Condensed bicycl [3.1.0] hex-4-en derivatives useful as anti bacterial agents
Номер патента: EP1608658A1
Опубликовано: 28-12-2005
Автор(ы): E. Aston Univ. Pharmacy LATTMANN, I. M. Fernandez
Принадлежит: Aston University
Опубликовано: 28-12-2005
Автор(ы): E. Aston Univ. Pharmacy LATTMANN, I. M. Fernandez
Принадлежит: Aston University
Реферат: According to a first aspect of the present invention there is provided a compound of formula (I): where, A is carbon, sulphur, oxygen or nitrogen B is carbon or nitrogen, X is oxygen or sulphur, Y is hydrogen, a halogen, a substituted or unsubstituted heterocyclic moiety, substituted or unsubstituted, linear or branched alkyl, alkyloxy, alkylcarbonyl, alkyloxycarbonyl, alkenyl, alkenyloxy, alkenylcarbonyl, alkenyloxycarbonyl, alkynyl, alkynyloxy, alkynylcarbonyl, alkynyloxycarbonyl, aryl, benzyl, arlyoxy, arylcarbonyl, aryloxycarbonyl and sulphur equivalents of said oxy, carbonyl and oxycarbonyl moieties Z is hydrogen, a halogen, a substituted or unsubstituted heterocyclic moiety, substituted or unsubstituted, linear or branched alkyl, alkylcarbonyl, alkyloxycarbonyl, alkenyl, alkenylcarbonyl, alkenyloxycarbonyl, alkynyl, alkynylcarbonyl, alkynyloxycarbonyl, aryl, benzyl, arylcarbonyl, aryloxycarbonyl, and sulphur equivalents of said carbonyl and oxycarbonyl moieties, excluding the compound where A and X are oxygen, B is nitrogen, Y is chlorine and Z is methyl. The invention also relates to the use of the compounds to prevent or ameliorate bacterial infections.
Condensed bicyclo`3.1.0!hex-4-en derivatives useful as antibacterial agents
Номер патента: WO2004074293A1. Автор: Eric Lattmann,Isidro Merino Fernandez. Владелец: Aston University. Дата публикации: 2004-09-02.