N-Phenpropylcyclopentyl-Substituted Glutaramide Derivatives as Inhibitors of Neutral Endopeptidase Enzyme (NEP) for Treating Female Sexual Dysfunction (FSAD)
Номер патента: GEP20063783B
Опубликовано: 10-04-2006
Автор(ы): Adam Thomas Gillmore, Alan Stobie, Andrew Simon Cook, David Cameron Pryde, Donald Stuart Middleton, Stephen Challenger
Принадлежит: Pfizer
Опубликовано: 10-04-2006
Автор(ы): Adam Thomas Gillmore, Alan Stobie, Andrew Simon Cook, David Cameron Pryde, Donald Stuart Middleton, Stephen Challenger
Принадлежит: Pfizer
Реферат: 1. Technical Result Increase in treatment efficiency. 2. Essence N-phenpropylcyclopentyl -substituted glutara- mide derivatives of formula 1 wherein R1, X, Y are provided in the description, pharmaceutically acceptable salts thereof, solvates, polymorphs or prodrugs thereof as inhibitors of neutral endopeptidase (NEP) for treatment of the disorders of Female Sexual Dysfunction (FSAD), methods for its production and pharmaceutical compositions on its basis. 3. Field of Application Medicine, pharmacology.
N-phenpropylcyclopentyl-substituted glutaramide derivatives as NEP inhibitors for FSAD
Номер патента: NZ527012A. Автор: Donald Stuart Middleton,Alan Stobie,Andrew Simon Cook,Stephen Challenger,Adam Thomas Gillmore,Davidcameron Pryde. Владелец: Pfizer. Дата публикации: 2005-03-24.