SELECTED SUBSTITUTED PYRAZOLE DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ B1 RECEPTOR ANTAGONISTS

18-11-2004 дата публикации

Номер:

WO2004099155A2

Автор: GAROFALO, Albert, W., TUNG, Jay, S., PLEISS, Michael, A., WU, Jing, WONE, David, W., G., GUINN, Ashley, C., DRESSEN, Darren, B., MARUGG, Jennifer, NEITZEL, Martin

Принадлежит: Elan Pharmaceuticals, Inc.

Контакты:

Номер заявки: US36-01-200455

Дата заявки: 30-04-2004

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Disclosed are compounds that are bradykinin B1 receptor antagonists and are useful for treating diseases, or relieving adverse symptoms associated with disease conditions, in mammals mediated by bradykinin B1 receptor. Certain of the compounds exhibit increased potency and are also expected to exhibit increased duration of action.

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CPC - классификация

A A6 A61 A61P A61P1 A61P1/A61P1/0 A61P1/04 A61P11 A61P11/A61P11/0 A61P11/02 A61P11/06 A61P15 A61P15/A61P15/0 A61P15/06 A61P17 A61P17/A61P17/0 A61P17/02 A61P19 A61P19/A61P19/0 A61P19/02 A61P2 A61P25 A61P25/A61P25/0 A61P25/00 A61P25/04 A61P25/06 A61P29 A61P29/A61P29/0 A61P29/00 A61P3 A61P31 A61P31/A61P31/0 A61P31/04 A61P4 A61P43 A61P43/A61P43/0 A61P43/00 C C0 C07 C07D C07D2 C07D23 C07D231 C07D231/C07D231/1 C07D231/16 C07D231/4 C07D231/40 C07D4 C07D40 C07D401 C07D401/C07D401/1 C07D401/12 C07D403 C07D403/C07D403/1 C07D403/12 C07D41 C07D417 C07D417/C07D417/1 C07D417/12

IPC - классификация

A A6 A61 A61P A61P1 A61P1/A61P1/0 A61P1/04 A61P2 A61P25 A61P25/A61P25/0 A61P25/06 A61P4 A61P43 A61P43/A61P43/0 A61P43/00 C C0 C07 C07D C07D2 C07D23 C07D231 C07D231/C07D231/1 C07D231/16 C07D231/4 C07D231/40 C07D4 C07D40 C07D401 C07D401/C07D401/1 C07D401/12 C07D403 C07D403/C07D403/1 C07D403/12 C07D41 C07D417 C07D417/C07D417/1 C07D417/12

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