Pesticidal 1 (4-phenoxyphenyl) - 3-benzoyl urea compounds and process for preparation.

PESTICIDAL 1-ARYLIMIDAZOLES

5-SUBSTITUTED-ALKYLAMINOPYRAZOLE DERIVATIVES AS PESTICIDES

PESTICIDAL BIPHENYLYLOXY AND BIPHENYLYLALKOXY ARYL ACYL UREA COMPOUNDS, A PROCESS FOR THEIR PREPARATION, PESTICIDAL COMPOSITIONS AND A METHOD OF CONTROLLING PESTS

PESTICIDES 1 (2-PYRIDYL) PYRAZOLE

1 (ALKYLPHENOXYARYL) - 3-BENZOYLHARNSTOFFE WITH PESTIZIDER EFFECT AND PROCEDURE FOR THEIR PRODUCTION.

5-SUBSTITUIERTE of ALKYLAMINOPYRAZOL DERIVATIVES AS PESTICIDES

Pesticides

Pesticidal 1-(2-pyridyl)pyrazoles

PESTICIDAL 1-(4-PHENOXYPHENYL)-3-BENZOYL UREA COMPOUNDS AND PROCESS FOR PREPARATION

5-SUBSTITUIERTE of ALKYLAMINOPYRAZOL DERIVATIVES AS PESTICIDES

PESTICIDAL 1-(4-PHENOXYPHENYL)-3-BENZOYL UREA COMPOUNDS AND PROCESS FOR PREPARATION

Control of arthropods in animals

PESTICIDAL 1-(2-PYRIDYL)PYRAZOLE

PURPOSE: To obtain a new compd. effective in controlling arthropods, nematodes, helminths or protozoa. CONSTITUTION: This is a new compd. of formula I (where X is halogen, nitro, alkylsulfinyl, etc.; Y is H, halogen, cyano, alkoxy, amino, etc.; Z is cyano or halogen; and R2-R5 are individually H, halogen, alkyl, alkoxy, cyano, nitro, etc., but at lest one of R2-R5 is other than H), e.g. 1-[2-(3-chloro-5- trifluoromethyl)pyridine]-5-amino-3-cyano-4-chlorodifluoromethylsulfenylpyrazole. The compd. of the formula I is obtd. by allowing a compd. of formula II (where R is 1-4C lower alkyl) to react with a sulfenyl halide and amidating the resultant sulfenyl compd. with ammonia. COPYRIGHT: (C)1993,JPO ...

1 (4-PHENOXYPHENYL) - 3-BENZOYLHARNSTOFFDERIVATE WITH PESTIZIDER EFFECT AND MANUFACTURING PROCESS.

PESTICIDES BIPHENYLYLOXY AND BIPHENYLYLALKOXYARYL ECYL UREA, PROCEDURES FOR THEIR PRODUCTION, PESTICIDES COMPOSITIONS AND PROCEDURES FOR THE FIGHT AGAINST PARASITS.

1- ALKYL-PHENOXYARYL -3-BENZOYL UREAS

PESTICIDAL 1-ARYLIMIDAZOLES

The invention describes novel 1-arylimidazoles of formula (I), wherein typically preferred substituents are: X is S(O)n R1, in which R1 is unsubstituted or halo-substituted alkyl a nd n is 0, 1 or 2; Y is hydrogen, halogen, alkyl, alkoxy, alkoxyalkylideneimino, alkylsulfenyl, alkylsulfinyl or alkylsulfonyl; Z is hydrogen or alkyl; R2 is halogen or alkylsulfenyl; R3 and R5 are hydrogen; R6 is halogen; and R4 is hydrogen, halogen, haloalkyl or haloalkoxy. The invention further describes processes to make the compounds, compositions of the compounds, and methods of use of the compounds for the control of arthropods (especially mites, aphids or insects), nematodes, helminths, or protozoa.

SULFONYLAMINOPYRAZOLE ALS PESTIZIDE

1-phenyl and 1-pyridylpyrazole derivatives and their use as pesticides

The invention relates to 1-(2,4,6-trisubstituted-phenyl)-5-amino-4-substituted-pyrazole derivatives of formula (I) or salts thereof wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

PESTICIDAL 1-(2-PYRIDYL)PYRAZOLES

Novel 1-(2-pyridyl)pyrazoles of formula (I) (see formula I) wherein: X is a halogen, nitro or unsubstituted or halo-substituted alkylsulfenyl, alkylsulfinyl or alkylsulfonyl, wherein the alkyl moiety is a linear or branched chain, containing one to four carbon atoms, and where substituted, is substituted by one of more halogen atoms, which are the same or different, up to full substitution of the alkyl moiety; Y is hydrogen, halogen, cyano, alkylsulfenyl, alkylsulfinyl, alkylsulfonyl, alkoxy, amino, alkylamino, dialkylamino, trialkylammanium salt, cyanoalkylamino, alkoxyalkylamino, alkoxycarbonylamino, alkylcarbonylamino, haloalkylcarbonylamino, alkylaminocarbonylamino, dialkylaminocarbonylamino or alkoxyalkylideneimino, wherein the alkyl and alkoxy moieties are linear or branched and contain one to four carbon atoms, and the haloalkyl moieties are substituted by one or more halogen atoms, which are the same or different, up to full substitution of the alkyl moiety; Z is cyano or halogen ...

ACYL UREAS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES

Pesticidal 1-arylimidazoles

PESTICIDAL 1-(4-PHENOXYPHENYL)-3-BENZOYL UREA COMPOUNDS AND PROCESS FOR PREPARATION

Pesticidal 5-substituted-oxyalkylamino-1-arylpyrazole derivatives

1-phenyl and 1-pyridylpyrazole derivatives and their use as pesticides

5-substituted-alkylaminopyrazole derivatives as pesticides

1- ALKYL-PHENOXYARYL -3-BENZOYL UREAS

Control of arthropods in animals

A method of controlling parasites in or on an animal comprising administering to the animal a parasiticidally effective, substantially non-emetic 1-arylpyrazole.

PESTICIDAL BIPHENYLYLOXY AND BIPHENYLYLALKOXY ARYL ACYL UREA DERIVATIVES

Pesticidal sulphonylaminopyrazoles

N-BENZOYL-N:-PYRIDYLOXY THIO PHENYL UREAS

Control of arthropods in animals

A method of controlling parasites in or on an animal comprising orally administering to the animal a parasiticidally effective, substantially non-emetic 1-arylpyrazole.

Pesticides

5-substituted-alkylaminopyrazole derivatives as pesticides

The invention relates to the use for the control of pests, of a compound which is a 5 ­substituted-alkylaminopyrazole derivative of formula (I) or a salt thereof: wherein the various symbols are as defined in the description, to novel 5-substituted-­alkylaminopyrazole derivatives and pesticidal compositions thereof, and to processes for their preparation.

5-SUBSTITUTED-ALKYLAMINOPYRAZOLE DERIVATIVES AS PESTICIDES

Control of arthropods in animals

PESTICIDAL BENZOYL UREAS AND PROCESS FOR THEIR PREPARATION

PESTICIDAL COMPOSITIONS

5-substituted-alkylaminopyrazole derivatives as pesticides

PESTICIDAL 1-(4-PHENOXYPHENYL)-3-BENZOYL UREA COMPOUNDS AND PROCESS FOR PREPARATION

N-BENZOYL-N:-PYRIDYLOXY THIO PHENYL UREAS

PESTICIDAL BIPHENYLYLOXY AND BIPHENYLYLALKOXY ARYL ACYL UREA DERIVATIVES

5-substituted-alkylaminopyrazole derivatives as pesticides

The invention relates to the use for the control of pests, of a compound which is a 5 ­substituted-alkylaminopyrazole derivative of formula (I) or a salt thereof: wherein the various symbols are as defined in the description, to novel 5-substituted-­alkylaminopyrazole derivatives and pesticidal compositions thereof, and to processes for their preparation.

Pestizide 1-(2-Pyridyl)pyrazole

PESTICIDAL 1-(4-PHENOXYPHENYL)-3-BENZOYL UREA COMPOUNDS AND PROCESS FOR PREPARATION

Pesticidal compositions

... 5-Substituted-sulfonylaminopyrazole derivatives of formula (I): or salts thereof, wherein the various symbols are as defined in the description, and pesticidal compositions thereof, processes for their preparation, and methods for their use for the control of arthropods (including insects and arachnids) and helminths (including nematodes).

1-phenyl and 1-pyridylpyrazole derivatives and their use as pesticides

The invention relates to 1-(2,4,6-trisubstituted-phenyl)-5-amino-4-substituted-pyrazole derivatives of formula (I) or salts thereof wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

1-PHENYL- UND 1-PYRIDYLPYRAZOLDERIVATE UND DEREN VERWENDUNG ALS PESTIZIDE

PESTICIDAL PHENOXYPHENYL AND PHENOXYPYRIDYL BENZOYL UREAS AND PROCESS FOR THEIR PREPARATION

1-PHENYL AND 1-PYRIDYLPYRAZOLE DERIVATIVES AND THEIR USE AS PESTICIDES

5-AMINOALKYLPYRAZOLDERIVATE ALS PESTIZIDE MITTEL

PESTICIDAL 1-(ALKYL-PHENOXYARYL)-3-BENZOYL UREAS AND PROCESS FOR PREPARATION

1-ARYLPYRAZOLDERIVATE ALS PESTIZIDMITTEL

Vinylaminopyrazole derivatives as pesticides

Disclosed are 5-(vinylamino)pyryazole derivatives of formula I or pesticidally acceptable salts thereof (I) wherein, for example, W is N, CH, CR6 or C(NH2)-, R6 is halogen or haloalkyl, R1 is cyano, halogen, alkyl, haloalkyl or CSNH2, R2 is alkyl or cycloalkyl, R3 is alkyl, alkenyl, alkynyl, cycloalkyl, aryl, heterocyclyl, aralkyl, heterocyclylalkyl, COOR9, COR10, SOR, SO2R12; R9, R10, R11 and R12 are for example organic groups, R4 is halogen or NH2, R5 is haloalkyl, haloalkoxy, halogen or SF5, and n is an integer selected from 0, 1 or 2. These compounds cab be used for controlling pests, especially by treatment of domestic animals.

PESTIZIDE

5-SUBSTITUTED-ALKYLAMINOPYRAZOLE DERIVATIVES AS PESTICIDES

5-substituted-alkylaminopyrazole derivatives as pesticides

The invention relates to the use for the control of pests, of a compound which is a 5-substituted-alkylaminopyrazole derivative of formula (I) or a salt thereof: wherein the various symbols are as defined in the description, to novel 5-substituted-alkylaminopyrazole derivatives and pesticidal compositions thereof, and to processes for their preparation.

Pestizide 1-(2-Pyridyl)pyrazole

Pesticidal agents

PESTICIDAL 1-ARYLIMIDAZOLES

PURPOSE: To provide a novel compd. that has high activity and is safe to the human body or environment as an insecticidal and acaricidal agent. CONSTITUTION: The compd. of formula I [X is (O)nR1 (R1 is a 1 to 4C alkyl, (n) is 0, 1, 2; Y is H, a halogen alkyl, etc.; Z is H, a 1 to 4C alkyl, R2 is a halogen, etc.; R3, R5 are each H; R6 is a halogen; R4 is H, a halogen, etc.]; for example, 1-(2,6-dichloro-4-fluoropheny)5-methylsulphenyl-4- chlorodifluoromethylsulphenylimdazole. The compd. is obtd. from the compd. obtd. by bringing the compd. of formula II into reaction with halogenated sulphenyl R1SHalo in an org. reaction medium, in the presence of an acid receptor, such as ternary amine at need and then bringing the same into reaction with chlorosulfonic acid, etc. COPYRIGHT: (C)1992,JPO ...

5-aminoalkylpyrazole derivatives as pesticidal agents

The invention relates to 5-aminoalkylaminopyrazole derivatives of formula (I) or salts thereof: wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

5-substituted-alkylaminopyrazole derivatives as pesticides

The invention relates to the use for the control of parasites in animals, of a compound which is a 5-substituted-alkylaminopyrazole derivative of formula (I) or a salt thereof, wherein the various symbols are as defined in the description, to novel 5-substituted-alkylaminopyrazole derivatives and pesticidal compositions thereof, and to processes for their preparation.

Chemical compounds, process for their preparation and use thereof

Pesticidal compounds

Control of arthropods in animals

A method of controlling parasites in or on an animal comprising administering to the animal a parasiticidally effective, substantially non-emetic 1-arylpyrazole.

Control of arthropods in animals

A method of controlling parasites in or on an animal comprising orally administering to the animal a parasiticidally effective, substantially non-emetic 1-arylpyrazole.

5-substituted-alkylaminopyrazole derivatives as pesticides

The invention relates to the use for the control of parasites in animals, of a compound which is a 5-substituted-alkylaminopyrazole derivative of formula (I) or a salt thereof: wherein the various symbols are as defined in the description, to novel 5-substituted-alkylaminopyrazole derivatives and pesticidal compositions thereof, and to processes for their preparation.

1-Phenyl and 1-Pyridylpyrazole Derivatives and Their Use as Pesticides

The invention relates to 1-(2,4,6-trisubstituted-phenyl)-5-amino-4-substituted-pyrazole derivatives of formula (I) or salts thereof wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

Pesticidal compounds

The invention relates to 5-(substituted dithio- or dioxy-alkylamino)pyrazole derivatives of formula (I) or salts thereof: , wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

Pesticidal agents

The invention relates to 5-(oximinoalkyl- and hydrazonoalkyl-amino)pyrazole derivatives of formula (I) or salts thereof: wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

5-substituted-alkylaminopyrazole derivatives as pesticides

Control of arthropods in animals

A method of controlling parasites in or on an animal comprising orally administering to the animal a parasiticidally effective, substantially non-emetic 1-arylpyrazole.

Pesticidal 5-substituted-oxyalkylamino-1-arylpyrazole derivatives

The invention relates to 5-sub-stituted-oxyalkylaminopyrazole derivatives of the formula or salts thereof wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests including arthropods and helminths.

Control of arthropods in animals

A method of controlling parasites in or on an animal comprising administering to the animal a parasiticidally effective, substantially non-emetic 1-arylpyrazole.

COMPOUND 1- (2-PYRIDIL) PINE PLANTS, PROCESS FOR YOUR PREPARATIONS, PESTICID COMPOSITIONS AND METHOD TO CONTROL ARTROPODES, NEMATODES, HELMINTAS OR PROTOZOARIOS

Control of arthropods in animals with 1-arylpyrazoles

A method of controlling parasites in or on an animal comprising administerin g to the animal a parasiticidally effecive, substantially non-emetic 1-arylpyrazole.

Control of arthropods in animals with 1-arylpyrazoles

A method of controlling parasites in or on an animal comprising administering to the animal a parasiticidally effecive, substantially non-emetic 1-arylpyrazole.

Pesticidal 1-(alkyl-phenoxyaryl)-3-benzoyl ureas and process for preparation

1-(alkylphenoxyphenyl)-3-benzoyl ureas and a process for their preparation are provided. The ureas are useful as the active toxicant in pesticidal composition. The ureas have the general formula: wherein X, X' are independently hydrogen, halogen, C 1 -C 4 alkyl, haloalkyl, polyhaloalkyl, alkoxy, polyhaloalkoxy Y represents oxygen or sulfur; m, n are independently 0-4; R, represents hydrogen, halogen, C 1 -C 4 alkyl, haloalkyl, polyhaloalkyl, or alkoxy, R 2 represents hydrogen, halogen, C 1 -C 4 alkyl, polyhaloalkyl, polyhaloalkoxy, C 1 -C 8 alkylsulfonyl, C 1 -C 8 alkoxy, C 1 -C 8 alkylthio, C 1 -C 8 dialkylamino, CN, NO 2 , C0 2 R 4 , or CONHR 4 wherein R 4 represents C 1 -C 8 alkyl; and R 3 represents C 1 -C 12 alkyl, with the proviso that m may not be 0 or 1 when n is less than 2.

5-SUBSTITUTED ALKYLAMINOPYRAZOL DERIVATIVES AS PESTICIDES

5-Substituted-alkylaminopyrazole derivatives as pesticides

Disclosed is a method for controlling parasites in or on a non-human animal comprising administering to the non-human animal a parasiticidally effective amount of a 5-substiuted-alkylaminopyrazole derivative of formula (I), wherein: R1 is CN, W is C-halogen, C-CH3 or N, R2 is H, halogen or CH3, R3 is haloalkyl, haloalkoxy or S(O)p-haloalkyl, R4 is H, alkenyl, halo-alkenyl, alkynyl, halo-alknynl, cycloalkyl, CO-(CH2)q-R7, COR8, CO-(CH2)q-R9, -CO-haloalkynyl, cycloalkyl, CO-(CH2)q-R7, COR8, CO-(CH2)q-R9, -CO-alkyl-alkoxy, -CO2-(CH2)q-R7, CO2R8, -CO2-(CH2)q-R9, -CO2-cycloalkyl, -CO2-alkyl-cycloalkyl, -CO2-alkyl-cycloalkyl, -CO2-alkenyl, -CO2-alknyl, CONR10R11, -CH2R7, -CH2R9, OR7, OR8 or OR9, or optionally substituted alkyl, and the remaining substituents are defined herein.

PESTICIDE 1- (2-PYRIDYL) PYRAZOLER.

PESTICIDE 1- (ALKYLPHENOXYARYL) -3-BENZOYLURIN INGREDIENTS

Pesticidal 1-(2-pyridyl)pyrazoles

Pesticidal sulphonylaminopyrazoles

5-Substituted-sulfonylaminopyrazole derivatives of formula (I) or salts thereof: wherein the various symbols are as defined in the description, processes for their preparation, compositions thereof, and their use for the control of pests, such as arthropods (insects and arachnids) and helminths (nematodes).

Pesticidal biphenylyloxy and biphenylylalkoxy aryl acyl urea compounds, a process for their preparation, pesticidal compositions and a method of controlling pests

Systemically controlling parasites of warm-blooded non-human animals with urea derivatives

Arylimidazole Compounds, Their Use, and Preparations Containing Such

Insecticide compositions containing aryl-imidazol derivatives as active components and process for producing the active components

Control of parasites in animals, the novel active ingredients applied and compositions containing the same

A találmány szerinti eljárás paraziták irtására szolgál állatban vagyállaton, amelynek megfelelően az állatnak egy (I) általános képletű 1-aril-pirazol vegyületnek vagy sójának parazitaellenes szempontbólhatékony, lényegében nern hánytató mennyiségét tartalmazó készítménytadagolják - a képletben R201 jelentése ciano-, -C(O)alkil, -C(S)NH2, -C NH)OR203, -C(NH)SR203, -C(=NOH)NH2, -C(=NNH2)NH2, -C(O)NH2, -C(O)NHR205 -C(O)NR205R206 alkil-, halogén-alkil- vagy adott esetbenszubsztituált 1,2,4-oxadiazol-3-il-; 1,3-oxazolidin-2-il-, 1,3-oxazol-2-il- vagy 1,3,4.-oxazin-2-il-csoport; R202 jelentése -S(O)hR2O3általános képletű csoport, alkenil-, halogén-alkenil-, cikloalkil-,halogén-cikloalkil-, cikloalkil-alkil-, alkinil-, nitrocsoport vagyadott esetben szubsztituált imidazol-2-il-csoport; R203 jelentésealkil- vagy halogén-alkil-csoport; R204 jelentése R205O-, HC(O)O-,R205C(O)O-, R205OC(O)O-, NH2C(O)O-, R205NHC(O)O-, R205R206NC(O)O-R205S(O)nC(O)O- R206SO2O-, R205R206N-C(NR205)-O- R205R206N-C(NH)-O-,R205NH-C(N205)-O- R205N=CH-O- R205N=C(R206)-O-, R205NH-C(S)-O- vagyR205R206N-C(S)-O- általános képletű csoport, vagy hidroxil-,oxacikloalkil-oxi- vagy aril-szulfonil-oxi-csoport; R205 jelentésealkenil-, alkinil-, adamantilcsoport, adott esetben szubsztituáltalkil-, cikloalkil-, aril- vagy heteroarilcsoport. R206 jelentéseadott esetben szubsztituált alkil-, cikloalkil-, aril- vagyheteroaril-csoport vagy R205 és R206 együtt a nitrogénatommal, melyhezkapcsolódnak, 3-7-tagú gyűrűt alkothat, amely adott esetben továbbiheteroatomként még egy vagy több nitrogén-, oxigénvagy kénatomottartalmaz; X1 jelentése nitrogénatom vagy -CR212 általános képletűcsoport; R211 és R212 jelentése egymástól függetlenül hidrogén-,halogénatom, ciano-, alkil- vagy nitrocsoport; R213 jelentésehalogénatom, halogén-alkil-, halogén-alkoxi-, -S(O)kCF3 vagy SF5képletű csoport, vagy R214-gyel gyűrűt alkot; R214 jelentésehidrogénatom, vagy R213-mal együtt -OCF2O-, -CF2OCF2-, -CF2OCF2O- vagy-CF2CF2O- képletű csoport, ...

Pesticidal n-phenylpyrazole derivatives

The invention relates to 5-(substituted dithio- or dioxy-alkylamino)pyrazole derivatives of formula (I) or salts thereof: wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

1-arylpyrazole derivatives as pesticidal agents

The invention relates to 5-(oximinoalkyl- and hydrazonalkyl-amino)pyrazole derivatives of formula (I) or salts thereof: formula (I), wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

Pesticide

Novel 1-(2-pyridyl)pyrazoles of formula (I) <CHEM> wherein: X is a halogen, nitro or unsubstituted or halo-substituted alkylsulfenyl, alkylsulfinyl or alkylsulfonyl, wherein the alkyl moiety is a linear or branched chain, containing one to four carbon atoms, and where substituted, is substituted by one of more halogen atoms, which are the same or different, up to full substitution of the alkyl moiety; Y is hydrogen, halogen, cyano, alkylsulfenyl, alkylsulfinyl, alkylsulfonyl, alkoxy, amino, alkylamino, dialkylamino, trialkylammonium salt, cyanoalkylamino, alkoxyalkylamino, alkoxycarbonylamino, alkylcarbonylamino, haloalkylcarbonylamino, alkylaminocarbonylamino, dialkylaminocarbonylamino or alkoxyalkylideneimino, wherein the alkyl and alkoxy moieties are linear or branched and contain one to four carbon atoms, and the haloalkyl moieties are substituted by one or more halogen atoms, which are the same or different, up to full substitution of the alkyl moiety; Z is cyano or halogen; and R2, R3, R4 and R5 are each individually hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, cyano or nitro, wherein the alkyl and alkoxy moieties are linear or branched and contain one to four carbon atoms, and the halo-substituted moieties are substituted by one or more halogen atoms, which are the same or different, up to full substitution of the alkyl and alkoxy moieties; at least one of R2 to R5 being other then hydrogen. The invention further relates to intermediates and processes to make the compounds, pesticidal compositions comprising the compounds, and methods of use of the compounds for the control of arthropods (mites, aphids or insects) nematodes, helminths or protozoa.

Control of arthropods in animals

Pesticidal 1-(2-pyridyl)pyrazoles

Novel 1-(2-pyridyl)pyrazoles of formula (I) (see formula I) wherein: X is a halogen, nitro or unsubstituted or halo-substituted alkylsulfenyl, alkylsulfinyl or alkylsulfonyl, wherein the alkyl moiety is a linear or branched chain, containing one to four carbon atoms, and where substituted, is substituted by one of more halogen atoms, which are the same or different, up to full substitution of the alkyl moiety; Y is hydrogen, halogen, cyano, alkylsulfenyl, alkylsulfinyl, alkylsulfonyl, alkoxy, amino, alkylamino, dialkylamino, trialkylammanium salt, cyanoalkylamino, alkoxyalkylamino, alkoxycarbonylamino, alkylcarbonylamino, haloalkylcarbonylamino, alkylaminocarbonylamino, dialkylaminocarbonylamino or alkoxyalkylideneimino, wherein the alkyl and alkoxy moieties are linear or branched and contain one to four carbon atoms, and the haloalkyl moieties are substituted by one or more halogen atoms, which are the same or different, up to full substitution of the alkyl moiety; Z is cyano or halogen; and R2, R3, R4 and R5 are each individually hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, cyano or vitro, wherein the alkyl and alkoxy moieties are linear or branched and contain one to four carbon atoms, and the halo-substituted moieties are substituted by one or more halogen atoms, which are the same or different, up to full substitution of the alkyl and alkoxy moieties; at least one of R2 to R5 being other then hydrogen. The invention further relates to intermediates and processes to make the compounds, pesticidal compositions comprising the compounds, and methods of use of the compounds for the control of arthropods (mites, aphids or insects) nematodes, helminths or protozoa.

Pesticidal phenoxyphenyl and phenoxypyridyl benzoyl ureas and process for their preparation

Phenoxyphenyl and phenoxypyridyl benzoyl ureas and a process for their preparation are provided. The ureas are useful as the active toxicant in pesticidal compositions and have the general formula: <CHEM> wherein: X is oxygen or sulfur; Y is CR3 or nitrogen; B is oxygen, sulfur, sulfinyl, sulfonyl, oxysulfonyl, sulfonyloxy or carbonyl; R1 and R2 are independently hydrogen, halogen, methoxy, alkyl (C1 - C4) or trifluoromethyl; R3, R4, R5 are independently hydrogen, methoxy, halogen, alkyl (C1-C4) or trifluoromethyl; R6 is hydrogen, halogen or alkyl (C1-C4) or trifluoromethyl; R7, R8 are independently hydrogen, halogen, alkyl (C1-C4), trifluoromethyl, alkylthio (C1-C4), alkylsulfinyl (C1-C4), alkylsulfonyl (C1-C4), or R7 and R8 can optionally be a substituted arylthio, a substituted arylsulfonyl, or a substituted arylsulfinyl, group, wherein said optional substituents are alkyl (C1-C4) or halogen and provided that when B is oxygen, and Y is CR3, at least two of R3-R5 are other than hydrogen.

Vinylminopyrazole derivatives as pesticides

Un compuesto que es un derivado de 5-(vinilamino)pirazol de fórmula I o una sal del mismo aceptable desde el punto de vista de pesticida **Fórmula** en el que W es >=N-, >=CH-, >=CR6- o >=C(NR7R8)-; R6 es halógeno o haloalquilo, R7 y R8 son independientemente entre sí hidrógeno, alquilo, cicloalquilo, arilo, heterociclilo, aralquilo o heterociclilalquilo, o uno de R7 o R8 es -CO-R7a, -CO-O-R8a, -SO-R7a o -SO2R7a, o R7 y R8 junto con el átomo N fijado forman un anillo heterocíclico de cinco a siete eslabones que contiene opcionalmente un átomo adicional de oxígeno, azufre o nitrógeno en el anillo o R7 y R8 junto con el átomo N fijado forman un grupo imina -N>=CR7bR8b o un grupo iminoéter -N>=CR7b(OR8b), R7a y R8a son alquilo, cicloalquilo, arilo, heterociclilo, aralquilo o heterociclilalquilo, R7b es hidrógeno, alquilo, cicloalquilo, arilo, heterociclilo, aralquilo o heterociclilalquilo, R8b es alquilo, cicloalquilo, arilo, heterociclilo, aralquilo o heterociclilalquilo, en los que los grupos R7, R8, R7a, R8a, R7b y R8b independientemente entre sí están sustituidos opcionalmente por uno o más átomos de halógeno, grupos hidroxilo, oxo, ciano, nitro, alquilo, alcoxi, alquiltio, cicloalquilo, arilo, heterociclilo, aralquilo o heterociclilalquilo o por amino, que está sustituido opcionalmente por grupos alquilo, alquenilo, alquinilo, arilo o heteroarilo; R1 es ciano; R2 es alquilo o cicloalquilo, en el que el grupo R2 está sustituido opcionalmente por uno o más átomos de halógeno, grupos hidroxilo, oxo, alquilo, alcoxi, alquiltio, cicloalquilo, arilo, heterociclilo, aralquilo o heterociclilalquilo; R3 es alquilo, alquenilo, alquinilo, cicloalquilo, arilo, heterociclilo, aralquilo, heterociclilalquilo, -CO-O-R9, -CO-R10, - SOR11, -SO2-R12; R9, R10, R11 y R12 son alquilo, haloalquilo, alquenilo, alquinilo, cicloalquilo, arilo, heterociclilo, aralquilo o heterociclilalquilo, en los que los grupos R3, R9, R10, R11 y R12 están sustituidos opcionalmente por ...

5-aminoalkylpyrazole derivatives as pesticidal agents

The invention relates to 5-aminoalkylaminopyrazole derivatives of formula (I) or salts thereof: wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

Arthropod control in animals

El uso de un compuesto de fórmula (II) o una sal del mismo para la fabricación de una composición veterinaria para administración oral o parenteral para el control de parásitos en o dentro de un animal. en la que: R21 es ciano, C(>=S)NH2, C(>=NOH)NH2 o C(>=NNH2)NH2; R22 es S(O)mR23; R23 es alquilo o haloalquilo; R24 es OH, HC(O)O-, R25C(O)O-, R25OC(O)O- o R25S(O)nC(O)OR25 es alquilo, haloalquilo, cicloalquilo, halocicloalquilo, alcoxialquilo, haloalcoxialquilo, adamantilo, aminoalquilo, alquilaminoalquilo, dialquilaminoalquilo, haloalquilaminoalquilo, di(haloalquil)aminoalquilo, arilo opcionalmente sustituido, hetarilo opcionalmente sustituido, arilalquilo opcionalmente sustituido, hetarilalquilo opcionalmente sustituido, alquenilo C2-C6, alquinilo C2-C6, o dos grupos R25 pueden formar junto con el átomo de nitrógeno al que están unidos un anillo de 3 a 7 miembros que puede contener adicionalmente uno o más heteroátomos seleccionados de nitrógeno, oxígeno y azufre; X se ha seleccionado de nitrógeno y C-R32; R31 y R32 se han seleccionado independientemente de halógeno, hidrógeno, CN, C1-C3 alquil y NO2; R33 se ha seleccionado de halógeno, haloalquilo, haloalcoxi, -S(O)rCF3, y -SF5 o forma un anillo junto con R34 ; R34 es hidrógeno o puede constituir junto con R33 un grupo de OCF2O, CF2OCF2, CF2OCF2O y CF2CF2O, que junto a los átomos de carbono a los que están unidos forman un anillo de cinco a seis miembros; m es 0, 1 o 2; r se ha seleccionado de 0, 1, y 2; y sales veterinariamente aceptables de los mismos. The use of a compound of formula (II) or a salt thereof for the manufacture of a veterinary composition for oral or parenteral administration for the control of parasites in or within an animal. wherein: R21 is cyano, C (> = S) NH2, C (> = NOH) NH2 or C (> = NNH2) NH2; R22 is S (O) mR23; R23 is alkyl or haloalkyl; R24 is OH, HC (O) O-, R25C (O) O-, R25OC (O) O- or R25S (O) nC (O) OR25 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkoxyalkyl, ...

Pesticidal 5-substituted-oxyalkylamino-1-arylpyrazole derivatives

The invention relates to 5-substituted-oxyalkylaminopyrazole derivatives of formula (I) or salts thereof wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

1-(substituted)phenylimidazoles process for their preparation and compositions containing them for the control of arthropodes nematodes helminths or protozoa

The invention describes novel 1-arylimidazoles of formula (I), <CHEM> wherein typically preferred substituents are: X is S(O)nR1, in which R1 is unsubstituted or halo-substituted alkyl and n is 0, 1 or 2; Y is hydrogen, halogen, alkyl, alkoxy, alkoxyalkylideneimino, alkylsulfenyl, alkylsulfinyl or alkylsulfonyl; Z is hydrogen or alkyl; R2 is halogen or alkylsulfenyl; R3 and R5 are hydrogen; R6 is halogen; and R4 is hydrogen, halogen, haloalkyl or haloalkoxy. The invention further describes processes to make the compounds, compositions of the compounds, and methods of use of the compounds for the control of arthropods (especially mites, aphids or insects), nematodes, helminths, or protozoa.

Pesticidal 1-arylimidazoles

The invention describes novel 1-arylimidazoles of formula (I), wherein typically preferred substituents are: X is S(O)n R1, in which R1 is unsubstituted or halo-substituted alkyl and n is 0, 1 or 2; Y is hydrogen, halogen, alkyl, alkoxy, alkoxyalkylideneimino, alkylsulfenyl, alkylsulfinyl or alkylsulfonyl; Z is hydrogen or alkyl; R2 is halogen or alkylsulfenyl; R3 and R5 are hydrogen; R6 is halogen; and R4 is hydrogen, halogen, haloalkyl or haloalkoxy. The invention further describes processes to make the compounds, compositions of the compounds, and methods of use of the compounds for the control of arthropods (especially mites, aphids or insects), nematodes, helminths, or protozoa.

1-phenylimidazole compound, processes of its preparation, composition in which the compound is comprised, method of controlling articulates and use of the compound for preparing preparation used in veterinary medicine

1-Arylimidazoly obecného vzorce I, ve kterém X zejména znamená S/O/.sub.n.n.R.sub.1.n., kde R.sub.1 .n.znamená nesubstituovanou nebo halogen-substituovanou alkylovou skupinu a n je rovno 0,1 nebo 2, Y, zejména znamená atom vodíku, atom halogenu, alkylovou skupinu, alkoxylovou skupinu, alkoxyalkylideniminovou skupinu, alkylsulfenylovou skupinu, alkylsulfinylovou skupinu nebo alkylsulfonylovou skupinu, Z znamená atom vodíku nebo alkylovou skupinu, R.sub.2 .sub..n.znamená atom halogenu nebo alkylsulfenylovou skupinu, R.sub.3 .n.a R.sub.5 .n.znamenají atom vodíku, R.sub.6 .sub..n.znamená atom halogenu a R.sub.4 .n.zejména znamená atom vodíku, atom halogenu, halogenalkylovou skupinu nebo halogenalkoxylovou skupinu. Dále se popisuje způsob přípravy těchto sloučenin, kompozice obsahující tyto sloučeniny a způsoby použití těchto sloučenin pro kontrolu členovců, zejména roztočů, mšic nebo hmyzu, dále hlístic, cizopasných červů a protozoí.ŕ 1-Arylimidazoles of the general formula I, wherein X in particular represents S (O) .sub.nnR.sub.1, wherein R.sub.1 is unsubstituted or halo-substituted alkyl and is equal to 0.1 or 2, Y, in particular a hydrogen atom, a halogen atom, an alkyl group, an alkoxy group, an alkoxyalkylidenimino group, an alkylsulfenyl group, an alkylsulfinyl group, or an alkylsulfonyl group, Z represents a hydrogen atom or an alkyl group, R.sub.2. is a halogen atom or an alkylsulfenyl group, R.sub.3 is hydrogen, R.sub.6 is halogen, and R.sub.4 is, in particular, is hydrogen, halogen, haloalkyl or haloalkoxy. Further disclosed is a process for the preparation of these compounds, compositions comprising these compounds, and methods of using the compounds for the control of arthropods, especially mites, aphids or insects, nematodes, parasitic worms, and protozoa.

Vinylaminopyrazole derivatives as pesticides

Disclosed are 5-(vinylamino)pyryazole derivatives of formula I or pesticidcally acceptable salts thereof (I) wherein, for example, W is =N-, =CH-, =CR6- or =C(NH2)-, R6 is halogen or haloalkyl, R1 is cyano, halogen, alkyl, haloalkyl or -CS-N H2, R2 is alkyl or cycloalkyl, R3 is alkyl, alkenyl, alkynyl, cycloalkyl, aryl, heterocyclyl, aralkyl, heterocyclylalkyl, -CO-O-R9, -CO-R10, -SO-R", -S02-R12; R9, R10,R11 and R12 are for example organic groups, R4 is halogen or -NH2, R5 is haloalkyl, haloalkoxy, halogen or -SF5, and n is an integer selected from 0, 1 or 2. These compounds cab be used for controlling pests, especially by treatment of domestic animals.

5-aminoalkylpyrazole derivatives as pesticidal agents

The invention relates to 5-aminoalkylaminopyrazole derivatives of formula (I) or salts thereof: wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

Pesticidal 5-substituted-oxyalkylamino-1-arylpyrazole derivatives

The invention relates to 5-substituted-oxyalkylaminopyrazole derivatives of formula (I) or salts thereof wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

1-phenyl and 1-pyridylpyrazole derivatives and their use as pesticides

Vinylaminopyrazole derivatives as pesticides

Disclosed are 5-(vinylamino)pyryazole derivatives of formula I or pesticidcally acceptable salts thereof (I) wherein, for example, W is =N-, =CH-, =CR6- or =C(NH2)-, R6 is halogen or haloalkyl, R1 is cyano, halogen, alkyl, haloalkyl or -CS-N H2, R2 is alkyl or cycloalkyl, R3 is alkyl, alkenyl, alkynyl, cycloalkyl, aryl, heterocyclyl, aralkyl, heterocyclylalkyl, -CO-O-R9, -CO-R10, -SO-R", -S02-R12; R9, R10,R11 and R12 are for example organic groups, R4 is halogen or -NH2, R5 is haloalkyl, haloalkoxy, halogen or -SF5, and n is an integer selected from 0, 1 or 2. These compounds cab be used for controlling pests, especially by treatment of domestic animals.

5-substituted-alkylaminopyrazole derivatives as pesticides

5-substituted-alkylaminopyrazole derivatives as pesticides

The invention relates to the use for the control of parasites in animals, of a compound which is a 5-substituted-alkylaminopyrazole derivative of formula (I) or a salt thereof:, wherein the various symbols are as defined in the description, to novel 5-substituted-alkylaminopyrazole derivatives and pesticidal compositions thereof, and to processes for their preparation.

Pesticidal agents on the basis of 1-aryl-aminopyrrol

Pesticidal Compounds The invention relates to 1-aryl-5-disubstituted-aminopyrrole derivatives of formula (I) or salts thereof: wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

Pestizide 1-(2-pyridyl)pyrazole

Pesticidal agents on the basis of 1-aryl-aminopyrrol

Pesticidal Compounds The invention relates to 1-aryl-5-disubstituted-aminopyrrole derivatives of formula (I) or salts thereof: wherein the various symbols are as defined in the description, to processes for their preparation, to compositions thereof, and to their use for the control of pests (including arthropods and helminths).

Pesticide 1-(4-fenyloksyfenyl)-3-benzoyl urinstofforbindelser og en fremgangsmaate for deres fremstilling.

5-substituierte alkylaminopyrazol-derivative als pestizide

5-substituierte alkylaminopyrazol-derivate als pestizide

5-υποκατεστημενα -αλκυλαμινοπυραζολικα παραγωγα ως παρασιτοκτονα

Η εφεύρεση σχετίζεται με τη χρήση για τον έλεγχο παρασίτων, μιας ένωσης η οποία είναι ένα 5 υποκατεστημένο-αλκυλαμινοπυραζολικό παράγωγο του τύπου (I) ή ενός άλατος αυτού: όπου τα διάφορα σύμβολα είναι όπως ορίζονται στην περιγραφή, με νέα 5-υποκατεστημένα-αλκυλαμινοπυραζολικά παράγωγα και παρασιτοκτόνες συνθέσεις αυτών, και με διαδικασίες για την παρασκευή τους.

Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals

Pesticide 1-(4-phenoxyphenyl)-3-benzoylurinstofforbindelser samt fremgangsmaade til fremstilling deraf

Pesticide 1-(4-phenoxyphenyl)-3-benzoylurinstofforbindelser samt fremgangsmaade til fremstilling deraf

Pesticide 1-(4-fenyloksyfenyl)-3-benzoyl urinstofforbindelser og en fremgangsmaate for deres fremstilling.

Chemical compounds, process for their preparation and use thereof

CHEMICAL COMPOUNDS, PROCESS FOR THEIR PREPARATION AND USE THEREOF 5 DISCLOSED ARE 5-(VINYLAMINO)PYRYAZOLE DERIVATIVES OF FORMULA I OR PESTICIDCALLY ACCEPTABLE SALTS THEREOF R2 O N S R H @N H 4 N N\ 3 H R "I@Z W R R I 0 WHEREIN, FOR EXAMPLE, W IS =N-, =CH-, =CR 6_ OR =C(NH2)-, R6 IS HALOGEN OR HALOALKYL, R' IS CYANO, HALOGEN, ALKYL, HALOALKYL OR -CS-NH2, R2IS ALKYL OR CYCLOALKYL, R3IS ALKYL, ALKENYL, ALKYNYL, CYCLOALKYL, ARYL, HETEROCYCLYL, ARALKYL, HETEROCYCLYLALKYL, -CO-0-R9, -CO-R'O, -SO-R", -SO2-R 12 ; R9, R10, R" AND R1 2ARE FOR 1 5 EXAMPLE ORGANIC GROUPS, R 4IS HALOGEN OR -NH2, R5 IS HALOALKYL, HALOALKOXY, HALOGEN OR -SF5, AND N IS AN INTEGER SELECTED FROM 0, 1 OR 2. THESE COMPOUNDS CAN BE USED FOR CONTROLLING PESTS, ESPECIALLY BY TREATMENT OF DOMESTIC ANIMALS. 20 CN

Pestizide 1-arylimidazole