23-01-2003 дата публикации
Номер: WO2003006424A1
The present invention relates to compounds of the general formula (I), wherein A is a non-aromatic ring system containing 4 to 8 carbon atoms, wherein the ring system comprises at least one double bond and wherein one or more of the carbon atoms in the ring can be substituted by a group X, wherein X is selected from the group consisting of S, O, N, NH, NHR4, SO or SO¿2?, and wherein one or more of the carbon atoms of the ring can carry a substituent R?1¿; D is O, S, SO¿2?, NH, NHR?4¿, or CH¿2; R?1 is independently H, halogen, CF¿3?, OCF3, or C1-C5-alkyl; R?2¿ is H, OH, OR6, NH2, NHR7; R6 is H, alkyl, cycloalkyl, aryl, arylalkyl, alkylaryl, alkoxyalkyl, acylmethyl, (acyloxy)alkyl, non-symmetrical(acyloxy)alkyldiester, dialkylphosphate; R7 is H, alkyl, aryl, O-alkyl, O-aryl, cycloalkyl or O-cycloalkyl; R8 is hydrogen or alkyl; R3 is H, cycloalkyl, aryl, O-alkyl, O-aryl or O-cycloalkyl; R4 is C1-C5-alkyl or an unsaturated or saturated carbocycle selected from the group consisting of cyclopentyl, cyclohexyl or aryl; Z?1 and Z2¿ are independent from each other O, S, NH or NR5; R5 is OH, O-alkyl, O-aryl, alkyl or aryl; Ar is a monocyclic or polycyclic substituted or unsubstituted ring system which may contain one or more groups X and which contains at least one aromatic ring; Y is hydrogen, halogen, CF¿3?, OCF3, substituted or unsubstituted alkyl; substituted or unsubstituted cycloalkyl, Ar, O-substituted or unsubstituted Ar, O-substituted or unsubstituted alkylaryl, O-substituted or unsubstituted arylalkyl or (Formula); m is 0 or 1; and q is 0 to 10; with the proviso that when ring A is an unsubstituted carbocyclus containing five carbon atoms and one double bond between the CZ?1 and CZ2-¿substituents with Z1 = Z2 = O and R2 = OH, the following compounds are excluded: q = 0; Y = hydrogen; Ar = phenylene or naphthylene, phenylene substituted with one or two chlorine atoms or with 2-methyl, 4-methyl, 4-methoxy, 4-ethoxy, 2, 6-diethyl, 2-chloro-4-methyl, 4-bromo, 4-cyano, 2 ...
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