24-06-2021 дата публикации
Номер: US20210188805A9
Автор:
CHRISTIAN Sven,
Eis Knut,
Ferrara Steven James,
Gradl Stefan Nikolaus,
GÜNTHER Judith,
Janzer Andreas,
KRÖBER Michael,
LIU Kery,
MERZ Claudia,
Müller Thomas,
Nguyen Duy,
Niehues Michael,
NISING Carl Friedrich,
Schäfer Martina,
SHEIKH Sherif El,
Stellfeld Timo,
SYKES David B.,
ZHAO Changjia,
ZHOU Han Jie,
Zimmermann Katja
Принадлежит:
The present invention provides triazolone compounds of general formula (I): 2. The method according to in which{'sup': '1', 'claim-text': [{'sub': 5', '8, 'a C-C-alkyl group,'}, {'sub': 2', '5, 'a C-C-haloalkyl group,'}, {'sub': 4', '5, 'claim-text': {'sup': 7', '8, 'claim-text': {'sub': 1', '3', '1', '4', '1', '3, 'wherein said phenyl substituent is optionally substituted, one, two or three times, each substituent independently selected from a halogen atom or a group selected from C-C-alkyl, C-C-haloalkyl, C-C-alkoxy and hydroxy,'}, 'wherein said cycloalkyl groups are optionally substituted, one or two times, each substituent independently selected from a halogen atom or a group selected from hydroxy, phenyl and —N(R)(R),'}, 'a C-C-cycloalkyl group,'}, {'sub': 1', '6', '3', '5, 'a C-C-alkyl group which is substituted with a C-C-cycloalkyl group,'}, {'sub': 2', '6, 'a C-C-alkyl group which is substituted with a cyano group, a hydroxy group or a phenyl group,'}, {'sub': 3', '6, 'a C-C-alkyl group which is substituted with a monocyclic- or bicyclic heteroaryl group,'}, {'sub': 2', '6', '2', '6, 'a (C-C-hydroxyalkyl)-O—(C-C-alky)-group,'}, {'sub': 3', '6, 'sup': 7', '8, 'a —(C-C-alkyl)-N(R)(R) group,'}, {'sub': 3', '5, 'sup': 7', '8, 'a —(C-C-cycloalkyl)-N(R)(R) group,'}, {'sub': 3', '6, 'sup': 7', '8, 'a —(C-C-alkyl)-C(═O)N(R)(R) group,'}, [{'sub': 1', '3', '1', '4', '1', '6', '3', '6', '2', '1', '6, 'claim-text': 'wherein said 5- to 6-membered heteroaryl substituent is optionally substituted, one, two or three times, each substituent independently selected from a halogen atom or a group selected from', 'which is optionally substituted one or two times, each substituent independently selected from a group selected from C-C-alkyl, 5- to 6-membered heteroaryl, —C(═O)O(C-C-alkyl), —C(═O)(C-C-alkyl), —C(═O)(C-C-cycloalkyl), —S(═O)(C-C-alkyl) and oxo (═O),'}, {'sub': 1', '3', '1', '4', '1', '3, 'C-C-alkyl, C-C-haloalkyl, C-C-alkoxy and hydroxy,'}, 'and wherein said- to 7- ...
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