'sub': '4', 'sup': '4', 'Arepresents CRor nitrogen,'}{'sub': 1', '4, 'but where not more than three of the chemical moieties Ato Asimultaneously represent nitrogen;'}{'sup': 2', '3', '4, 'sub': 1', '6', '3', '7', '1', '6', '1', '6', '1', '3', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6, 'R, Rand Rindependently of one another represent hydrogen, halogen, cyano, nitro, in each case optionally substituted C-C-alkyl, C-C-cycloalkyl, C-C-alkoxy, N—(C-C-alkoxy)imino-C-C-alkyl, C-C-alkylsulphanyl, C-C-alkylsulphinyl, C-C-alkylsulphonyl, N—(C-C-alkyl)amino, N,N-di(C-C-alkyl)amino, C-C-alkylsulphonylamino, or N—(C-C-alkyl)-C-C-alkylsulphonylamino;'}W represents oxygen or sulphur;{'sub': 1', '6', '1', '6', '2', '6', '2', '6', '3', '7', '1', '6', '3', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6, 'Q represents hydrogen, hydroxy, formyl or ...

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27-04-2017 дата публикации

HALOGEN-SUBSTITUTED COMPOUNDS

Номер: US20170114021A1
Принадлежит: Bayer Animal Health GmbH

The invention encompasses inter alia halogen-substituted compounds of the general formula (I) in which the radicals A-A, T, W, Q, Rand Z-Zhave the meanings given in the description. Also described are processes for preparing the compounds of the formula (I). The compounds according to the invention are especially suitable for controlling insects, arachnids and nematodes in agriculture, and ectoparasites in veterinary medicine. 2. Compound of formula (I) according to in which Zand Zindependently of one another represent perhalogenated C-C-alkyl and Zrepresents C-C-alkyl.3. Compound of formula (I) according to in which Zrepresents perfluorinated ethyl (CF) claim 1 , Zrepresents perfluorinated methyl (CF) and Zrepresents methyl.4. Compound of formula (I) according to claim 1 , in which T represents T3 (formula (Ic)) claim 1 , T6 (formula (If)) claim 1 , T7 (formula (Ig)) or T8 (formula (Ih)).5. Compound of formula (I) according to claim 1 , in which Q represents hydrogen claim 1 , C-C-alkyl claim 1 , C-C-cycloalkyl claim 1 , C-C-alkoxy or benzyl.6. Compound of formula (I) according to claim 1 , in whichT represents T3 (formula (Ic)), T6 (formula (If)), T7 (formula (Ig)) or T8 (formula (Ih)) and n in T represents 0;{'sub': 1', '2', '2, 'Arepresents CR, where Rrepresents hydrogen;'}{'sub': 2', '3', '3, 'Arepresents CR, where Rrepresents hydrogen;'}{'sub': 3', '4', '4', '1', '4', '1', '4, 'Arepresents CR, where Rrepresents hydrogen, halogen, (C-C)-alkyl or (C-C)-alkoxy;'}{'sub': 4', '5', '5, 'Arepresents CR, where Rrepresents hydrogen;'}W represents oxygen;n in T represents 0;{'sup': '1', 'sub': 1', '4, 'Zrepresents halogenated (C-C)-alkyl;'}{'sup': '2', 'sub': 1', '4, 'Zrepresents halogenated (C-C)-alkyl;'}{'sup': '3', 'sub': 1', '4, 'Zrepresents (C-C)-alkyl;'}{'sub': 1', '1', '4, 'Rrepresents hydrogen or C-C-alkyl;'}{'sup': 1', '1, 'sub': 1', '6', '3', '6, 'Q represents hydrogen or a group, optionally substituted by at least one radical M, selected from the group ...

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13-05-2021 дата публикации

HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20210139480A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. The compound according to claim 1 , wherein{'sup': '1', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '3', '6, 'Rrepresents (C-C)alkyl, (C-C)cyanoalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkyl, (C-C)alkenyl, (C-C)haloalkenyl, (C-C)alkynyl, (C-C)haloalkynyl or (C-C)cycloalkyl,'}{'sup': '2', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '3', '6', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Rrepresents hydrogen, (C-C)alkyl, (C-C)haloalkyl, (C-C)cyanoalkyl, (C-C)hydroxyalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkoxy-(C-C)alkyl, (C-C)cycloalkyl, (C-C)cycloalkyl-(C-C)cycloalkyl, (C-C)alkyl-(C-C)cycloalkyl, halo(C-C)cycloalkyl, cyano(C-C)cycloalkyl, (C-C)alkylthio-(C-C)alkyl, (C-C)haloalkylthio-(C-C)alkyl, (C-C)alkyl sulfinyl-(C-C)alkyl, (C-C)haloalkyl sulfinyl-(C-C)alkyl, (C-C)alkylsulfonyl-(C-C)alkyl or (C-C)haloalkylsulfonyl-(C-C)alkyl,'}{'sup': '3', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '2', '4', '2', '4', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Rrepresents aryl which is optionally mono- or disubstituted by identical or different substituents or represents a saturated, partially saturated or heteroaromatic ring which is optionally mono- or disubstituted by identical or different substituents, where at least one carbon atom is replaced by a heteroatom from the group consisting of N, O and ...

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05-05-2016 дата публикации

HETEROCYCLIC COMPOUNDS AS PEST CONTROL AGENTS

Номер: US20160122353A1
Принадлежит:

The present application relates to the use of known and novel heterocyclic compounds for controlling animal pests, to novel heterocyclic compounds, to processes for preparation thereof and to the use thereof for controlling animal pests. 4. Composition claim 1 , comprising a content of at least one compound of formula (I) according to and one or more customary extenders and/or surfactants.5. Composition claim 2 , comprising a content of at least one compound of formula (Ia) according to and one or more customary extenders and/or surfactants.6. Composition claim 3 , comprising a content of at least one compound of formula (Ib) according to and one or more customary extenders and/or surfactants.7. A compound of formula (Ia) according to capable of being used for controlling one or more pests.8. A compound of formula (Ib) according to capable of being used for controlling one or more pests. The present application relates to the use of known and novel heterocyclic compounds for controlling animal pests, to novel heterocyclic compounds, to processes for preparation thereof and to the use thereof for controlling animal pests.WO 2012/102387 A1 describes heterocyclic compounds which can be used particularly as insecticides and acaricides.Heterocyclic compounds for pharmaceutical applications are disclosed in WO 2004/009597 A2, WO 2008/107418 A1, WO 2009/068617 A1 and US 2004/242596 A1.WO 2004/099211 A1 describes 6-cyclylmethyl- and 6-alkylmethyl-substituted pyrazolopyrimidines for pharmaceutical applications.Bioorganic & Medicinal Chemistry Letters (2007), 17(15), 4303-4307 reports synthesis and pharmacological properties of particular pyrazolo[3,4-d]pyrimidin-4-ones.Modern crop protection compositions have to meet many demands, for example in relation to efficacy, persistence and spectrum of their action and possible use. Questions of toxicity and of combinability with other active ingredients or formulation auxiliaries play a role, as does the question of the cost and ...

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25-04-2019 дата публикации

SUBSTITUTED 2-ALKYLIMIDAZOLYLCARBOXAMIDES AS PESTICIDES

Номер: US20190119250A1
Принадлежит:

The present invention relates to compounds of the general formula (I) 3. A compound according to whereinQ represents oxygen or sulphur,V represents a radical from the group consisting of hydrogen, fluorine, chlorine, bromine, methyl, ethyl, difluoromethyl, trifluoromethyl, methoxy, ethoxy, difluoromethoxy, trifluoromethoxy and cyano,W represents a radical from the group consisting of hydrogen, fluorine, chlorine, bromine, methyl, ethyl, difluoromethyl, trifluoromethyl, methoxy, ethoxy, difluoromethoxy, trifluoromethoxy and cyano,{'sub': 1', '4', '3', '4', '3', '4', 'n', 'n', '3', '6', '3', '6', '1', '2', 'n, 'sup': '4', 'Y represents a radical from the group consisting of hydrogen; C-C-alkyl, C-C-alkenyl and C-C-alkynyl, optionally mono- to pentasubstituted independently of one another by fluorine, chlorine, bromine, methoxy, ethoxy, methyl-S(O)—, ethyl-S(O)—, cyano; C-C-cycloalkyl, optionally mono- or disubstituted independently of one another by fluorine, chlorine, bromine, methyl, ethyl, trifluoromethyl, methoxy, ethoxy, cyano; straight-chain or branched C-C-cycloalkyl-C-C-alkyl, optionally interrupted once or twice independently of one another by O, S(O), NRand optionally mono- to tetrasubstituted independently of one another by fluorine, chlorine, bromine, methyl, ethyl, trifluoromethyl, methoxy, ethoxy, cyano; and cyano,'}{'sub': 1', '6', '3', '6', '3', '6', 'n', 'n', '3', '6', '3', '6', '1', '2, 'A represents a radical from the group consisting of hydrogen; C-C-alkyl, C-C-alkenyl or C-C-alkynyl, optionally mono- to pentasubstituted independently of one another by fluorine, chlorine, bromine, methoxy, ethoxy, methyl-S(O)—, ethyl-S(O)— or cyano; C-C-cycloalkyl, optionally mono- or disubstituted independently of one another by fluorine, chlorine, bromine, methyl, ethyl, trifluoromethyl, methoxy, ethoxy or cyano; and straight-chain or branched C-C-cycloalkyl-C-C-alkyl, optionally mono- or disubstituted independently of one another by fluorine, chlorine, bromine, ...

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27-05-2021 дата публикации

HETEROARYL-TRIAZOLE AND HETEROARYL-TETRAZOLE COMPOUNDS AS PESTICIDES

Номер: US20210155608A1
Принадлежит:

The present invention relates to novel heteroaryl-triazole and heteroaryl-tetrazole compounds of the general formula (I), in which the structural elements Y, Q, Q, R, R, R, R, Rand Rhave the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals. 2. Compound according to claim 1 , in whichX is O or S;{'sup': 1', '2', '5', '1', '2, 'Qand Qare independently CRor N, provided at least one of Qand Qis N;'}{'sub': '2', 'Y is a direct bond or CH;'}{'sup': '1', 'sub': 1', '6', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3, 'claim-text': or', {'sub': 3', '6', '2', '1', '6', '1', '6', '3', '6', '1', '6', '2', '1', '4', '1', '4', '1', '4', '2, 'C-Ccycloalkyl optionally substituted with one or two substituents selected from the group consisting of halogen, CN, —COOH, —CONH, C-Calkyl, C-Chaloalkyl, C-Ccycloalkyl, C-Calkoxy, —COC-Calkyl, —CONH(C-Calkyl), and —CON(C-Calkyl);'}, 'or', {'sub': 1', '2', '2', '1', '6', '1', '6', '3', '6', '1', '6', '1', '6', '2', '1', '4', '1', '4', '1', '4', '2', '1', '6', '3', '6', '1', '3', '1', '4', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3, 'cyclopropyl-C-Calkyl wherein the cyclopropyl is substituted with one or two substituents each independently selected from the group consisting of halogen, CN, —COOH, —CONH, C-Calkyl, C-Chaloalkyl, C-Ccycloalkyl, C-Calkoxy, C-Chaloalkoxy, —COC-Calkyl, —CONH(C-Calkyl), —CON(C-Calkyl), and phenyl optionally substituted by one to three substituents independently selected from the group consisting of halogen, CN, C-Calkyl, C-Ccycloalkyl, C-Chaloalkyl, C-Calkoxy, C-Chaloalkoxy, C-Calkylthio, C-Calkylsulfinyl, C-Calkylsulfonyl, C-Chaloalkylthio, C-Chaloalkylsulfinyl, and C-Chaloalkylsulfonyl;'}, 'or', {'sub': 5', '6', '1', '2', '5', '6 ...

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12-05-2016 дата публикации

ARYL SULFIDE DERIVATIVES AND ARYL SULFOXIDE DERIVATIVES AS ACARICIDES AND INSECTICIDES

Номер: US20160130240A1
Принадлежит:

The present invention relates to aryl sulfoxide derivatives, to the use thereof as acaricides and insecticides for controlling animal pests and to processes and intermediates for preparation thereof. The aryl sulfide and aryl sulfoxide derivatives have the general structure (I) 3. The compound as claimed in in whichA and B together with the atoms to which they are attached represent a substructure selected from the group consisting of (I-A) to (I-D),where{'sup': 1', '2', '3, 'claim-text': {'sup': 11', '11, 'represent oxygen; sulfur, NRor a salt of NR;'}, 'V, Vand Veach independently of one another'}{'sup': 1', '1', '2, 'Qrepresents oxygen, sulfur, NRor CRR;'}{'sup': 2', '10', '8', '9, 'Qrepresents NRor CRR;'}{'sup': '1', 'claim-text': represents alkyl, cycloalkylalkyl, haloalkyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, aminoalkyl, alkoxycarbonylalkyl, alkylsulfanylalkyl, alkylsulfinylalkyl, alkylsulfonylalkyl, haloalkylsulfanylalkyl, haloalkylsulfinylalkyl, haloalkylsulfonylalkyl, alkoxyalkylsulfanylalkyl, alkoxyalkylsulfinylalkyl, alkoxyalkylsulfonylalkyl, phenylalkyl, phenoxyalkyl, phenylsulfanylalkyl, phenylsulfinylalkyl, phenylsulfonylalkyl, hetarylalkyl, hetaryloxyalkyl, hetarylthioalkyl, alkoxycarbonyl, aryloxycarbonyl, arylcarbamoyl, where the aforementioned radicals may each be saturated or unsaturated and/or optionally substituted; or', 'represents optionally substituted saturated or unsaturated cycloalkyl which may optionally be interrupted by one or more heteroatoms; or', 'represents haloalkylcarbonyl, hydroxyalkylcarbonyl, alkoxyalkylcarbonyl, phenylcarbonyl, hetarylcarbonyl, haloalkoxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, cycloalkylaminocarbonyl, dicycloalkylaminocarbonyl, cycloalkyl(alkyl)aminocarbonyl, arylaminocarbonyl, diarylaminocarbonyl, alkyl(aryl)aminocarbonyl, cycloalkyl(aryl)aminocarbonyl, alkylaminothiocarbonyl, dialkylaminothiocarbonyl or aminothiocarbonyl, where the aforementioned radicals may each be saturated ...

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18-05-2017 дата публикации

NOVEL HALOGEN-SUBSTITUTED COMPOUNDS

Номер: US20170137413A1
Принадлежит:

The invention relates inter alia to halogen-substituted compounds of the general formula (I) 7. A compound according to in which Zrepresents CFCF claim 6 , Zrepresents CF claim 6 , Zrepresents CH claim 6 , the radicals Rand Rrepresent hydrogen claim 6 , Aand Arepresent CH claim 6 , Arepresents CH or N claim 6 , Arepresents C—Cl claim 6 , W represents oxygen and Q represents 1-cyanocyclopropyl or cyclopropyl.8. A compound formula (I) according to for controlling one or more insects claim 1 , arachnids and/or nematodes.9. A pharmaceutical composition comprising at least one compound according to .10. A compound according to for use as a medicament.11. A compound according to for producing a pharmaceutical composition for controlling one or more parasites on animals.12. A process for producing a crop protection composition comprising mixing a compound according to and one or more customary extenders and/or surfactants.13. A method for controlling one or more pests claim 1 , comprising allowing a compound according to to act on the pests and/or a habitat thereof.14. A compound according to for protecting the propagation material of one or more plants. The present application relates to novel halogen-substituted compounds, to processes for their preparation and to their use for controlling animal pests, in particular arthropods and especially insects, arachnids and nematodes.It is known that similar compounds are used as FAAH inhibitors [WO2009-152025], LXR modulators [WO2007-002559] and ATP binding cassette transporter modulators [WO2004-080972].Modern crop protection compositions have to meet many demands, for example in relation to extent, persistence and spectrum of their action and possible use. Questions of toxicity and of combinability with other active compounds or formulation auxiliaries play a role, as does the question of the expense that the synthesis of an active compound requires. In addition, resistances can occur. For all these reasons, the search for ...

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10-06-2021 дата публикации

HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20210169080A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. Compound of formula (I) according to claim 1 , in which{'sup': '1', 'Arepresents N (nitrogen) or C(H),'}{'sup': '2', 'Arepresents N (nitrogen) or C(H),'}{'sup': '3', 'Arepresents oxygen or sulfur,'}{'sup': '1', 'sub': 1', '6', '1', '6', '2', '6', '2', '6', '2', '6', '2', '6', '3', '8', '3', '8', '3', '6', '1', '6', '3', '6', '1', '6', '1', '6', '3', '8', '1', '6', '3', '8', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6, 'Rrepresents (C-C)-alkyl, (C-C)-haloalkyl, (C-C)-alkenyl, (C-C)-haloalkenyl, (C-C)-alkynyl, (C-C)-haloalkynyl, (C-C)-cycloalkyl, halo-(C-C)-cycloalkyl, (C-C)-cycloalkyl-(C-C)-alkyl, (C-C)-cycloalkyl-(C-C)-haloalkyl, (C-C)-alkyl-(C-C)-cycloalkyl, (C-C)-haloalkyl-(C-C)-cycloalkyl, (C-C)-cyanoalkyl, (C-C)-hydroxyalkyl, (C-C)-alkoxy-(C-C)-alkyl, (C-C)-haloalkoxy-(C-C)-alkyl, (C-C)-alkylthio-(C-C)-alkyl, (C-C)-alkylsulfinyl-(C-C)-alkyl or (C-C)-alkylsulfonyl-(C-C)-alkyl,'}{'sup': 2', '3, 'sub': 1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6, 'claim-text': [{'sub': 1', '6', '3', '8', '1', '6', '3', '8', '1', '6', '3', '8', '1', '6', '3', '8', '3', '6', '1', '4', '3', '8', '3', '8', '4-12, 'represent (C-C)-haloalkyl-(C-C)-cycloalkyl, (C-C)-cyanoalkyl-(C-C)-cycloalkyl, (C-C)-haloalkyl-(C-C)-cyanocycloalkyl, (C-C)-haloalkyl-(C-C)-halocycloalkyl, cyano-(C-C)-cycloalkyl which is optionally mono- or polysubstituted by (C-C)-alkyl or halogen, spiro-(C-C)-cycloalkyl-(C-C)-cycloalkyl which is optionally mono- or polysubstituted by cyano or halogen or (C)-bicycloalkyl which is optionally mono- or polysubstituted by cyano or halogen,'}, {'sup': 2', '3, 'sub': 1', '6', '3', '8', '1', '6', '3', '8', '1', '6', '3', '8', '1', '6', '3', '8', '3', '6', '1', '4', '3', '8', '3', '8', '4', '12, 'where one of the radicals Ror Rmust be selected from (C-C)-haloalkyl-(C-C)-cycloalkyl, (C-C)-cyanoalkyl-(C-C)-cycloalkyl, (C-C)- ...

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26-05-2016 дата публикации

ARYL SULFIDE DERIVATIVES AND ARYL SULFOXIDE DERIVATIVES AS ACARICIDES AND INSECTICIDES

Номер: US20160145235A1
Принадлежит:

The present invention relates to aryl sulphide and aryl sulphoxide derivatives, to the use thereof as acaricides and insecticides for controlling animal pests and to processes and intermediates for preparation thereof. The aryl sulphide and aryl sulphoxide derivatives have the general structure (I) 3. Compound according to in whichA and B together with the atoms to which they are bonded are a substructure selected from the group consisting of I-A to I-G;{'sup': '1', 'claim-text': [{'sub': 1', '6', '3', '6', '1', '6', '2', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6, 'is (C-C)alkyl, (C-C)cycloalkyl(C-C)alkyl, halo(C-C)alkyl, cyano(C-C)alkyl, hydroxy(C-C)alkyl, (C-C)alkoxy(C-C)alkyl, amino(C-C)alkyl, (C-C)alkoxycarbonyl(C-C)alkyl, (C-C)alkylsulphanyl(C-C)alkyl, (C-C)alkylsulphinyl(C-C)alkyl, (C-C)alkylsulphonyl(C-C)alkyl, halo(C-C)alkylsulphanyl(C-C)alkyl, halo(C-C)alkylsulphinyl(C-C)alkyl, halo(C-C)alkylsulphonyl(C-C)alkyl, (C-C)alkoxy(C-C)alkylsulphanyl(C-C)alkyl, (C-C)alkoxy(C-C)alkylsulphinyl(C-C)alkyl, (C-C)alkoxy(C-C)alkylsulphonyl(C-C)alkyl, phenyl(C-C)alkyl, phenoxy(C-C)alkyl, phenylsulphanyl(C-C)alkyl, phenylsulphinyl(C-C)alkyl, phenylsulphonyl(C-C)alkyl, hetaryl(C-C)alkyl, hetaryloxy(C-C)alkyl, hetarylsulphanyl(C-C)alkyl, hetarylsulphinyl(C-C)alkyl, hetarylsulphonyl(C-C)alkyl, where the aforementioned radicals may each optionally be substituted and/or, under the condition that, in the case of an unsaturated radical, the defined minimum number of carbon atoms is 2, the radicals may be saturated or unsaturated; or'}, {'sub': 3', '6, 'is optionally substituted saturated or unsaturated (C-C)cycloalkyl which may optionally be ...

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25-05-2017 дата публикации

ARYL-TRIAZOLYL PYRIDINES AS PEST CONTROL AGENTS

Номер: US20170144988A1
Принадлежит:

The invention relates to novel aryltriazolylpyridines of the general formula (I). Also described are processes for preparing the compounds of the formula (I). The compounds according to the invention are especially suitable for controlling insects and arachnids in agriculture, and ectoparasites in veterinary medicine. 2. Compound of formula (I) and/or a salt claim 1 , N-oxide and/or a tautomeric form according to in which{'sup': '1', 'Rrepresents hydrogen, methyl, ethyl, n-propyl, isopropyl, n-butyl, isobutyl, s-butyl, t-butyl, methoxymethyl, ethoxymethyl, propoxymethyl, 2-propyn-1-yl, 2-propen-1-yl, methylcarbonyl, ethylcarbonyl, n-propylcarbonyl, isopropylcarbonyl, s-butylcarbonyl, t-butylcarbonyl, methoxycarbonyl, ethoxycarbonyl, n-propoxycarbonyl, isopropoxycarbonyl, s-butoxycarbonyl, t-butoxycarbonyl, cyanomethyl, 2-cyanoethyl, benzyl, 4-methoxybenzyl, pyrid-2-ylmethyl, pyrid-3-ylmethyl, pyrid-4-ylmethyl, 4-chloropyrid-3-ylmethyl, preferably hydrogen, methyl, ethyl, n-propyl, isopropyl, n-butyl, isobutyl, s-butyl or t-butyl;'}the chemical moieties{'sub': '1', 'sup': '2', 'Arepresents CRor nitrogen,'}{'sub': '2', 'Arepresents nitrogen,'}{'sub': '3', 'sup': '3', 'Arepresents CRor nitrogen, and'}{'sub': '4', 'sup': '4', 'Arepresents CRor nitrogen,'}{'sub': '1', 'sup': '5', 'Brepresents CRor N,'}{'sub': '2', 'sup': '6', 'Brepresents CRor N,'}{'sub': '3', 'sup': '7', 'Brepresents CRor N,'}{'sub': '4', 'sup': '8', 'Brepresents CRor N, and'}{'sub': '5', 'sup': '9', 'Brepresents CRor N,'}{'sub': 1', '4', '1', '5, 'but not more than two of the chemical moieties Ato Asimultaneously represent nitrogen and not more than two of the moieties Bto Bsimultaneously represent nitrogen;'}{'sup': 2', '4, 'Rand Rindependently of one another represent hydrogen, methyl, fluorine or chlorine; and'}{'sup': '3', 'Rrepresents hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro, methyl, ethyl, fluoromethyl, difluoromethyl, chlorodifluoromethyl, trifluoromethyl, 2,2,2-trifluoroethyl ...

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15-09-2022 дата публикации

5-AMINO-SUBSTITUTED PYRAZOLES AND TRIAZOLES AS PEST CONTROL AGENTS

Номер: US20220289691A1
Принадлежит: Bayer Aktiengesellschaft

The invention relates to novel compounds of the formula (I) 7. A formulation comprising at least one compound of the formula (I) according to .8. The formulation of claim 7 , further comprising at least one extender and/or at least one surface-active substance.9. The formulation of claim 7 , wherein the compound of the formula (I) is in a mixture with at least one further active compound.10. A method for controlling pests claim 1 , comprising applying a compound of formula (I) according to claim 1 , to the pests and/or their habitat.11. The method of claim 10 , wherein the pests are animal pests and comprise an insect claim 10 , an arachnid or a nematode claim 10 , or wherein the pests are insects claim 10 , arachnids or nematodes.12. A method for controlling pests claim 7 , comprising applying a formulation according to claim 7 , to the pests and/or their habitat.13. The method of claim 12 , wherein the pests are animal pests and comprise an insect claim 12 , an arachnid or a nematode claim 12 , or wherein the pests are insects claim 12 , arachnids or nematodes.14. A method for controlling animal pests in crops claim 12 , comprising applying a compound of formula (I) directly to the crop plant or crop plant parts claim 12 , or to their surroundings claim 12 , habitat or storage space.15. A method for protecting seed or a germinating plant from pests claim 1 , comprising contacting the seed with a compound of formula (I) according to .16. A seed obtained by a method according to .17. The method of claim 15 , wherein the pests are animal pests. The present invention relates to novel 5-amino-substituted pyrazoles and triazoles, to processes for their preparation and to their use for controlling animal pests, especially arthropods and in particular insects, arachnids and nematodes.Certain amino-substituted triazoles and pyrazoles having insecticidal action are already known (WO2002090335). Furthermore, triazoles and pyrazoles, substituted in the 5-position or ...

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17-06-2021 дата публикации

Hood Prop

Номер: US20210180383A1
Автор: Joseph Kugel
Принадлежит: Individual

A hood prop attaches to right and left side hoods and engages a receptacle plate attached to a fire wall. The hood prop includes a mounting plate attached to hood latch fasteners at a bottom rear position of each side hood. A mounting plate end of a prop arm is pivotally attached by a friction fit. The friction fit allows the arm to pivot on the rod but retain a position to reduce or eliminate any rattles. The arm includes at least one bend to align a firewall end of the prop arm with a receptacle reaching out from the receptacle plate.

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23-05-2019 дата публикации

SUBSTITUTED HALOGEN(THIO)ACYL COMPOUNDS

Номер: US20190150445A1
Принадлежит:

The present invention relates to novel substituted halogen(thio)acyl compounds according to formula(I), to processes for their preparation and to their use for controlling animal pests, especially arthropods, in particular insects. 2. A compound according to claim 1 , in which{'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'A represents pyrimidin-5-yl which is optionally substituted in the 2-position by halogen or C-C-alkyl, represents 1H-pyrazol-4-yl which is optionally substituted in the 1-position by C-C-alkyl and in the 3-position by halogen, represents 1H-pyrazol-5-yl which is optionally substituted in the 2-position by halogen or C-C-alkyl, represents isoxazol-5-yl which is optionally substituted in the 3-position by halogen or C-C-alkyl, represents 1,2,4-oxadiazol-5-yl which is optionally substituted in the 3-position by halogen or C-C-alkyl, represents 1-methyl-1,2,4-triazol-3-yl or represents 1,2,5-thiadiazol-3-yl, or'}n represents 0 or 1.D represents sulfur,G represents hydrogen,Q represents sulphur or NH,{'sup': '1', 'Rrepresents hydrogen,'}{'sup': '2', 'Rrepresents halogen,'}{'sup': '3', 'Rrepresents halogen,'}Z represents halogen or halogenalkyl.3. A compound according to claim 1 , in whichA represents one of the radicals 5,6-difluoropyrid-3-yl, 5-chloro-6-fluoropyrid-3-yl, 5-bromo-6-fluoropyrid-3-yl, 5-iodo-6-fluoropyrid-3-yl, 5-fluoro-6-chloropyrid-3-yl, 5, 6-dichloropyrid-3-yl, 5-bromo-6-chloropyrid-3-yl, 5-iodo-6-chloropyrid-3-yl, 5-fluoro-6-bromopyrid-3-yl, 5-chloro-6-bromopyrid-3-yl, 5, 6-dibromopyrid-3-yl, 5-iodo-6-bromopyrid-3-yl, 5-fluoro-6-iodopyrid-3-yl, 5-chloro-6-iodopyrid-3-yl, 5-bromo-6-iodopyrid-3-yl, 5, 6-diiodopyrid-3-yl, 5-methyl-6-fluoropyrid-3-yl, 5-methyl-6-chloropyrid-3-yl, 5-methyl-6-bromopyrid-3-yl, 5-methyl-6-iodopyrid-3-yl, 5-difluoromethyl-6-fluoropyrid-3-yl, 5-difluoromethyl-6-chloropyrid-3-yl, 5-difluoromethyl-6-bromopyrid-3-yl, 5-difluoromethyl-6-iodopyrid-3-yl .n represents 0 or 1.D represents oxygen,G represents ...

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14-05-2020 дата публикации

MESOIONIC IMIDAZOPYRIDINES AS INSECTICIDES

Номер: US20200146292A1
Принадлежит:

Provided are compounds of the formula (I) 3. The compound according to claim 1 , in which{'sup': 5a', '5b', '5c, 'sub': 2', '4', '3', '4', '3', '6', '2', '4', '3', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'claim-text': 'or', 'T represents hydrogen, C(R)(R)(R), C-C-alkenyl, C-C-alkynyl or C-C-cycloalkyl, where C-C-alkenyl, C-C-alkynyl or C-C-cycloalkyl may each optionally be mono- to trisubstituted and the substituents independently of one another are selected from the group consisting of halogen, and/or may each optionally be monosubstituted and the substituent is selected from the group consisting of cyano, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-haloalkoxy, C-C-alkylthio, C-C-alkylsulfinyl and C-C-alkylsulfonyl,'}{'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'claim-text': 'or', 'T represents phenyl, C-C-alkylenedioxyphenyl, naphthyl, furanyl, thienyl, pyrrolyl, pyrazolyl, imidazolyl, 1,2,3-triazolyl, 1,2,4-triazolyl, oxazolyl, isoxazolyl, thiazolyl, isothiazolyl, 1,2,3-oxadiazolyl, 1,2,4-oxadiazolyl, 1,3,4-oxadiazolyl, 1,2,5-oxadiazolyl, 1,2,3-thiadiazolyl, 1,2,4-thiadiazolyl, 1,3,4-thiadiazolyl, 1,2,5-thiadiazolyl, pyridyl, pyrimidyl, thiophenyl, pyridazinyl, pyrazinyl, 1,2,3-triazinyl, 1,2,4-triazinyl, 1,3,5-triazinyl, benzofuranyl, indolyl, benzothiazolyl, benzoxazolyl, benzimidazolyl, pyrazolopyridinyl, quinolinyl, isoquinolinyl, cinnolinyl, azetidinyl, azolidinyl, azinanyl, oxetanyl, oxolanyl, oxanyl, dioxanyl, thiethanyl, thiolanyl, thianyl, or dihydroisoxazolyl, where the radicals mentioned above may each optionally be mono- to tetrasubstituted and the substituents independently of one another are selected from the group consisting of fluorine and chlorine, and/or may each optionally be mono- to disubstituted and the substituents independently of one another are selected from the group consisting of bromine, nitro, cyano, C- ...

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14-05-2020 дата публикации

2-(HET)ARYL-SUBSTITUTED FUSED HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20200146293A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. Compound of formula (I) according to wherein{'sup': 1', '+', '−', '5, 'Ais nitrogen, ═N(O)— or ═C(R)—,'}{'sup': 2', '6, 'Ais —N(R)— or oxygen,'}{'sup': '1', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '3', '6', '3', '6', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '3', '6', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'claim-text': {'sub': 1', '4', '1', '4', '2', '4', '2', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'or is in each case optionally identically or differently mono- or di-aryl-, -hetaryl- or -heterocyclyl-substituted (C-C)alkyl, (C-C)alkoxy, (C-C)alkenyl, (C-C)alkynyl or (C-C)cycloalkyl, where aryl, hetaryl or heterocyclyl are each optionally identically or differently mono- or disubstituted by halogen, cyano, carbamoyl, aminosulfonyl, (C-C)alkyl, (C-C)cycloalkyl, (C-C)alkoxy, C-C)haloalkyl, (C-C)haloalkoxy, (C-C)alkylthio, (C-C)alkylsulfinyl, (C-C)alkylsulfonyl, (C-C)alkylsulfimino,'}, 'Ris (C-C)alkyl, (C-C)hydroxyalkyl, (C-C)haloalkyl, (C-C)cyanoalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkoxy-(C-C)alkyl, (C-C)alkenyl, (C-C)alkenyloxy-(C-C)alkyl, (C-C)haloalkenyloxy-(C-C)alkyl, (C-C)haloalkenyl, (C-C)cyanoalkenyl, (C-C)alkynyl, (C-C)alkynyloxy-(C-C)alkyl, (C-C)haloalkynyloxy-(C-C)alkyl, (C-C)haloalkynyl, (C-C)cyanoalkynyl, (C-C)cycloalkyl, (C-C)-halocycloalkyl, (C-C)-cyanocycloalkyl, (C-C)cycloalkyl(C-C)cycloalkyl, (C-C)alkyl-(C-C)cycloalkyl, halo(C-C)cycloalkyl, (C-C)alkylamino, di-(C-C)alkyl-amino, (C-C)cycloalkylamino, (C-C)alkylcarbonyl-amino, (C-C)alkylthio-(C-C)alkyl, (C-C)haloalkylthio-(C-C)alkyl, (C ...

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14-05-2020 дата публикации

2-(HET)ARYL-SUBSTITUTED FUSED HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20200148686A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. Compound of formula (I) according to claim 1 , wherein{'sup': 1', '+', '−', '5, 'Ais nitrogen, ═N(O)— or ═C(R)—,'}{'sup': 2', '6, 'Ais —N(R)— or oxygen,'}{'sup': '1', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '3', '6', '3', '6', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '3', '6', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Ris (C-C)alkyl, (C-C)hydroxyalkyl, (C-C)haloalkyl, (C-C)cyanoalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkoxy-(C-C)alkyl, (C-C)alkenyl, (C-C)alkenyloxy-(C-C)alkyl, (C-C)haloalkenyloxy-(C-C)alkyl, (C-C)haloalkenyl, (C-C)cyanoalkenyl, (C-C)alkynyl, (C-C)alkynyloxy-(C-C)alkyl, (C-C)haloalkynyloxy-(C-C)alkyl, (C-C)haloalkynyl, (C-C)cyanoalkynyl, (C-C)cycloalkyl, (C-C)halocycloalkyl, (C-C)cyanocycloalkyl, (C-C)cycloalkyl(C-C)cycloalkyl, (C-C)alkyl-(C-C)cycloalkyl, halo(C-C)cycloalkyl, (C-C)alkylamino, di-(C-C)alkyl-amino, (C-C)cycloalkylamino, (C-C)alkylcarbonyl-amino, (C-C)alkylthio-(C-C)alkyl, (C-C)haloalkylthio-(C-C)alkyl, (C-C)alkylsulfinyl-(C-C)alkyl, (C-C)haloalkylsulfinyl-(C-C)alkyl, (C-C)alkylsulfonyl-(C-C)alkyl, (C-C)alkylcarbonyl-(C-C)alkyl, (C-C)haloalkylcarbonyl-(C-C)alkyl, (C-C)alkylsulfonylamino,'}{'sub': 1', '4', '1', '4', '2', '4', '2', '4', '3', '6', '1', '4', '3', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'or is in each case optionally identically or differently mono- or di-aryl-, -hetaryl- or -heterocyclyl-substituted (C-C)alkyl, (C-C)alkoxy, (C-C)alkenyl, (C-C)alkynyl, (C-C)cycloalkyl, where aryl, hetaryl or heterocyclyl are each optionally identically or differently mono- or disubstituted by halogen, cyano, ...

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30-05-2019 дата публикации

ACTIVE COMPOUND COMBINATIONS AND METHODS TO PROTECT THE PROPAGATION MATERIAL OF PLANTS

Номер: US20190159451A1
Принадлежит:

The present invention relates to novel mixtures, to processes for preparing these mixtures, to compositions comprising these mixtures, and to the use thereof as biologically active compounds, especially for control of harmful microorganisms or pests in crop protection and in the protection of materials and as plant growth regulators. 2. The composition according to claim 1 , in whichX represents fluorine, bromine or chlorine;n=0; andQ=NH or S.3. The composition according to claim 1 , in whichX represents chlorine, fluorine or bromine;n=0; andQ=S.4. The composition according to claim 1 , in whichX represents chlorine or bromine;n=0; andQ=NH.5. The composition according to claim 1 , in whichX represents fluorine, chlorine or bromine;n=1; andQ=S or NH, optionally NH.6. The composition according to claim 1 , in whichX represents chlorine,n=0, 1; Q=NH or n=0; Q=S.8. The composition according to claim 1 , wherein the pest control agent is a fungicide selected from1) Inhibitors of the ergosterol biosynthesis, optionally (1.1) aldimorph, (1.2) azaconazole, (1.3) bitertanol, (1.4) bromuconazole, (1.5) cyproconazole, (1.6) diclobutrazole, (1.7) difenoconazole, (1.8) diniconazole, (1.9) diniconazole-M, (1.10) dodemorph, (1.11) dodemorph acetate, (1.12) epoxiconazole, (1.13) etaconazole, (1.14) fenarimol, (1.15) fenbuconazole, (1.16) fenhexamid, (1.17) fenpropidin, (1.18) fenpropimorph, (1.19) fluquinconazole, (1.20) flurprimidol, (1.21) flusilazole, (1.22) flutriafol, (1.23) furconazole, (1.24) furconazole-cis, (1.25) hexaconazole, (1.26) imazalil, (1.27) imazalil sulfate, (1.28) imibenconazole, (1.29) ipconazole, (1.30) metconazole, (1.31) myclobutanil, (1.32) naftifine, (1.33) nuarimol, (1.34) oxpoconazole, (1.35) paclobutrazol, (1.36) pefurazoate, (1.37) penconazole, (1.38) piperalin, (1.39) prochloraz, (1.40) propiconazole, (1.41) prothioconazole, (1.42) pyributicarb, (1.43) pyrifenox, (1.44) quinconazole, (1.45) simeconazole, (1.46) spiroxamine, (1.47) tebuconazole, (1.48 ...

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04-09-2014 дата публикации

Compounds with Nematicidal Activity

Номер: US20140249149A1
Принадлежит: Bayer Intellectual Property GmbH

The present invention relates to the use of known pyridyl carboxamide derivatives and novel pyridyl carboxamide derivatives as nematicides, compositions containing such compounds and methods for the control of nematodes. 4. A compound according to claim 3 , in which R claim 3 , R claim 3 , Rrepresent hydrogen claim 3 , n represents 2 and X represent 3-Cl and 6-CF.6. A Compound according to claim 5 , in which R claim 5 , R claim 5 , Rrepresent hydrogen claim 5 , n represents 2 and X represent 3-Cl and 6-CF.7. A compound according to claim 5 , in which R claim 5 , R claim 5 , Rrepresent hydrogen claim 5 , n represents 2 and X represent 3-Cl and 6-Cl.10. A compound according to claim 9 , in which R claim 9 , R claim 9 , Rrepresent hydrogen claim 9 , n represents 1 and X represents 6-Cl.27. A composition claim 1 , comprising an effective amount of at least one compound of formula (I) according to claim 1 , and at least one surfactant claim 1 , solid or liquid diluent. The present invention relates to the use of predominantly known pyridyl carboxamide derivatives as nematicides, compositions containing such compounds and methods for the control of nematodes.Nematodes cause a substantial loss in agricultural product including food and industrial crops and are combated with chemical compounds having nematicidal activity. To be useful in agriculture these compounds should have a high activity, a broad spectrum activity against different strains of nematodes and should not be toxic to non-target organisms.The use of certain N-2-(pyridyl)ethyl-carboxamide derivatives for controlling nematodes is described in EP 2 132 987 A1.Most of the compounds of formula (I) described below are known from WO 2001/011965 A1 (later, e.g. in the Tables, referred to as P1), WO 2005/058828 A1 (P2), WO2005/014545 A2 (P3), WO 2005/103004 A1 (P4), WO 2006/122952 A1 (P5), EP 2 289 880 A1 (P6), WO 2006/008191 A1 (P7) and WO 2006/008192 A1 (P8). There it is stated that they can be used as fungicides. ...

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11-09-2014 дата публикации

COMPOUNDS WITH NEMATICIDAL ACTIVITY

Номер: US20140256728A1
Принадлежит: Bayer Intellectual Property GmbH

The present invention relates to the use of predominantly known pyridyl carboxamide derivatives as nematicides, compositions containing such compounds and methods for the control of nematodes.

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23-06-2016 дата публикации

IMIDAZOTHIAZOLE SUFONAMIDES AS NEMATICIDES

Номер: US20160176898A1
Принадлежит:

Disclosed are compounds of formula (I) which possess nematicidal properties 8. A composition comprising at least one compound of formula (I) according to .9. A composition comprising an effective amount of at least one compound of formula (I) according to and at least one surfactant claim 1 , solid or liquid diluent.10. A composition according to which further comprises at least one additional active ingredient.11. A composition according to comprising a spray composition.12. A compound of the formula (I) according to capable of being used for controlling animal pests claim 1 , optionally parasitic nematodes claim 1 , in crop protection claim 1 , in the protection of materials and/or in the veterinary sector.13. A compound according to claim 12 , wherein the compound is applied by spray application.14. A method for controlling a parasitic nematode comprising contacting the parasitic nematode or an environment thereof with a biologically effective amount of a compound of formula (I) according to .15. A method for controlling a parasitic nematode comprising contacting the parasitic nematode or an environment thereof with a composition according to .16. A method according to wherein the compound is applied by spray application.17. A method for protecting a seed from a parasitic nematode comprising contacting the seed with a biologically effective amount of a compound of formula (I) according to .18. A seed obtained by a method according to . The present invention relates to imidazothiazole sulfonamides, their use for the control of nematodes in agricultures, compositions containing such compounds and methods for the control of nematodes. This invention relates to certain sulfonamides, their N-oxides, salts and compositions suitable for agronomic and nonagronomic uses, and methods of their use for controlling parasitic nematodes in both agronomic and nonagronomic environments.The present invention further relates to novel imidazothiazoles, processes and intermediate ...

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06-06-2019 дата публикации

SUBSTITUTED 2-HETEROCYCLYLIMIDAZOLYLCARBOXAMIDES AS PESTICIDES

Номер: US20190166837A1
Принадлежит:

The present invention relates to compounds of the general formula (I) 3. Compound according to in whichQ is oxygen or sulphur, 'trifluoromethoxy and cyano,', 'V is a radical from the group of hydrogen, fluorine, chlorine, bromine, methyl, ethyl, difluoromethyl, trifluoromethyl, methoxy, ethoxy, difluoromethoxy,'} 'trifluoromethoxy and cyano,', 'W is a radical from the group of hydrogen, fluorine, chlorine, bromine, methyl, ethyl, difluoromethyl, trifluoromethyl, methoxy, ethoxy, difluoromethoxy,'}{'sub': n', 'n', '1', '4', '3', '4', '3', '4', '3', '6', 'n', '3', '6', '1', '2, 'sup': '1', 'Y is a radical from the group of hydrogen, optionally independently mono- to penta-fluorine-, -chlorine-, -bromine-, -methoxy-, -ethoxy-, -methyl-S(O)—, -ethyl-S(O)and -cyano-substituted C-C-alkyl, C-C-alkenyl and C-C-alkynyl, optionally independently mono- or di-fluorine-, -chlorine-, -bromine-, -methyl-, -ethyl-, -trifluoromethyl-, -methoxy-, -ethoxy-, -cyano-substituted C-C-cycloalkyl, optionally independently singly or doubly O-, S(O)-, NR-interrupted, optionally independently mono- to tetra-fluorine-, -chlorine-, -bromine-, -methyl-, -ethyl-, -trifluoromethyl-, -methoxy-, -ethoxy-, -cyano-substituted, straight-chain or branched C-C-cycloalkyl-C-C-alkyl and cyano,'}{'sub': n', 'n', '1', '6', '3', '6', '3', '6', '3', '6', '3', '6', '1', '2, 'A is a radical from the group of hydrogen, optionally independently mono- to penta-fluorine-, -chlorine-, -bromine-, -methoxy-, -ethoxy-, -methyl-S(O)—, -ethyl-S(O)— and -cyano-substituted C-C-alkyl, C-C-alkenyl and C-C-alkynyl, optionally independently mono- or di-fluorine-, -chlorine-, -bromine-, -methyl-, -ethyl-, -trifluoromethyl-, -methoxy-, -ethoxy-, -cyano-substituted C-C-cycloalkyl, optionally independently mono- or di-fluorine-, -chlorine-, -bromine-, -methyl-, -ethyl-, -trifluoromethyl-, -methoxy-, -ethoxy-, -cyano-substituted, straight-chain or branched C-C-cycloalkyl-C-C-alkyl,'}T is oxygen or an electron pair,X is a partly ...

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11-06-2020 дата публикации

NOVEL ISOTHIAZOLO-BASED BICYCLES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS HERBICIDES AND/OR PLANT GROWTH REGULATORS

Номер: US20200178532A1
Принадлежит:

The invention relates to the technical field of the herbicides and/or plant growth regulators. Specifically, the invention primarily relates to novel substituted isothiazolopyridones, and compositions comprising said novel substituted isothiazolopyridones. Further, the present invention relates to processes for the preparation said novel substituted isothiazolopyridones and their use as herbicides and/or plant growth regulators. 2. Compound of the formulae (G1) and (G2) and/or salt thereof according to in which{'sup': 6', '7, 'A is CRR,'}x is 0, 1 or 2,{'sup': 1', '13', '14, 'sub': 3', '6', '3', '6', '3', '6', '1', '6', '3', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6, 'Ris hydrogen, (C-C)-cycloalkyl, (C-C)-cycloalkenyl, (C-C)-cycloalkyl-(C-C)-alkyl, (C-C)-cycloalkenyl-(C-C)-alkyl, phenyl, pyridinyl, furanyl, thienyl wherein all these residues are unsubstituted or substituted by one or more residues from the group consisting of halogen, nitro, hydroxyl, cyano, NRR, (C-C)-alkyl, (C-C)-haloalkyl, (C-C)-alkoxy, (C-C)-haloalkoxy, (C-C)-alkylthio, (C1-C6)-alkylsulphinyl, (C-C)-alkylsulphonyl,'}{'sup': 2', '3', '13', '14', '12, 'sub': 1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '2', '6', '2', '6', '1', '6', '1', '6', '1', '6', '1', '6', '2', '6', '3', '6', '3', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', 'm', 'n, 'R, Rare each independently hydrogen, (C-C)-alkoxyphenyl-(C-C)-alkyl, (C-C)-alkylthiocarbonyl, (C-C)-haloalkylthiocarbonyl, (C-C)-alkoxy-(C-C)-alkylcarbonyl, (C-C)-alkylthio-(C-C)-alkylcarbonyl, (C-C)-alkylsulphinyl-(C-C)-alkylcarbonyl, (C-C)-alkylsulphonyl-(C-C)-alkylcarbonyl, (C-C)-alkylcarbonyl, (C-C)-haloalkylcarbonyl, (C-C)-alkenylcarbonyl, (C-C)-alkynylcarbonyl, (C-C)-alkoxycarbonyl-(C-C)-alkylcarbonyl, (C-C)-alkoxycarbonyl, (C-C)- ...

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11-06-2020 дата публикации

HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20200181172A1
Принадлежит:

The present invention relates to novel fused bicyclic heterocycle derivatives of formula (I) 6. Compound of formula (I) according to claim 5 , wherein R{'sub': 1', '4', '3', '6', '1', '4', 'm, 'sup': 21', '21', '20', '21, 'claim-text': [{'sup': '20', 'where Rrepresents hydrogen,'}, {'sup': '21', 'sub': 3', '6', '1', '4', '1', '4, 'Rrepresents (C-C)-cycloalkyl, (C-C)-alkoxy or (C-C)-alkyl'}, 'and m represents 2,', 'or in the case that Q=Q7, Q8 or Q9, represents hydrogen., 'in the case that Q=Q1, represents 3-halogen, 3-(C-C)-haloalkyl, 3-(C-C)-cycloalkyl, 3-(C-C)-haloalkoxy, 3-S(═O)—R, —C(═O)—ORor 3-N(R)—C(═O)—R,'}8. Compound of formula (I) according to claim 7 , wherein R{'sub': 2', '3, 'in the case that Q=Q1, represents 3-iodine, 3-cyclopropyl, 3-S02-cyclopropyl, 3-trifluoromethyl, 3-OCHCF, 3—NHCOMe, 3-NHCOOMe, 3-COOMe or 3-NHCO-cyclopropyl, or'}in the case that Q=Q7, Q8 or Q9, represents hydrogen.9. Compound of the formula (I) according to claim 1 , wherein{'sup': 2', '3', '2', '3, 'sub': 1', '4', '1', '4', '1', '4', '1', '4, 'R, Rindependently of one another represent hydrogen, (C-C)-haloalkylthio, (C-C)-haloalkylsulfinyl, (C-C)-haloalkylsulfonyl or (C-C)-haloalkyl, where only one of the radicals Ror Rdoes not represent hydrogen.'}10. Compound of formula (I) according to claim 1 , wherein{'sup': '1', 'Aa represents nitrogen or C(R),'}{'sup': '2', 'Ab represents nitrogen or C(R),'}{'sup': '3', 'Ac represents nitrogen or C(R) and'}Ad represents CH,{'sup': 2', '3', '1', '3, 'where at most one of the radicals Aa, Ab or Ac represents nitrogen and at least one of the radicals Ror Rdoes not represent hydrogen and Rdoes not represent hydrogen only in the case where Rlikewise does not represent hydrogen.'}11. Compound of formula (I) according to claim 2 , where for Q=Q1 claim 2 , Q2 claim 2 , Q3 and Q4{'sup': 6', '7', 'x, 'sub': 3', '6', '2', '3', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '2, 'at least one of ...

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19-07-2018 дата публикации

NITROGEN-CONTAINING HETEROCYCLES AS PESTICIDES

Номер: US20180201600A1
Принадлежит:

The present application relates to novel heterocyclic compounds, to processes and intermediates for the preparation thereof, and their use for controlling animal pests. 5. Composition comprising at least one compound of the formula (I) according to and one or more customary extenders and/or surfactants.6. A product comprising a compound of formula (I) according to or a composition thereof for controlling pests. The present application relates to novel heterocyclic compounds, to processes and intermediates for the preparation thereof, and their use for controlling animal pests.DE 10024938 A1 describes the preparation of phenyliminoazines having herbicidal activity.US 2007/0259924 A1 describes imidazoles containing an N-[1-aryl-2(1H)-pyridinylidene]cyanamide fragment as factor Xa inhibitors.Crop protection agents, which also include pesticides, have to meet many demands, for example in relation to extent, persistence, and spectrum of their action and possible use. Questions of toxicity and of combinability with other active compounds or formulation auxiliaries play a role, as does the question of the expense that the synthesis of an active compound requires. In addition, resistances can occur. For all these reasons, the search for novel crop protection agents cannot be considered to be complete, and there is a constant need for novel compounds having properties which, compared to the known compounds, are improved at least in relation to individual aspects.It was an object of the present invention to provide compounds which widen the spectrum of the pesticides in various aspects.The object, and further objects which are not stated explicitly but can be discerned or derived from the connections discussed herein, are achieved by compounds of the formula (I)Preference is given to compounds of the formula (I)Particular preference is given to compounds of the formula (I)Very particular preference is given to compounds of the formula (I)The radical definitions or ...

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04-08-2016 дата публикации

CARBOXAMIDE DERIVATIVES AS PESTICIDAL COMPOUNDS

Номер: US20160221950A1
Принадлежит:

Disclosed are compounds of formula (I) which possess pesticidal, especially nematicidal properties wherein in the structural elements have the meaning as indicated in the description. 7. A compound according to to , wherein the phenyl ring bearing the substituent Ym preferably is in para-position.9. A compound according to claim 8 , wherein the phenyl ring bearing the substituent Ym preferably is in para-position.11. A formulation claim 8 , particularly an agrochemical formulation claim 8 , comprising at least one compound of formula (I) according to to .12. A formulation according to which further comprises at least one extender and/or at least one surfactant.13. A formulation according to or claim 11 , wherein the compound of the formula (I) is present in a mixture with at least one other active compound.14. A method for controlling an animal pest claim 11 , wherein a compound of formula (I) according to to or a formulation according to to is allowed to act on the animal pest and/or their habitat.15. A method according to claim 14 , wherein the animal pest comprises a nematode or is a nematode.16. Use of a compound of formula (I) according to to or a formulation according to to for controlling an animal pest.17. A use according to claim 16 , wherein the animal pest comprises a nematode or is a nematode.18. A use according to or in crop protection.19. A use according to or in the animal health field.20. A method for protecting a seed and/or a germinating plant from attack by a pest claim 16 , particularly a nematode claim 16 , comprising the step of contacting the seed with a compound of formula (I) according to to or with a formulation according to to .21. A seed obtained by a method according to . The present invention relates to certain pyridylalkyl carboxamide derivatives as to processes for their preparation, to compositions comprising those compounds and their use in agriculture and veterinary fields and fields relying on pest management. The compounds are ...

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02-08-2018 дата публикации

HETEROCYCLIC COMPOUNDS AS PESTICIDES

Номер: US20180213782A1
Принадлежит:

The present application relates to thiadiazole compounds, compositions containing such compounds, their use for controlling animal pests including arthropods, insects and nematodes, and to processes and intermediates for the preparation of the thiadiazole compounds. 8. Composition comprising claim 1 , at least one compound according to and one or more customary extenders and/or surfactants.9. Method for controlling one or more pests claim 1 , comprising allowing a compound of the formula (I) according to to act on the pests and/or a habitat thereof claim 1 , provided that methods for the therapeutic treatment of an animal body are excluded.10. A compound according to for controlling one or more arthropodal parasites on animals.11. 3-(2 claim 1 ,6-Difluorophenyl)-1 claim 1 ,2 claim 1 ,4-thiadiazol-5-amine.12. 3-(2-Chloropyridin-3-yl)-1 claim 1 ,2 claim 1 ,4-thiadiazol-5-amine. The present application relates to thiadiazole compounds, compositions containing such compounds, their use for controlling animal pests including arthropods, insects and nematodes, and to processes and intermediates for the preparation of the thiadiazole compounds.Certain thiadiazole compounds and their use for controlling pests are known from WO 01/40223 A2. Thiadiazole compounds with a pyridine moiety in the 3-position of the thiadiazole ring system and their use for controlling parasites are disclosed in WO 2015/073797 A1.Crop protection compositions, which also include pesticides, have to meet many demands, for example in relation to efficacy, persistence, spectrum, resistance breaking properties, pollinator and beneficial safety of their action and possible use. Questions of toxicity, the combinability with other active compounds or formulation auxiliaries play a role, as well as the question of the expense that the synthesis of an active compound requires. Furthermore, resistances may occur. For all these reasons, the search for novel crop protection compositions cannot be considered to ...

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11-08-2016 дата публикации

SUBSTITUTED QUINOXALINE DERIVATIVES AS PEST CONTROL AGENT

Номер: US20160227779A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. A compound of formula (I-L) as claimed in wherein{'sup': '2', 'sub': 1', '3', '1', '3', '2', '3', '2', '3', '2', '3', '2', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3, 'claim-text': represents phenyl or hetaryl from the group Q-1, Q-22, Q-36, Q-37, Q-41, Q-44, Q-45, Q-51, Q-64, Q-66, Q-67, each of which is optionally mono- or disubstituted by identical or different substituents,', {'sub': 1', '3', '1', '3', '2', '3', '2', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3, 'possible substituents being in each case: cyano, halogen, (C-C)-alkyl, (C-C)-haloalkyl, (C-C)-alkenyl, (C-C)-haloalkenyl, (C-C)-alkoxy, (C-C)-haloalkoxy, (C-C)-alkylsulfinyl, (C-C)-haloalkylsulfinyl, (C-C)-alkylsulfonyl, (C-C)-haloalkylsulfonyl, (C-C)-alkylthio,'}], 'Rrepresents hydrogen, cyano, halogen, (C-C)-alkyl, (C-C)-haloalkyl, (C-C)-alkenyl, (C-C)-haloalkenyl, (C-C)-alkynyl, (C-C)-haloalkynyl, (C-C)-alkoxy, (C-C)-haloalkoxy, (C-C)-alkylsulfinyl, (C-C)-haloalkylsulfinyl, (C-C)-alkylsulfonyl, (C-C)-haloalkylsulfonyl or'}{'sup': 3', '4', '5', '6, 'sub': 1', '3', '1', '3', '2', '3', '2', '3', '2', '3', '2', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '1', '3, 'R, R, Rand Rindependently of one another represent hydrogen, cyano, halogen, (C-C)-alkyl, (C-C)-haloalkyl, (C-C)-alkenyl, (C-C)-haloalkenyl, (C-C)-alkynyl, (C-C)-haloalkynyl, (C-C)-alkoxy, (C-C)-haloalkoxy, (C-C)-alkylsulfinyl, (C-C)-haloalkylsulfinyl, (C-C)-alkylsulfonyl, (C-C)-haloalkylsulfonyl,'}{'sup': 3', '4', '5', '6, 'with the proviso that R, R, Rand Rdo not simultaneously represent hydrogen or'}{'sup': 3', '4', '4', '5', '5', '6, 'sub': 1', '3, 'Rand R, or Rand R, or Rand Rtogether with the atoms to which they are attached form a saturated, optionally fluorine-, chlorine- or (C-C)-alkyl-substituted 5-membered ring which optionally contains one or two oxygen atoms (where the heteroatoms must not be directly adjacent ...

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23-10-2014 дата публикации

N-ARYLAMIDINE-SUBSTITUTED TRIFLUOROETHYL SULFIDE DERIVATIVES AS ACARICIDES AND INSECTICIDES

Номер: US20140315898A1
Принадлежит: Bayer CropScience AG

The present invention relates to novel N-arylamide-substituted trifluoroethyl sulfide derivatives of the formula (I) 13. An active compound composition comprising at least one compound as claimed in and at least one further insecticidally claim 1 , acaricidally or nematicidally active compound selected from the group consisting of(1) Acetylcholinesterase (AChE) inhibitors optionally comprisingcarbamates, optionally comprising alanycarb, aldicarb, bendiocarb, benfuracarb, butocarboxim, butoxycarboxim, carbaryl, carbofuran, carbosulfan, ethiofencarb, fenobucarb, formetanate, furathiocarb, isoprocarb, methiocarb, methomyl, metolcarb, oxamyl, pirimicarb, propoxur, thiodicarb, thiofanox, triazamate, trimethacarb, XMC and xylylcarb; ororganophosphates, optionally comprising acephate, azamethiphos, azinphos-ethyl, azinphos-methyl, cadusafos, chlorethoxyfos, chlorfenvinphos, chlormephos, chloropyrifos, chloropyrifos-methyl, coumaphos, cyanophos, demeton-S-methyl, diazinon, dichlorvos/DDVP, dicrotophos, dimethoate, dimethylvinphos, disulfoton, EPN, ethion, ethoprophos, famphur, fenamiphos, fenitrothion, fenthion, fosthiazate, heptenophos, imicyafos, isofenphos, isopropyl O-(methoxyaminothiophosphoryl)salicylate, isoxathion, malathion, mecarbam, methamidophos, methidathion, mevinphos, monocrotophos, naled, omethoate, oxydemeton-methyl, parathion, parathion-methyl, phenthoate, phorate, phosalone, phosmet, phosphamidon, phoxim, pirimiphos-methyl, profenofos, propetamphos, prothiofos, pyraclofos, pyridaphenthion, quinalphos, sulfotep, tebupirimfos, temephos, terbufos, tetrachlorvinphos, thiometon, triazophos, trichlorfon and vamidothion.(2) GABA-gated chloride channel antagonists optionally comprising,cyclodiene organochlorines, optionally comprising chlordane and endosulfan; orphenylpyrazoles (fiproles), optionally comprising ethiprole and fipronil.(3) Sodium channel modulators/voltage-dependent sodium channel blockers optionally comprising,pyrethroids, optionally comprising ...

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10-08-2017 дата публикации

Heterocyclic Compounds as Pesticides

Номер: US20170226107A1
Принадлежит:

The present application relates to novel heterocyclic compounds of the formula (I) 10. A composition claim 1 , comprising a content of at least one compound of the formula (I) according to and one or more customary extenders and/or surface-active substances.11. The compound of formula (I) according to for controlling pests. The present application relates to novel heterocyclic compounds, to processes and intermediates for the preparation thereof, and their use for controlling animal pests.WO 2012/102387 A1 describes heterocyclic compounds which can be used particularly as insecticides and acaricides.Heterocyclic compounds for pharmaceutical applications are disclosed in WO 2004/009597 A2, WO 2008/107418 A1, WO 2009/068617 A1 and US 2004/242596 A1.Bioorganic & Medicinal Chemistry Letters (2007), 17(15), 4303-4307 reports synthesis and pharmacological properties of particular pyrazolo[3,4-d]pyrimidin-4-ones.Modern crop protection compositions have to meet many demands, for example in relation to efficacy, persistence and spectrum of their action and possible use. Questions of toxicity, environmental properties, application rates, combinability with other active ingredients or formulation auxiliaries play a role, as does the question of the effort required for the synthesis of an active ingredient; furthermore, resistances may occur, to mention only some parameters. For all these reasons alone, the search for novel crop protection compositions cannot be considered complete, and there is a constant need for novel compounds having improved properties compared to the known compounds, at least in relation to individual aspects.It was an object of the present invention to provide compounds which widen the spectrum of the pesticides in various aspects.This object, and further objects which are not stated explicitly which can be discerned or derived from the connections discussed herein, are achieved by the provision of compounds of the formula (I)in whichPreferred ...

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27-08-2015 дата публикации

HETEROCYCLIC COMPOUNDS AS PESTICIDES

Номер: US20150239847A1
Принадлежит:

The present application relates to the use of heterocyclic compounds for controlling animal pests including arthropods, insects and nematodes, to novel heterocyclic compounds, to processes for their preparation and to intermediates for preparing the heterocyclic compounds. 7. A Composition claim 1 , comprising at least one compound of formula (I) as described in .8. A Composition comprising at least one compound of formula (I) as described in .9. Method for controlling one or more pests claim 1 , comprising allowing a compound of formula (I) according to to act on one or more pests and/or a habitat thereof.10. 2-(3 claim 1 ,5-Difluoropyridin-2-yl)-2H-1 claim 1 ,2 claim 1 ,3-triazole-4-amine11. 1-(3 claim 1 ,5-Difluoropyridin-2-yl)-1H-pyrazole-3-amine12. N-[1-(2 claim 1 ,6-Difluorophenyl)-4 claim 1 ,5-dihydro-1H-pyrazol-3-yl]acetamide13. N-[1-(2 claim 1 ,6-Difluorophenyl)-1H-pyrazol-3-yl]acetamide14. 1-(2 claim 1 ,6-Difluorophenyl)-1H-pyrazole-3-amine15. 1-(2 claim 1 ,6-Difluorophenyl)-4 claim 1 ,5-dihydro-1H-pyrazole-3-amine The present application relates to the use of heterocyclic compounds for controlling animal pests including arthropods, insects and nematodes, to novel heterocyclic compounds, to processes for their preparation and to intermediates for preparing the heterocyclic compounds.The heterocyclic compounds of the formulae (W) and (W2) are known (cf. for the compounds of the formula (W) Registry Numbers 1189645-25-7, 1189474-83-6, 1193202-69-5, 1172407-07-6, 1185158-40-0, 1185036-12-7, 1170986-74-9, 1193179-17-7, 1189458-68-1, 1189956-23-7, 1189915-26-1, 1170047-96-7). A use of these compounds has not been described.Derivatives of pyrazole-4-carboxamides are known from JP 2010-202649. The compounds described therein have bactericidal action against plant-damaging bacteria. Intermediates for their preparation are described in JP 2010-202648.Crop protection compositions, which also include pesticides, have to meet many demands, for example in relation to ...

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01-09-2016 дата публикации

SIX-MEMBERED C-N-LINKED ARYL SULFIDE DERIVATIVES AND ARYL SULFOXIDE ERIVATVES AS PEST CONROL AGENTS

Номер: US20160251321A1
Принадлежит:

The present invention relates to novel heterocyclic compounds, to processes for preparation thereof and to the use thereof for controlling animal pests, which include arthropods and especially insects and acarids. 2. The compound according to claim 1 , whereinD is a substructure of the formula (I-A);{'sup': 1', '2', '11, 'V, Vare each independently an oxygen, sulphur or N—R, especially oxygen;'}{'sup': 1', '2', '7', '1', '1, 'Qis CRRor N—R, especially N—R;'}{'sup': 3', '4', '4, 'Qis CRor nitrogen, especially CR;'}{'sup': 4', '5, 'Qis CRor nitrogen;'}{'sup': '1', 'claim-text': or alkyl, cycloalkylalkyl, haloalkyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, aminoalkyl, alkoxycarbonylalkyl, alkylthioalkyl, haloalkylthioalkyl, alkylsulphinylalkyl, haloalkylsulphinylalkyl, alkylsulphonylalkyl, haloalkylsulphonylalkyl, phenylalkyl, phenoxyalkyl, phenylsulphanylalkyl, phenylsulphinylalkyl, phenylsulphonylalkyl, hetarylalkyl, hetaryloxyalkyl, hetarylthioalkyl, where the aforementioned radicals may each be saturated or unsaturated and/or optionally substituted, and where one of the nitrogen atoms present in hetarylalkyl, hetaryloxyalkyl and hetarylthioalkyl may also be in the form of the N-oxide;', 'or optionally substituted saturated or unsaturated cycloalkyl which may optionally be interrupted by one or more heteroatoms;', 'or hydroxyl, alkoxy or haloalkoxy;', 'or alkylcarbonyl, haloalkylcarbonyl, hydroxyalkylcarbonyl, alkoxyalkylcarbonyl, phenylcarbonyl, hetarylcarbonyl, alkoxycarbonyl, haloalkoxycarbonyl, aryloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, cycloalkylaminocarbonyl, dicycloalkylaminocarbonyl, cycloalkyl(alkyl)aminocarbonyl, arylaminocarbonyl, diarylaminocarbonyl, alkyl(aryl)aminocarbonyl, cycloalkyl(aryl)aminocarbonyl, alkylaminothiocarbonyl, dialkylaminothiocarbonyl or aminothiocarbonyl, where the aforementioned radicals may each be saturated or unsaturated and/or optionally substituted, or is carbonyl or carboxyl; or', 'or optionally ...

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08-08-2019 дата публикации

FUSED BICYCLIC HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20190239510A1
Принадлежит: Bayer CropScience Aktiengesellschaft

The invention relates to novel compounds of the formula (I) 5. A compound of formula (I) according to in which{'sub': 'a', 'sup': '7', 'Arepresents ═C(R)—,'}{'sub': b', 'm, 'sup': '2', 'Arepresents —S(O)— or ═C(R)—,'}{'sub': 'c', 'sup': '3', 'Arepresents ═C(R)—,'}{'sub': d', 'm, 'sup': '8', 'Arepresents ═N—, —S(O)— or ═C(R)—,'}resulting in the following structural units: A9, A10, A14{'sup': '1', 'Rrepresents ethyl,'}{'sup': '2', 'Rrepresents hydrogen,'}{'sup': '3', 'Rrepresents hydrogen,'}{'sup': '7', 'Rrepresents hydrogen,'}{'sup': '8', 'Rrepresents hydrogen,'}Q represents a heteroaromatic 9-membered fused bicyclic ring system from the group consisting of Q2 and Q3,{'sup': '4', 'Rrepresents methyl,'}{'sup': '5', 'Rrepresents trifluoromethyl'}{'sup': '6', 'Rrepresents hydrogen,'}m represents 0,n represents 0, 1 or 2.6. A compound of formula (I) according to in whichQ represents a heteroaromatic 9-membered fused bicyclic ring system from the group consisting of Q2 and Q3.7. A compound of formula (I) according to in which{'sub': 'a', 'sup': '7', 'Arepresents ═C(R)—,'}{'sub': b', 'm, 'sup': '2', 'Arepresents —S(O)— or ═C(R)—,'}{'sub': 'c', 'sup': '3', 'Arepresents ═C(R)—,'}{'sub': d', 'm, 'sup': '8', 'Arepresents ═N—, —S(O)— or ═C(R)—,'}resulting in the following structural units: A9, A10, A14.8. A compound of formula (I) according to in which{'sub': 'a', 'sup': '7', 'Arepresents ═C(R)—,'}{'sub': b', 'm, 'sup': '2', 'Arepresents —S(O)— or ═C(R)—,'}{'sub': 'c', 'sup': '3', 'Arepresents ═C(R)—,'}{'sub': d', 'm, 'sup': '8', 'Arepresents ═N—, —S(O)— or ═C(R)—,'}resulting in the following structural units: A9, A10, A14and Q represents Q2 or Q3.9. Agrochemical formulation comprising a compound of formula (I) according to and one or more extenders and/or surfactants.10. Agrochemical formulation according to claim 9 , additionally comprising a further agrochemically active compound.11. Method for controlling one or more animal pests claim 1 , wherein a compound of formula (I) ...

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30-07-2020 дата публикации

2-(HET)ARYL-SUBSTITUTED FUSED HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20200236940A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. Compound of formula (I) according to claim 1 , wherein{'sup': 1', '+', '−', '5, 'Ais nitrogen, ═N—Oor ═C—R,'}{'sup': 2', '6, 'Ais —N(R)— or oxygen,'}{'sup': '1', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '3', '6', '3', '6', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '3', '6', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'claim-text': {'sub': 1', '4', '1', '4', '2', '4', '2', '4', '3', '6', '1', '4', '3', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'or is in each case optionally singly or doubly, identically or differently aryl-, hetaryl- or heterocyclyl-substituted (C-C)alkyl, (C-C)alkoxy, (C-C)alkenyl, (C-C)alkynyl, (C-C)cycloalkyl, where aryl, hetaryl or heterocyclyl may each optionally be mono- or disubstituted identically or differently by halogen, cyano, carbamoyl, aminosulfonyl, (C-C)alkyl, (C-C)cycloalkyl, (C-C)alkoxy, (C-C)haloalkyl, (C-C)haloalkoxy, (C-C)alkylthio, (C-C)alkylsulfinyl, (C-C)alkylsulfonyl, (C-C)alkylsulfimino,'}, 'Ris (C-C)alkyl, (C-C)hydroxyalkyl, (C-C)haloalkyl, (C-C)cyanoalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkoxy-(C-C)alkyl, (C-C)alkenyl, (C-C)alkenyloxy-(C-C)alkyl, (C-C)haloalkenyloxy-(C-C)alkyl, (C-C)haloalkenyl, (C-C)cyanoalkenyl, (C-C)alkynyl, (C-C)alkynyloxy-(C-C)alkyl, (C-C)haloalkynyloxy-(C-C)alkyl, (C-C)haloalkynyl, (C-C)cyanoalkynyl, (C-C)cycloalkyl, (C-C)halocycloalkyl, (C-C)cyanocycloalkyl, (C-C)cycloalkyl(C-C)cycloalkyl, (C-C)alkyl-(C-C)cycloalkyl, halo(C-C)cycloalkyl, (C-C)alkylamino, di(C-C)alkylamino, (C-C)cycloalkylamino, (C-C)alkylcarbonyl-amino, (C-C)alkylthio-(C-C)alkyl, (C-C)haloalkylthio-(C-C) ...

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08-08-2019 дата публикации

2-(HET)ARYL-SUBSTITUTED CONDENSED BICYCLIC HETEROCYCLE DERIVATIVES AS PEST CONTROL AGENTS

Номер: US20190241564A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. Compound of the formula (IIa) according to in which{'sup': '3', 'sub': 2', '2', '4', '2', '3', '2', '2', '2', '3', '2', '4', '2', '5', '3', '7', '3', '7', '2', '2', '2', '2', '2', '2', '2', '2', '2', '2', '3', '2', '1', '2', '3', '3', '2', '3', '2', '4', '2', '4', '2', '4', '2', '2', '4', '2', '3', '2', '2', '3', '2', '2', '3', '2', '2', '2', '3', '2', '2', '2', '3', '2', '2', '3', '2', '2', '3', '2', '2', '2', '3', '2', '4', '2', '4', '2', '4', '2', '2', '4', '2', '5', '2', '5', '2', '5', '2', '2', '5', '3', '7', '3', '7', '3', '7', '2', '3', '7', '3', '7', '3', '7', '3', '7', '2', '3', '7, 'Ris CHF, CHF, CHF, CHF, CHF, CF, n-CF, i-CF, OCHF, SCHF, SOCHF, SOCHF, OCHF, SCHF, SOCHF, SOCHF, OCF, OCFC, OCFCl, SCF, SOCF, SOCF, OCHF, SCHF, SOCHF, SOCHF, OCHF, SCHF, SOCHF, SOCHF, OCHF, SCHF, SOCHF, SOCHF, OCHF, SCHF, SOCHF, SOCHF, OCF, SCF, SOCF, SOCF, n-OCF, n-SCF, n-SOCF, n-SOCF, i- OCF, i-SCF, i-SOCFor i-SOCF.'}3. Compound of the formula (IIa) according to in which{'sup': '3', 'sub': 2', '3', '2', '4', '2', '3', '2', '2', '2', '3', '2', '4', '2', '5', '3', '3', '2', '3, 'Ris CHF, OCF, CHF, CHF, CHF, CHF, CF, SCF, SOCFor SOCF.'} This application is a Divisional Application of U.S. application Ser. No. 15/119,124, filed 15 Aug. 2016, which is a National Stage entry of International Application No. PCT/EP2015/052351, filed Feb. 5, 2015, which claims priority to European Patent Application No. 14155372.7, filed Feb. 17, 2014. The disclosures of the priority applications are incorporated in their entirety herein by reference.The present invention relates to novel 2-(het)aryl-substituted fused bicyclic heterocycle derivatives of the formula (I), to the use thereof as acaricides and/or insecticides for controlling animal pests, particularly arthropods and especially insects and arachnids, and to processes and intermediates for preparation thereof.2-(Het)aryl-substituted fused bicyclic heterocycle derivatives having ...

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15-08-2019 дата публикации

FUSED BICYCLIC HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20190248811A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. Compound of formula (I) according to in which{'sup': '10', 'Aa is nitrogen or ═C(R)—,'}{'sup': '11', 'Ab is nitrogen or ═C(R)—,'}{'sup': '12', 'Ac is nitrogen or ═C(R)—,'}{'sup': '13', 'Ad is nitrogen or ═C(R)—,'}where not more than two of Aa, Ab, Ac and Ad can be nitrogens,{'sup': '1', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '3', '6', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Ris (C-C)alkyl, (C-C)hydroxyalkyl, (C-C)haloalkyl, (C-C)cyanoalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkoxy-(C-C)alkyl, (C-C)alkenyl, (C-C)alkenyloxy-(C-C)alkyl, (C-C)haloalkenyloxy-(C-C)alkyl, (C-C)haloalkenyl, (C-C)cyanoalkenyl, (C-C)alkynyl, (C-C)alkynyloxy-(C-C)alkyl, (C-C)haloalkynyloxy-(C-C)alkyl, (C-C)haloalkynyl, (C-C)cyanoalkynyl, (C-C)cycloalkyl, (C-C)cycloalkyl(C-C)cycloalkyl, (C-C)alkyl-(C-C)cycloalkyl, halo(C-C)cycloalkyl, (C-C)alkylamino, di-(C-C)alkyl-amino, (C-C)cycloalkylamino, (C-C)alkylcarbonyl-amino, (C-C)alkylthio-(C-C)alkyl, (C-C)haloalkylthio-(C-C)alkyl, (C-C)alkylsulfinyl-(C-C)alkyl, (C-C)haloalkylsulfinyl-(C-C)alkyl, (C-C)alkylsulfonyl-(C-C)alkyl, (C-C)alkylcarbonyl-(C-C)alkyl, (C-C)haloalkylcarbonyl-(C-C)alkyl, (C-C)alkylsulfonylamino,'}{'sub': 1', '4', '1', '4', '2', '4', '2', '4', '3', '6', '1', '4', '3', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'or is in each case optionally identically or differently mono- or di-aryl-, -hetaryl- or -heterocyclyl-substituted (C-C)alkyl, (C-C)alkoxy, (C-C)alkenyl, (C-C)alkynyl, (C-C)cycloalkyl, where aryl, hetaryl or heterocyclyl are each optionally identically ...

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14-09-2017 дата публикации

BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS

Номер: US20170260183A1
Принадлежит:

The present application relates to novel bicyclic compounds, to compositions comprising these compounds, to their use for controlling animal pests and to processes and intermediates for their preparation. 3. Composition claim 1 , comprising a content of at least one compound of formula (I) according to and one or more customary extenders and/or surfactants.4. A compound of the formula (I) according for controlling pests. The present application relates to novel bicyclic compounds, to compositions comprising these compounds, to their use for controlling animal pests and to processes and intermediates for their preparation.Recently, bicyclic compounds having insecticidal properties have been disclosed (WO 2015/038503 A1).WO 2014/100695 A1 describes the preparation and pharmaceutical use of PRMTS inhibitors containing, inter alia, an N-substituted 2H-pyrazolo[3,4-b]pyridin-1-yl fragment. Furthermore, WO 2010/056999 describes the preparation of parasiticides containing an N-substituted 2H-pyrazolo[3,4-b]pyridin-1-yl fragment.Modern crop protection compositions have to meet many demands, for example in relation to extent, persistence and spectrum of their action and possible use. Questions of toxicity and of combinability with other active ingredients or formulation auxiliaries play a role, as does the question of the cost and complexity involved in the synthesis of an active ingredient. In addition, resistances can occur. For all these reasons alone, the search for novel crop protection compositions cannot be considered complete, and there is a constant need for novel compounds having improved properties compared to the known compounds, at least in relation to individual aspects.It was an object of the present invention to provide compounds which widen the spectrum of the pesticides under various aspects.The object, and further objects which are not stated explicitly but can be discerned or derived from the connections discussed herein, are achieved by compounds of the ...

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21-09-2017 дата публикации

BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS

Номер: US20170265474A1
Принадлежит: Bayer CropScience Aktiengesellschaft

The present application relates to novel bicyclic compounds, to compositions comprising these compounds, to their use for controlling animal pests and to processes and intermediates for their preparation.

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29-09-2016 дата публикации

NOVEL COMPOUNDS FOR CONTROLLING ARTHROPODS

Номер: US20160278379A1
Принадлежит:

The invention relates inter alia to compounds of the general formula (I) 8. A compound according to claim 1 , wherein Ris independently H and W is O.9. A compound according to claim 1 , wherein Ris independently H and W is O and B3 is C—R claim 1 , Ris halogen-substituted C-C-alkyl or halogen-substituted C-C-alkoxy.10. A compound according to claim 1 , wherein the Ato Aand Bto Bmoieties are as follows:{'sub': '1', 'Ais C—H,'}{'sub': '2', 'sup': '3', 'Ais CRor N,'}{'sub': '3', 'sup': '4', 'Ais CR,'}{'sub': '4', 'Ais C—H,'}{'sub': '1', 'sup': '6', 'Bis CRor N,'}{'sub': '2', 'Bis C—H,'}{'sub': '3', 'sup': '8', 'Bis CR,'}{'sub': '4', 'Bis C—H and'}{'sub': '5', 'sup': '10', 'Bis CRor N.'}11. A compound according to claim 1 , wherein Ris H.12. A compound according to claim 1 , wherein Q is C-C-alkyl claim 1 , cyclopropyl claim 1 , 1-(cyano)cyclopropyl claim 1 , 1-(perfluorinated C-C-alkyl)cyclopropyl claim 1 , 1-(C-C-alkyl)cyclopropyl claim 1 , 1-(thiocarbamoyl)cyclopropyl claim 1 , halogen-substituted C-C-alkyl claim 1 , thietan-3-yl claim 1 , N-methylpyrazol-3-yl or 2-oxo-2(2 claim 1 ,2 claim 1 ,2-trifluoroethylamino)ethyl.13. A compound according to claim 1 , wherein Ris fluorine-substituted C-C-alkoxy or fluorine-substituted C-C-alkyl.14. An insecticidal composition claim 1 , comprising a content of at least one compound according to and an extender and/or a surface-active substance. The present application relates to trifluoro novel compounds, to processes for preparation thereof and to use thereof for controlling animal pests, in particular arthropods and especially insects, arachnids and nematodes.It is known that particular halogen-substituted compounds have insecticidal activity (EP 1 911 751, WO2012/069366, WO2012/080376, WO2012/107434 and WO2012/175474).WO 2011/113756 discloses triazole derivatives having insecticidal activity.It is also known that particular halogen-substituted compounds have cytokine-inhibiting activities (WO 2000/07980).Modern crop ...

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08-10-2015 дата публикации

NOVEL HETEROCYCLIC COMPOUNDS AS PEST CONTROL AGENTS

Номер: US20150284380A1
Принадлежит:

The present invention relates to novel heterocyclic compounds, to processes for preparation thereof and to the use thereof for controlling animal pests, which also include arthropods and especially insects. 2. A Salt claim 1 , tautomeric and/or isomeric form and/or N-oxide of a compound of formula (I) according to .3. A Composition claim 1 , comprising at least one compound of formula (I) and/or salt claim 1 , tautomeric and/or isomeric form and/or N-oxide according to .4. Method for controlling pests claim 1 , comprising allowing a compound of formula (I) according to to act on a pest and/or a habitat thereof. The present application relates to novel heterocyclic compounds, to processes for preparation thereof and to the use thereof for controlling animal pests, which also include arthropods and especially insects.WO 2008/028903 A2, WO 2003/077918 A1 and WO 2003/029210 A2 disclose heterocyclic compounds for which pharmaceutical applications are described.Further heterocycles suitable for use in crop protection are described in WO 2009/149858, WO 2010/006713, WO2011/045240 and WO 2011/045224.Modern crop protection agents have to meet many demands, for example in relation to efficacy, persistence and spectrum of their action and possible use. Questions of toxicity and of combinability with other active compounds or formulation auxiliaries play a role, as does the question of the expense that the synthesis of an active compound requires. In addition, resistances can occur. For all these reasons alone, the search for novel crop protection agents cannot be considered complete, and there is a constant need for novel compounds having improved properties compared to the known compounds, at least in relation to individual aspects.It was an object of the present invention to provide compounds which widen the spectrum of the pesticides in various respects.This object, and further objects which are not stated explicitly but can be discerned or derived from the connections ...

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27-09-2018 дата публикации

PYRAZOLOPYRIDINE SULFONAMIDES AS NEMATICIDES

Номер: US20180273534A1
Принадлежит:

Disclosed are compounds of formula (I) which possess nematicidal properties This application is a divisional application of U.S. patent application Ser. No. 15/309,183, filed 6 Nov. 2016, which is a § 371 National Stage Application of PCT/EP2015/059776, filed 5 May 2015, which claims priority to EP 14167534.8, filed 8 May 2014. The above applications are each incorporated by reference in their entireties.The present invention relates to pyrazolopyridine sulfonamides, their use for the control of animal pests, especially nematodes, in agricultures, formulations containing such compounds and methods for the control of animal pests, especially nematodes. This invention relates to certain sulfonamides, their N-oxides, salts and formulations suitable for agronomic and nonagronomic uses, and methods of their use for controlling animal pests, especially nematodes, in both agronomic and nonagronomic environments. The present invention further relates to processes and intermediate compounds for the preparation of such pyrazolopyridine sulfonamides.Nematodes cause a substantial loss in agricultural product including food and industrial crops and are combated with chemical compounds having nematicidal activity. To be useful in agriculture these compounds should have a high activity, a broad spectrum activity against different strains of nematodes and should not be toxic to non-target organisms. Due to widespread development of resistance to anthelmintic agents in nematode parasites, nematodes continue to cause problems in livestock despite the available chemical therapeutic agents. The need continues for new compounds which are more effective, less costly, less toxic, environmentally safer or have different modes of action.European Patent Application Publication No. 0 244 166 A2 (referred to as P1) discloses compounds of formula (i) as herbicideswherein, inter alia, R is H or an organic substituent, W is O or S, L is an aryl or heteroaryl moiety, and A is selected from a list ...

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15-10-2015 дата публикации

PYRIDYLOXYALKYL CARBOXAMIDES AND USE THEREOF AS ENDOPARASITICIDES AND NEMATICIDES

Номер: US20150291524A1
Принадлежит:

The present application relates to novel pyridyloxyalkylcarboxamides of the formula (I) 6. Compound of formula (I) and/or a salt claim 1 , N-oxide and/or tautomeric form thereof according to for use as medicaments for controlling endoparasites in animals or humans.7. Compound of formula (I) and/or a salt claim 1 , N-oxide and/or tautomeric form thereof according to for controlling endoparasites in animals or humans.8. A compound and/or a salt claim 1 , N-oxide and/or tautomeric form thereof according to capable of being used for preparing medicaments for controlling endoparasites in animals or humans.9. Compound and/or a salt claim 1 , N-oxide and/or tautomeric form thereof according to for use in the control of endoparasites in animals claim 1 , wherein the compound and a salt claim 1 , N-oxide and/or tautomeric form is administered prophylactically and/or therapeutically to an animal and/or human.10. Endoparasiticidal composition comprising a compound of formula (I) and/or a salt claim 1 , N-oxide and/or tautomeric form thereof according to .11. A compound and/or a salt claim 1 , N-oxide and/or tautomeric form thereof according to capable of being used for controlling phytopathogenic nematodes.12. Method for controlling phytopathogenic nematodes claim 1 , comprising bringing a compound of formula (I) and/or a salt claim 1 , N-oxide and/or tautomeric form thereof according to into contact with a plant or plant part claim 1 , soil in which the plant grows and/or plant propagation material.13. Nematicidal or endoparasiticidal composition comprising one or more compounds of formula (I) and/or a salt claim 1 , N-oxide and/or tautomeric form thereof according to and one or more auxiliaries. The present application relates to novel pyridyloxyalkylcarboxamides and to their use as endoparasiticides against endoparasites in animals or humans, and to their use as nematicides for controlling phytopathogenic nematodes, and furthermore to endoparasiticides and nematicides ...

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16-12-2021 дата публикации

NOVEL HETEROARYL-TRIAZOLE AND HETEROARYL-TETRAZOLE COMPOUNDS AS PESTICIDES

Номер: US20210386070A1
Принадлежит:

The present invention relates to novel heteroaryl-triazole and heteroaryl-tetrazole compounds of the general formula (I), in which the structural elements Y, Q, Q, R, R, R, Rand Rhave the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals. 2. The compound according to claim 1 , in whichX is O or S;{'sup': 1', '2', '5', '1', '2, 'Qand Qare independently CRor N, provided at least one of Qand Qis N;'}{'sub': '2', 'Y is a direct bond or CH;'}{'sup': '1', 'sub': 1', '6', '2', '2', '3', '3', '1', '6', '2', '6', '2', '6', '2', '6', '2', '6', '3', '4', '1', '2', '3', '4', '2', '1', '3, 'Ris hydrogen; C-Calkyl optionally substituted with one substituent selected from —CN, —CONH, —COOH, —NOand —Si(CH); C-Chaloalkyl; C-Calkenyl; C-Chaloalkenyl; C-Calkynyl; C-Chaloalkynyl; C-Ccycloalkyl-C-Calkyl- wherein the C-Ccycloalkyl is optionally substituted with one or two halogen atoms; oxetan-3-yl-CH— or benzyl optionally substituted with halogen atoms or C-Chaloalkyl;'}{'sup': '2', 'sub': 1', '3', '1', '3', '1', '3', '1', '3', '1', '3', '2', '5', '2', '2, 'Ris phenyl, pyridine, pyrimidine, pyrazine or pyridazine, wherein the phenyl, pyridine, pyrimidine, pyrazine or pyridazine is optionally substituted with one to three substituents, provided the substituent(s) are not on either carbon adjacent to the carbon bonded to the C═X-group, each independently selected from the group consisting of C-Calkyl, C-Chaloalkyl, C-Chaloalkylthio, C-Calkoxy, C-Chaloalkoxy, halogen, —NO, —SF, —CN, —CONH, —COOH and —C(S)NH;'}{'sup': '3', 'sub': 1', '3', '1', '3, 'Ris C-Calkyl or C-Chaloalkyl;'}{'sup': '4', 'claim-text': [{'sub': 2', '2', '2', '2', '1', '6', '3', '6', '1', '3', '1', '4', '1', '3', '1', '6', '1', '6', '1', '6', '3', '6', '3', '6', '3', '6', '1', '3', '1', '3', '1', '3', '1', '4', '1', '4', '2 ...

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12-09-2019 дата публикации

2-[3-(ALKYLSULFONYL)-2H-INDAZOL-2-YL]-3H-IMIDAZO[4,5-B]PYRIDINE DERIVATIVES AND SIMILAR COMPOUNDS AS PESTICIDES

Номер: US20190274306A1
Принадлежит:

The invention relates to compounds of the formula (Ia) or (Ib), in which Aa, Ab, Ac, Ad, R, RR, R, R, R, R, R, R, Q, R4, R, Rand have the meanings indicated in the claims, and to agrochemical formulations containing the compounds according to formula (Ia) or (Ib) for use as acaricides and/or insecticides for combating animal pests, primarily arthropods and in particular insects and arachnids. 2-[3-(alkylsulfonyl)-2H-indazol-2-yl]-3H-imidazo[4,5-b]pyridine derivatives and similar compounds are particularly preferable. 3: The compound of formula (Ia) or (Ib) according to claim 2 , in which claim 2 ,{'img': {'@id': 'CUSTOM-CHARACTER-00028', '@he': '3.22mm', '@wi': '3.22mm', '@file': 'US20190274306A1-20190912-P00001.TIF', '@alt': 'custom-character', '@img-content': 'character', '@img-format': 'tif'}, 'if represent exclusively double bonds and hence Aa to Ad together with the carbon atoms adjacent to Aa and Ad in each case form an aromatic ring,'}{'sup': '10', 'Aa is nitrogen or C(R),'}{'sup': '11', 'Ab is nitrogen or C(R),'}{'sup': '12', 'Ac is nitrogen or C(R), and'}{'sup': '13', 'Ad is nitrogen or C(R),'}where not more than two of Aa, Ab, Ac and Ad are nitrogen,{'img': {'@id': 'CUSTOM-CHARACTER-00029', '@he': '3.22mm', '@wi': '3.22mm', '@file': 'US20190274306A1-20190912-P00001.TIF', '@alt': 'custom-character', '@img-content': 'character', '@img-format': 'tif'}, 'or, if represent exclusively single bonds,'}{'sup': 10', '14, 'Aa is C(R)(R),'}{'sup': 11', '15, 'Ab is C(R)(R),'}{'sup': 12', '16, 'Ac is C(R)(R) and'}{'sup': 13', '17, 'Ad is C(R)(R),'}{'sup': '1', 'sub': 1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Ris (C-C)alkyl, (C-C)hydroxyalkyl, (C-C)haloalkyl, (C-C)alkenyl, (C-C)haloalkenyl, (C-C)alkynyl, (C-C)haloalkynyl, (C-C)cycloalkyl, (C-C)alkylthio-(C-C)alkyl, (C-C)alkylsulfinyl-(C-C)alkyl or (C-C)alkylsulfonyl-(C-C)alkyl,'}{'sup': 10', '11', '12', '13', '14', '15', '16 ...

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04-10-2018 дата публикации

Mesoionic imidazole derivatives as insecticides

Номер: US20180282323A1
Принадлежит:

What are demonstrated are compounds of the formula (I) 3. Compound according to claim 1 , in which{'sup': 1', '2, 'Qand Qtogether are one of the A-1, A-4 or A-5 radicals which, together with the carbon and nitrogen atom to which they are bonded, form a 5- or 6-membered aromatic ring,'}{'sup': 5', '6', '7', '8', '7a', '7', '8, 'T is R, —OR, —N(R)(R) or —N(R)—N(R)(R),'}W is O,{'sup': 9', '10, 'G is a bond or is —C(R)(R)—,'}U is a cycle from the group of U-2, U-9, U-10 or U-23,{'sup': 'a', 'Xis halogen, cyano, methyl, ethyl, trifluoromethyl, methoxy, ethoxy, trifluoromethoxy, methylthio, methylsulphinyl, methylsulphonyl or methoxycarbonyl,'}n is 0, 1 or 2,{'sup': 1', '2', '3', '4, 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '3', '4', '3', '4', '1', '4', '1', '4', '1', '4, 'R, R, R, Rare each independently a radical from the group of hydrogen, halogen, cyano, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, C-C-haloalkoxy, C-C-alkoxy-C-C-alkyl, C-C-alkenyl, C-C-alkenyloxy, C-C-alkynyl, C-C-alkynyloxy, C-C-alkylthio, C-C-alkylsulphinyl or C-C-alkylsulphonyl,'}{'sup': '5', 'sub': '2', 'Ris CHY,'}{'sup': 51', '52', '53', '54, 'sub': 'p', 'Y is hydrogen, Cl, Br, —O—R, —S(O)—R, —N(R)(R) or is one of the Y-2, Y-3, Y-4, Y-5, Y-6 or Y-7 radicals,'}{'sup': 'b', 'Xis halogen, cyano, methyl, ethyl, trifluoromethyl, difluoromethyl, methylaminocarbonyl, methylcarbonylamino, methoxy, ethoxy, trifluoromethoxy, methylthio, ethylthio, methylsulphinyl, methylsulphonyl or methoxycarbonyl,'}m is 0, 1 or 2,p is 0, 1 or 2,{'sup': '51', 'claim-text': [{'sub': 1', '6', '2', '4', '2', '4', '3', '6', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'is C-C-alkyl, C-C-alkenyl, C-C-alkynyl or C-C-cycloalkyl, where the aforementioned radicals may optionally be mono- to trisubstituted by halogen or monosubstituted by cyano, C-C-cycloalkyl, C-C-alkoxy, C-C-haloalkoxy, C-C-alkylthio, C-C-alkylsulphinyl, C-C-alkylsulphonyl, C-C- ...

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04-10-2018 дата публикации

BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS

Номер: US20180282347A1
Принадлежит: Bayer CropScience Aktiengesellschaft

The present application relates to novel bicyclic compounds, to compositions comprising these compounds, to their use for controlling animal pests and to processes and intermediates for their preparation. 3. A composition claim 1 , comprising a content of at least one compound of the formula (I) according to and one or more customary extenders and/or surfactants.4. A compound of the formula (I) according to for controlling pests. The present application relates to novel bicyclic compounds, to compositions comprising these compounds, to their use for controlling animal pests and to processes and intermediates for their preparation.EP 2 772 485 A1 describes 5,6-bicyclic compounds for pharmaceutical and diagnostic applications.Recently, bicyclic compounds having insecticidal properties have been disclosed (WO 2015/038503 A1).Modern crop protection compositions have to meet many demands, for example in relation to extent, persistence and spectrum of their action and possible use. Questions of toxicity and of combinability with other active ingredients or formulation auxiliaries play a role, as does the question of the expense that the synthesis of an active ingredient requires. In addition, resistances can occur. For all these reasons alone, the search for novel crop protection compositions cannot be considered complete, and there is a constant need for novel compounds having improved properties compared to the known compounds, at least in relation to individual aspects.It was an object of the present invention to provide compounds which widen the spectrum of the pesticides under various aspects.This object, and further objects which are not stated explicitly but can be discerned or derived from the connections discussed herein, are achieved by novel compounds of the formula (I)in whichA represents an A radical from the group consisting of (A-b) to (A-f)in which the broken line denotes the bond to the carbon atom of the bicyclic system of the formula (I) andBrepresents ...

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13-10-2016 дата публикации

NOVEL COMPOUNDS FOR CONTROLLING ARTHROPODS

Номер: US20160297765A1
Принадлежит:

The invention relates inter alia to compounds of the general formula (I) 9. Compounds according to any of to , wherein Ris independently H and W is O.10. Compounds according to any of to , wherein Ris independently H and W is O and Bis C—R , Ris halogen-substituted C-C-alkyl or halogen-substituted C-C-alkoxy.11. Compound according to any of to , wherein the Ato Aand Bto Bmoieties are as follows:{'sub': '1', 'Ais C—H,'}{'sub': '2', 'sup': '3', 'Ais CRor N,'}{'sub': '3', 'sup': '4', 'Ais CR,'}{'sub': '4', 'Ais C—H,'}{'sub': '1', 'sup': '6', 'Bis CRor N,'}{'sub': '2', 'Bis C—H,'}{'sub': '3', 'sup': '8', 'Bis CR,'}{'sub': '4', 'Bis C—H and'}{'sub': '5', 'sup': '10', 'Bis CRor N.'}12. Compounds according to any of to , wherein Ris methyl.13. Compounds according to any of to , wherein Q is C-C-alkyl , cyclopropyl , 1-(cyano)cyclopropyl , 1-(perfluorinated C-C-alkyl)cyclopropyl , 1-(C-C-alkyl)cyclopropyl , 1-(thiocarbamoyl)cyclopropyl , halogen-substituted C-C-alkyl , thietan-3-yl , N-methylpyrazol-3-yl or 2-oxo-2(2 ,2 ,2-trifluoroethylamino)ethyl.14. Compounds according to any of to , wherein Ris fluorine-substituted C-C-alkoxy or fluorine-substituted C-C-alkyl.15. Insecticidal composition , characterized by a content of at least one compound of the formula (I) according to any of to and an extender and/or a surface-active substance. The present application relates to trifluoro novel compounds, to processes for preparation thereof and to use thereof for controlling animal pests, in particular arthropods and especially insects, arachnids and nematodes.It is known that particular halogen-substituted compounds have insecticidal activity (EP 1 911 751, WO2012/069366, WO2012/080376, WO2012/107434 and WO2012/175474).WO 2011/113756 discloses triazole derivatives having insecticidal activity.It is also known that particular halogen-substituted compounds have cytokine-inhibiting activities (WO 2000/07980).Modern crop protection compositions have to meet many demands, for example ...

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11-10-2018 дата публикации

NOVEL COMPOUNDS FOR CONTROLLING ARTHROPODS

Номер: US20180289007A1
Принадлежит: Bayer CropScience Aktiengesellschaft

The invention relates inter alia to compounds of the general formula (I). Also described are methods for preparing the compounds of the formula (I). The compounds according to the invention are especially suitable for controlling insects, arachnids and nematodes in agriculture, and ectoparasites in veterinary medicine and also as herbicides. 2. Compound according to claim 1 , wherein Rin T is H.3. Compound according to claim 1 , wherein T is T2 claim 1 , T3 or T7 claim 1 , optionally T3.4. Compound according to claim 1 , wherein Ais CR claim 1 , Ais CR claim 1 , Ais CR claim 1 , Ais CR claim 1 , Ais C and R claim 1 , Rand Rare in each case H.5. Compound according to claim 1 , wherein Bis CR claim 1 , Bis CR claim 1 , Bis CR claim 1 , Bis CRand Bis CR.6. Compound according to claim 1 , wherein Bis CRand Ris halogenated C-C-alkyl and Bis CRand Bis CRand Rand Rare each H.7. Compound according to claim 1 , wherein Bis CRand Bis CRand Rand Rare each optionally independently halogen claim 1 , C-C-alkyl or C-C-alkyl substituted by halogen claim 1 , C-C-alkoxy or C-C-alkoxy substituted by halogen.8. Compound according to claim 1 , wherein Ais CRand Ris H claim 1 , halogen claim 1 , optionally F or Cl claim 1 , optionally F or Rtogether with the carbon atom of CR claim 1 , Aand either C-Mor C-Mform a 5- or 6-membered ring optionally substituted by F claim 1 , Cl claim 1 , Br claim 1 , I claim 1 , C-C-alkyl claim 1 , which may contain 0 claim 1 , 1 or 2 nitrogen atoms and/or 0 claim 1 , 1 or 2 oxygen atoms and/or 0 claim 1 , 1 or 2 sulfur atoms claim 1 , optionally form a 5-membered carbon ring.9. Compound according to claim 1 , wherein Mand Mare each independently H or C-C-alkyl claim 1 , optionally H claim 1 , or C-Mor C-Mtogether with CRand Aform a 5- or 6-membered ring optionally substituted by F claim 1 , Cl claim 1 , Br claim 1 , I claim 1 , C-C-alkyl claim 1 , which may contain 0 claim 1 , 1 or 2 nitrogen atoms and/or 0 claim 1 , 1 or 2 oxygen atoms and/or 0 claim 1 , ...

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27-10-2016 дата публикации

Compounds with Nematicidal Activity

Номер: US20160309717A1
Принадлежит:

The present invention relates to the novel pyridyl carboxamide derivatives and their use as nematicides, compositions containing such compounds and methods for the control of nematodes. 2. A composition claim 1 , comprising an effective amount of at least one compound of formula (I) according to and at least one surfactant claim 1 , and/or solid or liquid diluent.3. A compound according to capable of being used for controlling nematodes.4. A compound according to capable of being used as an antihelminthic.5. A nematode control agent comprising a compound of .6. An antihelminthic comprising a compound of . The present invention relates to the novel pyridyl carboxamide derivatives and their use as nematicides, compositions containing such compounds and methods for the control of nematodes.Nematodes cause a substantial loss in agricultural product including food and industrial crops and are combated with chemical compounds having nematicidal activity. To be useful in agriculture these compounds should have a high activity, a broad spectrum activity against different strains of nematodes and should not be toxic to non-target organisms.The use of certain N-2-(pyridyl)ethyl-carboxamide derivatives for controlling nematodes is described in EP 2 132 987 A1.Compounds with nematicidal activity are disclosed in WO 2013/064460, WO 2013/064461, WO 2013/064521. See also WO 2012/118139.The present invention relates to novel compounds of formula (I)in which X, R, R, Rand A have the meanings listed in the following tableSurprisingly it has now been found that these compounds exhibit pronounced nematicidal activity.It was also found that the compounds of formula (I) exhibit activity against bacteria and viruses and can be used as bactericides and as virucides.The compounds of formula (I) can also be used as antihelminthics in the field of animal health.In particular the present invention relates to the use of compounds of formula (I) against phytopathogenic nematodes, i.e. against ...

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17-09-2020 дата публикации

SUBSTITUTED SULPHONAMIDES FOR CONTROLLING ANIMAL PESTS

Номер: US20200288710A1
Принадлежит:

The present invention relates to the use of a compound of the general formula (I)

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26-10-2017 дата публикации

HETEROCYCLIC COMPOUNDS AS PESTICIDES

Номер: US20170305864A1
Принадлежит:

The present application relates to the use of heterocyclic compounds for controlling animal pests including arthropods, insects and nematodes, to novel heterocyclic compounds, to processes for their preparation and to intermediates for preparing the heterocyclic compounds. 7. A composition comprising at least one compound of formula (I) as described in .8. A composition comprising at least one compound of formula (I) as described in .9. Method for controlling one or more pests claim 6 , comprising allowing a compound of formula (I) according to to act on one or more pests and/or a habitat thereof.10. 2-(3 claim 6 ,5-Difluoropyridin-2-yl)-2H-1 claim 6 ,2 claim 6 ,3-triazole-4-amine.11. 1-(3 claim 6 ,5-Difluoropyridin-2-yl)-1H-pyrazole-3-amine.12. N-[1-(2 claim 6 ,6-Difluorophenyl)-4 claim 6 ,5-dihydro-1H-pyrazol-3-yl]acetamide.13. N-[1-(2 claim 6 ,6-Difluorophenyl)-1H-pyrazol-3-yl]acetamide.14. 1-(2 claim 6 ,6-Difluorophenyl)-1H-pyrazole-3-amine.15. 1-(2 claim 6 ,6-Difluorophenyl)-4 claim 6 ,5-dihydro-1H-pyrazole-3-amine. This application is continuation of U.S. application Ser. No. 14/432,501, filed 31 Mar. 2015, which is a §371 National Stage Application of PCT/EP2013/070371, filed 30 Sep. 2013, which claims priority to EP 12186946.5, filed 2 Oct. 2012 and EP 13170565.9, filed 5 Jun. 2013, the contents of each are incorporated herein in their entireties.The present application relates to the use of heterocyclic compounds for controlling animal pests including arthropods, insects and nematodes, to novel heterocyclic compounds, to processes for their preparation and to intermediates for preparing the heterocyclic compounds.The heterocyclic compounds of the formulae (W) and (W2) are known (cf. for the compounds of the formula (W) Registry Numbers 1189645-25-7, 1189474-83-6, 1193202-69-5, 1172407-07-6, 1185158-40-0, 1185036-12-7, 1170986-74-9, 1193179-17-7, 1189458-68-1, 1189956-23-7, 1189915-26-1, 1170047-96-7). A use of these compounds has not been described. ...

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03-11-2016 дата публикации

SIX-MEMBERED C-N-BONDED ARYL SULPHIDE AND ARYL SULPHOXIDE DERIVATIVES AS PESTICIDES

Номер: US20160316751A1
Принадлежит: Bayer CropScience Aktiengesellschaft

Illustrated are compounds of the formula (I), which are suitable for controlling animal pests including arthropods and in particular insects and acarids 2. Compound according to claim 1 , in whichV represents oxygen;{'sup': '5', 'claim-text': {'sup': '5', 'sub': 1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '3', '6', '1', '6, 'Rrepresents hydrogen, halogen, amino, cyano, nitro, (C-C)-alkyl, (C-C)-haloalkyl, (C-C)-alkylsulphanyl, (C-C)-alkylsulphinyl, (C-C)-alkylsulphonyl, (C-C)-haloalkylsulphanyl, (C-C)-haloalkylsulphinyl, (C-C)-haloalkylsulphonyl, (C-C)-cycloalkyl or (C-C)-alkoxy;'}, 'Q represents C—Ror nitrogen, where'}{'sup': 3', '6, 'claim-text': represent hydrogen, halogen, cyano or nitro; or', {'sub': 1', '6', '1', '6', '2', '6', '2', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '5', '1', '5', '2', '6, 'represent (C-C)-alkyl, (C-C)-haloalkyl, (C-C)-alkenyl, (C-C)-alkynyl, (C-C)-alkoxy, (C-C)-haloalkoxy, (C-C)-haloalkylsulphanyl, (C-C)-haloalkylsulphinyl, (C-C)-haloalkylsulphonyl, (C-C)-alkylsulphanyl, (C-C)-alkylsulphinyl, (C-C)-alkylsulphonyl, (C-C)-alkylcarbonyl, (C-C)-haloalkylcarbonyl or (C-C)-alkoxycarbonyl; or'}, {'sub': 3', '6', '3', '6', '1', '3', '3', '6, 'represent (C-C)-cycloalkyl, (C-C)-cycloalkyl-(C-C)-alkyl or (C-C)-cycloalkenyl, where the radicals mentioned above may optionally be substituted by halogen, alkyl, cyano, nitro, alkoxy, haloalkyl or haloalkoxy; or'}, {'sub': 1', '3', '1', '3, 'represent phenyl, heteroaryl, phenyl-(C-C)-alkyl or heteroaryl-(C-C)-alkyl, where the radicals mentioned above may optionally be substituted by halogen, alkyl, cyano, nitro, alkoxy, haloalkyl or haloalkoxy; or'}, {'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '3', '4', '3', '4', '2', '4', '3', '4', '3', '4', '3', '4', '1', '4', '1', '4, 'where R′ and R″ independently of one another represent hydrogen, cyano, (C-C)-alkyl ...

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25-10-2018 дата публикации

2-(Het)aryl-substituted fused heterocycle derivatives as pesticides

Номер: US20180303097A1
Принадлежит:

The invention relates to novel compounds of the formula (I) 2. Compound of formula (I) according to in which{'sup': 1', '+', '−', '4, 'Arepresents nitrogen, ═N(O)— or ═C(R)—,'}{'sup': '1', 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '2', '4', '2', '4', '1', '4', '2', '4', '1', '4', '2', '4', '2', '4', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '3', '6', '1', '4', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Rrepresents (C-C)alkyl, (C-C)hydroxyalkyl, (C-C)haloalkyl, (C-C)cyanoalkyl, (C-C)alkoxy-(C-C)alkyl, (C-C)haloalkoxy-(C-C)alkyl, (C-C)alkenyl, (C-C)alkenyloxy-(C-C)alkyl, (C-C)haloalkenyloxy-(C-C)alkyl, (C-C)haloalkenyl, (C-C)cyanoalkenyl, (C-C)alkynyl, (C-C)alkynyloxy-(C-C)alkyl, (C-C)haloalkynyloxy-(C-C)alkyl, (C-C)haloalkynyl, (C-C)cyanoalkynyl, (C-C)cycloalkyl, (C-C)cycloalkyl(C-C)cycloalkyl, (C-C)alkyl-(C-C)cycloalkyl, halo(C-C)cycloalkyl, (C-C)alkylamino, di-(C-C)alkylamino, (C-C)cycloalkylamino, (C-C)alkylcarbonylamino, (C-C)alkylthio-(C-C)alkyl, (C-C)haloalkylthio-(C-C)alkyl, (C-C)alkylsulphinyl-(C-C)alkyl, (C-C)haloalkylsulphinyl-(C-C)alkyl, (C-C)alkylsulphonyl-(C-C)alkyl, (C-C)alkylcarbonyl-(C-C)alkyl, (C-C)haloalkylcarbonyl-(C-C)alkyl, (C-C)alkylsulphonylamino,'}{'sub': 1', '4', '1', '4', '2', '4', '2', '4', '3', '6', '1', '4', '3', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'or represents (C-C)-alkyl, (C-C)alkoxy, (C-C)alkenyl, (C-C)alkynyl, (C-C)cycloalkyl, each of which is optionally mono- or disubstituted by identical or different substituents from the group consisting of aryl, hetaryl and heterocyclyl, where aryl, hetaryl and heterocyclyl may in each case optionally be mono- or disubstituted by identical or different substituents from the group consisting of halogen, ...

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25-10-2018 дата публикации

N-(2-FLUORO-2-PHENETHYL)CARBOXAMIDES AS NEMATICIDES AND ENDOPARASITICIDES

Номер: US20180305299A1
Принадлежит:

The present invention relates to N-(2-halogen-2-phenethyl)carboxamides, a process for producing such compounds, their use for the control of nematodes in agricultures and their use as anthelmintics against endoparasites in animals or humans, compositions containing such compounds and methods for the control of nematodes and helminths. 2. The method according to claim 1 , wherein{'sup': 2', '3', '4', '5, 'Y, Y, Yand Yrepresent independently from each other hydrogen.'}3. The method according to claim 1 , wherein n represents 1.4. The method according to claim 1 , wherein n represents 0.5. The method according to claim 1 ,{'sup': 1', '2', '3, 'wherein Zrepresents fluorine and Zand Zrepresent hydrogen.'}7Cooperia curticei.. The method according to claim 1 , wherein the nematode is8Haemonchus contortus.. The method according to claim 1 , wherein the nematode is9Nippostrongylus brasiliensis.. The method according to claim 1 , wherein the nematode is10Heligmosomoides polygyrus.. The method according to claim 1 , wherein the nematode is11Trichostrongylus colubriformis.. The method according to claim 1 , wherein the nematode is12Dirofilaria immitis.. The method according to claim 1 , wherein the nematode is13Meloidogyne incognita.. The method according to claim 1 , wherein the nematode is14chrysanthemum. The method according to claim 1 , wherein the plant is selected from the group consisting of rice claim 1 , barley claim 1 , wheat claim 1 , rye claim 1 , oat claim 1 , corn claim 1 , soybean claim 1 , azuki bean claim 1 , broad bean claim 1 , pea claim 1 , apple claim 1 , citrus claim 1 , pear claim 1 , pineapple claim 1 , grape claim 1 , peach claim 1 , Japanese apricot claim 1 , cherry claim 1 , nut claim 1 , banana claim 1 , strawberry claim 1 , pome fruit claim 1 , stone fruit claim 1 , cabbage claim 1 , tomato claim 1 , spinach claim 1 , broccoli claim 1 , lettuce claim 1 , onion claim 1 , Welsh onion claim 1 , pepper claim 1 , carrot claim 1 , potato claim 1 , sweet ...

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25-10-2018 дата публикации

FUSED BICYCLIC HETEROCYCLE DERIVATIVES AS PESTICIDES

Номер: US20180305353A1
Принадлежит:

The invention relates to novel compounds of the formula (I) or (I′) 4. Compound of formula (I) or (I′) according to claim 1 , in which{'sup': '7', 'Aa is nitrogen or ═C(R)—,'}Ab is nitrogen or ═C(H)—,Ac is nitrogen or ═C(H)—,Ad is nitrogen or ═C(H)—,Ae is nitrogen or ═C(H)—,where Ab, Ac, Ad and Ae cannot all be nitrogen,optionally resulting in the following structural units: A1, A2, A4, A5, A7, A9, A11, A12, A13, A19, A20, A21, A22, A23, A24, A26, A27, A29, A31, A33, A34, A35, A41, A42, A43, A44,{'sup': '1', 'sub': 1', '4', '1', '4', '3', '6, 'Ris (C-C)-alkyl, (C-C)-haloalkyl or (C-C)-cycloalkyl,'}{'sup': 2', '3, 'sub': 1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'R, Rare independently hydrogen, cyano, halogen, (C-C)-alkyl, (C-C)-alkoxy, (C-C)-haloalkyl, (C-C)-haloalkoxy, (C-C)-alkylthio, (C-C)-alkylsulphinyl, (C-C)-alkylsulphonyl, (C-C)-haloalkylthio, (C-C)-haloalkylsulphinyl, (C-C)-haloalkylsulphonyl or NHCO—(C-C)-alkyl ((C-C)-alkylcarbonylamino),'}{'sup': '7', 'sub': 1', '4', '1', '4, 'Ris hydrogen, halogen, cyano, (C-C)alkyl or (C-C)haloalkyl,'}Q is a heteroaromatic 9-membered or 12-membered fused bicyclic or tricyclic ring system from the group of Q1, Q2, Q3, Q5, Q6, Q8, Q9, Q10, Q11, Q12, Q13, Q15, Q16, Q17, Q18, Q19 or Q20,{'sup': '4', 'sub': 1', '4', '1', '4', '1', '4, 'Ris hydrogen, (C-C)alkyl or (C-C)-alkoxy-(C-C)alkyl,'}{'sup': '5', 'sub': 1', '4', '1', '4', '3', '6', '3', '6', '3', '6', '1', '4', '3', '6', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4', '1', '4, 'Ris hydrogen, cyano, halogen, (C-C)alkyl, (C-C)haloalkyl, (C-C)cycloalkyl, (C-C)cycloalkyl-(C-C)cycloalkyl, (C-C)alkyl-(C-C)cycloalkyl, (C-C)alkoxy, (C-C)haloalkoxy, (C-C)alkoxyimino, (C-C)alkylthio, (C-C)haloalkylthio, (C-C)alkylsulphinyl, (C-C)haloalkylsulphinyl, (C-C)alkylsulphonyl, (C-C)haloalkylsulphonyl, (C-C) ...

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02-11-2017 дата публикации

Current-Mode Sense Amplifier

Номер: US20170316812A1
Принадлежит: International Business Machines Corp

A current sense amplifier is provided. The amplifier comprises a first cross coupled inverter, a second cross coupled inverter, and a transmission gate. The first cross coupled inverter has a first source coupled to sense current input. The second cross coupled inverter has a second source coupled to a reference current input. The transmission gate comprises a first transmission end, a second transmission end, and a gate input. The first transmission end is operatively coupled to a first input of the first cross coupled inverter. The second transmission end is operatively coupled to a second input of the second cross coupled inverter. The gate input is operatively coupled to the control line input. Each cross coupled inverter is configured for switching a coupling of the sense current input and the reference current input.

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09-11-2017 дата публикации

COMPOUNDS FOR USE IN ANTHELMINTHIC TREATMENT

Номер: US20170320848A1
Принадлежит: Bayer Animal Health GmbH

Disclosed are compounds of formula (I) which possess anthelminthic properties wherein the structural elements have the meaning as indicated in the description. Further disclosed are such compounds for the control, treatment and/or prevention of infections with helminths in animals and humans. 10. A pharmaceutical composition comprising at least one compound of formula (I) according to claim 1 , or a salt claim 1 , a solvate claim 1 , a solvate of a salt claim 1 , an N-oxide claim 1 , a metal complex claim 1 , or a metalloid complex thereof.11. A method for the control claim 10 , treatment claim 10 , or prevention of infections with helminths claim 10 , comprising administering to an animal or human in need thereof the pharmaceutical composition according to .1214-. (canceled)15. A method for the control claim 1 , treatment or prevention of infections with helminths claim 1 , comprising the step of administering an effective amount of a compound of formula (I) of anyone of claim 1 , or a salt claim 1 , a solvate claim 1 , a solvate of a salt claim 1 , an N-oxide claim 1 , a metal complex claim 1 , or a metalloid complex thereof claim 1 , to an animal or human in need thereof. The present invention relates to certain bisphenyl-ethyl carboxamide derivatives. Further, the present invention relates to the use of certain bisphenyl-ethyl carboxamide derivatives for the control, treatment and/or prevention of infections with helminths in animals and humans, formulations containing such compounds and methods for the control, treatment and/or prevention of infections with helminths in animals and humans.The occurrence of resistances against all commercial anthelmintics seems to be a growing problem in the area of veterinary medicine. Therefore, endoparasiticides with new molecular modes of action are urgently desired. The new active ingredients should perform with excellent efficacy against a broad spectrum of helminths, like nematodes, preferably without any adverse toxic ...

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16-11-2017 дата публикации

BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS

Номер: US20170325458A1
Принадлежит: Bayer CropScience Aktiengesellschaft

The present application relates to novel bicyclic compounds, to their use for controlling animal pests and to processes and intermediates for their preparation. 3. The compound of the formula (I) as claimed in in which A represents the radical (A-b).4. The compound of the formula (I) as claimed in in which A represents the radical (A-f).5. The compound of the formula (I) as claimed in in which A represents the radical (A-a).6. A composition comprising a content of at least one compound of the formula (I) as claimed in and one or more customary extenders and/or surfactants.7. A product comprising one or more compounds of the formula (I) as claimed in or a composition thereof for controlling pests. The present application relates to novel bicyclic compounds, to compositions comprising these compounds, to their use for controlling animal pests and to processes and intermediates for their preparation.Recently, bicyclic compounds having insecticidal properties have been disclosed (WO 2015/038503 A1).WO 2010/078408 A1 describes the preparation and pharmaceutical use of Raf kinase inhibitors and WO 2013/259064 A1 describes the synthesis of anti-HIV agents and their use for the treatment of HIV infections, which compounds contain, inter alia, an N-substituted 2H-pyrazolo[3,4-b]pyridin-1-yl fragment. WO 2010/056999 describes the preparation of parasiticides containing an N-substituted 2H-pyrazolo[3,4-b]pyridin-1-yl fragment.Modern crop protection compositions have to meet many demands, for example in relation to extent, persistence and spectrum of their action and possible use. Questions of toxicity and of combinability with other active compounds or formulation auxiliaries play a role, as does the question of the expense that the synthesis of an active compound requires. In addition, resistances can occur. For all these reasons alone, the search for novel crop protection compositions cannot be considered complete, and there is a constant need for novel compounds having ...

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