Настройки

Укажите год
-

Небесная энциклопедия

Космические корабли и станции, автоматические КА и методы их проектирования, бортовые комплексы управления, системы и средства жизнеобеспечения, особенности технологии производства ракетно-космических систем

Подробнее
-

Мониторинг СМИ

Мониторинг СМИ и социальных сетей. Сканирование интернета, новостных сайтов, специализированных контентных площадок на базе мессенджеров. Гибкие настройки фильтров и первоначальных источников.

Подробнее

Форма поиска

Поддерживает ввод нескольких поисковых фраз (по одной на строку). При поиске обеспечивает поддержку морфологии русского и английского языка
Ведите корректный номера.
Ведите корректный номера.
Ведите корректный номера.
Ведите корректный номера.
Укажите год
Укажите год

Применить Всего найдено 401. Отображено 138.
20-07-2017 дата публикации

N-(SUBSTITUTED)-5-FLUORO-4-IMINO-3-METHYL-2-OXO-3,4-DIHYDROPYRIMIDINE-1(2H)-CARBOXYLATE DERIVATIVES

Номер: US20170204069A1
Принадлежит: Adama Makhteshim Ltd.

This present disclosure is related to the field of N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-di-hydropyrimidine-1(2H)-carboxylates and their derivatives and to the use of these compounds as fungicides. Also provided are methods of controlling a fungal disease such as Septoria tritici , comprising administering an effective amount of the fungicide compound to at lease one surface associated with the plant, seed or soil.

Подробнее
12-10-2011 дата публикации

Use of 5-fluorocytosine as a fungicide

Номер: CN102215691A
Принадлежит:

The present disclosure is related to the field agrochemicals including 5-flurocytosine and its derivatives and their use as fungicides.

Подробнее
04-07-2012 дата публикации

5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives

Номер: CN102548979A
Принадлежит:

This present disclosure is related to the field of 5-fluoro-2-oxopyrimidine-1-(2H)-carboxylates and their derivatives and to the use of these compounds as fungicides.

Подробнее
24-08-2017 дата публикации

3-ALKYL-5-FLUORO-4-SUBSTITUTED-IMINO-3,4-DIHYDROPYRIMIDIN-2(1H)-ONE DERIVATIVES AS FUNGICIDES

Номер: US20170240540A1
Принадлежит: Adama Makhteshim Ltd.

This present disclosure is related to the field of 3-alkyl-5-fluoro-4-substituted-imino-3,4-5 dihydropyrimidin-2(1H)-ones and their derivatives and to the use of these compounds as fungicides. Also provided are methods of controlling a fungal disease such as , comprising administering an effective amount of the fungicide compound to at lease one surface associated with the plant, seed or soil. 2. A compound according to claim 1 , wherein Ris independently C-Calkyl claim 1 , C-Calkoxy claim 1 , alkylthio claim 1 , hydroxyl claim 1 , or deuterium.3. A compound according to claim 1 , wherein Ris C-Calkyl claim 1 , C-Chaloalkyl claim 1 , phenyl or benzyl wherein each of the phenyl or the benzyl may be optionally substituted with 1-3 R.4. A compound according to claim 1 , wherein Ris independently halogen claim 1 , C-Calkyl claim 1 , C-Chaloalkyl claim 1 , C-Calkoxy claim 1 , C-Calkylthio claim 1 , or deuterium.5. A compound according to claim 1 , wherein Ris C-Calkyl claim 1 , C-Chaloalkyl claim 1 , phenyl or benzyl wherein each of the phenyl or the benzyl may be optionally substituted with 1-3 R.6. A compound according to claim 1 , wherein Ris independently halogen claim 1 , C-Calkyl claim 1 , C-Chaloalkyl claim 1 , alkoxy claim 1 , C-Chaloalkoxy claim 1 , C-Calkylthio claim 1 , cyano claim 1 , or nitro.7. A compound according to claim 1 , wherein Ris phenyl optionally substituted with 1-3 R claim 1 , or a 5- or 6-membered saturated or unsaturated ring containing 1-3 heteroatoms optionally substituted with 1-3 R.8. A compound according to claim 7 , wherein Ris independently halogen claim 7 , C-Calkyl claim 7 , C-Calkoxy claim 7 , C-Chaloalkoxy.9. A compound according to claim 1 , wherein Ris C-Calkyl.10. A compound according to claim 1 , wherein Ris C-Calkyl claim 1 , —C(═O)R claim 1 , or —C(═O)OR.11. A compound according to claim 10 , wherein Ris C-Calkyl or phenyl.12. A compound according to claim 11 , wherein Ris C-Calkyl.14. A compound according to claim 13 , ...

Подробнее
29-06-2017 дата публикации

MACROCYCLIC PICOLINAMIDES COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20170183324A1
Принадлежит:

The invention relates to compounds of macrocyclic picolinamides of Formula I suitable to control or prevent growth of fungi. 2. The compound according to claim 1 , wherein X and Y are independently chosen from H claim 1 , C(O)R claim 1 , or CHOR.3. The compound according to claim 2 , wherein Ris chosen from H claim 2 , alkyl claim 2 , alkenyl claim 2 , phenyl claim 2 , —Si(R) claim 2 , or —C(O)R claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.4. The compound according to claim 3 , wherein Ris chosen from CHR claim 3 , phenyl claim 3 , alkyl claim 3 , or alkenyl claim 3 , each optionally substituted with 0 claim 3 , 1 claim 3 , or multiple R.5. The compound according to claim 4 , wherein Ris chosen from H claim 4 , alkyl claim 4 , alkenyl claim 4 , phenyl claim 4 , or heteroaryl claim 4 , each optionally substituted with 0 claim 4 , 1 claim 4 , or multiple R.6. A formulation for the control of a fungal pathogen claim 4 , comprising:{'claim-ref': {'@idref': 'CLM-00001', 'claim 1'}, 'at least one of the compounds of ; and'}a phytologically acceptable carrier material.7. The formulation according to claim 6 , wherein the formulation is suitable for treating plants.8. A formulation for the control of a fungal pathogen claim 6 , comprising:{'claim-ref': {'@idref': 'CLM-00001', 'claim 1'}, 'at least one of the compounds of ; and'}at least one agriculturally active ingredient selected from the group consisting of: fungicides, insecticides, nematocides, miticides, arthropodicides, bactericides and combinations thereof.9. The formulation according to claim 8 , wherein the formulation is suitable for treating plants.10. A formulation for the control of a fungal pathogen claim 8 , comprising:{'claim-ref': {'@idref': 'CLM-00006', 'claim 6'}, 'the formulation of ; and'}at least one agriculturally active ingredient selected from the group consisting of: fungicides, insecticides, nematocides, miticides, arthropodicides, bactericides and combinations thereof. ...

Подробнее
12-01-2017 дата публикации

5-FLUOROPYRIMIDINONE DERIVATIVES

Номер: US20170008855A1
Принадлежит: Adama Makhteshim Ltd.

This present disclosure is related to the field of 5-fluoropyrimidinones and their derivatives and to the use of these compounds as fungicides. 2. A composition for the control of a fungal pathogen including the compound of and a phytologically acceptable carrier material.3Venturia inaequalisSeptoria triticiCercospora beticolaCercospora arachidicolaCercosporidium personatumMycosphaerella fifiensis. The composition of wherein the fungal pathogen is Apple Scab () claim 2 , Leaf Blotch of Wheat () claim 2 , Leaf Spot of Sugarbeets () claim 2 , Leaf Spots of Peanut (and ) claim 2 , and Black Sigatoka of Banana ().4. A method for the control and prevention of fungal attack on a plant claim 2 , the method including the steps of:{'claim-ref': {'@idref': 'CLM-00001', 'claim 1'}, 'applying a fungicidally effective amount of at least one of the compounds of to at least one of the plant, an area adjacent to the plant, soil adapted to support growth of the plant, a root of the plant, foliage of the plant, and a seed adapted to produce the plant.'} This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/232,177 filed Aug. 7, 2009.Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less.The present disclosure relates to 5-fluoropyrimidinone compounds and their use as fungicides. The compounds of the present disclosure may offer protection against ascomycetes, basidiomycetes, deuteromycetes and oomycetes.One embodiment of the present disclosure may include compounds of Formula I:wherein Ris:Another embodiment of the present disclosure may include a fungicidal composition for the control or prevention of fungal attack comprising the compounds described below and a ...

Подробнее
30-03-2017 дата публикации

SYNERGISTIC FUNGICIDAL MIXTURES AND COMPOSITIONS FOR FUNGAL CONTROL

Номер: US20170086459A1
Принадлежит: Adama Makhteshim Ltd.

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. (canceled)3. The synergistic claim 1 , fungicidal mixture of wherein the concentration ratio of the Compound of I to the succinate dehydrogenase inhibitor is between 1:272 and 787:1.412-. (canceled)13. A synergistic claim 1 , fungicidal composition comprising a fungicidally effective amount of the mixture of and an agriculturally acceptable adjuvant or carrier.14. The synergistic claim 13 , fungicidal composition of wherein the succinate dehydrogenase inhibitor is selected from a group consisting of fluxapyroxad claim 13 , benzovindiflupyr claim 13 , penthiopyrad claim 13 , isopyrazam claim 13 , boscalid claim 13 , and fluopyram.1519-. (canceled)21. The method of claim 20 , wherein the synergistic claim 20 , fungicidal mixture is applied to the roots claim 20 , seeds or foliage of the plant.22. The method of claim 20 , wherein the plant is an agricultural crop.23. The method of claim 20 , wherein the synergistic claim 20 , fungicidal mixture is applied at a rate between 40 g/ha and 2600 g/ha of the compound of I and the succinate dehydrogenase inhibitor.24. The method of claim 23 , wherein compound of I is applied at a rate between 15 g/ha and 100 g/ha.25. The method of claim 23 , wherein the succinate dehydrogenase inhibitor is applied at a rate between 25 g/ha and 500 g/ha.26. The method of claim 23 , wherein the succinate dehydrogenase inhibitor is selected from a group consisting of fluxapyroxad claim 23 , benzovindiflupyr claim 23 , penthiopyrad claim 23 , isopyrazam claim 23 , boscalid claim 23 , and fluopyram.27. The method of claim 26 , wherein:a. the succinate dehydrogenate inhibitor is boscalid and the boscalid is applied a rate between 100 g/ha and 625 g/ha,b. the succinate dehydrogenate inhibitor is isopyrazam and the isopyrazam is applied a rate between 25 g/ha and 300 g/ha,c. the succinate dehydrogenate inhibitor is fluxapyroxad and the fluxapyroxad is ...

Подробнее
21-11-2012 дата публикации

Thiazolo[5,4-d] pyrimidines and their use as agrochemicals

Номер: CN102791135A
Принадлежит:

The present disclosure relates to thiazolo[5,4-d]pyrimidines and their use as agrochemicals and animal health products.

Подробнее
30-03-2017 дата публикации

SYNERGISTIC FUNGICIDAL MIXTURES AND COMPOSITIONS FOR FUNGAL CONTROL

Номер: US20170086460A1
Принадлежит: Adama Makhteshim Ltd.

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. (canceled)3. The synergistic claim 1 , fungicidal mixture of wherein the concentration ratio of the Compound of I to (i) the fungicidal multi-site inhibitor or (ii) the strobilurin fungicide is between 1:272 and 787:1.48-. (canceled)9. A synergistic claim 1 , fungicidal composition comprising a fungicidally effective amount of the mixture of and an agriculturally acceptable adjuvant or carrier.10. (canceled)11. The synergistic claim 9 , fungicidal composition of wherein the at least one additional fungicide is a fungicidal multi-site inhibitor selected from captan and folpet.1225-. (canceled)27. The method of claim 26 , wherein the synergistic claim 26 , fungicidal mixture is applied to the roots claim 26 , seeds or foliage of the plant.28. The method of claim 27 , wherein the plant is an agricultural crop.29. The method of claim 27 , wherein the synergistic claim 27 , fungicidal mixture is applied at a rate between 40 g/ha and 2600 g/ha of the compound of I and the fungicidal multi-site inhibitor.30. The method of claim 29 , wherein compound of I is applied at a rate between 15 g/ha and 100 g/ha.31. The method of claim 29 , wherein the multi-site inhibitor is applied at a rate between 1015 g/ha and 2600 g/ha.32. The method of claim 29 , wherein the fungicidal multi-site inhibitor is selected from a group consisting of chlorothalonil claim 29 , mancozeb claim 29 , captan and folpet.33. The method of claim 32 , wherein:a. the multi-site inhibitor is chrlorothalonil and the chlorothalonil is applied a rate between 1000 g/ha and 2500 g/ha,b. the multi-site inhibitor is mancozeb and the mancozeb is applied a rate between 1500 g/ha and 2000 g/ha,c. the multi-site inhibitor is captan and the captan is applied a rate between 1015 g/ha and 2600 g/ha, ord. the multi-site inhibitor is folpet and the folpet is applied a rate between 1015 g/ha and 2600 g/ha.34Mycosphaerella ...

Подробнее
21-08-2013 дата публикации

Flame-suppression and explosion-suppression cryogenic liquefaction device for low-concentration coal bed gas

Номер: CN103256786A
Принадлежит:

The invention discloses a flame-suppression and explosion-suppression cryogenic liquefaction device for low-concentration coal bed gas, which comprises a coal bed gas storage system, a coal bed gas compression system, a coal bed gas purification system, a coal bed gas liquefaction and separation system, an LNG (Liquefied Natural Gas) storage system and a refrigerating circulatory system, wherein driving explosion-suppression devices are arranged on the front side and the rear side of the coal bed gas storage system; a filler used for fractionating methane in the coal bed gas and having the explosion-suppression performance is filled in a rectifying tower; the rectifying tower is internally provided with a fire-retardance and explosion-suppression material; the fire-retardance and explosion-suppression material is a fire-retardance silk screen which is laid in the filler at intervals; and the driving explosion-suppression devices can effectively prevent flame from spreading to a gas holder ...

Подробнее
31-10-2012 дата публикации

2-aldoximino-5-fluoropyrimidine derivatives

Номер: CN102762210A
Принадлежит:

This present disclosure is related to the field of 2-aldoximino-5-fluoropyrimidines and their derivatives and to the use of these compounds as fungicides.

Подробнее
26-06-2013 дата публикации

Device for preparing liquefied natural gas (LNG) by low condensation coal bed methane oxygen bearing copious cooling liquefaction

Номер: CN103175380A
Принадлежит:

The invention discloses a device for preparing liquefied natural gas (LNG) by low condensation coal bed methane oxygen bearing copious cooling liquefaction. The device for preparing LNG by low condensation coal bed methane oxygen bearing copious cooling liquefaction comprises a main process system and a refrigerating system, wherein the main process system comprises a first level heat exchanger, a second level heat exchanger, a third level heat exchanger, a subcooler and a rectifying tower, a tower top condenser and a reboiler are arranged inside the rectifying tower, a nitrogen-oxygen outlet formed at the top of the rectifying tower is connected with the tower top condenser, and a condensate outlet is formed at the bottom of the rectifying tower. The refrigerating system comprises a mixing cryogen circulatory system and a nitrogen circulatory system, wherein the mixing cryogen circulatory system comprises a mixing cryogen compressor, a mixing cryogen cooler and a heavy hydrocarbon separator ...

Подробнее
02-01-2013 дата публикации

Synergistic fungicidal composition containing 5-fluorocytosine for fungal control in cereals

Номер: CN102858341A
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of a) a compound of Formula I and (b) at least one fungicide selected from the group consisting of epoxiconazole, prothioconazole, azoxystrobin, pyraclostrobin, penthiopyrad, isopyrazam, bixafen, boscalid, chlorothalonil and isobutyric acid (3S,6S,7R,8R)-8-benzyl-3-[(3-isobutyryloxymethoxy-4-methoxypyridine-2-carbonyl)-amino]-6-methyl-4,9-dioxo-[1,5]dioxonan-7-yl ester provides synergistic control of selected fungi.

Подробнее
27-12-2016 дата публикации

Synergistic fungicidal mixtures comprising 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1H)-one for fungal control in cereals

Номер: US0009526245B2

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1H)-one, and at least one fungicide selected from the group consisting of: prothioconazole, epoxiconazole, cyproconazole, myclobutanil, metconazole, difenoconazole, propiconazole, fluquinconazole, and flutriafol provides synergistic control.

Подробнее
23-10-2013 дата публикации

Synergistic fungicidal interactions of aminopyrimidines and other fungicides

Номер: CN103369960A
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of a) a compound of Formula I and (b) at least one fungicide selected from the group consisting of myclobutanil, fenbuconazole, difenoconazole, trifloxystrobin, penthiopyrad, fluopyram, boscalid, mancozeb, pyrimethanil, and bixafen provides synergistic control of selected fungi.

Подробнее
27-02-2013 дата публикации

5-FLUORO PYRIMIDINE DERIVATIVES AS FUNGICIDES

Номер: EP2562163A1
Принадлежит:

This present disclosure is related to the field of 5-fluoro pyrmidines and their derivatives and to the use of these compounds as fungicides.

Подробнее
12-06-2013 дата публикации

Device for producing LNG (liquefied natural gas) through PSA (pressure swing adsorption) deepening cold liquefying purification of CBM (coalbed methane) with low concentration

Номер: CN103148678A
Принадлежит:

The invention discloses a device for producing LNG through PSA deepening cold liquefying purification of CBM with low concentration. The device comprises a compression purifying system, a liquefying separation system and a CBM enrichment system, wherein the CBM enrichment system comprises a blower, a cooling device and a PSA device; the PSA device comprises at least four parallelly-arranged adsorption towers, air inlet pipes used for introducing air into the adsorption towers, vacuum pipes used for vacuum-pumping the adsorption towers, blow-down pipes used for releasing pressure of the adsorption towers, and pressure-boosting pipes used for boosting pressure of the adsorption towers; vacuum pumps used for vacuum-pumping are arranged on the vacuum pipes; closed valves are arranged on exhaust ports in the pressure-boosting pipes; a bottom port of each adsorption tower is connected with each air inlet pipe and each vacuum pipe through valves; a top port of each adsorption tower is connected ...

Подробнее
26-06-2013 дата публикации

Process for preparing liquefied natural gas (LNG) by low concentration coal bed methane oxygen bearing copious cooling liquefaction

Номер: CN103175381A
Принадлежит:

The invention discloses a process for preparing liquefied natural gas (LNG) by low concentration coal bed methane oxygen bearing copious cooling liquefaction. The process for preparing LNG by low concentration coal bed methane oxygen bearing copious cooling liquefaction comprises the following steps: (1), compression and purification process; (2), liquefaction and separation process which comprises a, main procedure process; b, refrigeratory process, wherein the refrigeratory process comprises b1, mixing cryogen process; and b2, nitrogen cryogen process. Nitrogen cryogen sequentially passes through a first level heat exchanger, a second level heat exchanger, a third level heat exchanger and a subcooler for cooling after being compressed and cooled, the nitrogen cryogen after throttling enters an overhead condenser to output cold quantity, and then the gaseous nitrogen cryogen sequentially passes through the subcooler, the third level heat exchanger, the second level heat exchanger, and ...

Подробнее
03-01-2017 дата публикации

Synergistic fungicidal mixtures comprising 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1H)-one for fungal control in cereals

Номер: US0009532570B2

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1H)-one, and at least one fungicide selected from the group consisting of fluxapyroxad, benzovindiflupyr, penthiopyrad, isopyrazam, boscalid, and fluopyram provides synergistic control of selected fungi.

Подробнее
18-04-2017 дата публикации

N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxylate derivatives

Номер: US0009622474B2

This present disclosure is related to the field of N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxylates and their derivatives and to the use of these compounds as fungicides. Also provided are methods of controlling a fungal disease such as Septoria tritici, comprising administering an effective amount of the fungicide compound to at lease one surface associated with the plant, seed or soil.

Подробнее
12-12-2017 дата публикации

N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide derivatives

Номер: US0009840475B2

This present disclosure is related to the field of to N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-di-hydropyrimidme-1(2H)-carboxamide compounds and their derivatives and to the use of these compounds as fungicides. This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/746,837 filed Dec. 28, 2012, which is expressly incorporated by reference herein. Background and Summary of the Invention Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less.

Подробнее
28-09-2017 дата публикации

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20170273303A1
Принадлежит:

This disclosure relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. The compound according to claim 1 , wherein X and Y are hydrogen.3. The compound according to claim 2 , wherein Ris alkyl or aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.4. The compound according to claim 2 , wherein Ris hydrogen or alkyl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.5. The compound according to claim 1 , wherein X is C(O)Rand Y is hydrogen.6. The compound according to claim 5 , wherein Ris alkyl or aryl claim 5 , each optionally substituted with 0 claim 5 , 1 or multiple R.7. The compound according to claim 5 , wherein Ris hydrogen or alkyl claim 5 , each optionally substituted with 0 claim 5 , 1 or multiple R.8. The compound according to claim 1 , wherein X is hydrogen and Y is Q.9. The compound according to claim 8 , wherein Ris alkyl or aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.10. The compound according to claim 8 , wherein Ris hydrogen or alkyl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.11. The compound according to claim 9 , wherein Ris hydrogen.12. The compound according to claim 9 , wherein Ris —C(O)R or —CHOC(O)R.13. The compound according to claim 12 , wherein Ris alkyl or alkoxy claim 12 , each optionally substituted with 0 claim 12 , 1 claim 12 , or multiple R.14. The compound according to claim 13 , wherein Ris —CH claim 13 , —CH(CH) claim 13 , —CHOCHCH claim 13 , or —CHCHOCH.15. A composition for the control of a fungal pathogen including at least one of the compounds of Formula I and at least one additional compound selected from the group consisting of: a phytologically acceptable carrier material claim 13 , a second fungicide claim 13 , an insecticide claim 13 , a nematocide claim 13 , a miticide claim 13 , an arthropodicide claim 13 , and a bactericide.16. The composition according to claim 15 , wherein the least one ...

Подробнее
30-10-2013 дата публикации

Synergistic fungicidal interactions of 5-fluorocytosine and other fungicides

Номер: CN103379826A
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of a) a compound of Formula I and (b) at least one fungicide selected from the group consisting of myclobutanil, fenbuconazole, difenoconazole, trifloxystrobin, pentiopyrad, fluopyram, boscalid, mancozeb, and pyrimethanil provides synergistic control of selected fungi.

Подробнее
28-09-2017 дата публикации

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20170273306A1
Принадлежит:

The disclosure relates to macrocyclic picolinamides of Formula (I) and to the use of these compounds as fungicides. 2. The compound according to wherein X is C(O)Rand Y is chosen from H or C(O)R.3. The compound according to wherein X and Y are C(O)Rand Ris independently chosen from alkyl claim 2 , alkoxy claim 2 , benzyl claim 2 , or benzyloxy claim 2 , each substituted with 0 claim 2 , 1 claim 2 , or multiple R claim 2 , wherein each Rmay be substituted with 0 claim 2 , 1 claim 2 , or multiple R.4. The compound according to wherein Rand Rare independently chosen from H claim 3 , alkyl claim 3 , alkenyl claim 3 , aryl claim 3 , or —C(O)R claim 3 , each substituted with 0 claim 3 , 1 or multiple R.5. The compound according to wherein Ris alkoxy and Rand Rare H.6. The compound according to wherein Ris tert-butoxy.7. The compound according to wherein Y is hydrogen.8. The compound according to wherein Rand Rare independently chosen from H claim 7 , alkyl claim 7 , alkenyl claim 7 , aryl claim 7 , or —C(O)R claim 7 , each substituted with 0 claim 7 , 1 or multiple R.9. The compound according to wherein Rand Rare independently alkyl claim 8 , alkenyl claim 8 , aryl claim 8 , or —C(O)R claim 8 , each substituted with 0 claim 8 , 1 or multiple R.10. The compound according to wherein Rand Rare independently alkyl claim 9 , or aryl claim 9 , each substituted with 0 claim 9 , 1 or multiple R.11. The compound according to wherein the amine is protonated to give an ammonium salt of a mineral acid independently chosen from hydrogen chloride claim 8 , hydrogen bromide claim 8 , or hydrogen iodide.12. The compound according to wherein the ammonium salt is the ammonium hydrochloride.13. The compound according to wherein X is C(O)Rand Y is Q.14. The compound according to wherein Rand Rare independently chosen from H claim 13 , alkyl claim 13 , alkenyl claim 13 , aryl claim 13 , or —C(O)R claim 13 , each substituted with 0 claim 13 , 1 claim 13 , or multiple R.15. The compound ...

Подробнее
18-09-2013 дата публикации

Anti-explosion rectifying tower for low-concentration coal seam gas liquefaction and concentration

Номер: CN103307854A
Принадлежит:

The invention discloses an anti-explosion rectifying tower for low-concentration coal seam gas liquefaction and concentration. The anti-explosion rectifying tower comprises a rectifying tower body, wherein the rectifying tower body is filled with filler used for fractionating methane in coal seam gas and provided with an explosion-suppression performance; fire-retardant explosion-suppression materials are also arranged in the rectifying tower body; and the fire-retardant explosion-suppression materials are fire-retardant silk nets paved in the filler at an interval. By setting the filler which meets the rectifying conditions and has the explosion-suppression performance, and the fire-retardant explosion-suppression materials in the rectifying tower body, in a coal seam gas rectifying and separating process, with extraction of methane, even if the explosion limit range of methane is reached, the coal seam gas is divided into a plurality of small size units under the action of the filler ...

Подробнее
28-08-2013 дата публикации

Method for extracting methane contained in low-concentration oxygen-containing coal-seam gas

Номер: CN103267402A
Принадлежит:

The invention discloses a method for extracting methane contained in a low-concentration oxygen-containing coal-seam gas, and the method comprises the following procedures of: (1) a coal-seam gas storage procedure: storing the low-concentration oxygen-containing coal-seam gas by adopting a gas holder; (2) a coal-seam gas compression procedure: pressurizing and compressing the coal-seam gas output from the gas holder to 0.35-0.4 MPG, and keeping the temperature of the coal-seam gas lower than 80 DEG C in a pressurizing and compressing process; (3) a coal-seam gas purifying procedure: sequentially carrying out demercuration, desulfuration, decarbonation and dewatering treatment on the coal-seam gas; (4) a coal-seam gas cooling procedure: cooling the coal-seam gas to -140-160 DEG C, wherein the liquid molar fraction is not more than 15%; (5) a coal-seam gas rectification and separation procedure: delivering the coal-seam gas into a rectification tower, accessing methane liquid obtained through ...

Подробнее
11-07-2012 дата публикации

N1-sulfonyl-5-fluoropyrimidinone derivatives

Номер: CN102574831A
Принадлежит:

This present disclosure is related to the field of N1-sulfonyl-5-fluoropyrimidinones and their derivatives and to the use of these compounds as fungicides.

Подробнее
12-06-2013 дата публикации

Technology for making LNG (Liquefied Natural Gas) from low-concentration coal bed gas through pressure swing adsorption and cryogenic liquefaction

Номер: CN103146449A
Принадлежит:

The invention discloses a technology for making LNG (Liquefied Natural Gas) from low-concentration coal bed gas through pressure swing adsorption and cryogenic liquefaction. The technology comprises the following steps of: (1) enrichment working procedure: to be specific, carrying out methane enrichment on the coal bed gas through a coal bed gas enrichment system, so that the content of methane in the coal bed gas is risen to 35-45% from 10-28%; (2) compression and purification working procedures: to be specific, compressing and purifying the coal bed gas obtained in the enrichment working procedure to obtain a purified coal bed gas; and (3) liquefaction and separation working procedures: to be specific, liquefying and separating a methane component in the coal bed gas to obtain a liquefied natural gas product. The enrichment working procedure is added in conventional working procedures, so that the content of methane is risen to 35-45% from 10-28%, and then the coal beg gas is concentrated ...

Подробнее
11-07-2012 дата публикации

Pteridines and Their use as agrochemicals

Номер: CN102574855A
Принадлежит:

The present disclosure relates to 1- or 2-(4-(aryloxy)-phenyl)ethylamino-, oxy- or sulfanyl)pteridines and 1- or 2-(4-(heteroaryloxy)-phenyl)ethylamino-, oxy- or sulfanyl)pteridines and their use as agrochemicals and animal health products.

Подробнее
09-05-2017 дата публикации

3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides

Номер: US0009642368B2

This present disclosure is related to the field of 3-alkyl-5-fluoro-4-substituted-imino-3,4-5 dihydropyrimidin-2(1H)-ones and their derivatives and to the use of these compounds as fungicides. Also provided are methods of controlling a fungal disease such as Septoria tritici, comprising administering an effective amount of the fungicide compound to at lease one surface associated with the plant, seed or soil.

Подробнее
04-07-2012 дата публикации

N1-acyl-5-fluoropyrimidinone derivatives

Номер: CN102548981A
Принадлежит:

This present disclosure is related to the field of N1-acyl-5-fluoropyrimidinones and their derivatives and to the use of these compounds as fungicides.

Подробнее
30-03-2017 дата публикации

SYNERGISTIC FUNGICIDAL MIXTURES AND COMPOSITIONS FOR FUNGAL CONTROL

Номер: US20170086458A1
Принадлежит: Adama Makhteshim Ltd.

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. (canceled)3. The synergistic claim 1 , fungicidal mixture of wherein the concentration ratio of the Compound of I to the sterol biosynthesis inhibitor is between 1:272 and 787:1.415-. (canceled)16. A synergistic claim 1 , fungicidal composition comprising a fungicidally effective amount of the mixture of and an agriculturally acceptable adjuvant or carrier.17. The synergistic claim 16 , fungicidal composition of wherein the sterol biosynthesis inhibitor is selected from a group consisting of epoxiconazole claim 16 , cyproconazole claim 16 , myclobutanil claim 16 , metconazole claim 16 , propiconazole claim 16 , fluquinconazole claim 16 , flutriafol claim 16 , difenoconazole and prothioconazole.18. (canceled)20. The method of claim 19 , wherein the synergistic claim 19 , fungicidal mixture is applied to the roots claim 19 , seeds or foliage of the plant.21. The method of claim 19 , wherein the plant is an agricultural crop.22. The method of claim 19 , wherein the synergistic claim 19 , fungicidal mixture is applied at a rate between 40 g/ha and 2600 g/ha of the compound of I and the sterol biosynthesis inhibitor.23. The method of claim 22 , wherein compound of I is applied at a rate between 15 g/ha and 100 g/ha.24. The method of claim 22 , wherein the sterol biosynthesis inhibitor is applied at a rate between 25 g/ha and 500 g/ha.25. The method of claim 22 , wherein the sterol biosynthesis inhibitor is selected from a group consisting of epoxiconazole claim 22 , cyproconazole claim 22 , myclobutanil claim 22 , metconazole claim 22 , propiconazole claim 22 , prothioconazole claim 22 , fluquinconazole claim 22 , flutriafol claim 22 , and difenoconazole.26. The method of claim 25 , wherein:a. the sterol biosynthesis inhibitor is epoxyconazole and the epoxyconazole is applied a rate between 50 g/ha and 250 g/ha,b. the sterol biosynthesis inhibitor is cyproconazole and the ...

Подробнее
04-07-2012 дата публикации

5-fluoropyrimidinone derivatives

Номер: CN102548980A
Принадлежит:

This present disclosure is related to the field of 5-fluoropyrimidinones and their derivatives and to the use of these compounds as fungicides.

Подробнее
06-03-2018 дата публикации

N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxylate derivatives

Номер: US0009908855B2

This present disclosure is related to the field of N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-di-hydropyrimidine-1(2H)-carboxylates and their derivatives and to the use of these compounds as fungicides. Also provided are methods of controlling a fungal disease such as Septoria tritici, comprising administering an effective amount of the fungicide compound to at lease one surface associated with the plant, seed or soil.

Подробнее
05-09-2017 дата публикации

Synergistic fungicidal compositions

Номер: US0009750248B2

A synergistic fungicidal mixture contains a fungicidally effective amount of a compound of Formula I, (3S,6S,7R,8R)-8-benzyl-3-(3-((isobutyryloxy)methoxy)-4-methoxypicolinamido)-6-methyl-4,9-dioxo-1,5-dioxonan-7-yl isobutyrate, and at least one triazole fungicide wherein Formula I is ...

Подробнее
04-09-2013 дата публикации

Device for extracting methane in low-concentration oxygen-containing coal-bed gases

Номер: CN103277978A
Принадлежит:

The invention discloses a device for extracting methane in low-concentration oxygen-containing coal-bed gases. The device comprises a heat exchange system, a rectifying separation system, a mixed coolant circulating system and a nitrogen coolant circulating system. The mixed coolant circulating system and the nitrogen coolant circulating system are arranged, on one side, the condensing temperature of the rectifying separation system is lower than minus 180 DEG C, and the mixed coolant circulating system can not supply the required cooling capacity; on the other side, if the nitrogen coolant circulating system is used for supplying the cooling capacity to the heat exchange system, the defects that the energy consumption is high and the refrigerating efficiency is low exist; and besides, the mixed coolant circulating system and the nitrogen coolant circulating system are independent of each other and do not interfere with each other, so that the reasonable distribution of the cooling capacity ...

Подробнее
10-01-2017 дата публикации

Synergistic fungicidal mixtures comprising 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1H)-one for fungal control in cereals

Номер: US0009538753B2

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1H)-one, and at least one fungicide selected from the group consisting of mancozeb, chlorothalonil, pyraclostrobin, fluoxastrobin, azoxystrobin, trifloxystrobin, picoxystrobin, and kresoxim-methyl provides synergistic control of selected fungi.

Подробнее
27-02-2013 дата публикации

N3-substituted-N1-sulfonyl-5-fluoropyrimidinone derivatives

Номер: CN102946730A
Принадлежит:

This present disclosure is related to the field of N3-substituted-N1-sulfonyl-5-fluoropyrimidinones and their derivatives and to the use of these compounds as fungicides.

Подробнее
03-10-2012 дата публикации

Synergistic fungicidal mixtures for fungal control in cereals

Номер: CN102711477A
Автор: Owen W. John, Yao Chenglin
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of a compound of Formula (I-V) and at least one fungicide selected from the group consisting of epoxiconazole, prothioconazole, azoxystrobin, pyraclostrobin, penthiopyrad, isopyrazam, bixafen, boscalid, prochloraz, and chlorothalonil provides synergistic control of selected fungi.

Подробнее
21-06-2012 дата публикации

SYNERGISTIC FUNGICIDAL INTERACTIONS OF 5-FLUOROCYTOSINE AND OTHER FUNGICIDES

Номер: US20120157485A1
Принадлежит: DOW AGROSCIENCES LLC

A fungicidal composition containing a fungicidally effective amount of a) a compound of Formula I and (b) at least one fungicide selected from the group consisting of myclobutanil, fenbuconazole, difenoconazole, trifloxystrobin, pentiopyrad, fluopyram, boscalid, mancozeb, and pyrimethanil provides synergistic control of selected fungi. 2. The mixture of in which the weight ratio of Compound I to myclobutanil is between about 1:5 and about 5:1.3. The mixture of in which the weight ratio of Compound I to claim 1 , fenbuconazole is between about 1:5 and about 5:1.4. The mixture of in which the weight ratio of Compound I to trifloxystrobin is between about 1:5 and about 5:1.5. The mixture of in which the weight ratio of Compound I to penthiopyrad is between about 1:5 and about 5:1.6. The mixture of in which the weight ratio of Compound I to bixafen is between about 1:5 and about 5:1.7. The mixture of in which the weight ratio of Compound I to fluopyram is between about 1:5 and about 5:1.8. The mixture of in which the weight ratio of Compound I to boscalid is between about 1:20 and about 1:1.9. The mixture of in which the weight ratio of Compound I to mancozeb is between about 1:200 and about 1:1.10. The mixture of in which the weight ratio of Compound I to pyrimethanil is between about 1:20 and about 1:1.11. A fungicidal composition comprising a fungicidally effective amount of the fungicidal mixture of and an agriculturally acceptable adjuvant or carrier. This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/423,857 filed Dec. 16, 2010, which is expressly incorporated by reference herein.This invention concerns a synergistic fungicidal composition containing (a) a compound of Formula I and (b) at least one fungicide selected from the group consisting of myclobutanil, fenbuconazole, trifloxystrobin, penthiopyrad, bixafen, fluopyram, boscalid, mancozeb, and pyrimethanil.Fungicides are compounds, of natural or synthetic origin, which act ...

Подробнее
21-06-2012 дата публикации

Synergistic fungicidal interactions of aminopyrimidines and other fungicides

Номер: US20120157486A1
Принадлежит: DOW AGROSCIENCES LLC

A fungicidal composition containing a fungicidally effective amount of a) a compound of Formula I and (b) at least one fungicide selected from the group consisting of myclobutanil, fenbuconazole, difenoconazole, trifloxystrobin, penthiopyrad, fluopyram, boscalid, mancozeb, pyrimethanil, and bixafen provides synergistic control of selected fungi.

Подробнее
17-01-2013 дата публикации

5,8-DIFLUORO-4-(2-(4-(HETEROARYLOXY)-PHENYL)ETHYLAMINO)QUINAZOLINES AND THEIR USE AS AGROCHEMICALS

Номер: US20130017950A1
Принадлежит: DOW AGROSCIENCES LLC

The present disclosure relates to 5,8-difluoro-4-(2-(4-(heteroaryloxy)-phenyl)ethylamino)quinazolines and their use as agrochemicals and animal health products. 2. The process according to claim 1 , wherein the compound of Formula I is applied to an area where control of pests is desired along with at least one other pesticide.3. The process according to claim 1 , wherein the compound of Formula I is applied to an area where control of pests is desired along with at least one herbicide or fungicide.4. The process according to claim 1 , wherein the compound of Formula I is applied to an area where control of pests is desired along with at least one agriculturally active agent selected from the group consisting of: antimicrobials claim 1 , bactericides claim 1 , defoliants claim 1 , safeners claim 1 , synergists claim 1 , algaecides claim 1 , attractants claim 1 , desiccants claim 1 , pheromones claim 1 , repellants claim 1 , avicides claim 1 , disinfectants claim 1 , semiochemicals claim 1 , and molluscicides.5. The process according to claim 1 , wherein the compound of Formula I is applied to an area where control of pests is desired along with at least one other agriculturally active compound selected from the group consisting of: an acetyl choline esterase inhibitor; a sodium channel modulator; a chitin biosynthesis inhibitor; a GABA-gated chloride channel antagonist; GABA claim 1 , a glutamate-gated chloride channel agonist; an acetyl choline receptor agonist; a MET I inhibitor; a Mg-stimulated ATPase inhibitor; a nicotinic acetylcholine receptor; a Midgut membrane disrupter; and an oxidative phosphorylation disrupter.6. The process according to claim 1 , wherein the compound of Formula I is applied to an area where control of pests is desired wherein the compound of Formula I is in the form of a bait claim 1 , a concentrated emulsion claim 1 , a dust claim 1 , an emulsifiable concentrate claim 1 , a fumigant claim 1 , a gel claim 1 , a granule claim 1 , a ...

Подробнее
21-02-2013 дата публикации

5-FLUORO-4-IMINO-3,4-DIHYDROPYRIMIDIN-2-(1H)-ONES DERIVATIVES

Номер: US20130045984A1
Принадлежит: DOW AGROSCIENCES LLC

This present disclosure is related to the field of 5-fluoro-4-imino-3-(substituted)-3,4-dihydropyrimidin-2(1H)ones and their derivatives and to the use of these compounds as fungicides. 2. A composition for the control of a fungal pathogen including the compound of and a phytologically acceptable carrier material.3Venturia inaequalisSeptoria triticiCercospora beticolaCercospora arachidicolaCercosporidium personatumMycosphaerella fijiensis. The composition of wherein the fungal pathogen is at least one of Apple Scab () claim 2 , Leaf Blotch of Wheat () claim 2 , Leaf Spot of Sugarbeets () claim 2 , Leaf Spots of Peanut (and ) claim 2 , and Black Sigatoka of Banana ().4. A method for the control and prevention of fungal attack on a plant claim 2 , the method including the steps of:{'claim-ref': {'@idref': 'CLM-00001', 'claim 1'}, 'applying a fungicidally effective amount of at least one of the compounds of to at least one of the plant, an area adjacent to the plant, soil adapted to support growth of the plant, a root of the plant, foliage of the plant, and a seed adapted to produce the plant.'} This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/524,506 filed Aug. 17, 2011, which is expressly incorporated by reference herein.Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less.The present disclosure relates to 3-alkyl-5-fluoro-4-imino-3,4-dihydropyrimidin-2(1H)one compounds and their use as fungicides. The compounds of the present disclosure may offer protection against ascomycetes, basidiomycetes, deuteromycetes and oomycetes.One embodiment of the present disclosure may include compounds of Formula I:wherein Ris:C-Calkyl optionally substituted with 1-3 R ...

Подробнее
21-02-2013 дата публикации

N-(5-FLUORO-2-((4-METHYLBENZYL)OXY)PYRIMIDIN-4-YL)BENZAMIDE DERIVATIVES

Номер: US20130045985A1
Принадлежит: DOW AGROSCIENCES LLC

This present disclosure is related to the field of N-(5-fluoro-2-((4-methylbenzyl)oxy)pyrimidin-4-yl)benzamides and their derivatives and to the use of these compounds as fungicides. 2. A composition for the control of a fungal pathogen including the compound of and a phytologically acceptable carrier material.3Venturia inaequalisSeptoria triticiCercospora beticolaCercospora arachidicolaCercosporidium personatumMycosphaerella fijiensis. The composition of wherein the fungal pathogen is at least one of Apple Scab () claim 2 , Leaf Blotch of Wheat () claim 2 , Leaf Spot of Sugarbeets () claim 2 , Leaf Spots of Peanut (and ) claim 2 , and Black Sigatoka of Banana ().4. A method for the control and prevention of fungal attack on a plant claim 2 , the method including the steps of:{'claim-ref': {'@idref': 'CLM-00001', 'claim 1'}, 'applying a fungicidally effective amount of at least one compound of to at least one of the plant, an area adjacent to the plant, soil adapted to support growth of the plant, a root of the plant, foliage of the plant, and a seed adapted to produce the plant.'} This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/524,509 filed Aug. 17, 2011, which is expressly incorporated by reference herein.Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less.The present disclosure relates to N-(5-fluoro-2-((4-methylbenzyl)oxy)pyrimidin-4-yl)benzamide compounds and their use as fungicides. The compounds of the present disclosure may offer protection against ascomycetes, basidiomycetes, deuteromycetes and oomycetes.One embodiment of the present disclosure may include compounds of Formula I:wherein Ris —N(R)R; Ris C-Calkyl, optionally substituted ...

Подробнее
13-06-2013 дата публикации

5-FLUOROCYTOSINE AS A SEED TREATMENT AGENT TO CONTROL PLANT DISEASE

Номер: US20130152233A1
Принадлежит: DOW AGROSCIENCES LLC

The present disclosure relates to the use of 5-fluorocytosine as a seed treatment to prevent or control plant diseases. 1. A plant seed , comprising:a seed; anda disease-inhibiting and phytologically acceptable amount of 5-fluorocytosine, wherein said seed is contacted with the disease-inhibiting and phytologically acceptable amount of 5-fluorocytosine to form a treated seed that germinates to form a plant wherein the plant that forms is more resistant to fungal attack than is a plant from a similar untreated seed that has not been contacted with the a disease-inhibiting and phytologically acceptable amount of 5-fluorocytosine.2. The plant seed of claim 1 , wherein said seed is contacted with the disease-inhibiting and phytologically acceptable amount of 5-fluorocytosine before the treated seed is planted.3. The plant seed of claim 1 , wherein said seed is contacted with the disease-inhibiting and phytologically acceptable amount of 5-fluorocytosine after the seed is planted.4. The plant seed of claim 1 , wherein the disease-inhibiting and phytologically acceptable amount of 5-fluorocytosine used to create the treated seed is in a liquid form or a solid form.5. The plant seed of claim 1 , wherein the disease-inhibiting and phytologically acceptable amount of 5-fluorocytosine is between about 0.5 g to about 500 g of 5-fluorocytosine per 100 kg of seed.6. The plant seed of claim 1 , wherein the disease-inhibiting and phytologically acceptable amount of 5-fluorocytosine is between about 1.8 g to about 16.5 g of 5-fluorocytosine per 100 kg of seed.7. The plant seed of claim 1 , wherein the disease-inhibiting and phytologically acceptable amount of 5-fluorocytosine is between about 5.5 g to about 16.5 g of 5-fluorocytosine per 100 kg of seed.8. The plant seed of claim 1 , wherein the disease-inhibiting and phytologically acceptable amount of 5-fluorocytosine is about 16.5 g of 5-fluorocytosine per 100 kg of seed.9. The plant seed of claim 1 , further including at least ...

Подробнее
26-09-2013 дата публикации

PTERIDINES AND THEIR USE AS AGROCHEMICALS

Номер: US20130252960A1
Принадлежит: DOW AGROSCIENCES LLC

The present disclosure relates to 1- or 2-(4-(aryloxy)-phenyl)ethylamino-, oxy- or sulfanyl)pteridines and 1- or 2-(4-(heteroaryloxy)-phenyl)ethylamino-, oxy- or sulfanyl)pteridines and their use as agrochemicals and animal health products. More specifically, the invention provides new compounds of the formula (I-A): This application is a divisional application and claims priority to U.S. patent application Ser. No. 12/551,008, filed on Aug. 31, 2009, which is incorporated herein by reference in its entirety.The present disclosure relates to 1- or 2-(4-(aryloxy)-phenyl)ethylamino-, oxy- or sulfanyl)pteridines and 1- or 2-(4-(heteroaryloxy)-phenyl)ethylamino-, oxy- or sulfanyl)pteridines and their use as agrochemicals and animal health products.The present disclosure provides novel organic compounds that may demonstrate activity as pesticides, meaning that they may control fungi, insects, mites, and/or animal parasites. The disclosure also provides novel pesticide methods and compositions utilizing the novel compounds.More specifically, the invention provides new compounds of the formula (I-A):wherein:R is H, CH, phenyl, or a heterocycle comprising a 5 or 6 membered single ring or a fused ring system comprising at least one 5 or 6 membered heterocycle optionally substituted with H, halo, lower alkyl, lower alkoxy, benzyloxy, lower alkenyl, lower alkynyl, haloalkyl, haloalkoxy, NO, CN, lower alkoxycarbonyl, lower alkylcarbonyl, lower alkyl-SO, and aldoximes and lower alkyloximes, optionally substituted on oxygen by lower alkyl.Z is H, a C—C single bond, CH, NH, O, S, CN, CHO, OCH, CHCHO, or OCHCH;m is 4;p is 0 or 1;q is an integer from 0 to 2;Ris independently H, halo, lower alkyl, lower alkenyl, lower alkynyl, hydroxy, lower alkoxy, haloalkyl, haloalkoxy, NO, CN, lower alkylcarbonyl, lower alkoxycarbonyl, mercapto, lower alkylthio, aldoximes and lower alkyloximes, optionally substituted on oxygen by lower alkyl;Y is a C—C single bond, C(R)O or C(R);n is 2; ...

Подробнее
07-11-2013 дата публикации

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20130296371A1
Принадлежит: DOW AGROSCIENCES LLC

The disclosure relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. The compound according to claim 1 , wherein:{'sub': 1', '3', '2', '3, 'Ris H, —C(O)R, or —CHOC(O)R;'}{'sub': 2', '5, 'Ris alkyl, alkenyl, or aryl, each substituted with 0, 1 or multiple R;'}{'sub': 3', '5, 'Ris alkyl or alkoxy, substituted with 0, 1, or multiple R;'}{'sub': 5', '6, 'Ris alkyl, alkenyl, halo, haloalkyl, alkoxy, haloalkoxy, arylalkoxy, cyano, aryl or heterocyclyl, each substituted with 0, 1 or multiple R; and'}{'sub': '6', 'Ris alkyl, alkenyl, halo, haloalkyl, alkoxy, haloalkoxy, arylalkoxy, cyano, aryl or heterocyclyl.'}3. A compound according to claim 3 , wherein:{'sub': 1', '3', '2', '3, 'Ris H, —C(O)R, or —CHOC(O)R;'}{'sub': 2', '5, 'Ris alkyl, alkenyl, or aryl, each substituted with 0, 1 or multiple R;'}{'sub': 3', '5, 'Ris alkyl or alkoxy, substituted with 0, 1, or multiple R; and'}{'sub': '5', 'Ris alkyl, halo, haloalkyl, or aryl.'}4. A compound according to claim 3 , wherein:{'sub': 1', '3', '2', '3, 'Ris H, —C(O)R, or —CHOC(O)R;'}{'sub': 2', '5, 'Ris alkyl, alkenyl, or aryl, each substituted with 0, 1 or multiple R;'}{'sub': '3', 'Ris alkyl; and'}{'sub': '5', 'Ris alkyl, halo, haloalkyl, or aryl.'}7Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformisMycosphaerella fujiensis. The compositions according to claim 6 , wherein the effective amount of the compound is effective against at least one plant pathogen selected from the group consisting of: Leaf Blotch of Wheat (; anamorph: ) claim 6 , Wheat Brown Rust () claim 6 , Stripe Rust () claim 6 , and Black Sigatoka ().8Septoria triticiPuccinia triticina. The composition according to claim 7 , wherein the plant pathogen is at least one organism selected from the group consisting of () and (). This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/643,623 filed May 7, 2012, which is expressly incorporated by reference herein.Fungicides are ...

Подробнее
07-11-2013 дата публикации

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20130296373A1
Принадлежит: DOW AGROSCIENCES LLC

The disclosure relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. The compound according to claim 1 , wherein X and Y are independently chosen from H or C(O)R.3. The compound according to claim 2 , wherein Ris independently chosen from H claim 2 , alkyl claim 2 , alkenyl claim 2 , aryl claim 2 , heterocyclyl claim 2 , silyl claim 2 , —C(O)R claim 2 , each substituted with 0 claim 2 , 1 or multiple R.4. The compound according to claim 3 , wherein Ris independently phenyl or cyclohexyl.5. The compound according to claim 4 , wherein Ris alkyl or aryl substituted with 0 claim 4 , 1 claim 4 , or multiple R.6. The compound according to claim 5 , wherein Ris alkoxy or benzyloxy substituted with 0 claim 5 , 1 claim 5 , or multiple R.7. The compound according to claim 6 , wherein Ris hydrogen or alkyl.8. The compound according to claim 1 , wherein X is H and Y is Q.10. The compound according to claim 9 , wherein Ris independently chosen from alkyl claim 9 , aryl claim 9 , or —C(O)R claim 9 , each substituted with 0 claim 9 , 1 or multiple R.11. The compound according to claim 10 , wherein Ris phenyl.12. The compound according to claim 11 , wherein Ris alkyl substituted with 0 claim 11 , 1 claim 11 , or multiple R.13. The compound according to claim 12 , wherein Ris alkyl claim 12 , aryl claim 12 , alkoxy claim 12 , or halo.14. A composition for the control of a fungal pathogen including at least one of the compounds according to and a phytologically acceptable carrier material.16Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformisVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPseudoperonospora cubensisPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The composition according to claim claim 1 , 14 wherein the plant pathogen is at least one ...

Подробнее
07-11-2013 дата публикации

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20130296375A1
Принадлежит: DOW AGROSCIENCES LLC

The invention relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. A compound according to claim 1 , wherein:{'sub': '6', 'wherein, R is H, C(O)R;'}{'sub': 1', '6, 'Ris H, C(O)R;'}{'sub': 2', '5, 'Ris independently or separately H, alkyl, alkenyl, aryl, each substituted with 0, 1 or multiple R;'}{'sub': '3', 'Ris independently or separately H, methyl;'}{'sub': '5', 'Ris alkyl, alkoxy, halo, haloalkyl, or aryl; and'}{'sub': '6', 'Ris alkoxy, benzyloxy.'}5Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformisVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPseudoperonospora cubensisPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The compositions according to claim 4 , wherein the plant pathogen is least one pathogen selected from the group consisting of: Leaf Blotch of Wheat (; anamorph: ) claim 4 , Wheat Brown Rust () claim 4 , Stripe Rust () claim 4 , Scab of Apple () claim 4 , Blister Smut of Maize () claim 4 , Powdery Mildew of Grapevine () claim 4 , Barley scald () claim 4 , Blast of Rice () claim 4 , Downy Mildew of Cucurbits () claim 4 , Rust of Soybean () claim 4 , Glume Blotch of Wheat () claim 4 , Powdery Mildew of Wheat (f. sp. ) claim 4 , Powdery Mildew of Barley (f. sp. ) claim 4 , Powdery Mildew of Cucurbits () claim 4 , Anthracnose of Cucurbits () claim 4 , Leaf Spot of Beet () claim 4 , Early Blight of Tomato () claim 4 , and Net Blotch of Barley ().6Septoria triticiPuccinia triticinaPhakopsora pachyrhizi. The composition according to claim 5 , wherein the fungal pathogen is at least one of Leaf Blotch of Wheat () claim 5 , Wheat Brown Rust () claim 5 , and Rust of Soybean ().8. The method according to claim 7 , wherein the compound is applied in a mixture with at least one additional compound selected from the group ...

Подробнее
09-01-2014 дата публикации

N1-SUBSTITUTED-5-FLUORO-2-OXOPYRIMIDINONE-1(2H)-CARBOXAMIDE DERIVATIVES

Номер: US20140011824A1
Принадлежит: DOW AGROSCIENCES LLC

This present disclosure is related to the field of N1-substituted-5-fluoro-2-oxopyrimidinone-1-(2H)-carboxamides and their derivatives and to the use of these compounds as fungicides. 2. A composition for the control of a fungal pathogen including the compound of and a phytologically acceptable carrier material.3Venturia inaequalisSeptoria triticiCercospora beticolaCercospora arachidicolaCercosporidium personatumMycosphaerella fijiensis. The composition of wherein the fungal pathogen is Apple Scab () claim 2 , Leaf Blotch of Wheat () claim 2 , Leaf Spot of Sugarbeets () claim 2 , Leaf Spots of Peanut (and ) claim 2 , and Black Sigatoka of Banana ().4. A method for the control and prevention of fungal attack on a plant claim 2 , the method including the steps of:{'claim-ref': {'@idref': 'CLM-00001', 'claim 1'}, 'applying a fungicidally effective amount of at least one of the compounds of to at least one of the plant, an area adjacent to the plant, soil adapted to support growth of the plant, a root of the plant, foliage of the plant, and a seed adapted to produce the plant.'} This application is a continuation of U.S. application Ser. No. 12/851,331, filed Aug. 5, 2010, which claims priority to U.S. Provisional Application No. 61/232,245, filed on Aug. 7, 2009, the disclosures of which are expressly incorporated by reference herein.Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less.The present disclosure relates to N1-substituted-5-fluoro-2-oxopyrimidinone-1(2H)-carboxamide compounds and their use as fungicides. The compounds of the present disclosure may offer protection against ascomycetes, basidiomycetes, deuteromycetes and oomycetes.One embodiment of the present disclosure may ...

Подробнее
23-01-2014 дата публикации

5-FLUORO PYRIMIDINE DERIVATIVES

Номер: US20140024616A1
Принадлежит: DOW AGROSCIENCES LLC

This present disclosure is related to the field of 5-fluoro pyrimidines and their derivatives and to the use of these compounds as fungicides. 15-. (canceled)7. The compound of claim 6 , wherein Rand Rare taken together to form a 5- or 6-membered saturated or unsaturated ring containing 1-3 heteroatoms wherein each ring may be optionally substituted with 1-3 R.8. The compound of claim 6 , wherein Ris —C(═NR)NRR.9. The compound of claim 6 , wherein Ris hydroxyl or amino.10. The compound of claim 6 , wherein Ris C-Calkenyl optionally substituted with 1-3 R.11. The compound of claim 6 , wherein Ris —(CHR)R claim 6 , or —Si(R).12. The compound of claim 6 , wherein Ris methylene-2-furanyl claim 6 , —CHRC(O)OR claim 6 , or benzyl optionally substituted with 1-3 R.13. The compound of claim 6 , wherein Ris benzothiazoyl claim 6 , quinazolinyl claim 6 , or a 5- or 6-membered saturated or unsaturated ring containing 1-3 heteroatoms wherein each ring may be optionally substituted with 1-3 R.14. The compound of claim 6 , wherein Ris C-Calkenyl claim 6 , 2-benzofuranyl claim 6 , or a 5- or 6-membered saturated or unsaturated ring containing 1-3 heteroatoms wherein each ring may be optionally substituted with 1-3 R.15. The compound of claim 6 , wherein Ris C-Calkenyl claim 6 , benzyl claim 6 , or a 5- or 6-membered saturated or unsaturated ring containing 1-3 heteroatoms wherein each ring may be optionally substituted with 1-3 R.161. The compound of claim claim 6 , wherein Ris benzoyl.17. A composition for the control of a fungal pathogen including the compound of and a phytologically acceptable carrier material.18Venturia inaequalisSeptoria triticiCercospora beticolaCercospora arachidicolaMycosphaerella fijiensis. The composition of wherein the fungal pathogen is Apple Scab () claim 17 , Leaf Blotch of Wheat () claim 17 , Leaf spot of sugarbeets () claim 17 , Leaf Spot of peanut () claim 17 , and Black Sigatoka ().19. A method for the control and prevention of fungal attack on a ...

Подробнее
06-01-2022 дата публикации

SYNERGISTIC FUNGICIDAL MIXTURES AND COMPOSITIONS COMPRISING 5-FLUORO-4-IMINO-3-METHYL-1-TOSYL-3,4-DIHYDROPYRIMIDIN-2(1H)-ONE FOR FUNGAL CONTROL (MSI)

Номер: US20220000114A1
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of chlorothalonil and mancozeb.3. The mixture of in which the concentration ratio of the Compound of Formula I to chlorothalonil is about 1:219.4. The mixture of in which the concentration ratio of the Compound of Formula I to mancozeb is about 1:272.5Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is one of Leaf Blotch of Wheat (; anamorph: ) claim 2 , Wheat Brown Rust () claim 2 , Stripe Rust (f. sp. ) claim 2 , Scab of Apple () claim 2 , Blister Smut of Maize () claim 2 , Powdery Mildew of Grapevine () claim 2 , Barley scald () claim 2 , Blast of Rice () claim 2 , Rust of Soybean () claim 2 , Glume Blotch of Wheat () claim 2 , Powdery Mildew of Wheat (f. sp. ) claim 2 , Powdery Mildew of Barley (f. sp. ) claim 2 , Powdery Mildew of Cucurbits () claim 2 , Anthracnose of Cucurbits () claim 2 , Leaf Spot of Beet () claim 2 , Early Blight of Tomato () claim 2 , and Net Blotch of Barley ().6Mycosphaerella graminicola; anamorph: Septoria tritici. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is Leaf Blotch of Wheat ().7Mycosphaerella graminicola; anamorph: Septoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria ...

Подробнее
04-01-2018 дата публикации

PICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20180000075A1
Принадлежит:

This disclosure relates to picolinamides of Formula I and their use as fungicides. 2. A compound according to claim 1 , wherein X and Y are hydrogen.3. A compound according to claim 2 , wherein Rand Rare independently chosen from hydrogen or alkyl.4. A compound according to claim 2 , wherein Rand Rare independently chosen from hydrogen or alkyl.5. A compound according to claim 2 , wherein Ris chosen from C-Calkyl claim 2 , aryl claim 2 , or alkenyl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.6. A compound according to claim 2 , wherein Ris chosen from alkyl or aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.7. A compound according to claim 2 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 2 , Rand Rare independently chosen from hydrogen or alkyl claim 2 , Ris chosen from C-Calkyl claim 2 , aryl claim 2 , or alkenyl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R claim 2 , and Ris chosen from alkyl or aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.8. A compound according to claim 1 , wherein X is C(O)Rand Y is hydrogen.9. A compound according to claim 8 , wherein Rand Rare independently chosen from hydrogen or alkyl.10. A compound according to claim 8 , wherein Rand Rare independently chosen from hydrogen or alkyl.11. A compound according to claim 8 , wherein Ris chosen from C-Calkyl claim 8 , aryl claim 8 , or alkenyl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.12. A compound according to claim 8 , wherein Ris chosen from alkyl or aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.13. A compound according to claim 8 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 8 , Rand Rare independently chosen from hydrogen or alkyl claim 8 , Ris chosen from C-Calkyl claim 8 , aryl claim 8 , or alkenyl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R claim 8 ...

Подробнее
04-01-2018 дата публикации

PICOLINAMIDES AS FUNGICIDES

Номер: US20180000080A1
Принадлежит:

This disclosure relates to picolinamides of Formula I and their use as fungicides. 2. A compound according to claim 1 , wherein X and Y are hydrogen.3. A compound according to claim 2 , wherein Rand Rare independently chosen from hydrogen or alkyl.4. (canceled)5. A compound according to claim 2 , wherein Ris aryl claim 2 , optionally substituted with 0 claim 2 , 1 or multiple R.6. A compound according to claim 2 , wherein Ris chosen from alkyl or aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.7. A compound according to claim 2 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 2 , Ris aryl claim 2 , optionally substituted with 0 claim 2 , 1 or multiple R claim 2 , and Ris chosen from alkyl or aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.8. A compound according to claim 1 , wherein X is C(O)Rand Y is hydrogen.9. A compound according to claim 8 , wherein Rand Rare independently chosen from hydrogen or alkyl.10. (canceled)11. A compound according to claim 8 , wherein Ris aryl claim 8 , optionally substituted with 0 claim 8 , 1 or multiple R.12. A compound according to claim 8 , wherein Ris chosen from alkyl or aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.13. A compound according to claim 8 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 8 , Ris aryl claim 8 , optionally substituted with 0 claim 8 , 1 or multiple R claim 8 , and Ris chosen from alkyl or aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.14. A compound according to claim 1 , wherein X is hydrogen and Y is Q.15. A compound according to claim 14 , wherein Ris hydrogen.16. A compound according to claim 15 , wherein Ris alkoxy.17. A compound according to claim 16 , wherein Rand Rare independently chosen from hydrogen or alkyl.18. (canceled)19. A compound according to claim 16 , wherein Ris aryl claim 16 , optionally substituted with 0 claim 16 , 1 or ...

Подробнее
04-01-2018 дата публикации

5-FLUORO-4-IMINO-3-(ALKYL/SUBSTITUTED ALKYL)-1-(ARYLSULFONYL)-3,4-DIHYDROPYRIMIDIN-2(1H)-ONE AS A SEED TREATMENT

Номер: US20180000082A1
Принадлежит: ADAMA MAKHTESHIM LTD.

The present disclosure relates to the use of a compound of Formula I as a seed treatment to prevent or control plant diseases. 2. The method of claim 1 , wherein Rand Rare each —CH.3. The method of claim 2 , wherein the compound of Formula I is applied at a rate from about 0.5 to about 500 grams per 100 kilograms of seed.4Triticum. The method of claim 1 , wherein the seed being treated is a wheat seed (sp.; TRZSS) claim 1 , sugar beet (BEAVA) claim 1 , or peanut (ARHHY).5Zymoseptoria triticiCercospora beticolaCercospora arachidicolaCercosporidium personatum. The method of claim 1 , wherein the fungal pathogen is selected from the group consisting of the causal agent of wheat leaf blotch () claim 1 , leaf spot of sugar beets () claim 1 , and leaf spot of peanut (and ).7. The plant seed or seedling of claim 6 , wherein the plant seed or seedling is further treated with one or more additional fungicides.8. The plant seed or seedling of further adapted to eradicate undesirable vegetation claim 6 , wherein the plant seed or seedling is treated with the compound of Formula I and one or more herbicides.9. The seed or seedling of claim 6 , wherein the plant seed or seedling is further treated with one or more additional plant health stimulators selected from the group consisting of organic compounds claim 6 , inorganic fertilizers or micronutrient donors claim 6 , biocontrol agents and inoculants.10. (canceled)11. (canceled)12. (canceled)13. (canceled)14. The plant seed or seedling of further adapted to produce a plant resistant to insect attack claim 6 , wherein the plant seed or seedling is treated with the compound of Formula I and one or more insecticides.15. (canceled)16. (canceled)17. (canceled)18. (canceled)20. The method of claim 19 , wherein Rand Rare each —CH.21. The method of claim 1 , wherein Rand Rare independently selected from C-Calkyl.22Triticum. The method of claim 1 , wherein the seed being treated is a wheat seed (sp.; TRZSS).23. The method of claim 1 , ...

Подробнее
04-01-2018 дата публикации

USE OF PICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20180000084A1
Принадлежит:

This disclosure relates to picolinamides of Formula I and their use as fungicides. 2. A composition according to claim 1 , wherein X is hydrogen and Y is Q.3. A composition according to claim 2 , wherein Ris alkoxy.4. A composition according to claim 3 , wherein Ris hydrogen.5. A composition according to claim 4 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 4 , optionally substituted with 0 claim 4 , 1 or multiple R.6. A composition according to claim 4 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 4 , each optionally substituted with 0 claim 4 , 1 or multiple R.7. A composition according to claim 4 , wherein Ris aryl claim 4 , optionally substituted with 0 claim 4 , 1 or multiple R.8. A composition according to claim 4 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 4 , optionally substituted with 0 claim 4 , 1 or multiple R claim 4 , Rand Rare independently chosen from hydrogen or alkyl claim 4 , each optionally substituted with 0 claim 4 , 1 or multiple R claim 4 , and Ris aryl claim 4 , optionally substituted with 0 claim 4 , 1 or multiple R.9. A composition according to claim 3 , wherein Ris chosen from —C(O)R claim 3 , or —CHOC(O)R.10. A composition according to claim 9 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 9 , optionally substituted with 0 claim 9 , 1 or multiple R.11. A composition according to claim 9 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 9 , each optionally substituted with 0 claim 9 , 1 or multiple R.12. A composition according to claim 9 , wherein Ris aryl claim 9 , optionally substituted with 0 claim 9 , 1 or multiple R.13. A composition according to claim 9 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 9 , Rand Rare independently chosen from hydrogen or alkyl claim 9 , each optionally substituted with 0 claim 9 , 1 or multiple R claim 9 , and Ris aryl claim 9 , optionally substituted with 0 claim ...

Подробнее
04-01-2018 дата публикации

USE OF PICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20180000085A1
Принадлежит:

This disclosure relates to picolinamides of Formula I and their use as fungicides. 2. The composition according to claim 1 , wherein X is hydrogen and Y is Q.3. The composition according to claim 2 , wherein Ris alkoxy.4. The composition according to claim 3 , wherein Ris hydrogen.5. The composition according to claim 4 , wherein Rand Rare independently chosen from hydrogen or alkyl.6. The composition according to claim 4 , wherein Rand Rare independently chosen from hydrogen or alkyl.7. The composition according to claim 4 , wherein Ris chosen from C-Calkyl claim 4 , aryl claim 4 , or alkenyl claim 4 , each optionally substituted with 0 claim 4 , 1 or multiple R.8. The composition according to claim 4 , wherein Ris chosen from alkyl or aryl claim 4 , each optionally substituted with 0 claim 4 , 1 or multiple R.9. The composition according to claim 4 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 4 , Rand Rare independently chosen from hydrogen or alkyl claim 4 , Ris chosen from C-Calkyl claim 4 , aryl claim 4 , or alkenyl claim 4 , each optionally substituted with 0 claim 4 , 1 or multiple R claim 4 , and Ris chosen from alkyl or aryl claim 4 , each optionally substituted with 0 claim 4 , 1 or multiple R.10. The composition according to claim 3 , wherein Ris chosen from —C(O)R claim 3 , or —CHOC(O)R.11. The composition according to claim 10 , wherein Ris alkyl claim 10 , optionally substituted with 0 claim 10 , 1 or multiple R.12. The composition according to claim 11 , wherein Rand Rare independently chosen from hydrogen or alkyl.13. The composition according to claim 11 , wherein Rand Rare independently chosen from hydrogen or alkyl.14. The composition according to claim 11 , wherein Ris chosen from C-Calkyl claim 11 , aryl claim 11 , or alkenyl claim 11 , each optionally substituted with 0 claim 11 , 1 or multiple R.15. The composition according to claim 11 , wherein Ris chosen from alkyl or aryl claim 11 , each optionally substituted with ...

Подробнее
04-01-2018 дата публикации

USE OF PICOLINAMIDES AS FUNGICIDES

Номер: US20180002288A1
Принадлежит:

This disclosure relates to picolinamides of Formula I and their use as fungicides. 2. A composition according to claim 1 , wherein X is hydrogen and Y is Q.3. A composition according to claim 2 , wherein Ris alkoxy.4. A composition according to claim 3 , wherein Ris hydrogen.5. A composition according to claim 4 , wherein Rand Rare independently chosen from hydrogen or alkyl.6. (canceled)7. A composition according to claim 4 , wherein Ris aryl claim 4 , optionally substituted with 0 claim 4 , 1 or multiple R.8. A composition according to claim 4 , wherein Ris chosen from alkyl or aryl claim 4 , each optionally substituted with 0 claim 4 , 1 or multiple R.9. A composition according to claim 4 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 4 , optionally substituted with 0 claim 4 , 1 or multiple R claim 4 , and Ris chosen from alkyl or aryl claim 4 , each optionally substituted with 0 claim 4 , 1 or multiple R.10. A composition according to claim 3 , wherein Ris chosen from —C(O)R claim 3 , or —CHOC(O)R.11. A composition according to claim 10 , wherein Ris alkyl claim 10 , optionally substituted with 0 claim 10 , 1 or multiple R.12. A composition according to claim 11 , wherein Rand Rare independently chosen from hydrogen or alkyl.13. (canceled)14. A composition according to claim 11 , wherein Ris aryl claim 11 , optionally substituted with 0 claim 11 , 1 or multiple R.15. A composition according to claim 11 , wherein Ris chosen from alkyl or aryl claim 11 , each optionally substituted with 0 claim 11 , 1 or multiple R.16. A composition according to claim 11 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 11 , Ris aryl claim 11 , optionally substituted with 0 claim 11 , 1 or multiple R claim 11 , and Ris chosen from alkyl or aryl claim 11 , each optionally substituted with 0 claim 11 , 1 or multiple R.17. A composition according to claim 16 , wherein Ris chosen from —CH claim 16 , —CHOCHCH claim 16 , —CHCHOCH claim 16 , — ...

Подробнее
04-01-2018 дата публикации

MACROCYCLIC PICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20180002319A1
Принадлежит:

This disclosure relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. The compound according to claim 1 , wherein X and Y are hydrogen.3. The compound according to claim 2 , wherein Ris selected from the group consisting of hydrogen claim 2 , alkyl claim 2 , alkenyl claim 2 , and aryl claim 2 , each optionally substituted with 0 claim 2 , 1 claim 2 , or multiple R.4. (canceled)5. The compound according to claim 2 , wherein Ris independently selected for Rand Rfrom the group consisting of hydrogen claim 2 , alkyl claim 2 , alkenyl claim 2 , and aryl claim 2 , each optionally substituted with 0 claim 2 , 1 claim 2 , or multiple R.6. The compound according to claim 1 , wherein X is C(O)Rand Y is hydrogen.7. The compound according to claim 6 , wherein Ris selected from the group consisting of hydrogen claim 6 , alkyl claim 6 , alkenyl claim 6 , and aryl claim 6 , each optionally substituted with 0 claim 6 , 1 claim 6 , or multiple R.8. (canceled)9. The compound according to claim 6 , wherein Ris independently selected for Rand Rfrom the group consisting of hydrogen claim 6 , alkyl claim 6 , alkenyl claim 6 , and aryl claim 6 , each optionally substituted with 0 claim 6 , 1 claim 6 , or multiple R.10. The compound according to claim 1 , wherein X is hydrogen and Y is Q.11. The compound according to claim 10 , wherein Ris alkoxy.12. The compound according to claim 11 , wherein Ris hydrogen.13. The compound according to claim 12 , wherein Ris selected from the group consisting of hydrogen claim 12 , alkyl claim 12 , alkenyl claim 12 , and aryl claim 12 , each optionally substituted with 0 claim 12 , 1 claim 12 , or multiple R.14. (canceled)15. The compound according to claim 12 , wherein Ris independently selected for Rand Rfrom the group consisting of hydrogen claim 12 , alkyl claim 12 , alkenyl claim 12 , and aryl claim 12 , each optionally substituted with 0 claim 12 , 1 claim 12 , or multiple R.16. The compound according to claim 11 , ...

Подробнее
04-01-2018 дата публикации

USE OF MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20180002320A1
Принадлежит:

This disclosure relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. A composition according to claim 1 , wherein X is hydrogen and Y is Q.3. A composition according to claim 2 , wherein Ris alkoxy.4. A composition according to claim 3 , wherein Ris hydrogen.5. A composition according to claim 4 , wherein Ris selected from the group consisting of hydrogen claim 4 , alkyl claim 4 , alkenyl claim 4 , and aryl claim 4 , each optionally substituted with 0 claim 4 , 1 claim 4 , or multiple R.6. (canceled)7. A composition according to claim 4 , wherein Ris independently selected for Rand Rfrom the group consisting of hydrogen claim 4 , alkyl claim 4 , alkenyl claim 4 , and aryl claim 4 , each optionally substituted with 0 claim 4 , 1 claim 4 , or multiple R.8. A composition according to claim 3 , wherein Ris selected from the group consisting of —C(O)Rand —CHOC(O)R.9. A composition according to claim 8 , wherein Ris alkyl claim 8 , optionally substituted with 0 claim 8 , 1 claim 8 , or multiple R.10. A composition according to claim 9 , wherein Ris selected from the group consisting of hydrogen claim 9 , alkyl claim 9 , alkenyl claim 9 , and aryl claim 9 , each optionally substituted with 0 claim 9 , 1 claim 9 , or multiple R.11. (canceled)12. A composition according to claim 9 , wherein Ris independently selected for Rand Rfrom the group consisting of hydrogen claim 9 , alkyl claim 9 , alkenyl claim 9 , and aryl claim 9 , each optionally substituted with 0 claim 9 , 1 claim 9 , or multiple R.13. A composition according to claim 12 , wherein Ris selected from the group consisting of —CH claim 12 , —CH(CH) claim 12 , and —CHOCHCH.14. A composition for the control of a fungal pathogen including at least one of the compositions of and a phytologically acceptable carrier material.15. A composition for the control of a fungal pathogen including at least one of the compositions of and a phytologically acceptable carrier material.16. (canceled)17. A ...

Подробнее
14-01-2016 дата публикации

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20160007601A1
Принадлежит:

This disclosure relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. The compound according to claim 1 , wherein X and Y are hydrogen.3. The compound according to claim 1 , wherein X is C(O)Rand Y is hydrogen.4. The compound according to claim 1 , wherein X is hydrogen and Y is Q.5. The compound according to claim 4 , wherein Ris hydrogen.6. The compound according to claim 4 , wherein Ris —C(O)Ror —CHOC(O)R.7. The compound according to claim 6 , wherein Ris alkyl or alkoxy claim 6 , each optionally substituted with 0 claim 6 , 1 claim 6 , or multiple R.8. The compound according to claim 7 , wherein Ris chosen from —CH claim 7 , —CH(CH) claim 7 , —CHOCHCH claim 7 , or —CHCHOCH.9. A composition for the control of a fungal pathogen including at least one of the compounds of and at least one additional compound selected from the group consisting of: a phytologically acceptable carrier material claim 1 , a second fungicide claim 1 , an insecticide claim 1 , a nematocides claim 1 , a miticide claim 1 , an arthropodicide claim 1 , a bactericide.10. The composition for the control of a fungal pathogen according to claim 9 , wherein the at least one additional compound is at least one phytologically acceptable carrier material.11Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformisVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The compositions according to claim 9 , wherein the fungal pathogen is at least one pathogen selected from the group consisting of: Leaf Blotch of Wheat (; anamorph: ) claim 9 , Wheat Brown Rust () claim 9 , Stripe Rust () claim 9 , Scab of Apple () claim 9 , Blister Smut of Maize () claim 9 , Powdery Mildew of Grapevine () claim 9 , Barley Scald () claim 9 , Blast of ...

Подробнее
14-01-2016 дата публикации

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20160007602A1
Принадлежит:

This disclosure relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. The compound according to claim 1 , wherein X and Y are hydrogen.3. The compound according to claim 2 , wherein Ris alkyl or aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.4. The compound according to claim 2 , wherein Ris hydrogen or alkyl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.5. The compound according to claim 1 , wherein X is C(O)Rand Y is hydrogen.6. The compound according to claim 5 , wherein Ris alkyl or aryl claim 5 , each optionally substituted with 0 claim 5 , 1 or multiple R.7. The compound according to claim 5 , wherein Ris hydrogen or alkyl claim 5 , each optionally substituted with 0 claim 5 , 1 or multiple R.8. The compound according to claim 1 , wherein X is hydrogen and Y is Q.9. The compound according to claim 8 , wherein Ris alkyl or aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.10. The compound according to claim 8 , wherein Ris hydrogen or alkyl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.11. The compound according to claim 9 , wherein Ris hydrogen.12. The compound according to claim 9 , wherein Ris —C(O)Ror —CHOC(O)R.13. The compound according to claim 12 , wherein Ris alkyl or alkoxy claim 12 , each optionally substituted with 0 claim 12 , 1 claim 12 , or multiple R.14. The compound according to claim 13 , wherein Ris —CH claim 13 , —CH(CH) claim 13 , —CHOCHCH claim 13 , or —CHCHOCH.15. A composition for the control of a fungal pathogen including at least one of the compounds of Formula I and at least one additional compound selected from the group consisting of: a phytologically acceptable carrier material claim 13 , a second fungicide claim 13 , an insecticide claim 13 , a nematocide claim 13 , a miticide claim 13 , an arthropodicide claim 13 , and a bactericide.16. The composition according to claim 15 , wherein the least one ...

Подробнее
08-02-2018 дата публикации

PICOLINAMIDES WITH FUNGICIDAL ACTIVITY

Номер: US20180037541A1
Принадлежит:

The invention relates to picolinamides of Formula I and their use as fungicides. 2. A composition according to claim 1 , wherein X is hydrogen and Y is Q.3. A composition according to claim 2 , wherein Ris hydrogen.4. A composition according to claim 3 , wherein Ris OCH.5. A composition according to claim 4 , wherein Ris chosen from hydrogen or methyl.6. A composition according to claim 3 , wherein Ris C(O)R claim 3 , or CHOC(O)R.7. (canceled)8. A composition according to claim 6 , wherein Ris chosen from hydrogen or methyl.9. A composition for the control of a fungal pathogen including at least one of the compositions of and a phytologically acceptable carrier material.10. A composition for the control of a fungal pathogen including at least one of the compositions of and a phytologically acceptable carrier material.11. A composition for the control of a fungal pathogen including mixtures of at least one of the compositions of and another pesticide including fungicides claim 5 , insecticides claim 5 , nematocides claim 5 , miticides claim 5 , arthropodicides claim 5 , bactericides and combinations thereof.12. A composition for the control of a fungal pathogen including mixtures of at least one of the compositions of and another pesticide including fungicides claim 8 , insecticides claim 8 , nematocides claim 8 , miticides claim 8 , arthropodicides claim 8 , bactericides and combinations thereof.13Zymoseptoria triticiPuccinia triticinaPuccinia striiformisVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisPyricularia oryzaePhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumColletotrichum lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The composition according to wherein the fungal pathogen is one of Leaf Blotch of Wheat () claim 1 , Wheat Brown Rust () claim 1 , Stripe Rust () claim 1 , Scab of Apple () claim 1 , Blister Smut of Maize () claim 1 , Powdery Mildew of ...

Подробнее
10-03-2022 дата публикации

SYNERGISTIC MIXTURES FOR FUNGAL CONTROLS IN CEREALS

Номер: US20220071212A1
Принадлежит: CORTEVA AGRISCIENCE LLC

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I, (S)-1,1-bis(4-fluorophenyl)propan-2-yl (3-acetoxy-4-methoxypicolinoyl)-L-alaninate, and at least one fungicide selected from the group consisting of epoxiconazole, prothioconazole, azoxystrobin, pyraclostrobin, fluxapyroxad, benzovindiflupyr, and chlorothalonil, provides synergistic control of selected fungi. 2. The mixture of wherein the sterol biosynthesis inhibitor (SBI) is selected from the group consisting of epoxiconazole and prothioconazole.3. The mixture of wherein a concentration ratio of the compound of Formula I to epoxiconazole is about 16:1.4. The mixture of wherein a concentration ratio of the compound of Formula I to prothioconazole is about 1:1.5. The mixture of wherein the respiration inhibitor is selected from the group consisting of azoxystrobin and pyraclostrobin.6. The mixture of wherein a concentration ratio of the compound of Formula I to azoxystrobin is from about 1:1 to about 1:16.7. The mixture of wherein a concentration ratio of the compound of Formula I to pyraclostrobin is from about 26:1 to about 1.6:1.8. The mixture of wherein at least the respiration inhibitor is selected from the group consisting of fluxapyroxad and benzovindiflupyr.9. The mixture of wherein a concentration ratio of the compound of Formula I to fluxapyroxad is from about 26:1 to about 6.5:1.10. The mixture of wherein a concentration ratio of the compound of Formula I to benzovindiflupyr is about 1:1.3.11. The mixture of wherein the multi-site inhibitor is chlorothalonil.12. The mixture of wherein a concentration ratio of the compound of Formula I to chlorothalonil is from about 1:8 to about 1:64.13Rhynchosporium secalis. The mixture of - claim 11 , wherein the mixture provides control of a fungal pathogen claim 11 , and the pathogen is the causal agent of barley scald ().14. A synergistic claim 11 , fungicidal composition comprising of a fungicidally effective amount of ...

Подробнее
01-03-2018 дата публикации

THIOPICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20180055051A1
Принадлежит: DOW AGROSCIENCES LLC

The present disclosure relates to thiopicolinamides of Formula I and their use as fungicides. 2. A compound according to claim 1 , wherein Ris hydrogen.3. A compound according to claim 2 , wherein Ris methyl.4. A compound according to claim 2 , wherein Ris C-Calkyl.5. A compound according to claim 2 , wherein Rand Rindependently aryl claim 2 , each optionally substituted with 0 claim 2 , 1 claim 2 , or multiple R.6. A compound according to claim 2 , wherein Ris methyl claim 2 , Ris C-Calkyl claim 2 , and Rand Rindependently aryl claim 2 , each optionally substituted with 0 claim 2 , 1 claim 2 , or multiple R.7. A compound according to claim 1 , wherein Ris —C(O)R claim 1 , or —CHOC(O)R.8. A compound according to claim 7 , wherein Ris methyl.9. A compound according to claim 7 , wherein Ris C-Calkyl.10. A compound according to claim 7 , wherein Rand Rindependently aryl claim 7 , each optionally substituted with 0 claim 7 , 1 claim 7 , or multiple R.11. A compound according to claim 7 , wherein Ris methyl claim 7 , Ris C-Calkyl claim 7 , and Rand Rindependently aryl claim 7 , each optionally substituted with 0 claim 7 , 1 claim 7 , or multiple R.12. A composition for the control of a fungal pathogen including mixtures of at least one of the compounds of and another pesticide including fungicides claim 1 , insecticides claim 1 , nematocides claim 1 , miticides claim 1 , arthropodicides claim 1 , bactericides claim 1 , and combinations thereof.13. A composition for the control of a fungal pathogen including mixtures of at least one of the compounds of and another pesticide including fungicides claim 2 , insecticides claim 2 , nematocides claim 2 , miticides claim 2 , arthropodicides claim 2 , bactericides claim 2 , and combinations thereof.14. A composition for the control of a fungal pathogen including mixtures of at least one of the compounds of and another pesticide including fungicides claim 7 , insecticides claim 7 , nematocides claim 7 , miticides claim 7 , ...

Подробнее
01-03-2018 дата публикации

THIOPICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20180055052A1
Принадлежит: DOW AGROSCIENCES LLC

This disclosure relates to thiopicolinamides of Formula I and their use as fungicides. 2. The composition according to claim 1 , wherein Ris hydrogen.3. The composition according to claim 2 , wherein Ris methyl claim 2 , Ris C-Calkyl claim 2 , Rand Rindependently aryl claim 2 , each optionally substituted with 0 claim 2 , 1 claim 2 , or multiple R.4. The composition according to claim 1 , wherein Ris is chosen from —C(O)R claim 1 , or —CHOC(O)R.5. The composition according to claim 4 , wherein Ris alkyl claim 4 , optionally substituted with 0 claim 4 , 1 claim 4 , of multiple R.6. The composition according to claim 5 , wherein Ris methyl claim 5 , Ris C-Calkyl claim 5 , Rand Rindependently aryl claim 5 , each optionally substituted with 0 claim 5 , 1 claim 5 , or multiple R.7. The compound according to claim 6 , wherein Ris chosen from —CH claim 6 , —CHOCHCH claim 6 , —CHCHOCH claim 6 , —CH(CH) claim 6 , —CHCHCHCH claim 6 , -cyclopropyl.8Zymoseptoria triticiPuccinia triticinaPuccinia striiformisVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisPyricularia oryzaePhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumColletotrichum lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The composition according to wherein the fungal pathogen is one of Leaf Blotch of Wheat () claim 1 , Wheat Brown Rust () claim 1 , Stripe Rust () claim 1 , Scab of Apple () claim 1 , Blister Smut of Maize () claim 1 , Powdery Mildew of Grapevine () claim 1 , Barley scald () claim 1 , Blast of Rice () claim 1 , Rust of Soybean () claim 1 , Glume Blotch of Wheat () claim 1 , Powdery Mildew of Wheat (f. sp. ) claim 1 , Powdery Mildew of Barley (f. sp. ) claim 1 , Powdery Mildew of Cucurbits () claim 1 , Anthracnose of Cucurbits () claim 1 , Leaf Spot of Beet () claim 1 , Early Blight of Tomato () claim 1 , and Net Blotch of Barley ().9Zymoseptoria triticiPuccinia triticinaVenturia ...

Подробнее
01-03-2018 дата публикации

PICOLINAMIDE N-OXIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20180055053A1
Принадлежит: DOW AGROSCIENCES LLC

This disclosure relates to picolinamide N-oxides of Formula I and their use as fungicides. 2. The composition according to claim 1 , wherein Rand Rare independently hydrogen or C-Calkyl.3. The composition according to claim 2 , wherein Ris C-Calkyl.4. The composition according to claim 2 , wherein Rand Rare independently aryl claim 2 , each optionally substituted with 0 claim 2 , 1 claim 2 , or multiple R.5. The composition according to claim 2 , wherein Ris hydrogen.6. The composition according to claim 2 , wherein Rand Rare independently hydrogen or C-Calkyl claim 2 , Ris C-Calkyl claim 2 , Rand Rare independently aryl claim 2 , each optionally substituted with 0 claim 2 , 1 claim 2 , or multiple Rand Ris hydrogen.7Zymoseptoria triticiPuccinia triticinaPuccinia striiformisVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisPyricularia oryzaePhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graminis ftriticiBlumeria graminis fhordeiErysiphe cichoracearumColletotrichum lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The composition according to wherein the fungal pathogen is one of Leaf Blotch of Wheat () claim 1 , Wheat Brown Rust () claim 1 , Stripe Rust () claim 1 , Scab of Apple () claim 1 , Blister Smut of Maize () claim 1 , Powdery Mildew of Grapevine () claim 1 , Barley scald () claim 1 , Blast of Rice () claim 1 , Rust of Soybean () claim 1 , Glume Blotch of Wheat () claim 1 , Powdery Mildew of Wheat (. sp. ) claim 1 , Powdery Mildew of Barley (. sp. ) claim 1 , Powdery Mildew of Cucurbits () claim 1 , Anthracnose of Cucurbits () claim 1 , Leaf Spot of Beet () claim 1 , Early Blight of Tomato () claim 1 , and Net Blotch of Barley ().8Zymoseptoria triticiPuccinia triticinaVenturia inaequalisRhynchosporium secalisPyricularia oryzaePhakopsora pachyrhiziLeptosphaeria nodorumColletotrichum lagenariumCercospora beticolaAlternaria solani. The compostion according to wherein the fungal pathogen is one of Leaf Blotch of Wheat () ...

Подробнее
01-03-2018 дата публикации

PYRIDO-1,3-OXAZINE-2,4-DIONE COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20180055056A1
Принадлежит: DOW AGROSCIENCES LLC

This disclosure relates to pyrido-1,3-oxazine-2,4-diones of Formula I and their use as fungicides. 2. The composition according to claim 1 , wherein Rand Rare independently hydrogen or C-Calkyl.3. The composition according to claim 2 , wherein Ris C-Calkyl.4. The composition according to claim 2 , wherein Rand Rare independently aryl claim 2 , each optionally substituted with 0 claim 2 , 1 claim 2 , or multiple R.5. The composition according to claim 2 , wherein Ris hydrogen.6. The composition according to claim 2 , wherein Rand Rare independently hydrogen or C-Calkyl claim 2 , Ris C-Calkyl claim 2 , and Rand Rare independently aryl claim 2 , each optionally substituted with 0 claim 2 , 1 claim 2 , or multiple R claim 2 , and Ris hydrogen.7Zymoseptoria triticiPuccinia triticinaPuccinia striiformisVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisPyricularia oryzaePhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumColletotrichum lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The composition according to wherein the fungal pathogen is one of Leaf Blotch of Wheat () claim 1 , Wheat Brown Rust () claim 1 , Stripe Rust () claim 1 , Scab of Apple () claim 1 , Blister Smut of Maize () claim 1 , Powdery Mildew of Grapevine () claim 1 , Barley scald () claim 1 , Blast of Rice () claim 1 , Rust of Soybean () claim 1 , Glume Blotch of Wheat () claim 1 , Powdery Mildew of Wheat (f. sp. ) claim 1 , Powdery Mildew of Barley (f. sp. ) claim 1 , Powdery Mildew of Cucurbits () claim 1 , Anthracnose of Cucurbits () claim 1 , Leaf Spot of Beet () claim 1 , Early Blight of Tomato () claim 1 , and Net Blotch of Barley ().8Zymoseptoria triticiPuccinia triticinaVenturia inaequalisRhynchosporium secalisPyricularia oryzaePhakopsora pachyrhiziLeptosphaeria nodorumColletotrichum lagenariumCercospora beticolaAlternaria solani. The composition according to wherein the fungal pathogen is one of ...

Подробнее
02-03-2017 дата публикации

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20170055528A1
Принадлежит:

This disclosure relates to macrocyclic picolinamides of Formula (I) and their use as fungicides. 2. A compound according to claim 1 , wherein X and Y are hydrogen.3. A compound according to claim 2 , wherein Ris chosen from alkyl or aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.4. A compound according to claim 2 , wherein Ris chosen from alkyl or aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.5. A compound according to claim 1 , wherein X is C(O)Rand Y is hydrogen.6. A compound according to claim 5 , wherein Ris chosen from alkyl or aryl claim 5 , each optionally substituted with 0 claim 5 , 1 or multiple R.7. A compound according to claim 5 , wherein Ris chosen from alkyl or aryl claim 5 , each optionally substituted with 0 claim 5 , 1 or multiple R.8. A compound according to claim 1 , wherein Xis hydrogen and Y is Q.9. A compound according to claim 8 , wherein Ris chosen from alkyl or aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.10. A compound according to claim 8 , wherein Ris chosen from alkyl or aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.11. A compound according to claim 9 , wherein Ris hydrogen.12. A compound according to claim 9 , wherein Ris —C(O)Ror —CHOC(O)R.13. A compound according to claim 12 , wherein Ris chosen from alkyl or alkoxy claim 12 , each optionally substituted with 0 claim 12 , 1 claim 12 , or multiple R.14. A compound according to claim 13 , wherein Ris chosen from —CH claim 13 , —CH(CH) claim 13 , —CHOCHCH claim 13 , or —CHCHOCH.15. A composition for the control of a fungal pathogen including at least one of the compounds of and a phytologically acceptable carrier material.16. A composition for the control of a fungal pathogen including mixtures of at least one of the compounds of with other pesticides including fungicides claim 1 , insecticides claim 1 , nematocides claim 1 , miticides claim 1 , arthropodicides claim 1 ...

Подробнее
04-03-2021 дата публикации

Synergistic Fungicidal Mixtures and Compositions Comprising 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1H)-One for Fungal Control (SDHI)

Номер: US20210059252A1
Принадлежит: ADAMA MAKHTESHIM LTD.

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of fluxapyroxad claim 1 , benzovindiflupyr claim 1 , penthiopyrad claim 1 , isopyrazam claim 1 , boscalid claim 1 , and fluopyram.3. The mixture of in which the concentration ratio of the Compound of Formula I to fluxapyroxad is between about 4.4:1 and about 6.3:1.4. The mixture of in which the concentration ratio of the Compound of Formula I to benzovindiflupyr is between about 1:3 and about 7.9:1.5. The mixture of in which the concentration ratio of the Compound of Formula I to penthiopyrad is between about 1:4.3 and about 1:1.9.6. The mixture of in which the concentration ratio of the Compound of Formula I to isopyrazam is between about 1:1.3 and about 1:1.7. The mixture of in which the concentration ratio of the Compound of Formula I to boscalid is between about 1:13.2 and about 1:1.3.8. The mixture of in which the concentration ratio of the Compound of Formula I to fluopyram is between about 1:27.6 and about 1:3.6.9Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is one of Leaf Blotch of Wheat (; anamorph: ) claim 2 , Wheat Brown Rust () claim 2 , Stripe Rust (f. sp. ) claim 2 , Scab of Apple () claim 2 , Blister Smut of Maize () claim 2 , Powdery Mildew of Grapevine () claim 2 , Barley scald () claim 2 , Blast of Rice () claim 2 , Rust of Soybean () claim 2 , Glume Blotch of Wheat () claim 2 , Powdery Mildew of Wheat (f. sp. ) claim 2 , Powdery ...

Подробнее
04-03-2021 дата публикации

Synergistic Fungicidal Mixtures and Compositions Comprising 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1H)-One for Fungal Control (MSI)

Номер: US20210059253A1
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of chlorothalonil and mancozeb.3. The mixture of in which the concentration ratio of the Compound of Formula I to chlorothalonil is about 1:219.4. The mixture of in which the concentration ratio of the Compound of Formula I to mancozeb is about 1:272.5Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is one of Leaf Blotch of Wheat (; anamorph: ) claim 2 , Wheat Brown Rust () claim 2 , Stripe Rust (f. sp. ) claim 2 , Scab of Apple () claim 2 , Blister Smut of Maize () claim 2 , Powdery Mildew of Grapevine () claim 2 , Barley scald () claim 2 , Blast of Rice () claim 2 , Rust of Soybean () claim 2 , Glume Blotch of Wheat () claim 2 , Powdery Mildew of Wheat (f. sp. ) claim 2 , Powdery Mildew of Barley (f. sp. ) claim 2 , Powdery Mildew of Cucurbits () claim 2 , Anthracnose of Cucurbits () claim 2 , Leaf Spot of Beet () claim 2 , Early Blight of Tomato () claim 2 , and Net Blotch of Barley ().6Mycosphaerella graminicolaSeptoria tritici. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is Leaf Blotch of Wheat (; anamorph: ).7Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe ...

Подробнее
01-03-2018 дата публикации

PICOLINAMIDES AS FUNGICIDES

Номер: US20180057460A1
Принадлежит: DOW AGROSCIENCES LLC

This disclosure relates to picolinamides of Formula I and their use as fungicides. 2. A compound according to claim 1 , wherein X and Y are hydrogen.3. A compound according to claim 2 , wherein Rand Rare independently hydrogen or alkyl.4. A compound according to claim 2 , wherein Rand Rare independently hydrogen or methyl.5. A compound according to claim 2 , wherein Ris aryl claim 2 , optionally substituted with 0 claim 2 , 1 or multiple R.6. A compound according to claim 2 , wherein Ris alkyl claim 2 , aryl claim 2 , or heteroaryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.7. A compound according to claim 2 , wherein Rand Rare independently hydrogen or alkyl claim 2 , Rand Rare independently chosen from hydrogen or methyl claim 2 , Ris aryl claim 2 , optionally substituted with 0 claim 2 , 1 or multiple R claim 2 , and Ris chosen from alkyl claim 2 , aryl claim 2 , or heteroaryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.8. A compound according to claim 1 , wherein X is C(O)Rand Y is hydrogen.9. A compound according to claim 8 , wherein Rand Rare independently hydrogen or alkyl.10. A compound according to claim 8 , wherein Rand Rare independently hydrogen or methyl.11. A compound according to claim 8 , wherein Ris aryl claim 8 , optionally substituted with 0 claim 8 , 1 or multiple R;12. A compound according to claim 8 , wherein Ris alkyl claim 8 , aryl claim 8 , or heteroaryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.13. A compound according to claim 8 , wherein Rand Rare independently hydrogen or alkyl claim 8 , Rand Rare independently chosen from hydrogen or methyl claim 8 , Ris aryl claim 8 , optionally substituted with 0 claim 8 , 1 or multiple R claim 8 , and Ris chosen from alkyl claim 8 , aryl claim 8 , or heteroaryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.14. A compound according to claim 1 , wherein X is hydrogen and Y is Q.15. A compound ...

Подробнее
01-03-2018 дата публикации

PICOLINAMIDES AS FUNGICIDES

Номер: US20180057461A1
Принадлежит: DOW AGROSCIENCES LLC

This disclosure relates to picolinamides of Formula I and their use as fungicides. 2. A composition according to claim 1 , wherein X is hydrogen and Y is Q.3. A composition according to claim 2 , wherein Ris alkoxy.4. A composition according to claim 3 , wherein W is O claim 3 , or S.5. A composition according to claim 4 , wherein Ris hydrogen.6. A composition according to claim 5 , wherein Rand Rare independently hydrogen or alkyl.7. A composition according to claim 5 , wherein Rand Rare independently hydrogen or methyl.8. A composition according to claim 5 , wherein Ris aryl claim 5 , optionally substituted with 0 claim 5 , 1 or multiple R;9. A composition according to claim 5 , wherein Ris alkyl claim 5 , aryl claim 5 , or heteroaryl claim 5 , each optionally substituted with 0 claim 5 , 1 or multiple R.10. A composition according to claim 5 , wherein Rand Rare independently hydrogen or alkyl claim 5 , Rand Rare independently hydrogen or methyl claim 5 , Ris aryl claim 5 , optionally substituted with 0 claim 5 , 1 or multiple R; and Ris alkyl claim 5 , aryl claim 5 , or heteroaryl claim 5 , each optionally substituted with 0 claim 5 , 1 or multiple R.11. A composition according to claim 4 , wherein Ris —C(O)R claim 4 , or —CHOC(O)R.12. A composition according to claim 11 , wherein Ris alkyl claim 11 , optionally substituted with 0 claim 11 , 1 or multiple R.13. A composition according to claim 12 , wherein Rand Rare independently hydrogen or alkyl.14. A composition according to claim 12 , wherein Rand Rare independently hydrogen or methyl.15. A composition according to claim 12 , wherein Ris aryl claim 12 , optionally substituted with 0 claim 12 , 1 or multiple R;16. A composition according to claim 12 , wherein Ris alkyl claim 12 , aryl claim 12 , or heteroaryl claim 12 , each optionally substituted with 0 claim 12 , 1 or multiple R.17. A composition according to claim 12 , wherein Rand Rare independently hydrogen or alkyl claim 12 , Rand Rare independently ...

Подробнее
01-03-2018 дата публикации

Picolinamide n-oxide compounds with fungicidal activity

Номер: US20180057463A1
Принадлежит: DOW AGROSCIENCES LLC

This disclosure relates to picolinamide N-oxides of Formula I and their use as fungicides.

Подробнее
01-03-2018 дата публикации

PYRIDO-1,3-OXAZINE-2,4-DIONE COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20180057508A1
Принадлежит: DOW AGROSCIENCES LLC

This disclosure relates to pyrido-1,3-oxazine-2,4-diones of Formula I and their use as fungicides. 2. A compound according to claim 1 , wherein Rand Rare independently hydrogen or C-Calkyl.3. A compound according to claim 2 , wherein Ris C-Calkyl.4. A compound according to claim 2 , wherein Rand Rare independently aryl claim 2 , each optionally substituted with 0 claim 2 , 1 claim 2 , or multiple R.5. A compound according to claim 2 , wherein Ris hydrogen.6. A compound according to claim 2 , wherein Rand Rare independently hydrogen or C-Calkyl claim 2 , Ris C-Calkyl claim 2 , and Rand Rare independently aryl claim 2 , each optionally substituted with 0 claim 2 , 1 claim 2 , or multiple R claim 2 , and Ris hydrogen.7. A composition for the control of a fungal pathogen including mixtures of at least one of the compounds of and another pesticide including fungicides claim 1 , insecticides claim 1 , nematocides claim 1 , miticides claim 1 , arthropodicides claim 1 , bactericides claim 1 , and combinations thereof.8. A composition for the control of a fungal pathogen including mixtures of at least one of the compounds of and another pesticide including fungicides claim 6 , insecticides claim 6 , nematocides claim 6 , miticides claim 6 , arthropodicides claim 6 , bactericides claim 6 , and combinations thereof.9. A method for the control and prevention of fungal attack on a plant claim 6 , the method including the step of:{'claim-ref': [{'@idref': 'CLM-00001', 'claims 1'}, {'@idref': 'CLM-00006', '6'}], 'Applying a fungicidally effective amount of at least one of the compounds of any of - to at least one of the plant, an area adjacent to the plant, soil adapted to support growth of the plant, a root of the plant, and foliage of the plant.'}10. A method for the control and prevention of fungal attack on a plant claim 6 , the method including the step of:{'claim-ref': [{'@idref': 'CLM-00007', 'claims 7'}, {'@idref': 'CLM-00008', '8'}], 'Applying a fungicidally effective ...

Подробнее
05-03-2015 дата публикации

SYNERGISTIC FUNGICIDAL MEXURES FOR FUNGAL CONTROL IN CEREALS

Номер: US20150065529A1
Автор: JR. W. John, Owen, Yao Chenglin
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of a compound of Formula I-V and at least one fungicide selected from the group consisting of epoxiconazole, prothioconazole, azoxystrobin, pyraclostrobin, penthiopyrad, isopyrazam, bixafen, boscalid, prochloraz, and chlorothalonil provides synergistic control of selected fungi. 2. The mixture of in which the weight ratio of Compound I-V to epoxiconazole is between about 1:10 and about 10:1.3. The mixture of in which the weight ratio of Compound I-V to prothioconazole is between about 1:10 and about 10:1.4. The mixture of in which the weight ratio of Compound I-V to azoxystrobin is between about 1:10 and about 10:1.5. The mixture of in which the weight ratio of Compound I-V to pyraclostrobin is between about 1:10 and about 10:1.6. The mixture of in which the weight ratio of Compound I-V to penthiopyrad is between about 1:10 and about 10:1.7. The mixture of in which the weight ratio of Compound I to isopyrazam is between about 1:10 and about 10:1.8. The mixture of in which the weight ratio of Compound I to bixafen is between about 1:10 and about 10:1.9. The mixture of in which the weight ratio of Compound I-V to boscalid is between about 1:10 and about 10:1.10. The mixture of in which the weight ratio of Compound I-V to prochloraz is between about 1:10 and about 10:1.11. The mixture of in which the weight ratio of Compound I-V to chlorothalonil is between about 1:50 and about 1:1.12. A fungicidal composition comprising a fungicidally effective amount of the fungicidal mixture of and an agriculturally acceptable adjuvant or carrier. This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/249,479, filed Oct. 7, 2009, which is expressly incorporated by reference herein.This invention concerns a synergistic fungicidal composition containing (a) a compound of Formula I, II, III, IV or V and (b) at least one fungicide selected from the group consisting of epoxiconazole, ...

Подробнее
28-02-2019 дата публикации

USE OF PICOLINAMIDE COMPOUNDS AS FUNGICIDES

Номер: US20190059383A1
Принадлежит:

This disclosure relates to picolinamides of Formula I and their use as fungicides. 2. The composition according to claim 1 , wherein X is hydrogen and Y is Q.3. (canceled)4. The composition according to claim 2 , wherein Ris alkoxy.5. The composition according to claim 4 , wherein Ris hydrogen.6. The composition according to claim 5 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 5 , Rand Rare independently aryl claim 5 , each optionally substituted with 0 claim 5 , 1 or multiple R claim 5 , and Ris H.7. The composition according to claim 4 , wherein Ris chosen from —C(O)R claim 4 , or —CHOC(O)R.8. The composition according to claim 7 , wherein Ris alkyl claim 7 , optionally substituted with 0 claim 7 , 1 or multiple R.9. The composition according to claim 8 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 8 , Rand Rare independently aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R claim 8 , and Ris H.10. The composition according to claim 9 , wherein Ris chosen from —CH claim 9 , —CHOCHCH claim 9 , —CHCHOCH claim 9 , —CH(CH) claim 9 , —CHCHCHCH claim 9 , -cyclopropyl.11Zymoseptoria triticiPuccinia triticinaPuccinia striiformisVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisPyricularia oryzaePhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graminis f.triticiBlumeria graminis f.hordeiErysiphe cichoracearumColletotrichum lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The composition according to wherein the fungal pathogen is one of Leaf Blotch of Wheat () claim 1 , Wheat Brown Rust () claim 1 , Stripe Rust () claim 1 , Scab of Apple () claim 1 , Blister Smut of Maize () claim 1 , Powdery Mildew of Grapevine () claim 1 , Barley scald () claim 1 , Blast of Rice () claim 1 , Rust of Soybean () claim 1 , Glume Blotch of Wheat () claim 1 , Powdery Mildew of Wheat (sp. ) claim 1 , Powdery Mildew of Barley (sp. ) claim 1 , Powdery Mildew of Cucurbits () claim 1 ...

Подробнее
12-03-2020 дата публикации

Use of an Acyclic Picolinamide Compound as a Fungicide for Control of Phytopathogenic Fungi in Row Crops

Номер: US20200077656A1
Принадлежит: DOW AGROSCIENCES LLC

The present disclosure is related to the field of agrochemicals, including compound I and its use to control fungal diseases in agriculturally useful row crops. 3. The method of claim 1 , wherein the composition further includes at least one additional agriculturally active ingredient selected from the group consisting of: an insecticide claim 1 , an herbicide claim 1 , and a fungicide.4Puccinia polysoraCercospora zeaemaydisMagnaporthe griseaCercosporaCercospora beticolaPyrenophora teresBlumeria graministriticiRamulariaRamularia collocygniBlumeria graministriticiSclerotium rolfsiiCercospora arachidicolaCercosporidium personatumCercospora sojina. The method of claim 1 , wherein the fungal pathogen is selected from the group consisting of the causal agents of: brown rust of corn () claim 1 , grey leaf spot of corn (-) claim 1 , rice panicle blast () claim 1 , leaf spot of sugar beet () claim 1 , net blotch of barley () claim 1 , powdery mildew of barley (f. sp. ) claim 1 , leaf spot of barley (-) claim 1 , powdery mildew of wheat (f. sp. ) claim 1 , white mold of peanut () claim 1 , early leaf spot of peanut () claim 1 , late leaf spot of peanut () claim 1 , and frogeye leaf spot of soybean ().5. The method of claim 2 , wherein the composition further includes at least one additional agriculturally active ingredient selected from the group consisting of: an insecticide claim 2 , an herbicide claim 2 , and a fungicide.6Puccinia polysoraCercospora zeaemaydisMagnaporthe griseaCercosporaCercospora beticolaPyrenophora teresBlumeria graministriticiRamulariaRamularia collocygniBlumeria graministriticiSclerotium rolfsiiCercospora arachidicolaCercosporidium personatumCercospora sojina. The method of claim 2 , wherein the fungal pathogen is selected from the group consisting of the causal agents of: brown rust of corn () claim 2 , grey leaf spot of corn (-) claim 2 , rice panicle blast () claim 2 , leaf spot of sugar beet () claim 2 , net blotch of barley () claim 2 , powdery ...

Подробнее
12-03-2020 дата публикации

Synergistic Mixtures for Fungal Control in Cereals

Номер: US20200077657A1
Принадлежит: DOW AGROSCIENCES LLC

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I, (S)-1,1-bis(4-fluorophenyl)propan-2-yl (3-acetoxy-4-methoxypicolinoyl)-L-alaninate, and at least one fungicide selected from the group consisting of tebuconazole, prothioconazole, difenconazole, epoxiconazole, mefentrifluconazole, benzovindiflupyr, penthiopyrad, fluxapyroxad, bixafen, fluopyram, picoxystrobin, pyraclostrobin, azoxystrobin, mancozeb and chlorothalonil, provides synergistic control of selected fungi. 2. The mixture of wherein the sterol biosynthesis inhibitor is selected from the group consisting of tebuconazole claim 1 , prothioconazole claim 1 , difenoconazole claim 1 , epoxiconazole claim 1 , and mefentrifluconazole.3. The mixture of wherein a concentration ratio of the compound of Formula I to tebuconazole is from about 2:1 to about 1:4.4. The mixture of wherein a concentration ratio of the compound of Formula I to prothioconazole is from about 1:6.4 to about 1:52.5. The mixture of wherein a concentration ratio of the compound of Formula I to difenoconazole is from about 2:1 to about 1:2.6. The mixture of wherein a concentration ratio of the compound of Formula I to epoxiconazole is from about 4:1 to about 1:2.7. The mixture of wherein a concentration ratio of the compound of Formula I to mefentrifluconazole is from about 4:1 to about 1:2.8. The mixture of wherein respiration inhibitor is selected from the group consisting of benzovindiflupyr claim 1 , penthiopyrad claim 1 , fluxapyroxad claim 1 , bixafen claim 1 , and fluopyram.9. The mixture of wherein a concentration ratio of the compound of Formula I to benzovindiflupyr is from about 1:1.2 to about 1:5.10. The mixture of wherein a concentration ratio of the compound of Formula I to penthiopyrad is from about 1:10 to about 1:160.11. The mixture of wherein a concentration ratio of the compound of Formula I to fluxapyroxad is from about 1:2.5 to about 1:40.12. The mixture of wherein a concentration ...

Подробнее
02-04-2015 дата публикации

USE OF MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20150094281A1
Принадлежит:

The invention relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. The method according to claim 1 , wherein X and Y are independently chosen from H claim 1 , C(O)R claim 1 , or CHOR.3. The method according to claim 2 , wherein Ris chosen from H claim 2 , alkyl claim 2 , alkenyl claim 2 , aryl claim 2 , —Si(R) claim 2 , or —C(O)R claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.4. The method according to claim 3 , wherein Ris chosen from CHR claim 3 , aryl claim 3 , alkyl claim 3 , or alkenyl claim 3 , each optionally substituted with 0 claim 3 , 1 claim 3 , or multiple R.5. The method according to claim 4 , wherein Ris chosen from H claim 4 , alkyl claim 4 , alkenyl claim 4 , aryl claim 4 , or heteroaryl claim 4 , each optionally substituted with 0 claim 4 , 1 claim 4 , or multiple R.6. The method according to claim 1 , wherein X is H and Y is Q.7. The method according to claim 6 , wherein Ris chosen from H claim 6 , alkyl claim 6 , alkenyl claim 6 , aryl claim 6 , —Si(R) claim 6 , or —C(O)R claim 6 , each optionally substituted with 0 claim 6 , 1 or multiple R.8. The method according to claim 7 , wherein Ris chosen from CHR claim 7 , aryl claim 7 , alkyl claim 7 , or alkenyl claim 7 , each optionally substituted with 0 claim 7 , 1 claim 7 , or multiple R.9. The method according to claim 8 , wherein Ris chosen from H claim 8 , alkyl claim 8 , alkenyl claim 8 , aryl claim 8 , or heteroaryl claim 8 , each optionally substituted with 0 claim 8 , 1 claim 8 , or multiple R.10. The method according to claim 9 , wherein Ris H claim 9 , —C(O)Ror —CHOC(O)R.11. The method according to claim 10 , wherein Ris chosen from —C(O)Ror —CHOC(O)R.12. The method according to claim 11 , wherein Ris chosen from alkyl or alkoxy claim 11 , each optionally substituted with 0 claim 11 , 1 claim 11 , or multiple R.13. The method according to wherein:at least one compound of said Formula I is applied in combination with a phytologically ...

Подробнее
02-04-2015 дата публикации

MACROCYCLIC PICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20150094339A1
Принадлежит:

The invention relates to compounds of macrocyclic picolinamides of Formula I suitable to control or prevent growth of fungi. 2. The compound according to claim 1 , wherein X and Y are independently chosen from H or C(O)R.3. The compound according to claim 2 , wherein Ris chosen from H claim 2 , alkyl claim 2 , alkenyl claim 2 , aryl claim 2 , —Si(R) claim 2 , or —C(O)R claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.4. The compound according to claim 3 , wherein Ris chosen from H claim 3 , alkyl claim 3 , aryl claim 3 , heteroaryl claim 3 , or arylalkyl claim 3 , each optionally substituted with 0 claim 3 , 1 or multiple R.5. The compound according to claim 1 , wherein X is H and Y is Q.6. The compound according to claim 5 , wherein Ris chosen from H claim 5 , alkyl claim 5 , alkenyl claim 5 , aryl claim 5 , —Si(R) claim 5 , or —C(O)R claim 5 , each optionally substituted with 0 claim 5 , 1 or multiple R.7. The compound according to claim 6 , wherein Ris chosen from H claim 6 , alkyl claim 6 , aryl claim 6 , heteroaryl claim 6 , or arylalkyl claim 6 , each optionally substituted with 0 claim 6 , 1 or multiple R.8. The compound according to claim 7 , wherein Ris H claim 7 , —C(O)R claim 7 , or —CHOC(O)R.9. The compound according to claim 8 , wherein Ris alkyl or alkoxy claim 8 , each optionally substituted with 0 claim 8 , 1 claim 8 , or multiple R.10. A formulation for the control of a fungal pathogen claim 8 , comprising:{'claim-ref': {'@idref': 'CLM-00001', 'claim 1'}, 'at least one of the compounds of ; and'}a phytologically acceptable carrier material.11. The formulation according to claim 10 , wherein the formulation is suitable for treating plants.12. A formulation for the control of a fungal pathogen claim 10 , comprising:{'claim-ref': {'@idref': 'CLM-00001', 'claim 1'}, 'at least one of the compounds of ; and'}at least one agriculturally active ingredient selected from the group consisting of: fungicides, insecticides, nematocides, ...

Подробнее
02-04-2015 дата публикации

Use of macrocyclic picolinamides as fungicides

Номер: US20150094340A1
Принадлежит: DOW AGROSCIENCES LLC

The invention relates to macrocyclic picolinamides of Formula I and their use as fungicides.

Подробнее
02-04-2015 дата публикации

MACROCYCLIC PICOLINAMIDES COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20150094341A1
Принадлежит:

The invention relates to compounds of macrocyclic picolinamides of Formula I suitable to control or prevent growth of fungi. 2. The compound according to claim 1 , wherein X and Y are independently chosen from H claim 1 , C(O)R claim 1 , or CHOR.3. The compound according to claim 2 , wherein Ris chosen from H claim 2 , alkyl claim 2 , alkenyl claim 2 , aryl claim 2 , —Si(R) claim 2 , or —C(O)R claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.4. The compound according to claim 3 , wherein Ris chosen from CHR claim 3 , aryl claim 3 , alkyl claim 3 , or alkenyl claim 3 , each optionally substituted with 0 claim 3 , 1 claim 3 , or multiple R.5. The compound according to claim 4 , wherein Ris chosen from H claim 4 , alkyl claim 4 , alkenyl claim 4 , aryl claim 4 , or heteroaryl claim 4 , each optionally substituted with 0 claim 4 , 1 claim 4 , or multiple R.6. The compound according to claim 1 , wherein X is H and Y is Q.7. The compound according to claim 6 , wherein Ris chosen from H claim 6 , alkyl claim 6 , alkenyl claim 6 , aryl claim 6 , —Si(R) claim 6 , or —C(O)R claim 6 , each optionally substituted with 0 claim 6 , 1 or multiple R.8. The compound according to claim 7 , wherein Ris chosen from CHR claim 7 , aryl claim 7 , alkyl claim 7 , or alkenyl claim 7 , each optionally substituted with 0 claim 7 , 1 claim 7 , or multiple R.9. The compound according to claim 8 , wherein Ris chosen from H claim 8 , alkyl claim 8 , alkenyl claim 8 , aryl claim 8 , or heteroaryl claim 8 , each optionally substituted with 0 claim 8 , 1 claim 8 , or multiple R.10. The compound according to claim 9 , wherein Ris H claim 9 , —C(O)Ror —CHOC(O)R.11. The compound according to claim 10 , wherein Ris chosen from —C(O)Ror —CHOC(O)R.12. The compound according to claim 11 , wherein Ris chosen from alkyl or alkoxy claim 11 , each optionally substituted with 0 claim 11 , 1 claim 11 , or multiple R.13. A formulation for the control of a fungal pathogen claim 11 , ...

Подробнее
19-03-2020 дата публикации

Use of an Acyclic Picolinamide Compound as a Fungicide for Control of Phytopathogenic Fungi in Vegetables

Номер: US20200085047A1
Принадлежит: DOW AGROSCIENCES LLC

The present disclosure is related to the field of agrochemicals, including compound I and its use to control fungal diseases in agriculturally useful vegetable crops. 3. The method of claim 1 , wherein the composition further includes at least one additional agriculturally active ingredient selected from the group consisting of: an insecticide claim 1 , an herbicide claim 1 , and a fungicide.4Alternaria brassicicolaSclerotiniaSclerotinia sclerotiorumColletotrichum capsiciErysiphe cichoracearumAlternaria solaniMycovellosiella fulvaStagonosporopsis cucurbitacearumBotrytis cinereaCorynespora cassiicolaColletotrichum coccodes. The method of claim 1 , wherein the fungal pathogen is selected from the group consisting of the causal agents of: black leaf spot of cabbage () claim 1 , rot of lettuce () claim 1 , anthracnose of hot pepper () claim 1 , powdery mildew of cucumber () claim 1 , early blight of tomato () claim 1 , leaf mold of tomato () claim 1 , gummy stem blight of watermelon () claim 1 , gray mold of broad bean () claim 1 , target spot of tomato () claim 1 , and anthracnose of tomato ().5. The method of claim 2 , wherein the composition further includes at least one additional agriculturally active ingredient selected from the group consisting of: an insecticide claim 2 , an herbicide claim 2 , and a fungicide.6Alternaria brassicicolaSclerotiniaSclerotinia sclerotiorumColletotrichum capsiciErysiphe cichoracearumAlternaria solaniMycovellosiella fulvaStagonosporopsis cucurbitacearumBotrytis cinereaCorynespora cassiicolaColletotrichum coccodes. The method of claim 2 , wherein the fungal pathogen is selected from the group consisting of the causal agents of: black leaf spot of cabbage () claim 2 , rot of lettuce () claim 2 , anthracnose of hot pepper () claim 2 , powdery mildew of cucumber () claim 2 , early blight of tomato () claim 2 , leaf mold of tomato () claim 2 , gummy stem blight of watermelon () claim 2 , gray mold of broad bean () claim 2 , target spot of ...

Подробнее
19-03-2020 дата публикации

Synergistic Mixtures for Fungal Controls in Cereals

Номер: US20200085048A1
Принадлежит: DOW AGROSCIENCES LLC

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I, (S)-1,1-bis(4-fluorophenyl)propan-2-yl (3-acetoxy-4-methoxypicolinoyl)-L-alaninate, and at least one fungicide selected from the group consisting of epoxiconazole, prothioconazole, azoxystrobin, pyraclostrobin, fluxapyroxad, benzovindiflupyr, and chlorothalonil, provides synergistic control of selected fungi. 2. The mixture of wherein the sterol biosynthesis inhibitor (SBI) is selected from the group consisting of epoxiconazole and prothioconazole.3. The mixture of wherein a concentration ratio of the compound of Formula I to epoxiconazole is about 16:1.4. The mixture of wherein a concentration ratio of the compound of Formula I to prothioconazole is about 1:1.5. The mixture of wherein the respiration inhibitor is selected from the group consisting of azoxystrobin and pyraclostrobin.6. The mixture of wherein a concentration ratio of the compound of Formula I to azoxystrobin is from about 1:1 to about 1:16.7. The mixture of wherein a concentration ratio of the compound of Formula I to pyraclostrobin is from about 26:1 to about 1.6:1.8. The mixture of wherein at least the respiration inhibitor is selected from the group consisting of fluxapyroxad and benzovindiflupyr.9. The mixture of wherein a concentration ratio of the compound of Formula I to fluxapyroxad is from about 26:1 to about 6.5:1.10. The mixture of wherein a concentration ratio of the compound of Formula I to benzovindiflupyr is about 1:1.3.11. The mixture of wherein the multi-site inhibitor is chlorothalonil.12. The mixture of wherein a concentration ratio of the compound of Formula I to chlorothalonil is from about 1:8 to about 1:64.13Rhynchosporium secalis. The mixture of - claim 11 , wherein the mixture provides control of a fungal pathogen claim 11 , and the pathogen is the causal agent of barley scald ().14. A synergistic claim 11 , fungicidal composition comprising of a fungicidally effective amount of ...

Подробнее
19-03-2020 дата публикации

Synergistic Mixtures for Fungal Control in Vegetables

Номер: US20200085049A1
Принадлежит: DOW AGROSCIENCES LLC

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I, (S)-1,1-bis(4-fluorophenyl)propan-2-yl (3-acetoxy-4-methoxypicolinoyl)-L-alaninate, and at least one fungicide selected from the group consisting of epoxiconazole, prothioconazole, difenoconazole, azoxystrobin, pyraclostrobin, picoxoystrobin, fluxapyroxad, benzovindiflupyr, penthiopyrad, bixafen, chlorothalonil, and mancozeb provides synergistic control of selected fungi. 2. The mixture of wherein the sterol biosynthesis inhibitor is selected from the group consisting of epoxiconazole claim 1 , prothioconazole and difenoconazole.3. The mixture of wherein a concentration ratio of the compound of Formula I to epoxiconazole is from about 10:1 to about 1:1.6.4. The mixture of wherein a concentration ratio of the compound of Formula I to prothioconazole is from about 10:1 to about 1.3:1.5. The mixture of wherein a concentration ratio of the compound of Formula I to difenoconazole is from about 5:1 to about 1:1.6.6. The mixture of wherein the respiration inhibitor is selected from the group consisting of azoxystrobin claim 1 , pyraclostrobin and picoxystrobin.7. The mixture of wherein a concentration ratio of the compound of Formula I to azoxystrobin is from about 50:1 to about 3.1:1.8. The mixture of wherein a concentration ratio of the compound of Formula I to pyraclostrobin is from about 50:1 to about 3.1:1.9. The mixture of wherein a concentration ratio of the compound of Formula I to picoxystrobin is from about 10:1 to about 1:1.6.10. The mixture of wherein the respiration inhibitor is selected from the group consisting of fluxapyroxad claim 1 , benzovindiflupyr claim 1 , penthiopyrad and bixafen.11. The mixture of wherein a concentration ratio of the compound of Formula I to fluxapyroxad is from about 50:1 to about 3.1:1.12. The mixture of wherein a concentration ratio of the compound of Formula I to benzovindiflupyr is from about 10:1 to about 1:1.6.13. The mixture of ...

Подробнее
19-03-2020 дата публикации

Acyclic Picolinamides as a Seed Treatment

Номер: US20200085050A1
Принадлежит: DOW AGROSCIENCES LLC

The present disclosure relates to the use of the compound of Formula I, (S)-1,1-bis(4-fluorophenyl)propan-2-yl (3-acetoxy-4-methoxypicolinoyl)-L-alaninate, as a seed treatment to prevent or control plant diseases. 2. The method of claim 1 , wherein the compound of Formula I is applied at a rate from about 0.5 to about 500 grams per 100 kilograms of seed.3Triticum. The method of claim 1 , wherein the seed being treated is a wheat seed (spp.; TRZSS).4Zymoseptoria triticiParastagonospora nodorumPuccinia triticinaBlumeria graministritici. The method of claim 1 , wherein the fungal pathogen is selected from the group consisting of the causal agent of wheat leaf blotch () claim 1 , wheat glume blotch () claim 1 , wheat brown rust () claim 1 , and wheat powdery mildew (f. sp. ).5Hordeum vulgare. The method of claim 1 , wherein the seed being treated is a barley seed (; HORVS).6Blumeria graminishordeiRhynchosporium secalis. The method of claim 1 , wherein the fungal pathogen is selected from the group consisting of the causal agent of barley powdery mildew (f. sp. ) claim 1 , and barley scald ().7Cucumis. The method of claim 1 , wherein the seed being treated is a cucurbit seed (spp.; CUMSS).8Erysiphe cichoracearumPodosphaera xanthiiColletotrichum lagenarium. The method of claim 1 , wherein the fungal pathogen is selected from the group consisting of the causal agent of cucumber powdery mildew (or ) claim 1 , and cucumber anthracnose ().9Oryza sativa;. The method of claim 1 , wherein the seed being treated is a rice seed (ORYSP).10Pyricularia oryzae. The method of claim 1 , wherein the fungal pathogen is the causal agent of rice blast ().11. A plant seed adapted to produce a plant resistant to fungal and insect attack claim 1 , wherein the plant seed is treated with the compound of Formula I and one or more insecticides.12. A plant seed adapted to produce a plant resistant to fungal attack claim 1 , wherein the plant seed is treated with the compound of Formula I and one or ...

Подробнее
23-04-2015 дата публикации

5-FLUOROPYRIMIDINONE DERIVATIVES

Номер: US20150111851A1
Принадлежит:

This present disclosure is related to the field of 5-fluoropyrimidinones and their derivatives and to the use of these compounds as fungicides. 2. A composition for the control of a fungal pathogen including the compound of and a phytologically acceptable carrier material.3Venturia inaequalisSeptoria triticiCercospora beticolaCercospora arachidicolaCercosporidium personatumMycosphaerella fijiensis. The composition of wherein the fungal pathogen is Apple Scab () claim 2 , Leaf Blotch of Wheat () claim 2 , Leaf Spot of Sugarbeets () claim 2 , Leaf Spots of Peanut (and ) claim 2 , and Black Sigatoka of Banana ().4. (canceled)5. The compound of claim 1 , wherein:{'sup': '1', 'Ris: H;'}{'sup': '2', 'Ris H;'}{'sup': 3', '6', '7, 'sub': m', '2', '6, 'Ris —(CHR)OR, C-Calkenyl, cyclopropylmethyl, or (tetrahydrofuran-2-yl)methyl,'}wherein m is an integer 1-4;{'sup': '5', 'sub': 1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '2', '6', '2', '6', '2', '6', '1', '6, 'Ris independently halogen, C-Calkyl, C-Chaloalkyl, C-Calkoxy, C-Chaloalkoxy, C-Calkylthio, C-Chaloalkylthio, halothio, amino, C-Calkylamino, C-Cdialkylamino, C-Calkoxycarbonyl, C-Calkylcarbonyl, C-Calkylsulfonyl, nitro, hydroxyl, or cyano;'}{'sup': 6', '5, 'sub': 1', '6', '1', '6', '1', '6, 'Ris H, C-Calkyl, C-Calkoxy, C-Calkoxycarbonyl, phenyl or benzyl wherein each of the phenyl or the benzyl may be optionally substituted with 1-3 R; and'}{'sup': 7', '5', '5', '5, 'sub': 1', '8', '2', '6', '3', '6', '1', '6', '1', '6', '2', '6', '2', '6', '2', '6', '1', '6, 'Ris H, C-Calkyl, C-Calkenyl, C-Calkynyl, C-Chaloalkyl, C-Calkoxyalkyl, C-Ctrialkylsilyl, C-Ctrialkylsilylalkyl C-Calkylcarbonyl, C-Calkoxycarbonyl, benzyl, phenyl or benzyl wherein each of the phenyl or the benzyl may be optionally substituted with 1-3 R, or with a 5- or 6-membered saturated or unsaturated ring system, or with a 5-6 fused ring system, or with a 6-6 fused ring system each containing 1-3 heteroatoms wherein each ring may be ...

Подробнее
03-07-2014 дата публикации

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20140187588A1
Принадлежит:

The disclosure relates to macrocyclic picolinamides of Formula (I) and to the use of these compounds as fungicides. 2. The composition according to wherein X and Y are independently chosen from H or C(O)R.3. The composition according to wherein X and Y are C(O)Rand Ris independently chosen from alkyl claim 2 , alkoxy claim 2 , benzyl claim 2 , or benzyloxy claim 2 , each substituted with 0 claim 2 , 1 claim 2 , or multiple R claim 2 , wherein each Rmay be substituted with 0 claim 2 , 1 claim 2 , or multiple R.4. The composition according to wherein Rand Rare independently chosen from H claim 3 , alkyl claim 3 , alkenyl claim 3 , aryl claim 3 , or —C(O)R claim 3 , each substituted with 0 claim 3 , 1 or multiple R.5. The composition according to wherein Ris alkoxy and Rand Rare H.6. The composition according to wherein Ris tert-butoxy.7. The composition according to wherein X and Y are hydrogen.8. The composition according to wherein Rand Rare independently chosen from H claim 7 , alkyl claim 7 , alkenyl claim 7 , aryl claim 7 , or —C(O)R claim 7 , each substituted with 0 claim 7 , 1 or multiple R.9. The composition according to wherein Rand Rare independently alkyl claim 8 , alkenyl claim 8 , aryl claim 8 , or —C(O)R claim 8 , each substituted with 0 claim 8 , 1 or multiple R.10. The composition according to wherein Rand Rare independently alkyl claim 9 , or aryl claim 9 , each substituted with 0 claim 9 , 1 or multiple R.1110. The composition according to claim 9 , claim 9 , and wherein the amine is protonated to give an ammonium salt of a mineral acid independently chosen from hydrogen chloride claim 9 , hydrogen bromide claim 9 , or hydrogen iodide.12. The composition according to wherein the ammonium salt is the ammonium hydrochloride.13. The composition according to wherein X is H and Y is Q.14. The composition according to wherein Rand Rare independently chosen from H claim 13 , alkyl claim 13 , alkenyl claim 13 , aryl claim 13 , or —C(O)R claim 13 , each ...

Подробнее
03-07-2014 дата публикации

SYNERGISTIC FUNGICIDAL COMPOSITIONS

Номер: US20140187590A1
Принадлежит: DOW AGROSCIENCES LLC

A synergistic fungicidal mixture contains a fungicidally effective amount of a compound of Formula I, (3S,6S,7R,8R)-8-benzyl-3-(3-((isobutyryloxy)methoxy)-4-methoxypicolinamido)-6-methyl-4,9-dioxo-1,5-dioxonan-7-yl isobutyrate, and at least one triazole fungicide wherein Formula I is 2. The mixture of claim 1 , wherein the at least one triazole fungicide is selected from the group consisting of tebuconazole claim 1 , propiconazole claim 1 , metconazole claim 1 , and cyproconazole.3. The mixture of wherein the at least one triazole fungicide is tebuconazole and wherein the weight ratio of Compound I to tebuconazole is between about 1:16 and about 64:1.4. The mixture of wherein the at least one triazole fungicide is propiconazole and wherein the weight ratio of Compound I to propiconazole is between about 1:64 and about 64:1.5. The mixture of wherein the at least one triazole fungicide is metconazole and wherein the weight ratio of Compound I to metconazole is between about 1:4 and about 16:1.6. The mixture of wherein the at least one triazole fungicide is cyproconazole and wherein the weight ratio of Compound I to cyproconazole is between about 1:16 and about 64:1.7. The mixture of which further comprises an agriculturally acceptable adjuvant or carrier.9. The method of claim 8 , wherein the at least one triazole fungicide is selected from the group consisting of tebuconazole claim 8 , propiconazole claim 8 , metconazole claim 8 , and cyproconazole.10. The method of which further comprises mixing an agriculturally acceptable adjuvant or carrier with the compound of Formula I and at least one triazole fungicide prior to applying. This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/747,464 filed Dec. 31, 2012, which is expressly incorporated by reference herein.This disclosure concerns a synergistic fungicidal composition containing a fungicidally effective amount of a compound of Formula I and at least one triazole.Fungicides are ...

Подробнее
02-04-2020 дата публикации

Synergistic Fungicidal Mixtures and Compositions Comprising 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1h)-One for Fungal Control

Номер: US20200100500A1
Принадлежит: ADAMA MAKHTESHIM LTD.

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of epoxiconazole claim 1 , cyproconazole claim 1 , myclobutanil claim 1 , metconazole claim 1 , propiconazole claim 1 , prothioconazole claim 1 , fluquinconazole claim 1 , flutriafol claim 1 , and difenoconazole.3. The mixture of in which the concentration ratio of the Compound of Formula I to prothioconazole is between about 1:21.6 and about 2:1.4. The mixture of in which the concentration ratio of the Compound of Formula I to epoxiconazole is between about 3.6:1 and about 20:1.5. The mixture of in which the concentration ratio of xe Compound of Formula I to cyproconazole is between about 1:3 and about 4.5:1.6. The mixture of in which the concentration ratio of the Compound of Formula I to myclobutanil is between about 1:27 and about 1:4.7. The mixture of in which the concentration ratio of the Compound of Formula I to metconazole is between about 2.2.1 and about 30:1.8. The mixture of in which the concentration ratio of the Compound of Formula I to difenoconazole is between about 120:1 and about 787:1.9. The mixture of in which the concentration ratio of the Compound of Formula I to propiconazole is between about 1:2.1 and about 30:1.10. The mixture of in which the concentration ratio of the Compound of Formula I to fluquinconzole is between about 1:1.3 and about 170:1.11. The mixture of in which the concentration ratio of the Compound of Formula I to flutriafol is between about 1:20.6 and about 5.1:1.12Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The ...

Подробнее
16-04-2020 дата публикации

Synergistic Fungicidal Mixtures and Compositions Comprising 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1H)-One for Fungal Control (SDHI)

Номер: US20200113182A1
Принадлежит: ADAMA MAKHTESHIM LTD.

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of fluxapyroxad claim 1 , benzovindiflupyr claim 1 , penthiopyrad claim 1 , isopyrazam claim 1 , boscalid claim 1 , and fluopyram.3. The mixture of in which the concentration ratio of the Compound of Formula I to fluxapyroxad is between about 4.4:1 and about 6.3:1.4. The mixture of in which the concentration ratio of the Compound of Formula I to benzovindiflupyr is between about 1:3 and about 7.9:1.5. The mixture of in which the concentration ratio of the Compound of Formula I to penthiopyrad is between about 1:4.3 and about 1:1.9.6. The mixture of in which the concentration ratio of the Compound of Formula I to isopyrazam is between about 1:1.3 and about 1:1.7. The mixture of in which the concentration ratio of the Compound of Formula I to boscalid is between about 1:13.2 and about 1:1.3.8. The mixture of in which the concentration ratio of the Compound of Formula I to fluopyram is between about 1:27.6 and about 1:3.6.9Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is one of Leaf Blotch of Wheat (; anamorph: ) claim 2 , Wheat Brown Rust () claim 2 , Stripe Rust (f. sp. ) claim 2 , Scab of Apple () claim 2 , Blister Smut of Maize () claim 2 , Powdery Mildew of Grapevine () claim 2 , Barley scald () claim 2 , Blast of Rice () claim 2 , Rust of Soybean () claim 2 , Glume Blotch of Wheat () claim 2 , Powdery Mildew of Wheat (f. sp. ) claim 2 , Powdery ...

Подробнее
16-04-2020 дата публикации

Synergistic Fungicidal Mixtures and Compositions Comprising 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1H)-One for Fungal Control (MSI)

Номер: US20200113183A1
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of chlorothalonil and mancozeb.3. The mixture of in which the concentration ratio of the Compound of Formula I to chlorothalonil is about 1:219.4. The mixture of in which the concentration ratio of the Compound of Formula I to mancozeb is about 1:272.5Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is one of Leaf Blotch of Wheat (; anamorph: ) claim 2 , Wheat Brown Rust () claim 2 , Stripe Rust (f. sp. ) claim 2 , Scab of Apple () claim 2 , Blister Smut of Maize () claim 2 , Powdery Mildew of Grapevine () claim 2 , Barley scald () claim 2 , Blast of Rice () claim 2 , Rust of Soybean () claim 2 , Glume Blotch of Wheat () claim 2 , Powdery Mildew of Wheat (f. sp. ) claim 2 , Powdery Mildew of Barley (f. sp. ) claim 2 , Powdery Mildew of Cucurbits () claim 2 , Anthracnose of Cucurbits () claim 2 , Leaf Spot of Beet () claim 2 , Early Blight of Tomato () claim 2 , and Net Blotch of Barley ().6Mycosphaerella graminicolaSeptoria tritici. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is Leaf Blotch of Wheat (; anamorph: ).7Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe ...

Подробнее
23-04-2020 дата публикации

PICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20200120936A1
Принадлежит:

This disclosure relates to picolinamides of Formula I and their use as fungicides. 130-. (canceled)2. A method for the control and prevention of fungal attack on a plant , the method including the step of:{'claim-ref': {'@idref': 'CLM-00001', 'claim 1'}, 'applying a fungicidally effective amount of the compound of to at least one of the plant, an area adjacent to the plant, soil adapted to support growth of the plant, a root of the plant, and foliage of the plant.'} This application claims the benefit of U.S. Provisional Patent Application Ser. Nos. 62/098120 filed Dec. 30, 2014 and 62/098122 filed Dec. 30, 2014, which are expressly incorporated by reference herein.Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less.The present disclosure relates to picolinamides and their use as fungicides. The compounds of the present disclosure may offer protection against ascomycetes, basidiomycetes, deuteromycetes and oomycetes.One embodiment of the present disclosure may include compounds of Formula I:in which: X is hydrogen or C(O)R;wherein: Z is N or CH;Another embodiment of the present disclosure may include a fungicidal composition for the control or prevention of fungal attack comprising the compounds described above and a phytologically acceptable carrier material.Yet another embodiment of the present disclosure may include a method for the control or prevention of fungal attack on a plant, the method including the steps of applying a fungicidally effective amount of one or more of the compounds described above to at least one of the fungus, the plant, and an area adjacent to the plant.It will be understood by those skilled in the art that the following terms may include generic “R”-groups ...

Подробнее
03-06-2021 дата публикации

Synergistic Fungicidal Mixtures and Compositions Comprising 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1h)-One for Fungal Control (SBI)

Номер: US20210161138A1
Принадлежит: ADAMA MAKHTESHIM LTD.

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of epoxiconazole claim 1 , cyproconazole claim 1 , myclobutanil claim 1 , metconazole claim 1 , propiconazole claim 1 , prothioconazole claim 1 , fluquinconazole claim 1 , flutriafol claim 1 , and difenoconazole.3. The mixture of in which the concentration ratio of the Compound of Formula I to prothioconazole is between about 1:21.6 and about 2:1.4. The mixture of in which the concentration ratio of the Compound of Formula I to epoxiconazole is between about 3.6:1 and about 20:1.5. The mixture of in which the concentration ratio of the Compound of Formula I to cyproconazole is between about 1:3 and about 4.5:1.6. The mixture of in which the concentration ratio of the Compound of Formula I to myclobutanil is between about 1:27 and about 1:4.7. The mixture of in which the concentration ratio of the Compound of Formula I to metconazole is between about 2.2:1 and about 30:1.8. The mixture of in which the concentration ratio of the Compound of Formula I to difenoconazole is between about 120:1 and about 787:1.9. The mixture of in which the concentration ratio of the Compound of Formula I to propiconazole is between about 1:2.1 and about 30:1.10. The mixture of in which the concentration ratio of the Compound of Formula I to fluquinconazole is between about 1:1.3 and about 170:1.11. The mixture of in which the concentration ratio of the Compound of Formula I to flutriafol is between about 1:20.6 and about 5.1:1.12Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The ...

Подробнее
17-06-2021 дата публикации

Synergistic Fungicidal Mixtures and Compositions Comprising 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1H)-One for Fungal Control (MSI)

Номер: US20210176989A1
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of chlorothalonil and mancozeb.3. The mixture of in which the concentration ratio of the Compound of Formula I to chlorothalonil is about 1:219.4. The mixture of in which the concentration ratio of the Compound of Formula I to mancozeb is about 1:272.5Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is one of Leaf Blotch of Wheat (; anamorph: ) claim 2 , Wheat Brown Rust () claim 2 , Stripe Rust (f. sp. ) claim 2 , Scab of Apple () claim 2 , Blister Smut of Maize () claim 2 , Powdery Mildew of Grapevine () claim 2 , Barley scald () claim 2 , Blast of Rice () claim 2 , Rust of Soybean () claim 2 , Glume Blotch of Wheat () claim 2 , Powdery Mildew of Wheat (f. sp. ) claim 2 , Powdery Mildew of Barley (f. sp. ) claim 2 , Powdery Mildew of Cucurbits () claim 2 , Anthracnose of Cucurbits () claim 2 , Leaf Spot of Beet () claim 2 , Early Blight of Tomato () claim 2 , and Net Blotch of Barley ().6Mycosphaerella graminicolaSeptoria tritici. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is Leaf Blotch of Wheat (; anamorph: ).7Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe ...

Подробнее
17-06-2021 дата публикации

Synergistic Fungicidal Mixtures and Compositions Comprising 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1H)-One for Fungal Control (SDHI)

Номер: US20210176990A1
Принадлежит: ADAMA MAKHTESHIM LTD.

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of fluxapyroxad claim 1 , benzovindiflupyr claim 1 , penthiopyrad claim 1 , isopyrazam claim 1 , boscalid claim 1 , and fluopyram.3. The mixture of in which the concentration ratio of the Compound of Formula I to fluxapyroxad is between about 4.4:1 and about 6.3:1.4. The mixture of in which the concentration ratio of the Compound of Formula I to benzovindiflupyr is between about 1:3 and about 7.9:1.5. The mixture of in which the concentration ratio of the Compound of Formula I to penthiopyrad is between about 1:4.3 and about 1:1.9.6. The mixture of in which the concentration ratio of the Compound of Formula I to isopyrazam is between about 1:1.3 and about 1:1.7. The mixture of in which the concentration ratio of the Compound of Formula I to boscalid is between about 1:13.2 and about 1:1.3.8. The mixture of in which the concentration ratio of the Compound of Formula I to fluopyram is between about 1:27.6 and about 1:3.6.9Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is one of Leaf Blotch of Wheat (; anamorph: ) claim 2 , Wheat Brown Rust () claim 2 , Stripe Rust (f. sp. ) claim 2 , Scab of Apple () claim 2 , Blister Smut of Maize () claim 2 , Powdery Mildew of Grapevine () claim 2 , Barley scald () claim 2 , Blast of Rice () claim 2 , Rust of Soybean () claim 2 , Glume Blotch of Wheat () claim 2 , Powdery Mildew of Wheat (f. sp. ) claim 2 , Powdery ...

Подробнее
02-07-2015 дата публикации

USE OF MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20150181867A1
Принадлежит:

The invention relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. A composition according to claim 1 , wherein X is hydrogen and Y is Q.3. A composition according to claim 2 , wherein Ris hydrogen.4. A composition according to claim 3 , wherein Ris chosen from alkyl and aryl claim 3 , each optionally substituted with 0 claim 3 , 1 or multiple R.5. A composition according to claim 3 , wherein Ris chosen from alkyl claim 3 , aryl claim 3 , and acyl claim 3 , each optionally substituted with 0 claim 3 , 1 or multiple R.6. A composition according to claim 3 , wherein Ris chosen from alkyl and aryl claim 3 , each optionally substituted with 0 claim 3 , 1 or multiple R claim 3 , and Ris chosen from alkyl claim 3 , aryl claim 3 , and acyl claim 3 , each optionally substituted with 0 claim 3 , 1 or multiple R.7. A composition according to claim 2 , wherein Ris —C(O)Ror —CHOC(O)R.8. A composition according to claim 7 , wherein Ris chosen from alkyl and alkoxy claim 7 , each optionally substituted with 0 claim 7 , 1 claim 7 , or multiple R.9. A composition according to claim 8 , wherein Ris chosen from alkyl and aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.10. A composition according to claim 8 , wherein Ris chosen from alkyl claim 8 , aryl claim 8 , and acyl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.11. A composition according to claim 8 , wherein Ris chosen from alkyl and aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R claim 8 , and Ris chosen from alkyl claim 8 , aryl claim 8 , and acyl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.12. A composition according to claim 11 , wherein Ris chosen from —CHand —CHOCHCH.13. A composition for the control of a fungal pathogen including at least one of the compositions of and a phytologically acceptable carrier material.14. A composition for the control of a fungal pathogen including at least ...

Подробнее
02-07-2015 дата публикации

USE OF MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20150181868A1
Принадлежит:

The invention relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. A composition according to claim 1 , wherein X is hydrogen and Y is Q.3. A composition according to claim 2 , wherein Ris hydrogen.4. A composition according to claim 3 , wherein Ris chosen from alkyl and aryl claim 3 , each optionally substituted with 0 claim 3 , 1 or multiple R.5. A composition according to claim 3 , wherein Ris chosen from hydrogen claim 3 , alkyl claim 3 , aryl claim 3 , and acyl claim 3 , each optionally substituted with 0 claim 3 , 1 or multiple R.6. A composition according to claim 3 , wherein Ris chosen from alkyl and aryl claim 3 , each optionally substituted with 0 claim 3 , 1 or multiple R claim 3 , and Ris chosen from hydrogen claim 3 , alkyl claim 3 , aryl claim 3 , and acyl claim 3 , each optionally substituted with 0 claim 3 , 1 or multiple R.7. A composition according to claim 2 , wherein Ris —C(O)Ror —CHOC(O)R.8. A composition according to claim 7 , wherein Ris chosen from alkyl and alkoxy claim 7 , each optionally substituted with 0 claim 7 , 1 claim 7 , or multiple R.9. A composition according to claim 8 , wherein Ris chosen from alkyl and aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.10. A composition according to claim 8 , wherein Ris chosen from hydrogen claim 8 , alkyl claim 8 , aryl claim 8 , and acyl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.11. A composition according to claim 8 , wherein Ris chosen from alkyl and aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R claim 8 , and Ris chosen from hydrogen claim 8 , alkyl claim 8 , aryl claim 8 , and acyl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.12. A composition according to claim 11 , wherein Ris chosen from —CH claim 11 , —CHOCHCH claim 11 , and —CHCHOCH.13. A composition for the control of a fungal pathogen including at least one of the compositions of and a ...

Подробнее
02-07-2015 дата публикации

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20150181869A1
Принадлежит:

The invention relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. A compound according to claim 1 , wherein X and Y are hydrogen.3. A compound according to claim 2 , wherein Ris chosen from alkyl and aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.4. A compound according to claim 2 , wherein Ris chosen from hydrogen claim 2 , alkyl claim 2 , aryl claim 2 , and acyl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.5. A compound according to claim 2 , wherein Ris chosen from alkyl and aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R claim 2 , and Ris chosen from hydrogen claim 2 , alkyl claim 2 , aryl claim 2 , and acyl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.6. A compound according to claim 1 , wherein X is C(O)Rand Y is hydrogen.7. A compound according to claim 6 , wherein Ris chosen from alkyl and aryl claim 6 , each optionally substituted with 0 claim 6 , 1 or multiple R.8. A compound according to claim 6 , wherein Ris chosen from hydrogen claim 6 , alkyl claim 6 , aryl claim 6 , and acyl claim 6 , each optionally substituted with 0 claim 6 , 1 or multiple R.9. A compound according to claim 6 , wherein Ris chosen from alkyl and aryl claim 6 , each optionally substituted with 0 claim 6 , 1 or multiple R claim 6 , and Ris chosen from hydrogen claim 6 , alkyl claim 6 , aryl claim 6 , and acyl claim 6 , each optionally substituted with 0 claim 6 , 1 or multiple R.10. A compound according to claim 1 , wherein X is hydrogen and Y is Q.11. A compound according to claim 10 , wherein Ris hydrogen.12. A compound according to claim 11 , wherein Ris chosen from alkyl and aryl claim 11 , each optionally substituted with 0 claim 11 , 1 or multiple R.13. A compound according to claim 11 , wherein Ris chosen from hydrogen claim 11 , alkyl claim 11 , aryl claim 11 , and acyl claim 11 , each optionally substituted with 0 claim 11 , 1 or multiple ...

Подробнее
02-07-2015 дата публикации

SYNERGISTIC FUNGICIDAL MIXTURES FOR FUNGAL CONTROL IN CEREALS

Номер: US20150181874A1
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of epoxiconazole claim 1 , cyproconazole claim 1 , myclobutanil claim 1 , metconazole claim 1 , propiconazole claim 1 , prothioconazole claim 1 , fluquinconazole claim 1 , flutriafol claim 1 , and difenoconazole.3. The mixture of in which the concentration ratio of the Compound of Formula I to prothioconazole is between about 1:21.6 and about 2:1.4. The mixture of in which the concentration ratio of the Compound of Formula I to epoxiconazole is between about 3.6:1 and about 20:1.5. The mixture of in which the concentration ratio of the Compound of Formula I to cyproconazole is between about 1:3 and about 4.5:1.6. The mixture of in which the concentration ratio of the Compound of Formula I to myclobutanil is between about 1:27 and about 1:4.7. The mixture of in which the concentration ratio of the Compound of Formula I to metconazole is between about 2.2:1 and about 30:1.8. The mixture of in which the concentration ratio of the Compound of Formula I to difenoconazole is between about 120:1 and about 787:1.9. The mixture of in which the concentration ratio of the Compound of Formula I to propiconazole is between about 1:2.1 and about 30:1.10. The mixture of in which the concentration ratio of the Compound of Formula I to fluquinconazole is between about 1:1.3 and about 170:1.11. The mixture of in which the concentration ratio of the Compound of Formula I to flutriafol is between about 1:20.6 and about 5.1:1.12Mycosphaerella graminicola;Septoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The ...

Подробнее
02-07-2015 дата публикации

SYNERGISTIC FUNGICIDAL MIXTURES FOR FUNGAL CONTROL IN CEREALS

Номер: US20150181875A1
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of fluxapyroxad claim 1 , benzovindiflupyr claim 1 , penthiopyrad claim 1 , isopyrazam claim 1 , boscalid claim 1 , and fluopyram.3. The mixture of in which the concentration ratio of the Compound of Formula I to fluxapyroxad is between about 4.4:1 and about 6.3:1.4. The mixture of in which the concentration ratio of the Compound of Formula I to benzovindiflupyr is between about 1:3 and about 7.9:1.5. The mixture of in which the concentration ratio of the Compound of Formula I to penthiopyrad is between about 1:4.3 and about 1:1.9.6. The mixture of in which the concentration ratio of the Compound of Formula I to isopyrazam is between about 1:1.3 and about 1:1.7. The mixture of in which the concentration ratio of the Compound of Formula I to boscalid is between about 1:13.2 and about 1:1.3.8. The mixture of in which the concentration ratio of the Compound of Formula I to fluopyram is between about 1:27.6 and about 1:3.6.9Mycosphaerella graminicola;Septoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The mixtures of claim 1 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is one of Leaf Blotch of Wheat (anamorph: ) claim 1 , Wheat Brown Rust () claim 1 , Stripe Rust (f. sp. ) claim 1 , Scab of Apple () claim 1 , Blister Smut of Maize () claim 1 , Powdery Mildew of Grapevine () claim 1 , Barley scald () claim 1 , Blast of Rice () claim 1 , Rust of Soybean () claim 1 , Glume Blotch of Wheat () claim 1 , Powdery Mildew of Wheat (f. sp. ) claim 1 , Powdery ...

Подробнее
02-07-2015 дата публикации

SYNERGISTIC FUNGICIDAL MIXTURES FOR FUNGAL CONTROL IN CEREALS

Номер: US20150181883A1
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of chlorothalonil and mancozeb.3. The mixture of in which the concentration ratio of the Compound of Formula I to chlorothalonil is about 1:219.4. The mixture of in which the concentration ratio of the Compound of Formula I to mancozeb is about 1:272.5Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The mixture of claim 1 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is one of Leaf Blotch of Wheat (; anamorph: ) claim 1 , Wheat Brown Rust () claim 1 , Stripe Rust (f sp. ) claim 1 , Scab of Apple () claim 1 , Blister Smut of Maize () claim 1 , Powdery Mildew of Grapevine () claim 1 , Barley scald () claim 1 , Blast of Rice () claim 1 , Rust of Soybean () claim 1 , Glume Blotch of Wheat () claim 1 , Powdery Mildew of Wheat (f. sp. ) claim 1 , Powdery Mildew of Barley (f. sp. ) claim 1 , Powdery Mildew of Cucurbits () claim 1 , Anthracnose of Cucurbits () claim 1 , Leaf Spot of Beet () claim 1 , Early Blight of Tomato () claim 1 , and Net Blotch of Barley ().6Mycosphaerella graminicolaSeptoria tritici. The mixture of claim 1 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is Leaf Blotch of Wheat (; anamorph: ).7Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe ...

Подробнее
02-07-2015 дата публикации

MACROCYCLIC PICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY

Номер: US20150183759A1
Принадлежит:

The invention relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. A compound according to claim 1 , wherein X and Y are hydrogen.3. A compound according to claim 2 , wherein Ris chosen from alkyl and aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.4. A compound according to claim 2 , wherein Ris chosen from hydrogen claim 2 , alkyl claim 2 , aryl claim 2 , and acyl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.5. A compound according to claim 2 , wherein Ris chosen from alkyl and aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R claim 2 , and Ris chosen from hydrogen claim 2 , alkyl claim 2 , aryl claim 2 , and acyl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.6. A compound according to claim 1 , wherein X is C(O)Rand Y is hydrogen.7. A compound according to claim 6 , wherein Ris chosen from alkyl and aryl claim 6 , each optionally substituted with 0 claim 6 , 1 or multiple R.8. A compound according to claim 6 , wherein Ris chosen from hydrogen claim 6 , alkyl claim 6 , aryl claim 6 , and acyl claim 6 , each optionally substituted with 0 claim 6 , 1 or multiple R.9. A compound according to claim 6 , wherein Ris chosen from alkyl and aryl claim 6 , each optionally substituted with 0 claim 6 , 1 or multiple R claim 6 , and Ris chosen from hydrogen claim 6 , alkyl claim 6 , aryl claim 6 , and acyl claim 6 , each optionally substituted with 0 claim 6 , 1 or multiple R.10. A compound according to claim 1 , wherein X is hydrogen and Y is Q.11. A compound according to claim 10 , wherein Ris hydrogen.12. A compound according to claim 11 , wherein Ris chosen from alkyl and aryl claim 11 , each optionally substituted with 0 claim 11 , 1 or multiple R.13. A compound according to claim 11 , wherein Ris chosen from hydrogen claim 11 , alkyl claim 11 , aryl claim 11 , and acyl claim 11 , each optionally substituted with 0 claim 11 , 1 or multiple ...

Подробнее
09-07-2015 дата публикации

N1-SULFONYL-5-FLUOROPYRIMIDINONE DERIVATIVES

Номер: US20150191436A1
Принадлежит:

This present disclosure is related to the field of N1-sulfonyl-5-fluoropyrimidinones and their derivatives and to the use of these compounds as fungicides. 2. A composition for the control of a fungal pathogen including the compound of and a phytologically acceptable carrier material.3Venturia inaequalisSeptoria triticiCercospora beticolaCercospora arachidicolaCercosporidium personatumMycosphaerella fijiensis. The composition of wherein the fungal pathogen is Apple Scab () claim 2 , Leaf Blotch of Wheat () claim 2 , Leaf Spot of Sugarbeets () claim 2 , Leaf Spots of Peanut (and ) claim 2 , and Black Sigatoka of Banana ().4. A method for the control and prevention of fungal attack on a plant claim 2 , the method including the steps of:{'claim-ref': {'@idref': 'CLM-00001', 'claim 1'}, 'applying a fungicidally effective amount of at least one of the compounds of to at least one of the plant, an area adjacent to the plant, soil adapted to support growth of the plant, a root of the plant, foliage of the plant, and a seed adapted to produce the plant.'}5. The compound of claim 1 , wherein Ris selected from the group consisting of:H;{'sub': 1', '6, 'sup': '4', 'C-Calkyl optionally substituted with 1-3 R;'}{'sub': 1', '6, 'sup': '4', 'C-Calkenyl optionally substituted with 1-3 R;'}{'sub': 3', '6, 'sup': '4', 'C-Calkynyl optionally substituted with 1-3 R; and'}{'sup': 5', '5', '5, 'phenyl or benzyl wherein each of the phenyl or the benzyl may be optionally substituted with 1-3 R, or with a 5- or 6-membered saturated or unsaturated ring system, or with a 5-6 fused ring system, or with a 6-6 fused ring system each containing 1-3 heteroatoms wherein each ring may be optionally substituted with 1-3 R, biphenyl or naphthyl optionally substituted with 1-3 R.'}6. The compound of claim 1 , wherein Ris C-Calkyl optionally substituted with R. This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/232,204 filed Aug. 7, 2009.Fungicides are compounds, of ...

Подробнее
18-09-2014 дата публикации

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20140275171A1
Принадлежит:

The invention relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. A compound according to claim 1 , wherein:{'sub': '6', 'wherein, R is H, or C(O)R;'}{'sub': 1', '6, 'Ris C(O)R;'}{'sub': 2', '5, 'Ris independently or separately H, alkyl, alkenyl, aryl, each substituted with 0, 1 or multiple R;'}{'sub': '3', 'Ris independently or separately H, methyl;'}{'sub': '5', 'Ris alkyl, alkoxy, halo, haloalkyl, or aryl; and'}{'sub': '6', 'Ris alkoxy, or benzyloxy.'}5Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformisVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPseudoperonospora cubensisPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The compositions according to claim 4 , wherein the plant pathogen is least one pathogen selected from the group consisting of: Leaf Blotch of Wheat ( claim 4 , anamorph: ) claim 4 , Wheat Brown Rust () claim 4 , Stripe Rust () claim 4 , Scab of Apple () claim 4 , Blister Smut of Maize () claim 4 , Powdery Mildew of Grapevine () claim 4 , Barley scald () claim 4 , Blast of Rice () claim 4 , Downy Mildew of Cucurbits () claim 4 , Rust of Soybean () claim 4 , Glume Blotch of Wheat () claim 4 , Powdery Mildew of Wheat (f. sp. ) claim 4 , Powdery Mildew of Barley (f. sp. ) claim 4 , Powdery Mildew of Cucurbits () claim 4 , Anthracnose of Cucurbits () claim 4 , Leaf Spot of Beet () claim 4 , Early Blight of Tomato () claim 4 , and Net Blotch of Barley ().6Septoria triticiPuccinia triticinaPhakopsora pachyrhizi. The composition according to claim 5 , wherein the fungal pathogen is at least one of Leaf Blotch of Wheat () claim 5 , Wheat Brown Rust () claim 5 , and Rust of Soybean ().8. The method according to claim 7 , wherein the compound is applied in a mixture with at least one additional compound selected from ...

Подробнее
07-07-2016 дата публикации

N-(SUBSTITUTED)-5-FLUORO-4-IMINO-3-METHYL-2-OXO-3,4-DIHYDROPYRIMIDINE-1(2H)-CARBOXYLATE DERIVATIVES

Номер: US20160192653A1
Принадлежит:

This present disclosure is related to the field of N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxylates and their derivatives and to the use of these compounds as fungicides. Also provided are methods of controlling a fungal disease such as , comprising administering an effective amount of the fungicide compound to at lease one surface associated with the plant, seed or soil. 2. A composition for the control of a fungal disease , a comprising a composition for the control of at least one fungal disease , said composition including a fungicidally effective amount of the compound of Formula I and a phytologically acceptable carrier material.3Septoria tritici.. The composition of wherein the fungal disease is4. A method for the control and prevention of fungal attack on a plant claim 2 , the method including the steps of:applying a fungicidally effective amount of at least one of the compounds of Formula I to at least one surface selected from the group of surfaces selected from the group consisting of: a portion of a plant, an area adjacent to a plant, soil in contact with a plant, soil adjacent to a plant, any surface adjacent to a plant, any surface in contact with a plant, a seed, and equipment used in agriculture.5. The method of claim 1 , wherein the fungicidally effective amount Formula I is applied to a surface in the range of about 0.01 g/mto about 0.45 g/mof Formula I. This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/747,086 filed Dec. 28, 2012, which is expressly incorporated by reference herein.Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less.The present disclosure relates to N-(substituted)-5-fluoro-4 ...

Подробнее
05-07-2018 дата публикации

Picolinamides as fungicides

Номер: US20180186742A1
Принадлежит: DOW AGROSCIENCES LLC

This disclosure relates to picolinamides of Formula I and their use as fungicides.

Подробнее
05-07-2018 дата публикации

PICOLINAMIDES AS FUNGICIDES

Номер: US20180186743A1
Принадлежит: DOW AGROSCIENCES LLC

This disclosure relates to picolinamides of Formula I and their use as fungicides. 2. The composition according to claim 1 , wherein X is hydrogen and Y is Q.3. The composition according to wherein Z is N.4. The composition according to wherein W is O.5. The composition according to claim 4 , wherein Ris alkoxy.6. The composition according to claim 5 , wherein Ris hydrogen.7. The composition according to claim 6 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 6 , Rand R′ are independently chosen from C-Calkyl or taken together to form a 3-6 membered saturated carbocycle claim 6 , each optionally substituted with 0 claim 6 , 1 or multiple R claim 6 , and Ris aryl claim 6 , optionally substituted with 0 claim 6 , 1 or multiple R.8. The composition according to claim 5 , wherein Ris chosen from —C(O)R claim 5 , or —CHOC(O)R.9. The composition according to claim 8 , wherein Ris alkyl claim 8 , optionally substituted with 0 claim 8 , 1 or multiple R.10. The composition according to claim 9 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 9 , Rand R′ are independently chosen from C-Calkyl or taken together to form a 3-6 membered saturated carbocycle claim 9 , each optionally substituted with 0 claim 9 , 1 or multiple R claim 9 , and Ris aryl claim 9 , optionally substituted with 0 claim 9 , 1 or multiple R.11Zymoseptoria triticiPuccinia triticinaPuccinia striiformisVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisPyricularia oryzaePhakopsora pachyrhiziParastagonospora nodorumBlumeria graminis f.triticiBlumeria graminis f.hordeiErysiphe cichoracearumColletotrichum lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The composition according to wherein the fungal pathogen is one of Leaf Blotch of Wheat () claim 1 , Wheat Brown Rust () claim 1 , Stripe Rust () claim 1 , Scab of Apple () claim 1 , Blister Smut of Maize () claim 1 , Powdery Mildew of Grapevine () claim 1 , Barley scald () claim 1 , ...

Подробнее
14-07-2016 дата публикации

N-(SUBSTITUTED)-5-FLUORO-4-IMINO-3-METHYL-2-OXO-3,4-DIHYDROPYRIMIDINE-1(2H)-CARBOXAMIDE DERIVATIVES

Номер: US20160198711A1
Принадлежит:

This present disclosure is related to the field of to N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-di-hydropyrimidme-1(2H)-carboxamide compounds and their derivatives and to the use of these compounds as fungicides. This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/1746,837 filed Dec. 28, 2012, which is expressly incorporated by reference herein. Background and Summary of the Invention Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less. 2. The compound of claim 1 , wherein Ris thieno or phenyl claim 1 , and Ris H claim 1 , wherein the phenyl may be optionally substituted with 1-3 R.3. The compound of claim 2 , wherein Ris phenyl and each Ris independently selected from Calkyl claim 2 , halo claim 2 , Calkoxy claim 2 , Chaloalkyl claim 2 , and cyano.4. A composition for the control of a fungal disease claim 1 , a comprising a composition for the control of at least one fungal disease claim 1 , said composition including a fungicidally effective amount of the compound of Formula I of and a phytologically acceptable carrier material.5Septoria tritici.. The composition of wherein the fungal disease is6. A method for the control and prevention of fungal attack on a plant claim 4 , the method including the steps of:{'claim-ref': {'@idref': 'CLM-00001', 'claim 1'}, 'applying a fungicidally effective amount of at least one of the compounds of Formula I of to at least one surface selected from the group of surfaces selected from the group consisting of: a portion of a plant, an area adjacent to a plant, soil in contact with a plant, soil adjacent to a plant, any surface adjacent to a plant, any surface in contact with a plant, a seed, and equipment ...

Подробнее
02-10-2014 дата публикации

USE OF 5-FLUOROCYTOSINE AS A FUNGICIDE

Номер: US20140296065A1
Принадлежит:

The present disclosure is related to the field agrochemicals including 5-fluorocytosine and its derivatives and their use as fungicides. 16-. (canceled)7. A plant seed , comprising:a seed; anda fungicidally effective amount of 5-fluorocytosine or a 5-fluorocytosine derivative.8. The plant seed of claim 7 , wherein the 5-fluorocytosine or 5-fluorocytosine derivative is 5-fluorocytosine.9. The plant seed of claim 7 , wherein the 5-fluorocytosine or 5-fluorocytosine derivative has a concentration from about 0.1 to about 1000 parts per million.10. The plant seed of claim 7 , wherein the 5-fluorocytosine or 5-fluorocytosine derivative has a concentration from about 1 to about 500 parts per million.11. The plant seed of claim 7 , further comprising a second pesticidal compound.12. The plant seed of claim 11 , wherein the second pesticidal compound is selected from the group consisting of fungicides claim 11 , insecticides claim 11 , herbicides claim 11 , nematicides claim 11 , miticides claim 11 , arthropodicides claim 11 , bactericides claim 11 , or combinations thereof13. The plant seed of claim 11 , wherein the second pesticidal compound is an additional fungicide.13. The plant seed of claim 11 , wherein the weight ratio of the 5-fluorocytosine or 5-fluorocytosine derivative to the second pesticidal compound is from 1:100 to 100:1.14. A plant seedling claim 11 , comprisinga plant seedling; anda fungicidally effective amount of 5-fluorocytosine or a 5-fluorocytosine derivative.15. The plant seedling of claim 14 , wherein the 5-fluorocytosine or 5-fluorocytosine derivative is 5-fluorocytosine.16. The plant seedling of claim 14 , wherein the 5-fluorocytosine or 5-fluorocytosine derivative has a concentration from about 0.1 to about 1000 parts per million.17. The plant seedling of claim 14 , wherein the 5-fluorocytosine or 5-fluorocytosine derivative has a concentration from about 1 to about 500 parts per million.18. The plant seedling of claim 14 , further comprising a ...

Подробнее
16-08-2018 дата публикации

Picolinamide compounds with fungicidal activity

Номер: US20180228159A1
Принадлежит: DOW AGROSCIENCES LLC

This disclosure relates to picolinamides of Formula I and their use as fungicides.

Подробнее
16-07-2020 дата публикации

Synergistic Fungicidal Mixtures and Compositions Comprising 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1h)-One for Fungal Control (SBI)

Номер: US20200221698A1
Принадлежит: Adama Makhteshim Ltd

5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1H)-one, and at least one fungicide to provide synergistic control of selected fungi wherein the at least one fungicide is a fungicidal sterol biosynthesis-inhibitor.

Подробнее
23-07-2020 дата публикации

Synergistic Fungicidal Mixtures and Compositions Comprising 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1H)-One for Fungal Control (SDHI)

Номер: US20200229438A1
Принадлежит: ADAMA MAKHTESHIM LTD.

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of fluxapyroxad claim 1 , benzovindiflupyr claim 1 , penthiopyrad claim 1 , isopyrazam claim 1 , boscalid claim 1 , and fluopyram.3. The mixture of in which the concentration ratio of the Compound of Formula I to fluxapyroxad is between about 4.4:1 and about 6.3:1.4. The mixture of in which the concentration ratio of the Compound of Formula I to benzovindiflupyr is between about 1:3 and about 7.9:1.5. The mixture of in which the concentration ratio of the Compound of Formula I to penthiopyrad is between about 1:4.3 and about 1:1.9.6. The mixture of in which the concentration ratio of the Compound of Formula I to isopyrazam is between about 1:1.3 and about 1:1.7. The mixture of in which the concentration ratio of the Compound of Formula I to boscalid is between about 1:13.2 and about 1:1.3.8. The mixture of in which the concentration ratio of the Compound of Formula I to fluopyram is between about 1:27.6 and about 1:3.6.9Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia stritformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is one of Leaf Blotch of Wheat (; anamorph: ) claim 2 , Wheat Brown Rust () claim 2 , Stripe Rust (f. sp. ) claim 2 , Scab of Apple () claim 2 , Blister Smut of Maize () claim 2 , Powdery Mildew of Grapevine () claim 2 , Barley scald () claim 2 , Blast of Rice () claim 2 , Rust of Soybean () claim 2 , Glume Blotch of Wheat () claim 2 , Powdery Mildew of Wheat (f. sp. ) claim 2 , Powdery ...

Подробнее
09-09-2021 дата публикации

Synergistic Fungicidal Mixtures and Compositions Comprising 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1h)-One for Fungal Control (SBI)

Номер: US20210274785A1
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of epoxiconazole claim 1 , cyproconazole claim 1 , myclobutanil claim 1 , metconazole claim 1 , propiconazole claim 1 , prothioconazole claim 1 , fluquinconazole claim 1 , flutriafol claim 1 , and difenoconazole.3. The mixture of in which the concentration ratio of the Compound of Formula I to prothioconazole is between about 1:21.6 and about 2:1.4. The mixture of in which the concentration ratio of the Compound of Formula I to epoxiconazole is between about 3.6:1 and about 20:1.5. The mixture of in which the concentration ratio of the Compound of Formula I to cyproconazole is between about 1:3 and about 4.5:1.6. The mixture of in which the concentration ratio of the Compound of Formula I to myclobutanil is between about 1:27 and about 1:4.7. The mixture of in which the concentration ratio of the Compound of Formula I to metconazole is between about 2.2:1 and about 30:1.8. The mixture of in which the concentration ratio of the Compound of Formula I to difenoconazole is between about 120:1 and about 787:1.9. The mixture of in which the concentration ratio of the Compound of Formula I to propiconazole is between about 1:2.1 and about 30:1.10. The mixture of in which the concentration ratio of the Compound of Formula I to fluquinconazole is between about 1:1.3 and about 170:1.11. The mixture of in which the concentration ratio of the Compound of Formula I to flutriafol is between about 1:20.6 and about 5.1:1.12Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The ...

Подробнее
30-08-2018 дата публикации

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20180242582A1
Принадлежит:

This disclosure relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. The compound according to claim 1 , wherein X and Y are hydrogen.3. The compound according to claim 1 , wherein X is C(O)Rand Y is hydrogen.48.-. (canceled)9. A composition for the control of a fungal pathogen including at least one of the compounds of and at least one additional compound selected from the group consisting of: a phytologically acceptable carrier material claim 1 , a second fungicide claim 1 , an insecticide claim 1 , a nematocides claim 1 , a miticide claim 1 , an arthropodicide claim 1 , a bactericide.10. The composition for the control of a fungal pathogen according to claim 9 , wherein the at least one additional compound is at least one phytologically acceptable carrier material.11Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformisVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The compositions according to claim 9 , wherein the fungal pathogen is at least one pathogen selected from the group consisting of: Leaf Blotch of Wheat (; anamorph: ) claim 9 , Wheat Brown Rust () claim 9 , Stripe Rust () claim 9 , Scab of Apple () claim 9 , Blister Smut of Maize () claim 9 , Powdery Mildew of Grapevine () claim 9 , Barley Scald () claim 9 , Blast of Rice () claim 9 , Rust of Soybean () claim 9 , Glume Blotch of Wheat () claim 9 , Powdery Mildew of Wheat (f sp. ) claim 9 , Powdery Mildew of Barley (f. sp. ) claim 9 , Powdery Mildew of Cucurbits () claim 9 , Anthracnose of Cucurbits () claim 9 , Leaf Spot of Beet () claim 9 , Early Blight of Tomato () claim 9 , and Net Blotch of Barley ().12Septoria triticiPuccinia triticinaPhakopsora pachyrhizi. The composition according to wherein the fungal pathogen is ...

Подробнее
30-08-2018 дата публикации

Synergistic fungicidal mixtures for fungal control in cereals

Номер: US20180242583A1
Автор: Chenglin Yao, W. John OWEN
Принадлежит: DOW AGROSCIENCES LLC

A fungicidal composition containing a fungicidally effective amount of a compound of Formula I-V and at least one fungicide selected from the group consisting of epoxiconazole, prothioconazole, azoxystrobin, pyraclostrobin, penthiopyrad, isopyrazam, bixafen, boscalid, prochloraz, and chlorothalonil provides synergistic control of selected fungi.

Подробнее
06-08-2020 дата публикации

Synergistic Fungicidal Mixtures and Compositions Comprising 5-Fluoro-4-Imino-3-Methyl-1-Tosyl-3,4-Dihydropyrimidin-2(1H)-One for Fungal Control (MSI)

Номер: US20200245623A1
Принадлежит:

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of chlorothalonil and mancozeb.3. The mixture of in which the concentration ratio of the Compound of Formula I to chlorothalonil is about 1:219.4. The mixture of in which the concentration ratio of the Compound of Formula I to mancozeb is about 1:272.5Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is one of Leaf Blotch of Wheat (; anamorph: ) claim 2 , Wheat Brown Rust () claim 2 , Stripe Rust (f. sp. ) claim 2 , Scab of Apple () claim 2 , Blister Smut of Maize () claim 2 , Powdery Mildew of Grapevine () claim 2 , Barley scald () claim 2 , Blast of Rice () claim 2 , Rust of Soybean () claim 2 , Glume Blotch of Wheat () claim 2 , Powdery Mildew of Wheat (f. sp. ) claim 2 , Powdery Mildew of Barley (f. sp. ) claim 2 , Powdery Mildew of Cucurbits () claim 2 , Anthracnose of Cucurbits () claim 2 , Leaf Spot of Beet () claim 2 , Early Blight of Tomato () claim 2 , and Net Blotch of Barley ().6Mycosphaerella graminicola; anamorph: Septoria tritici. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is Leaf Blotch of Wheat ().7Mycosphaerella graminicola; anamorph: Septoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria ...

Подробнее
15-10-2015 дата публикации

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

Номер: US20150289508A1
Принадлежит:

The disclosure relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. The compound according to claim 1 , wherein:{'sub': 1', '3', '2', '3, 'Ris H, —C(O)R, or —CHOC(O)R;'}{'sub': 2', '5, 'Ris alkyl, alkenyl, or aryl, each substituted with 0, 1 or multiple R;'}{'sub': 3', '5, 'Ris alkyl or alkoxy, substituted with 0, 1, or multiple R;'}{'sub': 5', '6, 'Ris alkyl, alkenyl, halo, haloalkyl, alkoxy, haloalkoxy, arylalkoxy, cyano, aryl or heterocyclyl, each substituted with 0, 1 or multiple R; and'}{'sub': '6', 'Ris alkyl, alkenyl, halo, haloalkyl, alkoxy, haloalkoxy, arylalkoxy, cyano, aryl or heterocyclyl.'}3. A compound according to claim 3 , wherein:{'sub': 1', '3', '2', '3, 'Ris H, —C(O)R, or —CHOC(O)R;'}{'sub': 2', '5, 'Ris alkyl, alkenyl, or aryl, each substituted with 0, 1 or multiple R;'}{'sub': 3', '5, 'Ris alkyl or alkoxy, substituted with 0, 1, or multiple R; and'}{'sub': '5', 'Ris alkyl, halo, haloalkyl, or aryl.'}4. A compound according to claim 3 , wherein:{'sub': 1', '3', '2', '3, 'Ris H, —C(O)R, or —CHOC(O)R;'}{'sub': 2', '5, 'Ris alkyl, alkenyl, or aryl, each substituted with 0, 1 or multiple R;'}{'sub': '3', 'Ris alkyl; and'}{'sub': '5', 'Ris alkyl, halo, haloalkyl, or aryl.'}7Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformisMycosphaerella fujiensis. The compositions according to claim 6 , wherein the effective amount of the compound is effective against at least one plant pathogen selected from the group consisting of: Leaf Blotch of Wheat (; anamorph: ) claim 6 , Wheat Brown Rust () claim 6 , Stripe Rust () claim 6 , and Black Sigatoka ().8Septoria triticiPuccinia triticina. The composition according to claim 7 , wherein the plant pathogen is at least one organism selected from the group consisting of () and (). This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/643,623 filed May 7, 2012, which is expressly incorporated by reference herein.Fungicides are ...

Подробнее
12-09-2019 дата публикации

PICOLINAMIDES AS FUNGICIDES

Номер: US20190276404A1
Принадлежит: DOW AGROSCIENCES LLC

This disclosure relates to picolinamides of Formula I and their use as fungicides. 3. The compound according to claim 2 , wherein Rand Rare independently chosen from hydrogen or alkyl.4. The compound according to claim 2 , wherein Ris aryl claim 2 , optionally substituted with 0 claim 2 , 1 or multiple R.5. The compound according to claim 2 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 2 , and Ris aryl claim 2 , optionally substituted with 0 claim 2 , 1 or multiple R.7. The compound according to claim 6 , wherein Rand Rare independently chosen from hydrogen or alkyl.8. The compound according to claim 6 , wherein Ris aryl claim 6 , optionally substituted with 0 claim 6 , 1 or multiple R.9. The compound according to claim 6 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 6 , and Ris aryl claim 6 , optionally substituted with 0 claim 6 , 1 or multiple R.11. The compound according to wherein Z is N.12. The compound according to wherein W is O.13. The compound according to claim 12 , wherein Ris alkoxy.14. The compound according to claim 13 , wherein Ris hydrogen.15. The compound according to claim 14 , wherein Rand Rare independently chosen from hydrogen or alkyl.16. The compound according to claim 14 , wherein Ris aryl claim 14 , optionally substituted with 0 claim 14 , 1 or multiple R.17. The compound according to claim 14 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 14 , and Ris aryl claim 14 , optionally substituted with 0 claim 14 , 1 or multiple R.18. The compound according to claim 13 , wherein Ris chosen from —C(O)Ror —CHOC(O)R.19. The compound according to claim 18 , wherein Rand Rare independently chosen from hydrogen or alkyl.20. The compound according to claim 18 , wherein Ris aryl claim 18 , optionally substituted with 0 claim 18 , 1 or multiple R.21. The compound according to claim 18 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 18 , and Ris aryl claim 18 , ...

Подробнее
12-10-2017 дата публикации

Picolinamide compounds with fungicidal activity

Номер: US20170290333A1
Принадлежит: DOW AGROSCIENCES LLC

This disclosure relates to picolinamides of Formula I and their use as fungicides.

Подробнее
19-10-2017 дата публикации

USE OF PICOLINAMIDE COMPOUNDS AS FUNGICIDES

Номер: US20170295792A1
Принадлежит:

This disclosure relates to picolinamides of Formula I and their use as fungicides. 2. The composition according to claim 1 , wherein X is hydrogen and Y is Q.3. The composition according to claim 2 , wherein Z is N.4. The composition according to claim 3 , wherein Ris alkoxy.5. The composition according to claim 4 , wherein Ris hydrogen.6. The composition according to claim 5 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 5 , Rand Rare independently aryl claim 5 , each optionally substituted with 0 claim 5 , 1 or multiple R claim 5 , and Ris H.7. The composition according to claim 4 , wherein Ris chosen from —C(O)R claim 4 , or CHOC(O)R.8. The composition according to claim 7 , wherein Ris alkyl claim 7 , optionally substituted with 0 claim 7 , 1 or multiple R.9. The composition according to claim 8 , wherein Rand Rare independently chosen from hydrogen or alkyl claim 8 , Rand Rare independently aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R claim 8 , and Ris H.10. The composition according to claim 9 , wherein Ris chosen from —CH claim 9 , —CHOCHCH claim 9 , —CHCHOCH claim 9 , —CH(CH) claim 9 , —CHCHCHCH claim 9 , -cyclopropyl.11Zymoseptoria triticiPuccini triticinaPuccinia striiformisVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisPyricularia oryzaePhakopsora pachyrhiziLeposphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumColletotrichum lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. composition according to wherein the fungal pathogen is one of Leaf Blotch of Wheat () claim 1 , Wheat Brown Rust () claim 1 , Stripe Rust () claim 1 , Scab of Apple () claim 1 , Blister Smut of Maize () claim 1 , Powdery Mildew of Grapevine () claim 1 , Barley scald () claim 1 , Blast of Rice () claim 1 , Rust of Soybean () claim 1 , Glume Blotch of Wheat () claim 1 , Powdery Mildew of Wheat (f. sp. ) claim 1 , Powdery Mildew of Barley (f. sp. ) claim 1 , ...

Подробнее
25-10-2018 дата публикации

SYNERGISTIC FUNGICIDAL MIXTURES AND COMPOSITIONS FOR FUNGAL CONTROL

Номер: US20180303094A1
Принадлежит: ADAMA MAKHTESHIM LTD.

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of epoxiconazole claim 1 , cyproconazole claim 1 , myclobutanil claim 1 , metconazole claim 1 , propiconazole claim 1 , prothioconazole claim 1 , fluquinconazole claim 1 , flutriafol claim 1 , and difenoconazole.3. The mixture of in which the concentration ratio of the Compound of Formula I to prothioconazole is between about 1:21.6 and about 2:1.4. The mixture of in which the concentration ratio of the Compound of Formula I to epoxiconazole is between about 3.6:1 and about 20:1.5. The mixture of in which the concentration ratio of the Compound of Formula I to cyproconazole is between about 1:3 and about 4.5:1.6. The mixture of in which the concentration ratio of the Compound of Formula I to myclobutanil is between about 1:27 and about 1:4.7. The mixture of in which the concentration ratio of the Compound of Formula I to metconazole is between about 2.2:1 and about 30:1.8. The mixture of in which the concentration ratio of the Compound of Formula I to difenoconazole is between about 120:1 and about 787:1.9. The mixture of in which the concentration ratio of the Compound of Formula I to propiconazole is between about 1:2.1 and about 30:1.10. The mixture of in which the concentration ratio of the Compound of Formula I to fluquinconazole is between about 1:1.3 and about 170:1.11. The mixture of in which the concentration ratio of the Compound of Formula I to flutriafol is between about 1:20.6 and about 5.1:1.12Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The ...

Подробнее
25-10-2018 дата публикации

Synergistic fungicidal mixtures and compositions for fungal control

Номер: US20180303095A1
Принадлежит: Adama Makhteshim Ltd

5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1H)-one, and at least one fungicide to provide synergistic control of selected fungi, wherein the at least one fungicide is a succinate dehydrogenase-inhibitor.

Подробнее
25-10-2018 дата публикации

SYNERGISTIC FUNGICIDAL MIXTURES AND COMPOSITIONS FOR FUNGAL CONTROL

Номер: US20180303096A1
Принадлежит: ADAMA MAKHTESHIM LTD.

A fungicidal composition containing a fungicidally effective amount of the compound of Formula I: 2. The mixture of in which the at least one additional fungicide is selected from the group consisting of chlorothalonil and mancozeb.3. The mixture of in which the concentration ratio of the Compound of Formula I to chlorothalonil is about 1:219.4. The mixture of in which the concentration ratio of the Compound of Formula I to mancozeb is about 1:272.5Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe cichoracearumGlomerella lagenariumCercospora beticolaAlternaria solaniPyrenophora teres. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is one of Leaf Blotch of Wheat (; anamorph: ) claim 2 , Wheat Brown Rust () claim 2 , Stripe Rust (f. sp. ) claim 2 , Scab of Apple () claim 2 , Blister Smut of Maize () claim 2 , Powdery Mildew of Grapevine () claim 2 , Barley scald () claim 2 , Blast of Rice () claim 2 , Rust of Soybean () claim 2 , Glume Blotch of Wheat () claim 2 , Powdery Mildew of Wheat (f. sp. ) claim 2 , Powdery Mildew of Barley (f. sp. ) claim 2 , Powdery Mildew of Cucurbits () claim 2 , Anthracnose of Cucurbits () claim 2 , Leaf Spot of Beet () claim 2 , Early Blight of Tomato () claim 2 , and Net Blotch of Barley ().6Mycosphaerella graminicolaSeptoria tritici. The mixtures of - claim 2 , wherein the mixture provides control of a fungal pathogen and the fungal pathogen is Leaf Blotch of Wheat (; anamorph: ).7Mycosphaerella graminicolaSeptoria triticiPuccinia triticinaPuccinia striiformistriticiVenturia inaequalisUstilago maydisUncinula necatorRhynchosporium secalisMagnaporthe griseaPhakopsora pachyrhiziLeptosphaeria nodorumBlumeria graministriticiBlumeria graminishordeiErysiphe ...

Подробнее
12-11-2015 дата публикации

Macrocyclic picolinamides as fungicides

Номер: US20150322051A1
Принадлежит:

This disclosure relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. A compound according to claim 1 , wherein X and Y are hydrogen.3. A compound according to claim 2 , wherein Ris chosen from alkyl or aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.4. A compound according to claim 2 , wherein Ris chosen from alkyl or aryl claim 2 , each optionally substituted with 0 claim 2 , 1 or multiple R.5. A compound according to claim 1 , wherein X is C(O)Rand Y is hydrogen.6. A compound according to claim 5 , wherein Ris chosen from alkyl or aryl claim 5 , each optionally substituted with 0 claim 5 , 1 or multiple R.7. A compound according to claim 5 , wherein Ris chosen from alkyl or aryl claim 5 , each optionally substituted with 0 claim 5 , 1 or multiple R.8. A compound according to claim 1 , wherein X is hydrogen and Y is Q.9. A compound according to claim 8 , wherein Ris chosen from alkyl or aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.10. A compound according to claim 8 , wherein Ris chosen from alkyl or aryl claim 8 , each optionally substituted with 0 claim 8 , 1 or multiple R.11. A compound according to claim 9 , wherein Ris hydrogen.12. A compound according to claim 9 , wherein Ris —C(O)Ror —CHOC(O)R.13. A compound according to claim 12 , wherein Ris chosen from alkyl or alkoxy claim 12 , each optionally substituted with 0 claim 12 , 1 claim 12 , or multiple R.14. A compound according to claim 13 , wherein Ris chosen from —CH claim 13 , —CH(CH) claim 13 , —CHOCHCH claim 13 , or —CHCHOCH.15. A composition for the control of a fungal pathogen including at least one of the compounds of and a phytologically acceptable carrier material.16. A composition for the control of a fungal pathogen including mixtures of at least one of the compounds of with other pesticides including fungicides claim 1 , insecticides claim 1 , nematocides claim 1 , miticides claim 1 , arthropodicides claim 1 ...

Подробнее
03-12-2015 дата публикации

1-(SUBSTITUTED-BENZOYL)-5-FLUORO-4-IMINO-3-METHYL-3,4-DIHYDROPYRIMIDIN-2(1H)-ONE DERIVATIVES

Номер: US20150342188A1
Принадлежит:

This present disclosure is related to the field of 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-ones and their derivatives and to the use of these compounds as fungicides. Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less. The present disclosure relates to 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one compounds and their use as fungicides. The compounds of the present disclosure may offer protection against fungi and fungi like organisms including ascomycetes, basidiomycetes, deuteromycetes, and oomycetes. 3. A composition for the control of a fungal disease , a comprising a composition for the control of at least one fungal disease , said composition including a fungicidally effective amount of the compound of Formula I and a phytologically acceptable carrier material.4Septoria tritici.. The composition of wherein the fungal disease is5. A method for the control and prevention of fungal attack on a plant claim 3 , the method including the steps of:{'claim-ref': {'@idref': 'CLM-00001', 'claim 1'}, 'applying a fungicidally effective amount of at least one of the compounds of Formula (I) of to at least one surface selected from the group of surfaces selected from the group consisting of: a portion of a plant, an area adjacent to a plant, soil in contact with a plant, soil adjacent to a plant, any surface adjacent to a plant, any surface in contact with a plant, a seed, and equipment used in agriculture.'}6. The method of claim 5 , wherein the fungicidally effective amount Formula I is applied to a surface in the range of about 0.01 g/mto about 0.45 g/mof Formula I. This application claims the benefit of U.S. Provisional ...

Подробнее
23-11-2017 дата публикации

Macrocyclic picolinamides as fungicides

Номер: US20170334934A1
Принадлежит: DOW AGROSCIENCES LLC

This disclosure relates to macrocyclic picolinamides of Formula I and their use as fungicides. 2. A compound according to claim 1 , wherein X and Y are hydrogen.3. A compound according to claim 2 , wherein Ris alkyl claim 2 , aryl claim 2 , or acyl each optionally substituted with 0 claim 2 , 1 or multiple R.4. A compound according to claim 2 , wherein Ris chosen from —(CH)Rwhere n is an integer between 0 and 4 and Ris hydrogen or alkyl claim 2 , optionally substituted with 0 claim 2 , 1 or multiple R.5. A compound according to claim 1 , wherein X is C(O)Rand Y is hydrogen.6. A compound according to claim 5 , wherein Ris chosen from hydrogen claim 5 , alkyl claim 5 , aryl claim 5 , acyl claim 5 , or silyl each optionally substituted with 0 claim 5 , 1 or multiple R.7. A compound according to claim 5 , wherein Ris chosen from —(CH)Rwhere n is an integer between 0 and 4 and Ris hydrogen or alkyl claim 5 , optionally substituted with 0 claim 5 , 1 or multiple R.8. A compound according to claim 1 , wherein X is hydrogen and Y is Q.9. A compound according to claim 8 , wherein Ris chosen from alkyl claim 8 , aryl claim 8 , or acyl each optionally substituted with 0 claim 8 , 1 or multiple R.10. A compound according to claim 8 , wherein Ris chosen from —(CH)Rwhere n is an integer between 0 and 4 and Ris hydrogen or alkyl claim 8 , optionally substituted with 0 claim 8 , 1 or multiple R.11. A compound according to and claim 8 , wherein Ris hydrogen.12. A compound according to and claim 8 , wherein Ris —C(O)Ror —CHOC(O)R.13. A compound according to claim 12 , wherein Ris chosen from alkyl or alkoxy claim 12 , each optionally substituted with 0 claim 12 , 1 claim 12 , or multiple R.14. A compound according to claim 13 , wherein Ris chosen from —CHor —CH(CH).15. A composition for the control of a fungal pathogen including at least one of the compounds of - and a phytologically acceptable carrier material.16. A composition for the control of a fungal pathogen including mixtures ...

Подробнее
10-12-2015 дата публикации

N-(SUBSTITUTED)-5-FLUORO-4-IMINO-3-METHYL-2-OXO-3,4-DIHYDROPYRIMIDINE-1(2H)-CARBOXAMIDE DERIVATIVES

Номер: US20150353506A1
Принадлежит:

This present disclosure is related to the field of to N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-di-hydropyrimidine-1(2H)-carboxamide compounds and their derivatives and to the use of these compounds as fungicides. This application claims the benefit of U.S. Provisional Patent Application Ser. No. 61/746,837 filed Dec. 28, 2012, which is expressly incorporated by reference herein. Background and Summary of the Invention Fungicides are compounds, of natural or synthetic origin, which act to protect and/or cure plants against damage caused by agriculturally relevant fungi. Generally, no single fungicide is useful in all situations. Consequently, research is ongoing to produce fungicides that may have better performance, are easier to use, and cost less. 2. The compound of claim 1 , wherein Ris thieno or phenyl claim 1 , and Ris H claim 1 , wherein the phenyl may be optionally substituted with 1-3 R.3. The compound of claim 2 , wherein Ris phenyl and each Ris independently selected from Calkyl claim 2 , halo claim 2 , Calkoxy claim 2 , Chaloalkyl claim 2 , and cyano.4. A composition for the control of a fungal disease claim 1 , a comprising a composition for the control of at least one fungal disease claim 1 , said composition including a fungicidally effective amount of the compound of Formula I of and a phytologically acceptable carrier material.5Septoria tritici.. The composition of wherein the fungal disease is6. A method for the control and prevention of fungal attack on a plant claim 4 , the method including the steps of:{'claim-ref': {'@idref': 'CLM-00001', 'claim 1'}, 'applying a fungicidally effective amount of at least one of the compounds of Formula I of to at least one surface selected from the group of surfaces selected from the group consisting of: a portion of a plant, an area adjacent to a plant, soil in contact with a plant, soil adjacent to a plant, any surface adjacent to a plant, any surface in contact with a plant, a seed, and equipment ...

Подробнее
17-12-2015 дата публикации

3-ALKYL-5-FLUORO-4-SUBSTITUTED-IMINO-3,4-DIHYDROPYRIMIDIN-2(1H)-ONE DERIVATIVES AS FUNGICIDES

Номер: US20150359225A1
Принадлежит:

This present disclosure is related to the field of 3-alkyl-5-fluoro-4-substituted-imino-3,4-5 dihydropyrimidin-2(1H)-ones and their derivatives and to the use of these compounds as fungicides. Also provided are methods of controlling a fungal disease such as , comprising administering an effective amount of the fungicide compound to at lease one surface associated with the plant, seed or soil. 2. A compound according to claim 1 , wherein Ris independently C-Calkyl claim 1 , C-Calkoxy claim 1 , C-Calkylthio claim 1 , hydroxyl claim 1 , or deuterium.3. A compound according to claim 1 , wherein Ris C-Calkyl claim 1 , C-Chaloalkyl claim 1 , phenyl or benzyl wherein each of the phenyl or the benzyl may be optionally substituted with 1-3 R.4. A compound according to claim 1 , wherein Ris independently halogen claim 1 , C-Calkyl claim 1 , C-Chaloalkyl claim 1 , C-Calkoxy claim 1 , C-Calkylthio claim 1 , or deuterium.5. A compound according to claim 1 , wherein Ris C-Calkyl claim 1 , C-Chaloalkyl claim 1 , phenyl or benzyl wherein each of the phenyl or the benzyl may be optionally substituted with 1-3 R.6. A compound according to claim 1 , wherein Ris independently halogen claim 1 , C-Calkyl claim 1 , C-Chaloalkyl claim 1 , C-Calkoxy claim 1 , C-Chaloalkoxy claim 1 , C-Calkylthio claim 1 , cyano claim 1 , or nitro.7. A compound according to claim 1 , wherein Ris phenyl optionally substituted with 1-3 Ror a 5- or 6-membered saturated or unsaturated ring containing 1-3 heteroatoms optionally substituted with 1-3 R.8. A compound according to claim 7 , wherein Ris independently halogen claim 7 , C-Calkyl claim 7 , C-Calkoxy claim 7 , C-Chaloalkoxy.9. A compound according to claim 1 , wherein Ris C-Calkyl.10. A compound according to claim 1 , wherein Ris C-Calkyl claim 1 , —C(═O)R claim 1 , or —C(═O)OR.11. A compound according to claim 10 , wherein Ris C-Calkyl or phenyl.12. A compound according to claim 11 , wherein Ris C-Calkyl.14. A compound according to claim 13 , wherein ...

Подробнее