20-03-2014 дата публикации
Номер: US20140080862A1
Принадлежит:
The present invention relates to novel aryloazol-2-yl-cyanoethylamino derivatives of formula (I): 3. The aryloazol-2-yl-cyanoethylamine of claim 2 , wherein{'sub': 2', '8', '9', '10', '11', '1', '6', '2', '6', '2', '6', '3', '7', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '3', '7', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '2', '1', '6', '2', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6, 'R, R, R, Rand Reach, independently of one another, is hydrogen, amino, amido, cyano, nitro, halogen, C-C-alkyl, C-C-alkenyl, C-C-alkynyl, C-C-cycloalkyl, hydroxy-C-C-alkyl, halo-C-C-alkyl, C-C-alkylthio, halo-C-C-alkylthio arylthio, C-C-alkoxy, phenoxy, C-C-alkoxy-C-C-alkoxy, C-C-cycloalkyloxy, halo-C-C-alkoxy, C-C-alkylcarbonyl, halo-C-C-alkylcarbonyl, C-C-alkylsulfinyl, halo-C-C-alkylsulfinyl, C-C-alkylsulfonyl, C-C-alkylamino, di(C-C-alkyl)amino, C-C-alkylcarbonylamino, C-C-alkylamino-C-C-alkoxy, di-C-C-alkylamino-C-C-alkoxy, C-C-alkylamino-C-C-alkyl, di-C-C-alkylamino-C-C-alkyl, amino-C-C-alkyl, formyl, HOC—, C-C-alkyl-OC—, unsubstituted or substituted aryl or unsubstituted or substituted phenoxy, whereby the substituents may each be independent of one another and are selected from the group consisting of cyano, nitro, halogen, C-C-alkyl, halo-C-C-alkyl, C-C-alkylthio, halo-C-C-alkylthio, arylthio, C-C-alkoxy, halo-C-C-alkoxy, C-C-alkylcarbonyl, halo-C-C-alkylcarbonyl, C-C-alkylsulfinyl, halo-C-C-alkylsulfinyl, C-C-alkylsulfonyl and halo-C-C-alkylsulfonyl;'}{'sub': 3', '4', '6, 'R, Rand Rare H;'}{'sub': '5', 'Ris methyl;'}{'sub': 7', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', '6', '1', ...
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